Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
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07/20/2006 | WO2006075139A2 Novel process for the preparation of substituted indoles |
07/20/2006 | WO2006054162A8 Azabicyclic muscarinic receptor antagonists |
07/20/2006 | WO2006015060A3 Isoindoline compounds and methods of their use |
07/20/2006 | WO2005121130A3 Chemical compounds and pharmaceutical compositions containing them for the treatment of inflammatory disorders |
07/20/2006 | WO2004091382A3 Monitoring circadian activity |
07/20/2006 | US20060161006 Asymmetric urea compound and process for producing asymmetric compound by asymmetric conjugate addition reaction with the same as catalyst |
07/20/2006 | US20060161002 Tetrahydrocarbazole derivatives and their pharmaceutical use |
07/20/2006 | US20060160894 Benzamides as ppar modulators |
07/20/2006 | US20060160884 N-{[4-(but-2-ynyloxy)phenyl]sulfonyl}-1-(2-fluorobenzyl)-5-methoxy-2-methyltryptophan; for treatment of rheumatoid arthritis, juvenile rheumatoid arthritis, ulcerative colitis, or Crohn's disease |
07/20/2006 | US20060160882 Indoline derivatives |
07/20/2006 | US20060160880 2-(1H-indolylsulfanyl)-benzyl amine derivatives as SSRI |
07/20/2006 | US20060160879 Indoles useful in the treatment of inflammation |
07/20/2006 | US20060160876 Indole derivatives |
07/20/2006 | US20060160856 Diarylurea derivatives and their use as chloride channel blockers |
07/20/2006 | US20060160847 2,4-Dihalogen-6-(c2-c3alkyl)-phenyl substituted tetramic acid derivatives |
07/20/2006 | US20060160840 Tetrahydroisoquinolines as factor Xa inhibitors |
07/20/2006 | US20060160818 Ocular hypotensive agent |
07/20/2006 | US20060160798 3-Cyclohexyl-1-methyl-2-pyridin-2-yl-1H-indole-6-carboxylic acid methyl ester; hepatitis C virus infection; synergistic with another inhibitor of HCV polymerase or immunomodulatory agent such as interferons |
07/20/2006 | US20060159956 Fluorene-based derivative and organic electroluminescence device employing the same |
07/20/2006 | CA2594391A1 Process for the preparation of substituted indoles |
07/20/2006 | CA2593450A1 Indole derivatives for treating viral infections |
07/19/2006 | EP1680411A2 Modulators of atp-binding cassette transporters containing cycloalkyl or pyranyl groups |
07/19/2006 | EP1680401A2 Indolinone derivatives and their use in treating disease-states such as cancer |
07/19/2006 | EP1680397A2 Novel compounds and their use as antidiabetic and hypolipidemic agents, process for their preparation and pharmaceutical compositions containing them |
07/19/2006 | EP1680124A2 Bicyclic [3.1.0] derivatives as glycine transporter inhibitors |
07/19/2006 | EP1680109A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
07/19/2006 | EP1056452B1 Indole-3-propionic acids, salts and esters thereof used as medicaments |
07/19/2006 | CN1805972A Novel method for the synthesis of perindopril and the pharmaceutically acceptable salts thereof |
07/19/2006 | CN1805959A Cycloalkanepyrrolopyridines as DP receptor antagonists |
07/19/2006 | CN1805932A Process and intermediates for the preparation of (1r,2s,5s)-3-azabicyclo[3,1,0]hexane-2-carboxamide, n-[3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl]-3-[(2s)-2-[[[1,1-dimethylethyl]amino]carbonylamino |
07/19/2006 | CN1805931A Process and intermediates for the preparation of (1r,2s,5s)-6,6-dimethyl-3-azabicyclo[3,1,0]hexane-2-carboxylates or salts thereof |
07/19/2006 | CN1805930A Hydroxamic acids useful in the treatment of hyper-proliferative disorders |
07/19/2006 | CN1805928A Prodrugs of mitotic kinesin inhibitors |
07/19/2006 | CN1803800A Method for preparing 5-bromine-6-fluoro-8-methyl-1-ethyl-1,3,4,9- tetrahydropyrane[3,4-e] indole-1-ethyl acetate |
07/19/2006 | CN1803784A 4-phenyl-1-piperazinyl, -piperidinyl and -tetrahydropyridyl derivatives |
07/19/2006 | CN1264848C Pyrrolo[2,1-b] [1,3] benzothiazepines and their use for preparation of medicaments with antipsychotic activity |
07/19/2006 | CN1264841C Preparation of anti-cancer active material in camptothecinum cell and method for restraining cancer cell |
07/18/2006 | USRE39197 diaryl sulfides, substituted with cinnamides, such as (2,4-Dichlorophenyl)[2-(E-((6-hydroxyhexylamino)carbonyl)ethenyl)phenyl]sulfide, used for treating inflammatory and immune diseases in mammals |
07/18/2006 | US7078567 Forming c-n bonds; isomerization |
07/18/2006 | US7078535 Method for the production of 6-(4-chlorophenyl)-2,2-dimethyl-7-phenyl-2,3-dihydro-1h-pyrrolizin-5-ylacetic acid |
07/18/2006 | US7078534 Activation the corresponding keto ester; reacting with cysteamine; hydrogenation; crystallization in solvent |
07/18/2006 | US7078521 By reaction of pyrrolobenzothiazepin-9-one with amine to give the corresponding enamine, which is subsequently transformed into the final compound |
07/18/2006 | US7078429 Substituted 3-carbonyl-1H-indol-1-yl acetic acid derivatives for treating conditions resulting from fibrinolytic disorders, such as deep vein thrombosis and coronary heart disease, and pulmonary fibrosis; Alzheimer's disease |
07/18/2006 | US7078428 3-(Guanidinylcarbonylmethyl)-substituted; inhibit the cellular sodium-proton antiporter, in particular NHE1; antiarrhythmic agents;cardioprotective for infarction prophylaxis and treatment; preventing ischemia-induced damage |
07/18/2006 | US7078427 Bioavailability; anticancer agents; viricides |
07/18/2006 | US7078425 4-(2-substituted aminocarbonyl-2-substituted aminoethyl)-7-carboxymethoxy- indole, indazole, indoline, benzotriazole or benzoimidazole derivatives, e.g., 4-[2-Benzenesulfonylamino-2-(4-phenyl-butylcarbamoyl)-ethyl]-1H-indazol-7-yloxy}-acetic acid; treating or preventing Type II Diabetes Mellitus |
07/18/2006 | CA2356320C Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds |
07/18/2006 | CA2325781C New amino pyrrolin compounds, their preparation process and the pharmaceutical compositions therein |
07/18/2006 | CA2309771C New substitute dimeric derivatives, their preparation process and the pharmaceutical compositions that contain them |
07/13/2006 | WO2006072736A1 N- (heteroaryl) -1h-indole-2-carb0xamide derivatives and their use as vanilloid trpv1 receptor ligands |
07/13/2006 | WO2006048893A3 A process for synthesis of large particle size statin compounds |
07/13/2006 | WO2005112945A3 Synthesis of tetracyclines and analogues thereof |
07/13/2006 | WO2005090302A3 Palladium catalyzed indolization of 2-bromo or chloroanilines |
07/13/2006 | WO2004065367A8 Viral polymerase inhibitors |
07/13/2006 | US20060154872 chemical intermediate for Hemiasterlin, first isolated from the sponge Hemiasterella; anticarcinogenic agent for treatment of colon cancer, tumor; prevention of restenosis of blood vessels subject to traumas such as angioplasty and stenting |
07/13/2006 | US20060154343 Simultaneous isomerization at position 2 of monatin having different configurations at positions 2 and 4 in the presence of an aldehyde in a solvent mixture of alcohol and water and crystallization to produce an optical isomer of monatin that has the same configurations at positions 2 and 4 or salt . |
07/13/2006 | CA2594418A1 N-(heteroaryl)-1h-indole-2-carb0xamide derivatives and their use as vanilloid trpv1 receptor ligands |
07/12/2006 | EP1679303A1 Process for preparing 1-alkoxycarbonyl-3-phenylpropyl derivative |
07/12/2006 | EP1679302A1 Aromatic amino acid labeled with stable isotope, method for incorporating the same into target protein and method for analyzing protein structure using nmr |
07/12/2006 | EP1679301A1 Esters of nonsteroidal anti-inflammatory drugs and methods of their preparation |
07/12/2006 | EP1679072A1 Process for for synthesis of (2S,3aS,7aS)-1-(S)-alanyl-octahydro-1H-indole-2- carboxylic acid derivatives and use in the synthesis of perindopril |
07/12/2006 | EP1678258A1 Cyanine dye labelling reagents |
07/12/2006 | EP1678170A1 Use of a compound of formula (i) as an inhibitor of aromatase for therapeutic purposes and compounds of formula (1) thereas |
07/12/2006 | EP1678154A1 Arylalkyl- and cycloalkylalkyl-piperazine derivatives and methods of their use |
07/12/2006 | EP1678145A2 Benzimidazoles useful as modulators of ion channels |
07/12/2006 | EP1678137A1 Compositions and methods for viral inhibition |
07/12/2006 | EP1678136A1 Process for preparing an azabicyclo[3.1.0]hexane compound |
07/12/2006 | EP1678135A1 Process for the preparation of n-amino substituted heterocyclic compounds |
07/12/2006 | EP1678123A1 Tetrahydro-naphthalene and urea derivatives |
07/12/2006 | EP1678121A2 Tao kinase modulators and methods of use |
07/12/2006 | EP1677794A2 Methods of treating disorder |
07/12/2006 | EP1677783A2 Fibrinogen receptor antagonists and their use |
07/12/2006 | EP1394156B1 Chromene compound |
07/12/2006 | EP1335923B1 Condensed pyridoindole derivatives |
07/12/2006 | CN1802384A Method for synthesis of perindopril and its pharmaceutically acceptable salts |
07/12/2006 | CN1802354A Tetrahydrocarbazole derivatives and their pharmaceutical use |
07/12/2006 | CN1802353A Fluoroalkoxy-substituted 1,3-dihydro-isoindolyl compounds and their pharmaceutical uses |
07/12/2006 | CN1802091A Use of isoindolinone derivatives as insecticides |
07/12/2006 | CN1800183A One-step synthesis process for pemetrexed disodium key intermediate |
07/12/2006 | CN1800145A Substituted 2-dialkylaminoalkylbiphenyl derivatives |
07/12/2006 | CN1263745C Aryl fused azapolycyclic compounds |
07/11/2006 | US7075582 Methods for identifying and using MarR family polypeptide binding compounds |
07/11/2006 | US7074952 Synthesis of taxol enhancers |
07/11/2006 | US7074939 Indole derivatives as anti-inflammatory agents |
07/11/2006 | US7074938 Method for the synthesis of soritin compounds |
07/11/2006 | US7074934 Serine protease inhibitors |
07/11/2006 | US7074837 Acetalization of aldehydes in the presence of acid catalysts, then aminating, cyanating, reducing and cyclization to form heterocyclic amines used as chemical intermediates or bactericides |
07/11/2006 | US7074817 For treating conditions resulting from fibrinolytic disorders such as deep vein thrombosis and coronary heart disease, and pulmonary fibrosis |
07/11/2006 | US7074814 Antiinflammatory agents; cardiovascular disorders; anticancer agents; antiarthritic agents ; psoriasis |
07/11/2006 | US7074806 Antiinflammatory agents, antiallergens, antiproliferative agents, immunosuppressants, antidiabetic agents, cardiovascular disorders |
07/11/2006 | US7074805 Especially isoquinolin-5-ylurea derivatives; treating pain, inflammatory thermal hyperalgesia, urinary incontinence and bladder overactivity. |
07/11/2006 | US7074800 Quinazoline derivatives as angiogenesis inhibitors |
07/11/2006 | US7074796 High affinity for D4 receptors; treatment of psychological disorders such as schizophrenia, generalised anxiety disorder, panic disorder, and obsessive compulsive disorder. |
07/11/2006 | US7074782 Administering to a patient suffering from caspase mediated diseses, an effective amount of a mono,bi or tri-heterocyclic ring containing nitrogen atom attached to ester or thioester to form carbamate group, as caspase inhibitor |
07/11/2006 | US7074534 Polymeric charge transport compositions and electronic devices made with such compositions |
07/11/2006 | CA2376876C New isoindoloindolone derivatives, the process for preparing them and the pharmaceutical compounds that contain them |
07/11/2006 | CA2344255C Novel derivatives of heterocycloalkylbenzocyclobutane and heteroarylbenzocyclobutane, process for preparing them and pharmaceutical compositions containing them |
07/11/2006 | CA2325779C New derivatives of 12,13-(pyranosyl)-indolo[2,3-a]pyrrolo[3,4-c]carbzole and 12,13 (pyranosyl)-furo[3,4-c]indol[2,3-a]carbazole, their preparation process and the pharmaceutical compositions therein |
07/11/2006 | CA2246783C Mcbi analogs of cc-1065 and the duocarmycins |
07/11/2006 | CA2227984C Aza-anthracyclinone derivatives |