Patents
Patents for C07D 223 - Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom (8,732)
04/2004
04/21/2004CN1146455C 1,2,4,5-tetrahydro-benzo[d] azepine compound
04/15/2004WO2004031248A1 Novel nitrosation polymer in organic synthesis
04/15/2004WO2004031155A1 ENANTIOSELECTIVE PROCESS FOR THE PREPARATION OF BOTH ENANTIOMERS OF 10,11-DIHYDRO-10-HYDROXY-5H-DIBENZ [b,f]AZEPINE-5-CARBOXAMIDE AND NEW CRYSTAL FORMS THEREOF
04/15/2004WO2004031154A1 Novel lactams and uses thereof
04/15/2004WO2004014391B1 Use of carboxamides for the treatment of tinnitus
04/15/2004CA2501237A1 Enantioselective process for the preparation of both enantiomers of 10,11-dihydro-10-hydroxy-5h-dibenz [b,f]azepine-5-carboxamide and new crystal forms thereof
04/15/2004CA2500754A1 Novel nitrosation polymer in organic synthesis
04/14/2004EP1131297B1 Certain substituted caprolactams, pharmaceutical compositions containing them and their use in treating tumors
04/14/2004EP1109781B1 Process to continuously prepare an aqueous mixture of epsilon-caprolactam and epsilon-caprolactam precursors
04/14/2004CN1145612C New 1-aza-2-alkyl-6-aryl-cyclanes compound, its producing process and medical composition containing them
04/08/2004WO2004028538A1 Small organic molecules that increase the activity of gelatinase a in ocular cells
04/08/2004WO2003068732A3 Benzenesulfonamide derivatives and their use as dopamine d3 and d2 receptor liga ds
04/08/2004US20040068017 Small organic molecules that increase the activity of Gelatinase A in ocular cells
04/08/2004US20040067981 Acetylcholinesterase inhibitor; Alzheimer's diseases, Hubtington disease, antidepressants
04/08/2004CA2500200A1 Small organic molecules that increase the activity of gelatinase a in ocular cells
04/07/2004CN1144788C Bicycle vasporession agonists
04/06/2004US6716977 Method for making caprolactam from impure ACN wherein ammonia and water are removed from crude caprolactam in a simple separation step and then THA is removed from the resulting caprolactam melt
04/01/2004WO2003066597A3 Guanidino compounds
04/01/2004US20040063725 Binding neuropeptide Y receptors; hypertension, angina, atherosclerosis, depression, anxiety, inflammation, allergies
04/01/2004US20040063699 Gpr14 antagonist
03/2004
03/31/2004CN1486309A Tetrahydroazepine derivatives useful as dopamine d3 receptor modulators (antipsychotic agents)
03/31/2004CN1486184A Lactam compound to inhibit beta-amyloid peptide release or synthesis
03/30/2004US6713476 Substituted cycloalkyls as inhibitors of a beta protein production
03/30/2004US6713471 Such as tert-butyl-1-methyl-6,7,9,12-tetrahydro-5h-pyrido-(4,3-b)(1,4) thiazepino(2,3,4-hi)indole-11(10h)-carboxylate; serotonin agonists and antagonists; central nervous system disorders
03/30/2004US6713467 Anticoagulants in treating and preventing cardiovascular diseases, as anti-inflammatory agents, and metastasis inhibitors in treating cancer
03/30/2004US6713036 Mixing feed stream and oxidant using small scale multilamination mixing to yield reactant stream having characteristic mixing time; reacting with characteristic reaction time in reaction zone in presence of catalyst
03/25/2004WO2004024702A1 Novel carboxamide compounds having an mch-antagonistic effect, medicaments containing said compounds, and methods for the production thereof
03/25/2004WO2003086306B1 5ht2c receptor modulators
03/25/2004WO2003082260A3 Tuberculosis treatment using pleuromutilin derivatives
03/25/2004US20040058912 Psychological disorders; eating disorders; dietetics
03/25/2004US20040058900 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
03/25/2004CA2496563A1 New carboxamide compounds having mch-antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture
03/24/2004EP1399431A2 Novel nitriles useful as reversible inhibitors of cysteine proteases
03/24/2004EP1399424A1 Method for preparation of 10,11-dihydro-10-hydroxy-5h-dibenz/b,f/azepine-5-carboxamide and 10,11-dihydro-10-0x0-5h-dibenz/b,f/azepine-5-carboxamide
03/24/2004CN1484636A Method for storing and transporting N-vinyl caprolactam
03/24/2004CN1484633A N (phenylsulphonyl) glycine derivatives and their therapentic use
03/24/2004CN1483725A Method for producing cycloheximide and technology thereof
03/24/2004CN1142916C Dopamine D1 receptor agonist compounds
03/24/2004CN1142911C Compounds with growth hormone releasing properties
03/24/2004CN1142907C Process to continuously prepare aqueous mixture of epsi-caprolacta and epsi caprolactam precursors
03/23/2004US6710058 Use as anticoagulant agents for therapy and prophylaxis ofthromboembolic disorders
03/18/2004WO2003079975A3 Process for the manufacture of optically active 3-substituted lactams by asymmetric hydrogenation of 3-alkylidenelactams
03/18/2004US20040053933 Ligands of melanocortin receptors and compositions and methods related thereto
03/18/2004US20040053920 Administering to a patient suffering from caspase mediated diseses, an effective amount of a mono,bi or tri-heterocyclic ring containing nitrogen atom attached to ester or thioester to form carbamate group, as caspase inhibitor
03/18/2004US20040053826 Uses of polypeptides
03/17/2004EP1397340A2 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors
03/17/2004EP1240140B1 Method for the production of n-alkenyl amides
03/17/2004EP1140936B1 Tricyclic inhibitors of poly(adp-ribose) polymerases
03/17/2004CN1142139C Hydrofinishing method of caprolactam
03/16/2004CA2096460C Dual action inhibitors
03/11/2004US20040049038 N-substituted with a methylene-bridged nonaromatic ring system, e.g., N-(2-(benzyloxy)-5,6,7,8,9,10-hexahydro-6,9-methanobenzo(a)(8)annulen-11-yl)-N'-(2,2,2-trifluoroethyl)-sulfamide; preventing or treating Alzheimer's Disease
03/11/2004US20040048851 Amidinophenylalanine derivatives as thrombin inhibitors
03/11/2004US20040048346 Synthesis of chiral intermediates useful in preparing pharmacologically active compounds
03/11/2004DE10238865A1 New carboxamides are melanin-concentrating hormone receptor antagonists, useful for treating e.g. metabolic diseases, diabetes, eating disorders, cardiovascular disease, emotional disorders, reproductive and memory disorders
03/10/2004EP1395560A1 2-oxo-piperidinyl- and 2-oxo-azepanyl alkanoic acid derivativ es for the treatment of epilepsy and other neurological disorders
03/10/2004CN2606105Y Electric foreign ions remover with caprolactam
03/10/2004CN1481380A Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists
03/10/2004CN1481377A Cyclic Beta-amino acid derivatives as inhibitors of matrix metalloproteases and TNF alhpa
03/10/2004CN1481358A Carboxylic acid amide derivatives and their use in treatment of thromboembolic diseases and tumours
03/10/2004CN1481241A Therapeutic combination of amlodipine and benazepril/benazeprilat
03/09/2004US6703501 Porous catalyst for preparing epsilon-caprolactam from cyclohexanone oxime in vapor phase, comprising layered silicate and metal oxides pillared between silicate layers, having specified interlayer distance and surface area
03/04/2004WO2004018432A1 Substituted azepines as histamine h3 receptor antagonists, preparation and therapeutic uses
03/04/2004WO2004017911A2 Protease inhibitors
03/04/2004US20040044201 Bone disorders; osteoporosis; oral diseases; antiarthritic agents
03/04/2004US20040044200 Method of preparing a 5H-dibenz(b,f)azepine-5-carboxamide
03/04/2004US20040043977 Alzheimer's disease
03/03/2004EP1394870A2 Organic light emitting device
03/03/2004EP1392317A2 Substituted 1-benzazepines and derivatives thereof
03/03/2004EP1392307A1 Tartrate salts of 5,8,14-triazatetracyclo[10.3.1.02,11.04,9]-hexadeca-2(11),3,5,7,9-pentaene
03/02/2004US6699988 By reacting phosgene and lactam in the presence of a non-nucleophilic aliphatic tertiary amine, such as n,n-diisopropylethylamine; high purity, good yields
02/2004
02/26/2004US20040038962 Treatment of nocturnal enuresis, nocturia, polyuria resulting from central diabetes insipidus, urinary incontinence or bleeding disorders such a hemophilia
02/26/2004US20040038858 Carboxamide derivatives and their use in the treatment of thromboembolic diseases and tumours
02/25/2004EP1390366A1 The citrate salt of 5,8,14,-triazatetracyclo(10.3.1.02,11.04,9)-hexadeca-2(11),3,5,7,9-pentaene
02/19/2004WO2004014391A1 Use of carboxamides for the treatment of tinnitus
02/19/2004WO2003086306A3 5ht2c receptor modulators
02/19/2004US20040034250 Nitrosylating (with nitrosyl tetrafluoroborate) in presence of base then hydrolyzing to give hydroxy-imino derivative, followed by hydrogenation; for production of benazepril
02/19/2004US20040034018 2-amino-trihydroindole or tetrahydronapthalene-2-yl derivatives, useful for disease state associated with smooth muscle disorders, such as gastrointestinal and urogenital disorders
02/19/2004US20040034015 Administering to a human patient suffering from addictive behavior associated with 5HT2C receptor modulation, a fused tetra or pentaheterocyclic compound containing nitrogen in the rings
02/19/2004US20040033986 Anti tubercular drug: compositions and methods
02/19/2004CA2494660A1 Use of carboxamides for the treatment of tinnitus
02/18/2004EP1389189A2 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
02/18/2004EP1389103A2 Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic agents
02/18/2004CN1476434A Novel compounds
02/12/2004WO2004013105A1 Crystalline polymorphic and amorphous forms of benazepril hydrochloride
02/12/2004WO2004012726A2 Methods for treatment and prevention of gastrointestinal conditions
02/12/2004US20040030129 NF-kappaB inhibitor comprising phenylmethyl benzoquinone as an active ingredient
02/12/2004US20040029905 Using codeine, hydrocodeine, meptazinol, tilidine, propoxyphene
02/12/2004US20040029863 Carboxylic acid substituted heterocycles, derivatives thereof and methods of use
02/12/2004US20040029862 Alzheimer's disease
02/12/2004CA2494284A1 Methods for treatment and prevention of gastrointestinal conditions
02/12/2004CA2492949A1 Crystalline polymorphic and amorphous forms of benazepril hydrochloride
02/10/2004US6689784 Controlling cell apoptosis
02/10/2004CA2180301C Substituted dihydrodibenzo/b,f/azepines, method of their preparation, their use in the treatment of some central nervous system disorders, and pharmaceutical compositions containing them
02/10/2004CA2176836C The preparation of caprolactam
02/05/2004WO2004011431A1 Pleuromutilin derivatives as antimicrobbials
02/04/2004EP1385826A1 Method for preparation of (s)-(+)- and (r)-(-)-10,11-dihydro-10-hydroxy-5h-dibenz/b,f/azepine-5-carboxamide
02/04/2004EP1385818A2 Biurethane derivatives
02/04/2004EP1385517A1 Novel oral general anesthetics and metabolitically resistant anticonvulsants
02/04/2004EP1098875B1 Method for cyclizing hydrolysis of an aminonitrile compound into lactam
02/03/2004US6686477 Multistep chemical synthesis, including asymmetric hydrogenation of a lactam-enamide to produce an intermediate that can be used to make unspecified pharmaceuticals
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