Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
11/2009
11/05/2009WO2009134666A1 Indazole compounds as ccr1 receptor antagonists
11/05/2009WO2009133831A1 Phenylpropionic acid derivative and use thereof
11/05/2009WO2009133687A1 Cyclopentylacrylic acid amide derivative
11/05/2009WO2009133179A2 Method for the production of halogen-substituted 2-(aminomethylidene)-3- oxobutyric acid esters
11/05/2009WO2009133178A1 Process for preparing 2-(aminomethylidene)-4,4-difluoro-3-oxobutyric esters
11/05/2009WO2009132453A1 Cyclylamine derivatives as calcium channel blockers
11/05/2009WO2009077844A3 Inhibitors of biofilm formation of gram-positive and gram-negative bacteria
11/05/2009US20090275619 Amide Substituted Indazole and Benzotriazole Derivatives as Poly(ADP-Ribose)Polymerase (PARP) Inhibitors
11/05/2009US20090275617 such as 3-[(1S,3R)-3-fluorocyclopentylamino]methyl-5-(5-fluoro-6-methylpyridin-3-yl)-1-isopropyl-4-methyl-1H-pyrazole, having opioid receptor antagonistic activity, used analgesics or for the treatment of diabetes, neurodegenerative diseases, drug abuse, hypotension, schizophrenia , dementia or obesity
11/05/2009US20090275598 Conformationally constrained 3-(4-hydroxy-phenyl)-substituted-propanoic acids useful for treating metabolic disorders
11/05/2009US20090275588 Novel sulfonamide compounds
11/05/2009US20090275524 Novel hypocholesterolemic compounds
11/05/2009CA2722923A1 Indazole compounds as ccr1 receptor antagonists
11/05/2009CA2722733A1 Cyclopentylacrylamide derivative
11/05/2009CA2722704A1 Cyclylamine derivatives as calcium channel blockers
11/04/2009EP2113501A1 5-Methyl-1-(naphthalen-2-YL)-1H-Pyrazoles useful as sigma receptor inhibitors
11/04/2009EP1727804B1 N1 - ((pyrazol-1-ymethyl) -2-methylphenyl)- phatalamide derivatives and related compounds insecticides
11/04/2009EP1641465B1 Combinations of an aryl aniline beta-2 adrenergic receptor agonist and a corticosteroid
11/04/2009EP1617806B1 Selective spirocyclic glucocorticoid receptor modulators
11/04/2009CN101573339A Novel cannabinoid receptor ligands, pharmaceutical compositions containing them, and processes for their preparation
11/04/2009CN101573035A Herbicide containing benzoylpyrazole compound
11/03/2009US7612201 Pyrazole compounds
11/03/2009US7612106 Fused pyrazole derivatives and methods of treatment of metabolic-related disorders thereof
11/03/2009US7612105 3-arylphenyl sulfide derivative and insecticide and miticide
11/03/2009US7612069 Acyl guanidines as beta-secretase inhibitors
10/2009
10/29/2009WO2009131886A1 Processes for producing n-alkylpyrazole
10/29/2009WO2009131096A1 Compound having npy y5 receptor antagonist activity
10/29/2009WO2009131065A1 Long-chain fatty acid elongation enzyme inhibitor comprising arylsulfonyl derivative as active ingredient
10/29/2009WO2009130331A1 5-methyl-1-(naphthalen-2-yl)-1h-pyrazoles useful as sigma receptor inhibitors
10/29/2009WO2009130314A1 Process for the preparation of naphthalen-2-yl-pyrazol-3-one intermediates useful in the synthesis of sigma receptor inhibitors
10/29/2009WO2009130310A1 1-aryl-3-aminoalkoxy pyrazoles as sigma ligands enhancing analgesic effect of opioids and attenuating the dependency thereof
10/29/2009WO2009130242A1 Low molecular weight derivatives and use thereof in treatment of prostaglandin e synthase related diseases
10/29/2009WO2009106980A3 Indazole derivatives
10/29/2009WO2009035951A3 Soluble epoxide hydrolase inhibitors
10/29/2009US20090270460 Fxr agonists
10/29/2009US20090270365 such as N-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-2-(piperidin-1-ylmethyl)biphenyl-4-carboxamide, having vanilloid receptor 1 antagonistic activity, used as analgesics
10/29/2009US20090270361 Substituted pyrazole derivatives and use thereof
10/29/2009US20090270359 Substituted pyrazole derivatives
10/29/2009CA2722345A1 1-aryl-3-aminoalkoxy pyrazoles as sigma ligands enhancing analgesic effect of opioids and attenuating the dependency thereof
10/29/2009CA2722256A1 5-methyl-1-(naphthalen-2-yl)-1h-pyrazoles useful as sigma receptor inhibitors
10/29/2009CA2722250A1 Process for the preparation of naphthalen-2-yl-pyrazol-3-one intermediates useful in the synthesis of sigma receptor inhibitors
10/29/2009CA2722075A1 Long-chain fatty acyl elongase inhibitor comprising arylsulfonyl derivative as active ingredient
10/29/2009CA2721805A1 Processes for producing n-alkylpyrazole
10/29/2009CA2721576A1 Compound having npy y5 receptor antagonist activity
10/29/2009CA2720818A1 Substituted phenoxybenzamides
10/28/2009EP2112139A1 Process for the preparation of naphthalen-2-yl-pyrazol-3-one intermediates useful in the synthesis of sigma receptor inhibitors
10/28/2009EP2111394A1 Compounds with a combination of cannabinoid-cb1 antagonism and serotonin reuptake inhibition
10/28/2009EP1786779B1 4-arylazo-3,5-diamino-pyrazole compounds and use thereof
10/28/2009CN101568525A Cb1 receptor modulators
10/28/2009CN101565403A Preparation method of 1, 3-diphenyl-2-pyrazoline nano particle with laminar structure
10/28/2009CN101565344A Method for preparing aldehyde or alkone by oxygen catalysis and alcohol oxidation under mild condition
10/27/2009US7608739 2,3-Dihydrooxadiazoles such as 3-acetyl-5-(2,5-difluorophenyl)-2-phenyl-2,3-dihydro-1,3,4-oxadiazole and 3-[3-acetyl-5-(2,5-difluorophenyl)-2-phenyl-2,3-dihydro-1,3,4-oxadiazol-2-yl]-N,N-dimethylpropan-1-amine that are useful for treating cancer
10/27/2009US7608718 4,5-dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity
10/27/2009US7608635 Pyrazole compounds that modulate HSP90 activity
10/27/2009US7608633 1-(4-Octylphenoxy)-3-(pyrrol-1-yl)propan-2-one, for example; for preventing and treating diseases caused by an increased activity of this enzyme, such as inflammation, pain, fever, allergies, asthma, psoriasis and endotoxic shock
10/27/2009US7608632 Sulfonamide inhibitors of aspartyl protease
10/27/2009US7608631 1-(4-{3-[2,6-Dichloro-4-(3,3-dichloro-allyloxy)-phenoxy]-propoxy}-phenyl)-1H-pyrrole, for example; protecting soybean plants against pests such as caterpillars
10/27/2009US7608618 1-(2,2,2-trifluoroethanoyl)pyrrolidine-2-carboxylic acid [4-methoxy-3-(3-pyrazin-2-yl-ureido)phenyl]-amide; 4-Methoxy-N-(3-methylamino-propyl)-3-(3-pyrazin-2-yl-ureido)-benzamide; checkpoint kinase Chk1 inhibitor; chemosensitizing agents useful in the treatment of diseases related to DNA damage
10/27/2009US7608564 Herbicide; in crops such as wheat, rice, maize, soybeans and cotton they act against broad-leaved weeds and grass weeds without damaging the crop plants; compounds are based on 3-(5,5-disubstituted 2-isoxazolin-3-yl)benzoic acid, esters, thioesters and pyrazolyl ketones thereof
10/27/2009CA2493359C Novel polymorph of n-methyl-n-(3-{3-[2-thienylcarbonyl]-pyrazol-[1,5-.alpha.]-pyrimidin-7-yl}phenyl)acetamide and compositions and methods related thereto
10/27/2009CA2318976C Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives
10/22/2009WO2009128521A1 Cysteine protease inhibitor
10/22/2009WO2009127726A1 Novel microbiocides
10/22/2009WO2009127722A1 Novel microbiocides
10/22/2009WO2009127718A2 Novel microbiocides
10/22/2009WO2009127612A1 Novel pyrazole derivatives
10/22/2009WO2009127338A1 Oxo-heterocyclic substituted carboxylic acid derivates and the use thereof
10/22/2009US20090264468 Methods for treating a disease in which Rho kinase is involved
10/22/2009US20090264424 Vanilloid receptor ligands and their use in treatments
10/22/2009US20090264414 Amide Derivatives and Pharmaceutical Use Thereof
10/21/2009EP2109602A2 Tetracycline derivatives for the treatment of bacterial, viral and parasitic infections
10/21/2009EP1381366B9 Indole, azaindole and related heterocyclic amidopiperazine derivatives
10/21/2009CN101563347A Vasopressin V1a antagonists
10/21/2009CN101560191A Alpha-menaphthyl substituted spiro bis(oxazoline) ligands, synthetic method and application thereof in synthesizing pyrazolidine derivatives
10/20/2009US7605273 P38 map kinase inhibitors; inflammatory bowel disease, rheumatoid arthritis, psoriasis, multiple sclerosis, endotoxin shock, osteoporosis, Alzheimer's disease, and congestive heart failure
10/20/2009US7605272 N-{2-[2-(1H-indazol-3-yl)vinyl]-5-(4-methylpiperazin-1-ylmethyl)phenyl}-3-methylthiophene-2-carboxamide; type I insulin-like growth factor receptor inhibitors; anticarcinognenic agents; colon, pancreatic cancers; antitumor agents; hematopoietic tumors; industrial scale
10/20/2009US7605266 Azaindole inhibitors of Aurora kinases
10/20/2009US7605175 Inhibitors of cyclin-dependent kinases, compositions and uses related thereto
10/20/2009US7605111 Herbicides
10/15/2009WO2009125861A1 Cysteine protease inhibitor
10/15/2009WO2009124950A2 4-methyl-4,5-dihydro-1h-pyrazole-3-carboxamide useful as a cannabinoid cb1 neutral antagonist
10/15/2009WO2009015000A8 Pyrazole urea derivatives used as kinase inhibitors
10/15/2009US20090258912 N-(1-Alkyl-2-Phenylethyl)-Carboxamide Derivatives and Use Thereof as Fungicides
10/15/2009US20090258892 Fused pyrazole derivatives and methods of treatment of metabolic-related disorders thereof
10/15/2009US20090258884 Substituted amides
10/14/2009EP2108644A1 N-(methyl)-pyridin-2-amine derivatives for the treatment of diseases associated with amyloid or amyloid-like proteins
10/14/2009EP2108643A1 4-methyl-4, 5-dihydro-1H-pyrazole-3-carboxamide useful as a cannabinoid CB1 neutral antagonist
10/14/2009EP2108012A2 Substituted n-(4-cyano-1h-pyrazol-3-yl)methylamine derivatives, preparation thereof and therapeutic use thereof
10/14/2009EP1877367B1 Acetylene derivatives
10/14/2009EP1720829B1 Derivatives of heteroaryl-alkylcarbamates, preparation method thereof and use of same as faah enzyme inhibitors
10/14/2009CN101558058A Modulators of CB1 receptors
10/14/2009CN101558056A Process for production of anthranilamide compound
10/14/2009CN101558044A Process for preparing fluoromethyl-substituted heterocyclic compounds
10/14/2009CN101555257A Synthesizing method of 1-aryl-3, 5-dimethyl pyrazole-4-formic acid organotin derivatives and applications
10/14/2009CN101555228A Fipronil compound, preparation method and application thereof
10/14/2009CN100549003C 3-aminophenol derivatives and dyes that contain these compounds while serving to dye keratin fibers
10/14/2009CN100548989C Pyrazole derivatives and process for the production thereof
10/13/2009US7601859 Organometallic complexes
10/13/2009US7601847 Preparation and purification of 4-(indazol-3-yl)phenols
10/13/2009CA2560510C N-(1-arylpyrazol-4yl) sulfonamides and their use as parasiticides
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