Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
05/2006
05/31/2006CN1257892C New indole derivatives with 5-HT6 receptor affinity
05/31/2006CN1257886C Dehydroamino acids compounds
05/30/2006US7053234 Antibacterial agents
05/30/2006US7053211 Process for the preparation of α-aminosubstituted carboxylic acid amides
05/30/2006US7053122 Brain disorders; central nervous system disorders; anxiolytic agents; analgesics; sleep disorders
05/30/2006US7053109 Aminediols for the treatment of Alzheimer's disease
05/30/2006US7053104 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases
05/30/2006US7053088 Vanilloid receptor ligands and their use in treatments
05/30/2006US7053078 Serine protease inhibitors
05/30/2006US7053071 Induction of apoptosis in cancer cells
05/26/2006WO2006055725A2 Substituted amino acids as protein tyrosine phosphatase inhibitors
05/26/2006WO2006055463A2 2-amino-3-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
05/26/2006WO2006055462A1 2-amino-4-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
05/26/2006WO2006055435A1 2-aminonaphthalene derivatives and related glycogen phosphorylase inhibitors
05/26/2006WO2006055187A1 Sulfonyl-substituted bicyclic compounds as modulators of ppar
05/26/2006WO2006054491A1 Process for producing n-(3-chloro-1h-indol-7-yl)-4-sulfamoylbenzenesulfonamide
05/26/2006WO2006054456A1 Crystal of two-ring heterocyclic sulfonamide compound
05/26/2006WO2006054162A1 Azabicyclic muscarinic receptor antagonists
05/26/2006WO2006053700A1 Agonists and antagonists of the somatostatin receptor
05/26/2006WO2006053440A1 New processes for the preparation of optically pure indoline-2-carboxylic acid and n-acetyl-indoline-2-carboxylic acid
05/26/2006WO2006012162A3 Methods for producing and purifying 2-hydrocarbyl-3,3-bis(4-hydroxyaryl)phthalimidine monomers and polycarbonates derived therefrom
05/26/2006WO2006002361A3 2-methylpropanamides and their use as pharmaceuticals
05/26/2006WO2005108358A3 Pyrrolidine derivatives useful as bace inhibitors
05/26/2006CA2588776A1 Substituted amino carboxylic acids
05/26/2006CA2585172A1 Sulfonyl-substituted bicyclic compounds as modulators of ppar
05/26/2006CA2582384A1 Agonists and antagonists of the somatostatin receptor
05/25/2006US20060111427 Indole derivatives useful as progesterone receptor modulators
05/25/2006US20060111426 Indole-3-sulphur derivaties
05/25/2006US20060111425 To treat diseases of respiratory, urinary and gastrointestinal systems; highly selective; significant potency; (2R,2S)(1 alpha ,5 alpha ,6 alpha )-N-{-[4-(1,3-dioxo-1,3-dihydro-isoindol-2-yl)-butyl]-3-azabicyclo[3.1.0]hex-6-yl-methyl}-2-hydroxy-2-cyclopentyl-2-phenylacetamide
05/25/2006US20060111424 Treating nuclear hormone receptor-associated conditions such as cancer and immune disorders; (3a alpha ,4 alpha ,7 alpha ,7a alpha )-2-(3-Chloro-4-hydroxyphenyl)hexahydro-4,7-methano-1H-isoindole-1,3(2H)-dione
05/25/2006US20060111339 Novel oral general anesthetics and metabolitically resistant anticonvulsants
05/25/2006US20060111304 For therapy of pancreatitus, bilioecholic, gastroesophical relux (GERD), irritable bowel syndrome (IBS), non ulcerous dyspepsia
05/25/2006US20060111303 N-[(1S)-3-{(2Z)-2-[(4R)-3,4-dimethyl-1,3-thiazolidin-2-ylidene]hydrazino}-2,3-dioxo-1-(tetrahydro-2H-pyran-4-yl)propyl]cycloheptanecarboxamide; cysteine protease inhibitors; for the treatment of inflammatory, immune, ischemic, respiratory,circulatory, neuronal, blood, hepatic and metabolic diseases
05/24/2006EP1658267A2 Inhibitors of cathepsin s
05/24/2006EP1658068A1 Novel cycloalkyl'b! condensed indoles
05/24/2006EP1658067A1 Indolamide derivatives which possess glycogen phosphorylase inhibitory activity
05/24/2006EP1658066A2 Adamantylglycine- based inhibitors of dipeptidyl peptidase iv for the treatment of diabetes
05/24/2006EP1370526B1 Diamides which inhibit tryptase and factor xa activity
05/24/2006EP1334106B1 Imidazole derivatives, production method thereof and use thereof
05/24/2006EP1212298B1 Isolation of natural l-beta-3-indolylalanine and enrichment of natural aliphatic amino acid mixtures with natural l-beta-3-indolylalanine
05/24/2006EP1100492B1 INDOLE sPLA2 INHIBITORS
05/24/2006DE10347386B4 Tetrahydronaphthalinderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Entzündungshemmer Tetrahydronaphthalene derivatives, processes for their preparation and their use as anti-inflammatories
05/24/2006CN1777583A Methods for producing cyclic benzamidine derivatives
05/24/2006CN1777582A Substituted indoline and indole derivatives
05/24/2006CN1775763A Carboxyl acylamide compound and its preparing method and use
05/24/2006CN1775759A Bicyclic androgen and progesterone receptor modulator compounds and methods
05/24/2006CN1775754A Indole preparing method
05/24/2006CN1256998C Sublimation purifying method and apparatus
05/23/2006US7049468 Method for modulating the activity of a Rho C enzyme, comprising: contacting said Rho C enzyme with an effective amount of a compound of formula 1:
05/23/2006US7049448 Reacting cyclohexanedione with diol in halogenated solvent in presence of acid catalyst
05/23/2006US7049445 for treating or preventing diabetes, obesity, hyperlipidemia, digestive diseases, depression or urinary disturbances; beta 3-agonist
05/23/2006US7049444 3-azabicyclo[3.1.0]hexane derivatives useful in therapy
05/23/2006US7049335 3-azabicyclo[3.1.0]hexane derivatives
05/23/2006US7049330 Cycloalkyl-substituted aryl-piperazines, piperidines and tetrahydropyridines as serotonergic agents
05/23/2006US7049326 Altering a drug's distribution, metabolism and elimination properties, especially by modifying with aralkyl ester moieties to increase rate of metabolism to inactive and nontoxic metabolites when exposure is halted; surgery, riots
05/23/2006US7049316 Prodrugs of CC-1065 analogs
05/23/2006US7049314 Cyclopentyl indole derivatives
05/23/2006CA2339630C Carboline derivatives as cgmp phosphodiesterase inhibitors
05/23/2006CA2173747C Calcium receptor-active arylalkyl amines
05/22/2006CA2488324A1 Optical resolution of n-acetyl-indoline-2-carboxylic acid with phenylglycinol
05/18/2006WO2006051399A1 Piperazine derivatives useful as adrenergic receptor antagonists
05/18/2006WO2006051374A2 Arylpiperazines useful as adrenergic receptor antagonists
05/18/2006WO2006051047A1 N-substituted imides as polymerization initiators
05/18/2006WO2006034480A3 Sulfonamide bicyclic compounds
05/18/2006WO2006012504A3 Compounds and methods for treatment of thrombosis
05/18/2006WO2005051301A3 Heterocyclic inhibitors of mek and methods of use thereof
05/18/2006US20060106256 e.g. 1-[(benzylamino)methyl]-3-(3,5-difluorophenyl)-2-({3-[(dipropylamino)carbonyl]benzoyl}amino)propyl 4-nitrophenyl carbonate; secretase inhibitors; neurodegenerative disorders; Alzheimer's, Parkinson's diseases, Down syndrom, Hereditary Cerebral Hemorrhage with Amyloidosis of the Dutch-Type
05/18/2006US20060106227 3-'2-(Dimethylamino) ethyl!-n-methyl-1h-indole-5-methanesulfonamide and the succinate thereof
05/18/2006US20060106226 Isolation of amino acids and related isolates
05/18/2006US20060106086 Preparation of tegaserod and tegaserod maleate
05/18/2006US20060106067 Androgen receptor agonist; prostate cancer, hypogonadism; 4-[4-(hydroxymethyl)-1-piperidinyl]-1-naphthonitrile; 4-(4-hydroxy-2-methyl-1-pyrrolidinyl-1-benzothiophene-7-carbonitrile
05/18/2006US20060106053 Therapy of adenocarcinoma of the colon and rectum
05/18/2006US20060105441 Process for the preparation of indole derivatives by enzymatic acylation
05/18/2006US20060105257 Indolenine compound, near infrared absorber, and toner containing the same
05/17/2006EP1656348A1 Acetylene derivatives as inhibitors of histone deacetylase
05/17/2006EP1656347A1 Substituted indole derivatives for pharmaceutical composition for treating respiratory diseases
05/17/2006EP1656346A1 Novel substituted 3-sulfur indoles
05/17/2006EP1656141A1 Treatment for alzheimer s disease and related conditions
05/17/2006EP1656134A1 Indoline-sulfanilic acid amides used as ppar delta modulators
05/17/2006CN1256325C Process for cascade reaction preparation of N-acetyl-DL-tryptophan
05/16/2006US7045544 Myocardium; angina pectoris
05/16/2006US7045532 ACE-2 modulating compounds and methods of use thereof
05/16/2006US7045521 Cyclic amide derivative as monocyte chemotactic protein modulator; prevention and treatment of rheumatoid arthritis, multiple sclerosis, atherosclerosis and asthma; antiinflammatory agents
05/16/2006US7045360 Method for analysis of reaction products
05/16/2006CA2237752C Novel substituted aryl compounds useful as modulators of acetylcholine receptors
05/16/2006CA2192797C Indolinone compounds for the treatment of disease
05/11/2006WO2006050120A2 Synthesis of cox-2 and faah inhibitors
05/11/2006WO2006049889A1 Indole derivatives useful as progesterone receptor modulators
05/11/2006WO2006049835A2 Indole and benzimidazole derivatives
05/11/2006WO2006048893A2 A process for synthesis of large particle size statin compounds
05/11/2006WO2006048727A1 Piperazinylphenalkyl lactam/amine ligands for the 5ht1b receptor
05/11/2006WO2006048236A1 Process for the preparation of alkyl 5- (dicarboximido) levulinate and alkyl 4-oxo-pentenoate
05/11/2006WO2006047888A1 2-substituted indoles, their precursors and novel processes for the preparation thereof
05/11/2006US20060100283 Phenylcyclohexylpropanolamine derivatives, preparation and therapeutic application thereof
05/11/2006US20060100266 3-(2-Dimethylaminoethyl)-7-fluoro-1-methyl-1H-indol-4-ol; Obsessive Compulsive Disorder; appetite suppressants
05/11/2006US20060100265 4-(1-(sulfonyl)-1h-indol-2-yl)-4-(hydroxy)-cyclohexa-2,5-dienone compounds and analogs thereof as therapeutic agents
05/11/2006US20060100230 Indolin phenylsulfonamide derivatives
05/11/2006US20060100202 Novel compounds
05/11/2006US20060100196 Substituted amines for the treatment of alzheimer's disease
05/11/2006US20060099638 incorporating indolium ring moiety substituted at 3-position improves spectral properties; for detection of ligands; hybridization probes