Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
11/1995
11/23/1995WO1995031436A1 PROCESS AND DIASTEREOMERIC SALTS USEFUL FOR THE OPTICAL RESOLUTION OF RACEMIC α-[4-(1,1-DIMETHYLETHYL)PHENYL]-4-(HYDROXYDIPHENYLMETHYL)-1-PIPERIDINEBUTANOL AND DERIVATIVE COMPOUNDS
11/22/1995EP0683166A1 3-Indolylpiperidines
11/22/1995EP0682514A1 Use of topical anesthetics for the manufacture of a medicament for the treatment of bronchial asthma
11/22/1995CN1112104A Acetic acid derivatives
11/22/1995CN1030353C Nonlinear optical materials
11/21/1995US5468753 Use of a 1-(2-naphthylethyl)-4-(3-trifluoromethylphenyl)-1,2,3,6-tetrahydropyridine for the manufacture of a medicament for the treatment of cerebral and neuronal diseases
11/21/1995US5468746 Compounds active on the cardiovascular system
11/21/1995US5468733 For treating cancer
11/16/1995WO1995030661A1 Substituted aromatic thiocarboxylic acid amides and their use as herbicides
11/15/1995EP0682015A1 Piperidine derivates and anti-platelet agents containing the same
11/14/1995US5466698 Substituted tetrahydrophyridines and hydroxypiperidines as central nervous system agents
11/14/1995US5466684 7-(substituted)-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
11/09/1995WO1995029926A1 Guanidino-substituted compounds
11/09/1995WO1995029892A1 Hydroxamic acid and amino acid derivatives and their use as anti-arthritic agents
11/09/1995DE19500439A1 Substituierte aromatische Thiocarbonsäureamide Substituted aromatic Thiocarbonsäureamide
11/08/1995EP0680988A2 Carbamate compounds and coating compositions comprising same
11/08/1995EP0680952A1 Process for the preparation of optically pure 1,4-dihydropyridines
11/08/1995EP0680484A1 OPTICALLY ACTIVE $g(b)-AMINOALKOXYBORANE COMPLEX
11/08/1995EP0680470A1 Diarylalkyl piperidines useful as multi-drug resistant tumor agents.
11/08/1995EP0680469A1 Aminoacid derivates, medicaments containing these compounds and process for preparing the same
11/08/1995CN1111239A Preparation of 3,4,4-trisubstituted-piperidinyl-N-alkycarboxylates and intermediates
11/08/1995CN1111237A Preparation of amides and peptides
11/07/1995US5464840 Tricyclic derivatives, compositions and methods of use
11/07/1995US5464788 Tocolytic oxytocin receptor antagonists
11/02/1995WO1995029160A1 Cationic bleach activators
11/02/1995WO1995029158A1 Heterocyclylbenzonitriles
11/02/1995WO1995029155A1 Novel antitumour compounds with antimitotic activity
11/02/1995WO1995029152A1 Benzamide derivatives as vasopressin antagonists
11/02/1995WO1995028931A1 Spiro-substituted azacycles as neurokinin-3 antagonists
11/02/1995EP0679619A2 Process for cross-coupling of aromatic boron compounds with aromatic halogen compounds or perfluoroalkyl sulphonates
11/02/1995DE4414568A1 Heterocyclylbenzonitrile Heterocyclylbenzonitriles
11/02/1995CA2188031A1 Spiro-substituted azacycles as neurokinin-3 antagonists
10/1995
10/31/1995US5463122 Arylthio compounds
10/31/1995US5463105 Therapy for cardiovascular, nervous system disorders
10/31/1995US5463064 Vasodilating and hypotensive activity
10/31/1995US5463063 Preparation of thalidomide; inhibitor of tumor necrosis factor
10/31/1995US5463011 Allophanic acid derivatives from reacting amines with isocyanate components; anticoagulants; inhibits binding of fibrinogen to glycoprotein IIa/IIIb
10/31/1995US5462947 Nervous system disorders
10/31/1995US5462945 N-substituted trifluoromethylphenyltetrahydropyridines, process for the preparation thereof, intermediates in said process and pharmaceutical compositions containing them
10/26/1995WO1995028157A1 Use of alpha-1c specific compounds to treat benign prostatic hyperplasia
10/26/1995CA2187773A1 Use of alpha-1c specific compounds to treat benign prostatic hyperplasia
10/25/1995EP0678503A1 Delta-amino-gamma-hydroxy-omega-aryl alkanoic acid amides with enzyme especially renin inhibiting activities
10/24/1995US5461167 Heterocyclic compounds
10/24/1995US5461154 HIV protease inhibitors
10/24/1995US5461066 Antiarrthythmic agent
10/24/1995US5461059 Derivatives of terbutylphenyl-1-amino-4-hydroxybutane their preparation processes and the pharmaceutical compositions containing them
10/24/1995CA1337418C 4-aryl-4-piperiding (or pyrrolidine or hexahydroazepine) carbinols and heterocyclic analogs thereof
10/21/1995CA2147429A1 Piperidine derivatives and anti-platelet agents containing the same
10/19/1995WO1995027727A2 Process for peptide segment condensation
10/19/1995CA2186605A1 Process for peptide segment condensation
10/18/1995EP0677514A1 New cyclopropyl derivatives, preparation method thereof and applications
10/17/1995US5459270 Tachykinin antagonist for central nervous systum disorders and cardiovascular disorders
10/17/1995US5459151 N-acyl substituted phenyl piperidines as bronchodilators and antiinflammatory agents
10/13/1995CA2146818A1 Pipecolic acid derivatives; process for preparing them and their use as synthesis intermediates
10/12/1995WO1995026953A1 Benzoic acid compound and use thereof as medicine
10/12/1995WO1995025091A3 Nipecotic acid derivatives as antithrombic compounds
10/12/1995CA2186623A1 Benzoic acid compound and use thereof as medicine
10/11/1995EP0676200A2 Use of eliprodil and of its enantiomers in the preparation of medicaments for the treatment of peripheral neuropathies and or central neurodegenerative diseases
10/11/1995EP0675924A1 Cyclic-substituted unsymmetrical cyanine dyes
10/11/1995EP0654025A4 Method of preparing optically pure precursors of paroxetine.
10/11/1995CN1109875A Phenyl-substituted 1,4-dihydropyridines
10/11/1995CN1109874A Isopropyl 2-methoxyethyl 4-(2-chloro-3-cyano-phenyl)-1,4-dihydro-2,6-dimethyl-pyridine3,5-dicarboxylate
10/11/1995CN1029964C Novel N-(4-piperidinyl) bicyclic condensed 2-imiolazolamine derivatives
10/11/1995CN1029960C Neuroprotective 3-piperidino-4-hydroxychroman derivatives
10/10/1995USRE35059 Monomer for polycarbonates
10/10/1995US5457204 Tetraalkyl-4-(2,3-epoxypropoxy) piperidine compounds as stabilizers
10/10/1995US5457143 Stabilization of polymeric organic materials by using synergistic mixtures comprising sterically hindered cyclic amines and derivatives of 3-pyrazolidinone or 1,2,4-triazolidine-3,5-dione
10/10/1995US5457096 Antibiotic
10/10/1995CA1337295C Dihydropyridine derivatives and their preparation and pharmaceutical formulation
10/05/1995WO1995026338A1 Neurokinin receptor antagonists
10/05/1995WO1995026337A1 Novel carbamates and ureas as modifiers of multi-drug resistance
10/05/1995WO1995026336A1 N-(benzhydryloxyalkyl)-4-(carboxy/carbamoyl-methyl)-piperidine derivatives as antidepressants
10/05/1995WO1995026335A1 Novel n-arylaliphatic-n-alkyl-functionalised amides, method for their preparation and pharmaceutical compositions containing same
10/05/1995WO1995026325A2 Enhancement of the efficacy of drugs by deuteration
10/05/1995DE19509353A1 New 4-aminopiperidine cpds., useful in e.g. plant protection
10/05/1995CA2186460A1 N-(benzhydryloxyalkyl)-4-(carboxy/carbamoyl-methyl)-piperidine derivatives as antidepressants
10/05/1995CA2186371A1 Enhancement of the efficacy of dihydropyridines by deuteration
10/04/1995EP0675105A1 Polyiodinated compounds, process for their preparation and diagnostic composition
10/04/1995EP0674623A1 Bicyclic fibrinogen antagonists
10/04/1995EP0674514A1 Use of aryloxyalkyl substituted cyclic amines as calcium channel antagonists and new phenyloxyalkyl piperidin derivatives
10/03/1995US5455258 Useful as inhibitors of matrix-degrading metalloproteinase enzymes such as stromelysin and/or collegenase
10/03/1995US5455250 Treating central nervous system disorders
10/03/1995US5455246 Treating neuropsychiatric disorders
10/03/1995US5455243 Fibrinogen receptor antagonists for inhibiting aggregation of blood platelets
09/1995
09/28/1995WO1995025722A1 Separation of the enantiomers of amlodipine via their diastereomeric tartrates
09/28/1995WO1995025721A1 New 1,4-disubstituted piperidine derivatives useful as medicaments acting on the glutamate receptor
09/28/1995WO1995025720A1 Piperidyl-4-substituted thyrosine derivatives as scintigraphic imaging agents for the diagnosis of thrombosis
09/28/1995WO1995025443A1 Tocolytic oxytocin receptor antagonists
09/28/1995DE4410822A1 Neue Piperidin-Derivate New piperidine derivatives
09/28/1995CA2186129A1 Tocolytic oxytocin receptor antagonists
09/28/1995CA2186010A1 New 1,4-disubstituted piperidine derivatives useful as medicaments acting on the glutamate receptor
09/27/1995EP0673928A1 Novel N-(3,4-dichlorophenyl-propyl)-piperidine derivatives as selective human NK3-receptor antagonists
09/27/1995EP0673927A1 4-[2-indanyl-1-one]alkylpiperidines as anticholinergic agents
09/27/1995EP0673367A1 4-aminomethyl/thiomethyl/sulfonylmethyl-4-phenylpiperidines as tachykinin receptor antagonists
09/27/1995EP0673247A1 Fibrinogen receptor antagonists
09/27/1995EP0510003B1 Piperidine and pyrrolidine derivatives
09/27/1995CN1109051A 3-(phenylalkyl aminoalkyloxy)-5-phenlpyrazol, production, medium and pharmaceutical of same
09/26/1995US5453511 Bis-piperidinium compounds
09/26/1995US5453509 Functionalization of acyl pyridinium salts
09/26/1995US5453422 Animal growth promoters