Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
06/1995
06/24/1995CA2138840A1 Epoxidation process and catalyst therefore
06/21/1995EP0658539A1 Excitatory amino acid receptor antagonists
06/21/1995CN1028988C Certain glyoxyl-cyclohexendions
06/15/1995WO1995015962A1 Substituted benzimidazole, processes for its preparation and its pharmaceutical use
06/15/1995WO1995015959A1 Tricyclic derivatives and their use in pharmaceuticals
06/15/1995WO1995015949A1 Tricyclic derivatives and their use in pharmaceuticals
06/15/1995WO1995015948A1 Novel 2-arylalkenyl-azacycloalkane derivatives as sigma receptor ligands, preparation method therefor and therapeutical use thereof
06/15/1995CA2177739A1 Novel 2-arylalkenyl-azacycloalkane derivatives as sigma receptor ligands, preparation method therefor and therapeutical use thereof
06/14/1995EP0657434A1 Arylsubstituted -alkoxy-1,4-dihydropyridin-5-carbonic acid esters with cerebral activity
06/14/1995EP0657433A1 Dihydropyridines with substituted esters showing cerebral activity
06/14/1995EP0657432A1 Phenyl-substituted 1,4-dihydropyridines with cerebral activity
06/14/1995EP0657431A1 4-Phenyl-3-substituted 1,4-dihydropyridine esters with cerebral activity
06/14/1995EP0657430A1 Isopropyl-(2-methoxyethyl)-4-(2-chloro-3-cyano-phenyl)-1,4-dihydro-2,6-dimethyl-piridine-3,5-dicarboxylate
06/14/1995EP0657429A1 Optically active 1,4-dihydropyridine compound and process for producing the same
06/14/1995EP0657428A1 Preparation of 3,4,4-trisubstitutedpiperidinyl-n-alkylcarboxylates and intermediates, useful as opioid antagonists
06/14/1995EP0657425A1 Process for the preparation of chiral aminoalcohols
06/14/1995EP0657029A1 Calcium receptor active molecules
06/14/1995EP0656887A1 Hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
06/14/1995DE4342194A1 New pyridine-3,5-di:carboxylic acid deriv.
06/13/1995US5424435 1-hydroxy-6-substituted-2-pyridones
06/13/1995US5424318 Treating dementia, cerebrovascular diseases
06/13/1995US5423998 Bleaching agent for detergent
06/11/1995CA2137524A1 Aryl-substituted alkoxycarbonyl-1,4-dihydropyridine-5- carboxylic acid esters
06/11/1995CA2137519A1 4-phenyl-3-substituted 1,4-dihydropyridine esters
06/11/1995CA2137518A1 Dihydropyridines with substituted esters
06/09/1995CA2137446A1 3-(phenylalkylaminoalkyloxy)-5-phenylpyrazole compounds, intermediates for their preparation and pharmaceutical compositions containing them
06/08/1995WO1995015309A1 Dp-iv-serine protease inhibitors
06/08/1995CA2178066A1 Dp-iv-serine protease inhibitors
06/07/1995EP0656348A2 Aceric acid derivatives as medicaments
06/07/1995EP0655996A1 Substituted benzylamino nitrogen containing non-aromatic heterocycles
06/07/1995EP0655950A1 Chiral catalysts and epoxidation reactions catalyzed thereby.
06/06/1995US5422358 Muscarinic receptor antagonists
06/06/1995US5422356 Piperidine opioid antagonists
06/06/1995US5422353 Tetrahydropyridine derivatives
06/06/1995CA1335815C Piperidine or azepine peroxy compounds and derivatives useful as bleaching agents
06/04/1995CA2136904A1 Excitatory amino acid receptor antagonists
06/01/1995WO1995014791A1 Design of drugs involving receptor-ligand-dna interactions
06/01/1995WO1995014688A1 Derivatives of 2,3,5,6-tetrafluorobenzoic acid and their use in combating pests
06/01/1995WO1995014468A1 Blocking utilization of tetrahydrobiopterin to block induction of nitric oxide synthesis
06/01/1995CA2177388A1 Design of drugs involving receptor-ligand-dna interactions
06/01/1995CA2176251A1 Blocking utilization of tetrahydrobiopterin to block induction of nitric oxide synthesis
05/1995
05/31/1995EP0655469A1 Functional oligomeric vinylformamides and vinylamines
05/31/1995EP0655439A2 5,6-Bicyclic glycoprotein IIb IIIa antagonists useful in inhibition of platelet aggregation
05/31/1995EP0655247A1 Use of vincristine for the evaluation of substances at the neuroral level
05/31/1995EP0655056A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
05/31/1995EP0573467B1 NEUROLEPTIC PERHYDRO-1H-PYRIDO 1,2-a]PYRAZINES
05/31/1995CN1028592C Substituted guanidine derivatives their preparation and use
05/30/1995US5420283 Reacting s-1-cyclohexylethylamine with a racemic mixture of 2-benzylsuccinic acid 4-(4-/n-tert-butoxycarbonylmethylamino/ piperidine)amide
05/30/1995US5420280 Chemical intermediates for analgesics
05/30/1995US5420272 7-(substituted)-8-(substituted)-9-](substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
05/30/1995US5420142 For treatment of cardiovascular conditions which require an increase in contractility of the heart
05/26/1995WO1995014027A1 Anti-viral guanidino-substituted compounds
05/26/1995WO1995014017A1 Non-peptide tachykinin receptor antagonists
05/26/1995WO1995014012A1 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents
05/26/1995WO1995014011A2 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents
05/26/1995CA2176760A1 Anti-viral guanidino-substituted compounds
05/26/1995CA2176735A1 Non-peptide tachykinin receptor antagonists
05/26/1995CA2176043A1 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents
05/26/1995CA2176041A1 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents
05/24/1995EP0654025A1 Method of preparing optically pure precursors of paroxetine
05/24/1995CN1028531C 2-oxa-1-oxo-8-azaspiro ¾4,5 decane derivatives, pharmaceutical compositions containing them and process for preparing same
05/24/1995CN1028521C Therapeutic agents
05/23/1995US5418241 Antiserotonin agents
05/18/1995WO1995013066A1 Pharmaceutical emulsion
05/18/1995CA2175564A1 Cathepsin d is an amyloidogenic protease in alzheimer's disease
05/17/1995EP0652866A1 Azacyclic compounds
05/17/1995EP0652750A1 Use of alpha,omega-dicarboxylic acids as fibrinogen reducers
05/17/1995EP0377633B1 Peroxide free radical initiators containing hindered amine light stabilizer groups
05/17/1995CN1102649A Piperidines and piperazines
05/17/1995CN1102640A Alpha, omega-diarylalkane derivatives, their preparation and their use in the treatment and prevention of circulatory diseases and psychosis
05/16/1995US5416216 Tetramethylpiperidine compounds for use as stabilizers for organic materials
05/16/1995US5416215 Oxidation of 2,2,6,6-tetramethylpiperidine and it's 4-position substituted derivatives using hydrogen peroxide in the presence of a metal salt
05/16/1995US5416117 Cyclopropenone derivatives
05/13/1995CA2134192A1 5, 6-bicyclic glycoprotein iib/iiia antagonists
05/11/1995WO1995012584A1 Novel benzoyl guanidines, their production and their use in medicaments
05/11/1995WO1995012578A1 Short-acting dihydropyridines
05/11/1995WO1995012577A1 Novel 4-piperidinyl substituted lactames as neurokinin 2 receptor antagonists for the treatment of asthma
05/11/1995WO1995012576A1 New cyclopropyl derivatives, preparation method thereof and applications
05/11/1995WO1995012394A1 Use of nitric oxide releasing compounds as protective agents in ischemia reperfusion injury
05/11/1995CA2175838A1 Novel benzoyl guanidines, their production and their use in medicaments
05/11/1995CA2175467A1 Use of nitric oxide releasing compounds as protective agents in ischemia reperfusion injury
05/11/1995CA2172377A1 Novel 4-piperidinyl substituted lactames as neurokinin 2-receptor antagonists for the treatment of asthma
05/10/1995EP0651744A1 4-(4-fluorophenylmethyl)-piperidines having sigma and d2-receptor affinity
05/10/1995EP0651639A1 Methods of using (+) cisapride for the treatment of gastro-esophageal reflux disease and other disorders
05/09/1995US5414089 Useful for modifying enzymes or proteins
05/09/1995US5413999 HIV protease inhibitors useful for the treatment of AIDS
05/09/1995US5413997 Triphenylmethane derivatives
05/04/1995WO1995011895A1 N-benzoyl-4-oxy/thio-2-substituted piperidines as substance-p receptor antagonists
05/03/1995EP0650477A1 Light-activable 1-(2-nitrobenzyl)-substituted 1,4-dihydropyridines
05/03/1995EP0650476A1 Peripheral vasodilating agent containing n-acylated 4-amino piperidine derivatives as active ingredients
05/03/1995EP0650475A1 4-amino-n --(4-methyl-4-piperidinyl)-2-methoxybenzamides
05/03/1995EP0650474A1 Novel piperidyl amides, sulfonamides and sulfoxamides as inhibitors of cholesterol biosynthesis
05/02/1995US5412096 Treatment of senile dementia, Alzheimer*s disease, cholinergic activators
05/02/1995US5411972 Arylamide derivatives for treating hyperlipemia
05/02/1995US5411971 N-alkylenepiperidino compounds, their enantiomers and pharmaceutical compositions
05/02/1995US5411970 Method of inhibiting lentivirus
04/1995
04/27/1995WO1995011234A1 Radiolabelled ligands for muscarinic receptors
04/27/1995WO1995011233A1 Substituted pyridine-2-ones and substituted pyridine-2-thiones as biocides
04/27/1995WO1995011231A1 Amidino derivatives useful as nitric oxide synthase inhibitors
04/27/1995WO1995011228A1 2,3-diaminopropionic acid derivative