Patents
Patents for C07D 223 - Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom (8,732)
02/2002
02/21/2002DE10038747A1 Simplified purification of alkenyl compounds to low APHA color indexes, involves at least two distillations with time gap of at least one day after the first distillation
02/20/2002CN1336915A Urea of N-heterocyclic carboxylic acid or the isostere of carboxylic acid and aminocarboxylic acid ester
02/14/2002WO2002012196A2 Lactam compounds and their use as inhibitors of serine proteases and method
02/14/2002WO2001051479A3 Tricyclic compounds with antiviral activity
02/14/2002US20020019540 Conformationally constrained compounds as pharmaceutical agents
02/14/2002US20020019389 3-(N-(5,6-dimethyl-2-methoxypyridin-3-yl)aminocarbonyl)-7,8-dimethoxy-1-phenyl-2,3,4,5-tetrahydro-3H-benzazepine, for example
02/14/2002DE10038007A1 Neue Amino-und Amido-Diphenylether für Arzneimittel New amino and amido diphenyl ether for drugs
02/14/2002CA2418995A1 Lactam compounds and their use as inhibitors of serine proteases and method
02/13/2002EP1179341A1 Remedies or preventives for diseases in association with chemokines
02/13/2002EP0861250B1 Amidine and isothiourea derivatives as inhibitors of nitric oxide synthase
02/12/2002US6346527 Guanidine derivatives
02/12/2002CA2067877C Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions in which they are present
02/07/2002WO2002010146A1 Carboxamide compounds and their use as antagonists of a human 11cby receptor
02/07/2002WO2002010139A1 Hexahydro-7-1h-azepin-2-yl-haxanoic acid derivatives as inhibitors of inducible nitric oxide synthase
02/07/2002US20020016337 Heterocyclic analgesic compounds and methods of use thereof
02/07/2002US20020016336 Treatment of rheumatoid and osteoarthritis, corneal, epidermal or gastric ulceration, tumor metastasis or invasion, periodontal disease and bone disease
02/07/2002US20020016010 Synthesis of compounds and libraries of compounds
02/07/2002CA2417638A1 Carboxamide compounds and their use as antagonists of a human 11cby receptor
02/07/2002CA2415851A1 Hexahydro-7-1h-azepin-2-yl-haxanoic acid derivatives as inhibitors of inducible nitric oxide synthase
02/06/2002EP0891325B1 Para-substituted phenylpropanoic acid derivatives as integrin antagonists
02/06/2002EP0882024B1 Retroviral protease inhibiting compounds
02/06/2002CN1078889C Non-pepitde tachykinin receptor antagonists
02/05/2002US6344486 Anticoagulants
02/05/2002US6344466 Antithrombotic activity, use in inhibiting loss of blood platelets, inhibiting formation of blood platelet aggregates, inhibiting formation of fibrin, anticoagulants
02/05/2002US6344450 Lactam compounds and their use as inhibitors of serine proteases and method
01/2002
01/31/2002WO2001014328A3 Substituted ureas as cell adhesion inhibitors
01/31/2002US20020013245 Cyclic carbamate, lactonoxy or lactam structure and/or oxime esters and inert porous carrier of given surface area; storage stable solid, free-flowing form
01/30/2002EP1175405A1 LACTAM INHIBITORS OF FXa AND METHOD
01/29/2002CA2089880C Process for producing azacycloalkane derivatives
01/24/2002WO2002006241A1 1, 2, 3, 5 -tetrahydrobenzo`c!azepin-4-one derivatives having muscarinic antagonist activity
01/24/2002WO2002006232A1 Cyclic amine phenyl beta-3 adrenergic receptor agonists
01/24/2002WO2002006220A1 Free-flowing flakes of vinyl caprolactam monomer and process for making same
01/24/2002WO2001056992A3 Dibenzo (b,f) azepine intermediates
01/24/2002WO2001023357A3 Fused cycloheptane and fused azacycloheptane compounds and their use as integrin receptor antagonists
01/24/2002US20020010329 Solvent extraction; purification; pouring melt of raw materials into solvent
01/24/2002US20020010172 Lactams as inhibitors of A-beta protein production
01/24/2002US20020010171 New compounds, their preparation and use
01/24/2002CA2416245A1 Cyclic amine phenyl beta-3 adrenergic receptor agonists
01/23/2002CN1332159A Prep. of N-(3-halogeno-propyl)-imino stilbene
01/23/2002CN1332158A Prep. of epsilon-hexanolactam
01/22/2002US6340753 Cationic quaternary ammonium compounds dehydrohalogenation of compounds to form amines
01/22/2002US6340752 Cleavage of thio group from carbonyl and conversion to lactam ester
01/22/2002CA2049882C Process for iodinating or brominating the alpha-methylenic carbon of a secondary amide
01/17/2002US20020007075 Neurological disorders including physically damaged nerves and neurodegenerative diseases, and for treating alopecia and promoting hair growth; Alzheimer's, Parkinson's disease; amyotrophic lateral sclerosis
01/16/2002EP1171438A1 Compounds, their preparation and use
01/16/2002CN1331673A Semihydrogenation method for dinitriles
01/16/2002CN1331074A Process for hydrorefining caprolactam
01/16/2002CN1077886C Amidino derivatives useful as nitric oxide synthase inhibitors
01/10/2002WO2002002531A1 Nonpeptide substituted spirobenzoazepines as vasopressin antagonists
01/10/2002WO2002002530A1 Gpr14 antagonist
01/10/2002WO2002002520A2 Compounds to treat alzheimer's disease
01/10/2002WO2002002512A2 Compounds to treat alzheimer's disease
01/10/2002WO2001025212A3 Cyclic biphenyls, method for the production thereof, and their use as medicaments
01/10/2002US20020004503 Viricides
01/10/2002US20020004501 Therapy for muscular disorders, urogenital disorders, gastrointestinal disorders, respiratory system disorders
01/10/2002US20020004500 Drug mixture for cardiovascular disorders
01/10/2002US20020004494 Muscular disorders, gastrointestinal disorders, respiratory system disorders
01/10/2002CA2414976A1 Gpr14 antagonistic agent
01/10/2002CA2410651A1 Compounds to treat alzheimer's disease
01/09/2002EP1170289A2 Retroviral protease inhibiting compounds
01/09/2002EP1169290A1 Process to separate linear alkyl 5-formylvalerate
01/09/2002EP1169041A2 Use of carbamic acid derivatives for the treatment of viral infections
01/09/2002CN1330631A Amide derivatives which are useful as cell factor inhibitors
01/03/2002WO2002000626A1 Fused azepine derivatives and their use as antidiuretic agents
01/03/2002DE10027514A1 Liganden von Integrinrezeptoren Ligands of integrin
01/03/2002CA2412555A1 Fused azepine derivatives and their use as antidiuretic agents
01/02/2002EP1167350A1 Process for producing epsilon-caprolactam
01/02/2002EP1165532A1 Antibacterial agents
01/02/2002EP0964847B1 Method for separating an imine from a mixture containing an amine and an imine
01/02/2002CN1329609A Tetrahydrobenza epine derivatives useful as modulators of dopamine D3 receptors (antipsychotic agents)
01/02/2002CN1328824A Compound for curing female sexual disorder
01/01/2002US6335329 Carboxylic acid substituted heterocycles, derivatives thereof and methods of use
01/01/2002US6335327 1-benzazepine derivatives; agonists or antagonists of vasopressin and/or oxytocin
01/01/2002CA2051830C Tricyclic heterocycles
12/2001
12/27/2001WO2001098273A1 Novel compounds
12/20/2001WO2001096331A1 Lactam inhibitors of factor xa and method
12/20/2001WO2001095911A1 Protease inhibitors
12/20/2001WO2001095856A2 Urea derivative useful as an anti-cancer agent and process for preparing same
12/20/2001DE10028950A1 High yield caprolactam production by catalytic hydrogenation of a cyanovaleric acid derivative, followed by catalytic cyclization of the aminocaproic acid derivative-containing mixture obtained
12/20/2001CA2412353A1 Protease inhibitors
12/20/2001CA2412216A1 Lactam inhibitors of factor xa and method
12/19/2001EP1163225A1 Compounds and methods for modulation of estrogen receptors
12/19/2001CN1327468A Organic electroluminescent element
12/19/2001CN1327383A Pharmaceutical for treatment of neurological and neuropsychiatric disorders
12/18/2001US6331640 Diaminopropionic acid derivatives
12/18/2001US6331624 Process for preparing 6-aminocaproamide
12/13/2001WO2001094304A1 Process for the production of sulfonic esters
12/13/2001WO2001094294A1 Fungicides
12/12/2001EP1161233A2 Lxr modulators
12/12/2001CN1326445A Certain substituted caprolactams, pharmaceutical compositions containing them and their use in treating tumors
12/12/2001CN1326439A Phenyl-substituted cyclic enaminones
12/12/2001CN1326438A Method for treating lactams and method for purifying lactam
12/12/2001CN1076017C Process for producing caprolactane
12/11/2001CA2213108C 2-aminobenzazapine derivatives
12/11/2001CA2200336C Processes and intermediates for preparing 3-amino-benzo(b)azepinones
12/11/2001CA2053709C Piperazine derivatives
12/06/2001WO2001092235A1 LACTAMS SUBSTITUTED BY CYCLIC SUCCINATES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
12/06/2001WO2001092226A1 Heterocyclic analgesic compounds and method of use thereof
12/06/2001WO2001051474A3 Polypharmacophoric agents
12/06/2001WO2001010847A8 Novel integrin receptor antagonists
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