Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
01/1996
01/17/1996EP0691956A1 3-phenyl-1,2,5,6-tetrahydropyridine derivatives as sedatives
01/17/1996EP0691955A1 Process for preparing 3-methylpiperidine and 3-methylpyridine by catalytic cyclisation of 2-methyl-1,5-diaminopentane
01/17/1996EP0691953A1 1-amidinophenyl-pyrrolidones piperidinones azetinones as platelet aggregation inhibitors
01/16/1996US5484926 HIV protease inhibitors
01/16/1996US5484799 Antifungal dorrigocin derivatives
01/16/1996US5484797 Naphthly compounds, intermediates, processes, compositions, and method for inhibiting endometrosis
01/16/1996US5484796 Naphthyl compounds, intermediates, processes, compositions, and method of inhibiting aortal smooth muscle cell proliferation
01/16/1996US5484795 Naphthyl compounds, intermediates, processes, compositions, and method of inhibiting restenosis
01/16/1996CA1337938C Hydrophilic modifier monomers
01/14/1996CA2153726A1 .alpha.-(4-chlorophenyl)-4-[(4-fluorophenyl)-methyl]piperidine-1- ethanol esters, their preparation and their therapeutic application
01/11/1996WO1996000720A1 Aryl and heteroaryl alkoxynaphthalene derivatives
01/11/1996DE4424294A1 Prodn. of poly:ene-carbonyl cpds. with high all-E content
01/11/1996DE4423445A1 Rapid high yield prodn. of nifedipin
01/10/1996EP0690844A1 Process to prepare herbicidal bicyclic triazoles
01/10/1996CN1114651A 3-indolylpiperidine
01/09/1996US5482986 Benzopyran compound and use of the same
01/09/1996US5482938 Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment
01/09/1996US5482921 Herbicides
01/09/1996CA1337909C Non-peptide renin inhibitors
01/04/1996WO1996000214A1 Arylsulfonamido-substituted hydroxamic acids as matrix metalloproteinase inhibitors
01/04/1996WO1996000064A1 Therapeutical compositions comprising 3-phenyl-3-hydroxypiperidines
01/04/1996WO1996000063A1 Utilisation of derivatives of 1,2,5,6-tetrahydropyridine for the preparation of sedative medicaments
01/04/1996CA2193695A1 Therapeutical compositions comprising 3-phenyl-3-hydroxypiperidines
01/04/1996CA2193397A1 Utilisation of derivatives of 1,2,5,6-tetrahydropyridine for the preparation of sedative medicaments
01/03/1996EP0690039A2 Poly-perfluoroalkyl-substituted alcohols and acids, and derivatives thereof
01/03/1996EP0689549A1 New urea derivates, their preparation and their use
01/03/1996EP0689536A1 Naphthalene derivatives
01/03/1996EP0619806B1 Preparation of substituted piperidines
01/02/1996US5481036 Renin inhibitors, hypotensive agents
12/1995
12/28/1995WO1995035309A1 New thrombin inhibitors, their preparation and use
12/28/1995WO1995035303A1 Synthesis of conduritol epoxides and aziridines and methods of using such to synthesize higher disaccharides
12/28/1995WO1995035280A1 Methods of synthesis of peptidyl argininals
12/28/1995CA2193133A1 Novel thrombin inhibitors, the preparation and use thereof
12/28/1995CA2192697A1 Methods of synthesis of peptidyl argininals
12/27/1995EP0688752A1 Trifluoro-2-(trans-4-substituted cyclohexyl) ethylenes and process for their production
12/27/1995EP0688317A1 Process for preparing acryl-piperidine carbinols
12/26/1995US5478942 Cyclic urea derivatives and pharmaceutical compositions containing these compounds
12/26/1995US5478848 Inhibition of arthritis by L-type calcium channel antagonists nimodipine, nisoldipine and nifedipine
12/26/1995US5478846 1-piperidinyl alkanoylanyl sulfonamides for treatment of cardiac arrhythmia
12/26/1995US5478828 Piperazinyl-and piperidinyl-cyclohexanols
12/26/1995CA1337817C Heterocyclic spiro compounds and methods for preparing the same
12/21/1995WO1995034539A1 4-carbamoyloxy-piperidine-1-carboxylic acid esters: inhibitors of cholesterol absorption
12/21/1995WO1995034530A1 2-acylaminopropanol compound and medicinal composition
12/21/1995CA2192459A1 4-carbamoyloxy-piperidine-1-carboxylic acid esters: inhibitors of cholesterol absorption
12/20/1995EP0687268A1 Spiroazacyclic derivatives as substance p antagonists
12/20/1995EP0687252A1 2-phenoxyethylamine derivatives, their preparation and their therapeutical use
12/20/1995EP0687249A1 Balanoids
12/20/1995CN1113454A Epoxidation process and catalyst therefore
12/20/1995CN1113437A A process for preparing a pharmaceutical composition containing benzothiazole compounds
12/19/1995US5476934 Oxidation a nitrogen-containing perfluoroacyl halide
12/19/1995US5476859 Antiviral compounds
12/19/1995CA1337764C 1,4-dihydropyridine derivatives and pharmaceutical composition thereof
12/14/1995WO1995033731A1 Hydroxamic acid derivatives
12/14/1995WO1995033729A1 Serotonin 5-ht1a and dopamin d2 receptor ligands
12/14/1995WO1995033723A1 Phenoxyalkyl substituted piperidines, pyrrolidines, morpholines and thiomorpholines as calcium channel antagonists
12/14/1995WO1995033722A1 Phenoxyalkyl substituted piperidines, pyrrolidines, morpholines and tiomorpholines as calcium channel antagonists
12/14/1995WO1995033721A1 4-aryl-1-(indanmethyl, dihydrobenzofuranmethyl or dihydrobenzothiophenemethyl)piperidines, tetrahydropyridines or piperazines
12/14/1995WO1995026325A3 Enhancement of the efficacy of drugs by deuteration
12/14/1995CA2192113A1 Serotonin 5-ht 1a and dopamin d2 receptor ligands
12/14/1995CA2192112A1 4-aryl-1-(indanmethyl, dihydrobenzofuranmethyl or dihydrobenzothiophenemethyl)piperidines, tetrahydropyridines or piperazines
12/13/1995EP0686642A2 Modified guanidino and amidino thrombin inhibitors
12/13/1995EP0686629A2 Cyclohexyl tachykinine receptor antagonists
12/13/1995EP0686625A1 Anthranilic acid derivative
12/13/1995EP0686151A1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors
12/13/1995EP0573473B1 4-[(2-benzothiazolyl)methylamino]-alpha-[(3,4-difluorophenoxy)methyl]-1-piperidineethanol
12/12/1995US5475132 Fungicide intermediates
12/12/1995US5475111 Process for the preparation of dihydropyridinecarboxylic acids
12/12/1995US5475109 Useful in prevention or treatment of infection by influenza virus
12/11/1995CA2151412A1 Modified guanidino and amidino thrombin inhibitors
12/11/1995CA2150992A1 Cyclohexyl tachykinin receptor antagonists
12/07/1995WO1995032947A1 Chiral compounds and their resolution
12/07/1995CA2191363A1 Chiral compounds and their resolution
12/06/1995EP0685465A1 Butine- or hexadiine linked hindered amines as stabilizer
12/06/1995EP0685457A1 Glycerol derivative, device and pharmaceutical composition
12/06/1995EP0685234A1 Drug composition containing nucleic acid copolymer
12/06/1995EP0684947A1 Amide compounds with pharmacological activity
12/06/1995EP0684816A1 5-ht 2? receptor antagonist compositions useful in treating venous conditions
12/06/1995CN1030452C Preparation of novel 2-aminopyrimidinone derivatives
12/06/1995CN1030450C Preparation of analgesic carboxylic acid amides derivative
12/05/1995US5473070 Substituted long chain alcohol xanthine compounds
12/05/1995US5472984 1,2-ethanediol derivative and salt thereof and cerebral function-improving agent comprising the same
12/05/1995US5472969 Administering N-alkyl-1,5-dideoxy-1,5-imino-D-glucitol
12/05/1995US5472966 Antidepressant heteroarylaminoalkyl derivatives of naphthyl-monazines
12/05/1995CA1337695C Process for the production of 4,5,6,7-tetrahydrothieno-¬3,2-c|-pyridines
12/03/1995CA2150644A1 Butyne-linked or hexadiyne-linked hindered amines as stabilisers
11/1995
11/30/1995WO1995032200A1 Oxathiolanes, method for their preparation and pharmaceutical compositions containing same
11/30/1995WO1995031977A1 Novel potent inducers of terminal differentiation and methods of use thereof
11/30/1995CA2167930A1 Oxathiolanes, method for their preparation and pharmaceutical compositions containing same
11/29/1995EP0684238A2 Process for the manufacture of dicarboxamides
11/29/1995EP0684233A1 Pipecolic acid derivatives, their preparation and use as intermediates
11/29/1995EP0684227A2 Process for the manufacture of guanidines
11/29/1995EP0683770A1 Substituted tetrahydropyridazine carboxamides
11/29/1995EP0683767A1 Azacyclic compounds, compositions containing them and their use as tachykinin antagonists
11/29/1995CN1112560A Piperidine derivatives and anti-platelet agents containing the same
11/29/1995CN1112550A 4-amino-1-piperidylbenzoylguanidine
11/29/1995CN1112548A Polyiodinated compounds, process for preparing them and diagnostic compositions
11/28/1995US5470981 Process for trans-6-[2-(substituted-pyrrol-1-yl)alkyl]pyran-2-one inhibitors of cholesterol synthesis
11/28/1995US5470980 Light stabilizers for polymers that can be grafted to polymers
11/28/1995US5470878 Cell signaling inhibitors
11/23/1995WO1995031437A1 Processes for preparing anhydrous and hydrate forms of antihistaminic piperidine derivatives, polymorphs and pseudormophs thereof