Patents
Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273)
05/2003
05/01/2003US20030083502 Preparation of 4-haloalkylnicotinic esters
05/01/2003US20030083500 Imidazonaphthyridines
05/01/2003US20030083489 Method of synthesizing polynucleotides using ionic liquids
05/01/2003US20030083476 Morphine-6-glucuronide synthesis
05/01/2003US20030083382 Orally administered dosage forms of GABA analog prodrugs having reduced toxicity
05/01/2003US20030083374 NAALADase inhibitors useful as pharmaceutical compounds and compositions
05/01/2003US20030083359 Treating pain, urinary incontinence and bladder overactivity; P2X receptors are cation-permeable ion channels
05/01/2003US20030083357 Oxime derivatives for the treatment of dyslipidemia and hypercholesteremia
05/01/2003US20030083356 Statine derivatives for the treatment of Alzheimer's disease
05/01/2003US20030083353 Beta-secretase inhibitors
05/01/2003US20030083345 Method of treatment and/or prevention of brain, spinal or nerve injury
05/01/2003US20030083341 2,3,5-Substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
05/01/2003US20030083335 CCR1 receptor antagonists; inhibitors of MIP-1 alpha (CCL3) binding to its receptor CCR1 found on inflammatory and immunomodulatory cells; macrophage inflammatory protein (MIP)
05/01/2003US20030083333 1,4-Disubstituted benzo-fused compounds
05/01/2003US20030083332 N-heterocyclic derivatives as NOS inhibitors
05/01/2003US20030083331 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity
05/01/2003US20030083312 Borating and demetallization by reacting a pyridine Grignard reagent with an alkoxydialkylborane or a trialkylborane; in situ preparing the pyridine Grignard reagent by reacting alkyl magnesium halide with a halopyridine
05/01/2003US20030083269 Nictoinamide adenine dinucleotide (NAD); microbiocides; antiseptics; plant safening agents; antibiotic resistance; agriculture; food treatment
05/01/2003US20030083267 For inhibiting the binding of ligands to antigens; prophylaxis and treatment of inflammatory and autoimmune diseases such as asthma, arthritis, psoriasis, transplantation rejection, multiple sclerosis, diabetes, and inflammatory bowel disease
05/01/2003US20030082631 Detecting modulator of peroxisome proliferator-activated receptor; obtain sample contain proxisome receptor, incubate with test agent, monitor sample for adjustment in receptor activity
05/01/2003CA2464256A1 Novel dipeptidyl peptidase iv (dp-iv) inhibitors as anti-diabetic agents
05/01/2003CA2464254A1 Inhibitors of post-proline cleaving proteases
05/01/2003CA2463290A1 Zwitterionic imides
04/2003
04/30/2003CN1414966A Process and intermediates for preparation of imidazolidinone alpha U protein antagonists
04/30/2003CN1414956A Substituted piperazine derivatives as MIP inhibitors
04/30/2003CN1414849A Carboxylic acid amides, medicaments containing these compounds and the use and preparation thereof
04/30/2003CN1107061C Chemotaxis cell factor receptor-3 receptor antagonists
04/30/2003CN1107054C Method of preparation and separation of 2,4'-dipyridyl derivatives and its application
04/30/2003CN1107049C Benzyloxy substituted aromatics and their use as fungicides and insecticides
04/29/2003US6555700 1,3-propane diol esters and ethers and methods for their use in drug delivery
04/29/2003US6555684 Pyrimidinyl compounds for treatment of central nervous system disorders
04/29/2003US6555663 Prodrugs for selective drug delivery
04/29/2003US6555580 Treating arteriosclerosis and hypercholesterolaemia
04/29/2003US6555577 Compounds, their preparation and use
04/29/2003US6555572 Benzylated PDE4 inhibitors
04/29/2003US6555570 Growth hormone secretagogous with improved bioavailability
04/29/2003US6555566 Methods and materials for treating and preventing inflammation of mucosal tissue
04/29/2003US6555562 2-Carboxybenzoyl-(N'-3,5-dichloroisonicotinoyl)-L-4aminophenyl alanine, for example; inhibit the binding of alpha-4 integrins to their ligands, use to treat immune or inflammatory disorders
04/29/2003US6555561 Diaminopyridine-containing thiourea inhibitors of herpes viruses
04/29/2003US6555557 2,3-disubstituted pyridine derivatives, process for the preparation thereof, drug compositions containing the same and intermediates for the preparation
04/29/2003CA2059069C Method for preparing n-fluoropyridinium salt
04/24/2003WO2003033490A1 Synthesis of 4-[(z)-(4-bromophenyl)(ethoxyimino)methyl]-1'-[2,4-dimethyl-1-oxido-3-pyridinyl)carbonyl]-4'methyl-1,4'bipiperidine
04/24/2003WO2003033484A1 Substituted piperazine cyclohexane carboxilic acid amides and the use thereof
04/24/2003WO2003033483A1 Biphenylcarboxylic amide derivatives as p38 kinase inhibitors
04/24/2003WO2003033471A1 Novel pyridone derivative and remedial agent for circulatory disease containing the same
04/24/2003WO2003033470A1 Arylsulfanyl and heteroarylsulfanyl derivatives for treating pain
04/24/2003WO2003033469A1 A process for preparing beta-ketoester compound
04/24/2003WO2003033468A1 PROCESS FOR PREPARATION OF (S)-α-HALOMETHYLPYRIDINE- METHANOL DERIVATIVES
04/24/2003WO2003033467A1 Nitroso diphenylamine derivatives as nitrogen monoxide generating agents
04/24/2003WO2003033461A1 Synthesis of oxygen-substituted benzocycloheptenes, used as valuable intermediate products for producing tissue-selective oestrogens
04/24/2003WO2003033457A1 Biphenyl-derivatives as p38-kinase inhibitors
04/24/2003WO2003032999A1 Alkyne matrix metalloproteinase inhibitors
04/24/2003WO2003032980A1 5'-carbamoyl-1,1'-biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors
04/24/2003WO2003032972A1 5’-carbamoyl-1,1-biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors
04/24/2003WO2003032971A1 5’-acylamino-1,1’-biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors
04/24/2003WO2003032970A1 5'-carbamoyl-2'-methyl-1,1'-biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors
04/24/2003WO2003032921A2 Treatment of neurodegenerative diseases and cancer of the brain
04/24/2003WO2003032912A2 Treatment of cns disorders using cns target modulators
04/24/2003WO2003016282A3 Substituted 1h-dihydropyrazoles, their preparation and use
04/24/2003WO2003000679A3 Herbicidal substituted pyridines, method for producing the same and their use as herbicidal agents and plant growth regulators
04/24/2003WO2002058690A3 Methods for the treatment of diseases using malonyl-coa decarbox ylase inhibitors
04/24/2003US20030078302 As carriers for delivering active agents such as peptides, drugs by administration, such as oral, subcutaneous, sublingual, and intranasal administration
04/24/2003US20030078287 For controlling plant and animal pests
04/24/2003US20030078276 Matrix metalloproteinase inhibitors
04/24/2003US20030078266 Powder of 30-90% a water-soluble cycloxygenase inhibitor, 5-60% of a buffer and 0-10% of other excipients
04/24/2003US20030078265 Inhibitors of nitric oxide synthase (nos)
04/24/2003US20030078264 Treating atherosclerosis and other coronary artery diseases
04/24/2003US20030078261 Prostaglandin agonists
04/24/2003US20030078259 Nicotinic acetylcholine receptor activators; treating neurodegenerative disorders
04/24/2003US20030078249 VLA-4 inhibitor compounds
04/24/2003US20030078236 Arylsulfanyl and heteroarylsulfanyl derivatives for treating pain
04/24/2003US20030078235 Treatment of central nervous system disorders; anticonvulsants, antiepileptics, neuroprotective agents and muscle relaxants
04/24/2003US20030077405 Liquid crystal compounds having bis(trifluoromethyl) phenyl rings, liquid crystal compositions and liquid crystal display devices
04/24/2003CA2464435A1 Synthesis of oxygen-substituted benzocycloheptenes, used as valuable intermediate products for producing tissue-selective oestrogens
04/24/2003CA2463579A1 Treatment of cns disorders using cns target modulators
04/24/2003CA2463511A1 Synthesis of 4-[(z)-(4-bromophenyl)(ethoxyimino)methyl]-1'-[2,4-dimethyl-1-oxido-3-pyridinyl)carbonyl]-4'methyl-1,4'bipiperidine
04/24/2003CA2463426A1 Substituted piperazine cyclohexane carboxilic acid amides and the use thereof
04/24/2003CA2462442A1 Alkyne matrix metalloproteinase inhibitors
04/23/2003EP1304322A2 Carboxylic acid compound and use thereof
04/23/2003EP1304108A2 Anti-arrhythmic composition and methods of treatment
04/23/2003EP1304101A1 Composition and method for use of pyridinium derivatives in cosmetic and therapeutic applications
04/23/2003EP1303509A1 Beta3 adrenergic agonists
04/23/2003EP1303503A2 Aniline derivatives
04/23/2003EP1303494A2 Potassium channel inhibitors
04/23/2003EP1303490A1 N-oxides as nk1 receptor antagonist prodrugs of 4-phenyl-pyridine derivatives
04/23/2003EP1303489A2 Alpha,alpha-dibromo-alpha-chloro-acetophenones as synthons
04/23/2003EP1303483A1 Novel thiourea derivatives and the pharmaceutical compositions containing the same
04/23/2003EP1303482A2 N-substituted-1-amino-1,1-dialkylcarboxylic acid derivatives
04/23/2003EP1303479A2 7-, 8- and 9-substituted tetracycline compounds
04/23/2003EP1303308A2 Aldosterone antagonist and cyclooxygenase-2 inhibitor combination therapy to prevent or treat inflammation-related cardiovascular disorders
04/23/2003EP1303271A1 Ophthalmic formulation of a selective cyclooxygenase-2 inhibitory drug
04/23/2003EP1303249A1 Antimycotic nail varnish composition
04/23/2003EP1100783B1 Improved method for producing 2-halopyridine-n-oxide
04/23/2003EP1007032B1 4-cyano-4-deformylsordaricin derivatives
04/23/2003EP0993442B1 Hydrazine derivatives
04/23/2003EP0980236B1 Colourant and method for producing temporary hair colours
04/23/2003EP0882715B1 Novel n-(unsubstituted or substituted)-4-substituted-6-(unsubstituted or substituted)phenoxy-2-pyridinecarboxamides or thiocarboxamides, processes for producing the same, and herbicides
04/23/2003EP0882712B1 Process for preparing acid salts of gamma-(piperidyl)butyric acid
04/23/2003CN1413208A Novel derivatives of 3-imino-1,2,-dithioles, method for producing them and pharmaceutical compositions containing the same
04/23/2003CN1413195A Immunoassay detection method for neonicotinyl insecticides