Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
09/2004
09/30/2004US20040192673 Obesity, non-insulin-dependent diabetes,strokes, sleep disorders; antiischemic and antiemetic agents
09/30/2004CA2519440A1 Substituted piperidine and piperazine derivatives as melanocortin-4 receptor modulators
09/30/2004CA2519372A1 Substituted cyclohexyl and piperidinyl derivates as melanocortin-4 receptor modulators
09/30/2004CA2519220A1 Amino cyclobutylamide modulators of chemokine receptor activity
09/30/2004CA2518728A1 Cathepsin s inhibitors
09/30/2004CA2518707A1 Compounds, a process for their preparation and their use as dyes and pigments
09/30/2004CA2518447A1 Synthesis of aryl-substituted piperidines by hydrogenation of aryl-substituted pyridines
09/29/2004EP1462104A1 Optically pure (-) norcisapride for treating digestive tract disorders
09/29/2004EP1461384A1 Novel flame retarding compounds
09/29/2004EP1461313A1 Human adam-10 inhibitors
09/29/2004EP1461038A1 Arylsulfonamide derivatives for use as ccr3 antagonists in the treatment of inflammatory and immunological disorders
09/29/2004EP1181278B1 Cyclic amine derivatives and their uses
09/29/2004EP1028961B1 Pleuromutilin derivatives as antimicrobials
09/29/2004EP0993439B1 4-bromo or 4-iodo phenylamino benzhydroxamic acid derivatives and their use as mek inhibitors
09/29/2004EP0969813B1 Topical pharmaceutical composition comprising a cholinergic agent or a calcium channel blocker
09/29/2004CN1533377A Method for preparing 4-amino-4-phenylpiperidines
09/29/2004CN1168717C Novel intermediates for prepn. of antihisatminic piperidine derivatives
09/29/2004CN1168715C Novel benzene amine compound, its prepn. process and medicinal compsns. contg. them
09/29/2004CN1168714C Arylpiperazine derivatives useful as uroselective alpha-adrenoceptor blockers
09/29/2004CN1168700C Cyclic amine substd. phenylalkanone and preparing method thereof
09/28/2004US6797826 Acylating a starting compound containing carboxy or amide or ester-isopropylbenzene compound with an chlorobutanoylhalide to form mixture of regioisomer, hydrolyzing to form second mixture and recovering substantially pure rgioismor
09/28/2004US6797820 Succinate compounds, compositions and methods of use and preparation
09/28/2004US6797700 Antithrombotic azacycloalkylalkanoyl peptides and pseudopeptides
09/28/2004CA2224125C Pharmaceutical composition comprising a proteinase inhibitor and a monoglyceride
09/23/2004WO2004080966A1 Nitrogen-containing heterocyclic derivatives and drugs containing the same as the active ingredient
09/23/2004WO2004080959A2 Process for the preparation of dexmethylphenidate hydrochloride
09/23/2004WO2004080952A1 Phenylsulfonamide derivatives for treating alzheimer's disease
09/23/2004WO2004080947A1 Imino ether derivative compounds and drugs containing the compounds as the active ingredient
09/23/2004WO2004080583A2 PROCESS FOR THE PREPARATION OF threo-METHYLPHENIDATE HYDROCHLORIDE
09/23/2004WO2004080460A1 SUBSTITUTED PIPERIDINES AS NOVEL MDM2-p53 INHIBITORS
09/23/2004WO2004080377A2 Kcnq channel modulating compounds and their pharmaceutical use
09/23/2004WO2004050613A3 2-substituted-3-propenamide derivatives and methods of using the same
09/23/2004WO2004043913A3 Hetero-substituted benzimidazole compounds and antiviral uses thereof
09/23/2004WO2003082268A3 Hemiasterlin derivatives and uses thereof in the treatment of cancer
09/23/2004US20040186287 heterocyclic imines such as 2-(2,6-difluorophenyl)-5-phenyl-3,4-dihydro-2H-pyrrole, formed by cyclocondensation, for use as insecticides or miticides
09/23/2004US20040186148 E.g., 1-(pyrid-2-yl-so2-),2-((4-(isopropylphenyl)-so2-),5-(isopropoxy)benzene; antiinflammatory agents; immunomodulatory activity rheumatoid arthritis, asthma, allergy, psoriasis, Crohn's disease, systemic lupus erythematosus, multiple sclerosis, diabetes, cancer, glaucoma, osteoporosis, renal ischemia
09/23/2004US20040186145 Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
09/23/2004US20040186140 Cyclic derivatives as modulators of chemokine receptor activity
09/23/2004US20040186138 E.g., 4-[4-(4-fluoro)phenoxy]pheny-1-(2-phenyl-2-oxoethyl)-4-piperidinol; antiischemic agents; antiepilptic agents; relief of symptoms form seizures and migraines; calcium channel blockers (T-type Ca2+ channel); brain disorders; cardiovascular disorders
09/23/2004US20040186137 Heating a solution of a racemic mixture of terfenadine, carboxyterfenadine or an ester derivative and an equimolar amount of optically active resolving agent, (+)-di-para-toluoyltartaric acid or mandelic acid to solubilize the diastereomeric salt;cooling to precipitate the target salt; hydrolysis
09/23/2004US20040186135 Substituted piperidine compounds
09/23/2004US20040186134 Inhibitors of Factor Xa are useful as anticoagulants in the treatment of cardiovascular disorders associated with thromboses; e.g., 1,1-dimethylethyl 1-[1-(-2-(-3-[2-(5-Chloro-thiophen-2-yl)-ethenesulfonylamino]-2-oxo-piperidin-1-yl)-acetyl)-pyrrolidin-2- yl-methyl]-pyrrolidin-3-yl}-methyl-carbamate
09/23/2004US20040186098 Method for preventing and treating hearing loss using sensorineurotrophic compounds
09/23/2004US20040186097 such as N-phenyl-3-[[4-(phenylmethyl)-1-piperidinyl]methyl]-1-piperidinecarboxamide for prevention of asthma and allergies
09/23/2004US20040186080 Beta 2-adrenergic receptor agonists
09/23/2004DE10341535A1 New N,N-disubstituted (hetero)arylsulfonamide derivatives are gamma-secretase inhibitors useful for treatment or prophylaxis of Alzheimer's disease
09/23/2004CA2518986A1 Imino ether derivative compounds and drugs containing the compounds as the active ingredient
09/23/2004CA2516145A1 Substituted piperidines as novel mdm2-p53 inhibitors
09/22/2004EP1460069A1 Substituted cyclohexyl and piperidinyl derivatives as melanocortin-4 receptor modulators
09/22/2004EP1460062A1 Nitrogenous cyclic ketone derivative, process for producing the same, and use
09/22/2004EP1460061A1 Process for producing 1-alkoxycarbonyl nitrogenous saturated heterocyclic derivative
09/22/2004EP1458743A1 Tetrahydrobenzfluorene derivatives
09/22/2004EP1458689A1 Aryloxyphenyl and arylsulfanylphenyl derivatives
09/22/2004EP1458684A2 Therapeutic heterocycles
09/22/2004EP1458682A1 1,4-dihydro-1,4-diphenylpyridine derivatives
09/22/2004EP1458681A1 Hydrophilic (s)-amlodipine salts or their hydrates and pharmaceutical compositions
09/22/2004EP1458375A2 Compositions for decreasing activity of hormone-sensitive lipase
09/22/2004EP1458374A2 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
09/22/2004EP1157989B1 Fluorides of 4-substituted piperidine derivatives
09/22/2004EP1124801B1 Piperidine and pyrrolidine derivatives comprising a nitric oxide donor for treating stress
09/22/2004EP1100781B1 High affinity ligands for nociceptin receptor orl-1
09/22/2004EP1100503B1 Non-imidazole alkylamines as histamine h 3?-receptor ligands and their therapeutic applications
09/22/2004EP1030841B1 Process for the preparation of 1,4-dihydropyridines and compounds used in this process
09/22/2004CN1530107A Insulin resistance treatment by growth hormone secretory hormone
09/22/2004CN1167682C Muscarinic antagonists
09/22/2004CN1167673C Fluorovinyloxyacetamides, process for preparing the same and herbicidal composition comprising the same
09/21/2004US6794519 Reacting an amino alcohol derivative with a sulfonyl halide in a mixed solvent composed of an aprotic organic solvent and water in the presence of a non- water-prohibiting inorganic base to produce sulfonic acid ester derivative
09/21/2004US6794511 An enzyme inhibitors of metalloprotease; treating connective tissue degradation caused by inflammation or tumor
09/21/2004US6794510 Processes for the preparation of peripheral opioid antagonist compounds and intermediates thereto
09/21/2004US6794507 Compounds that inhibit factor Xa activity
09/21/2004US6794399 Beta-adrenoreceptor and calcium channel blocking agent; induced vasorelaxing effect
09/21/2004US6794392 Cell differentiation inducer
09/21/2004US6794386 β-amino acid compounds as integrin antagonists
09/21/2004US6794378 Heterocyclic compounds and medical use thereof
09/21/2004CA2155843C Novel urea derivatives, their preparation and use
09/16/2004WO2004078988A1 Process for production of aromatic diols
09/16/2004WO2004078717A1 Acylated piperazine derivatives as melanocortin-4 receptor agonists
09/16/2004WO2004078716A1 Acylated piperazine derivatives as melanocortin-4 receptor agonists
09/16/2004WO2004078715A1 Nitrogenous heterocyclic derivative having 2,6-disubstituted styryl
09/16/2004WO2004071445A3 2-(aminomethyl)arylamide analgesics
09/16/2004WO2004064972A9 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions
09/16/2004WO2004062562A3 Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof
09/16/2004WO2004058148A3 Mitotic kinesin inhibitors
09/16/2004WO2004010943A3 Substituted benzanilides as modulators of the ccr5 receptor
09/16/2004WO2003096989A3 Anti tubercular drug: compositions and methods
09/16/2004WO2003028729A3 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
09/16/2004WO2002028833A3 Process for the synthesis of 2,2,6,6-tetramethyl-4-oxopiperidine
09/16/2004US20040181071 Method for preparing 4-methylamino-4-phenylpiperidine
09/16/2004US20040181070 Which are the melanocortin-4 receptor agonists;halogenating the benzonitrile or benzoic acid or benzamide; Grignard; arylation of the pyridinium; hydrogenation; 4-phenylpiperidine-1-carboxcylic acid esthers
09/16/2004US20040181067 Tri(cyclo) substituted amide compounds
09/16/2004US20040180964 anti-obestic activity; Neuropeptide Y antagonist
09/16/2004US20040180929 Nitrogen compounds such as 4-Benzyloxy-4-(4-chlorophenyl)-3-(3,4-difluorobenzyloxy)-piperidine, administered as oncoprotein or ubiquitin-conjugating enzyme antagonists for prophylaxis of cancer; anticarcinogenic agents
09/16/2004US20040180928 Process for the preparation of dexmethylphenidate hydrochloride
09/16/2004US20040180927 Inhibitors of cysteine protease
09/16/2004US20040180926 Derivatives of 3-phenyl-n-(2-(4-benzyl)-piperidin-1-yl)-ethyl)-acrylamid with ccr-3-receptor antagonistic activity for use in the treatment of inflammations and allergic conditions
09/16/2004US20040180892 control of cardiovascular homeostasis is achieved through a combination of both direct neuronal control and systemic neurohormonal activation
09/16/2004US20040180886 Cathepsin S inhibitors
09/16/2004US20040180880 Piperazine and piperidine derivatives
09/16/2004US20040180871 Anti-inflammatory compositions and methods
09/16/2004US20040180863 Novel, nitric oxide-releasing amidine- and enamine-derived diazeniumdiolates, compositions and uses thereof and method of making same