Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
01/2009
01/20/2009CA2337770C Amide derivatives which are useful as cytokine inhibitors
01/20/2009CA2331758C Method for the stereochemically controlled production of isomerically pure highly substituted azacyclic compounds
01/20/2009CA2325526C Aryl phenyl substituted cyclic ketoenols
01/20/2009CA2235797C Process for purification of almost completely anhydrous organic liquids
01/15/2009WO2009008913A2 P1-nonepimerizable ketoamide inhibitors of hcv ns3 protease
01/15/2009WO2009007396A1 Nonsteroidal progesterone receptor modulators
01/15/2009WO2008140251A3 Cyclooxygenase-2 inhibitors
01/15/2009WO2008132142A3 New heterocyclic derivatives useful for the treatment of cns disorders
01/15/2009WO2008101914A3 N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
01/15/2009US20090018311 Methods and compounds for producing dipeptidyl peptidase iv inhibitors and intermediates thereof
01/15/2009US20090018183 N-phenylpyrrole guanidine derivatives as melanocortin receptor ligands
01/15/2009US20090018182 Crystalline forms of atorvastatin
01/15/2009US20090018167 angiogenesis inhibitors such as 1-phenyl-3-pyridin-2-ylprop-2-en-1-one, having antitumor and anticarcinogenic activity; treatment of skin disorders such as psoriasis, acne, rosacea, warts, eczema, hemangiomas, and lymphangiogenesis, as well as chronic inflammatory disease such as arthritis
01/15/2009US20090018116 Therapeutic Compounds
01/15/2009US20090018058 Vitamin D Receptor Modulators
01/15/2009US20090017489 Methods For Modulating The Development Of Dopamine Neuron By The Dopamine D2 Receptor And Compositions Thereof
01/15/2009US20090017004 Polymeric drug delivery systems containing an aromatic allylic acid
01/15/2009DE112007000484T5 Stabil isotopenmarkierte aliphatische Aminosäuren, Verfahren zum Einbringen von diesen in ein Zielprotein und Verfahren zur NMR-Konformationsanalyse von Proteinen Stable isotope-labeled aliphatic amino acids, methods for introducing these into a target protein, and NMR method for the conformation of proteins
01/15/2009CA2681624A1 P1-nonepimerizable ketoamide inhibitors of hcv ns3 protease
01/14/2009EP2014645A1 Pleuromutilin derivatives and their use as antimicrobials
01/14/2009EP2014285A1 NPYY5 antagonists
01/14/2009EP2013168A1 Alkoxyalkyl-substituted cyclic ketoenols
01/14/2009EP2013167A2 Total synthesis of salinosporamide a and analogs thereof
01/14/2009EP2013166A2 N-carbamoylmethyl-4(r)-phenyl-2-pyrrolidinone, method of its preparation and pharmaceutical use
01/14/2009EP2013163A1 Tetrasubstituted ureas as modulators of 11-beta hydroxyl steroid dehydrogenase type 1
01/14/2009EP1809600A4 Cyclic b-amino acid derivatives as factor xa inhibitors
01/14/2009EP1567518B1 Oxime ester photoinitiators with heteroaromatic groups
01/14/2009EP1463728B1 Fused cyclic modulators of nuclear hormone receptor function
01/14/2009CN101346351A Alkoxyalkyl spirocyclic tetramic acids and tetronic acids
01/14/2009CN101346350A Method for production of heteroaromatic ring compound having n-rf group
01/14/2009CN100450994C Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors
01/14/2009CN100450477C Novel pyrroles having hypolipidemic hypocholesteremic activities, process for their preparation and pharmaceutical compositions containing them and their use in medicine
01/13/2009US7476747 Substituted gamma lactams as therapeutic agents
01/13/2009US7476688 Cyclic amidine derivatives
01/13/2009US7476686 e.g. 1-(Benzofuran-2-carbonyl-3-(3-phenoxy-phenyl)-thiourea; viricides; Hepatitis C infection
01/13/2009US7476680 e.g. 1-[2-hydroxy-3-(quinolin-5-yloxy)-propyl]-piperidine-4-carboxylic acid [4-phenyl-1-(3-phenyl-propyl)-butyl]-amide; multidrug resistance protein or P-glycoprotein modulator; with other therapeutic agent: anticarcinogenic, antibacterial, antiviral, antifungal agents
01/13/2009US7476672 Acetylenic compounds useful in treating inflammatory disorders
01/13/2009CA2271276C Pure enantiomer basic aryl-cycloalkyl-hydroxycarboxylic acid esters, process for preparing the same and their use in medicaments
01/08/2009WO2008119457A3 Lactam-substituted dicarboxylic acids and use thereof
01/08/2009WO2008109055A8 Cyanopyrrole sulfonamides useful for modulation of the progesterone receptor
01/08/2009US20090012314 Process for Production of Lasofoxifene or Analogue Thereof
01/08/2009US20090012313 3-Carboxy-2-Oxo-1-Pyrrolidine Derivatives and Their Uses
01/08/2009US20090012312 Process for Preparing Pyrrole Derivatives and Intermediates
01/08/2009US20090012151 Novel Compounds 951
01/08/2009US20090012149 Prodrug of an ice inhibitor
01/08/2009US20090012144 Optically active 2,5-bisaryl-delta¹ -pyrrolines and their use as pest control agents
01/08/2009US20090012120 Synthesis of N-heterocycles, beta-amino acids, and allyl amines via aza-payne mediated reaction of ylides and hydroxy aziridines
01/08/2009US20090012070 Pesticidal heterocycles
01/08/2009US20090010860 used for protecting human hair and skin against the damaging effect of ultraviolet radiation
01/08/2009CA2692145A1 Antiviral compounds
01/07/2009EP2011800A2 Inhibitors of caspase
01/07/2009EP2010486A2 Diazeniumdiolated non-steroidal anti-inflammatory drugs, compositions thereof, and related methods
01/07/2009EP2010477A2 Poly (ethylene glycol) containing chemically disparate endgroups
01/07/2009EP2010475A2 Heterofunctional poly(ethylene glycol) containing acid-labile amino protecting groups and uses thereof
01/07/2009EP1928821B1 Carboxamide derivatives as muscarinic receptor antagonists
01/07/2009EP1807072B1 Cycloalkyl lactam derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
01/07/2009EP1667966A4 N-alkylated diaminopropane derivatives as modulators of chemokine receptor activity
01/07/2009EP1569916B1 Substituted aralkyl derivatives
01/07/2009EP1431285B1 Reverse hydroxamic acid derivatives
01/07/2009EP1345896B1 Crystalline forms of atorvastatin
01/07/2009CN101340959A Process for the treatment of an aqueous mixture comprising a dipolar aprotic compound
01/07/2009CN101337920A Phenylalanyl pyrrolidine derivates, preparation method and application thereof
01/07/2009CN100448877C 3-phenyl substituted 3-substituted-4ketolactams and ketolactones
01/07/2009CN100448876C Heterocyclocarboxamide derivatives
01/06/2009US7473795 Blends of quinone alkide and nitroxyl compounds as polymerization inhibitors
01/06/2009US7473779 e.g. 2-amino-N-(4-{[amino(2-thienyl)methylidene]amino}phenethyl)-5-methoxybenzamide; nitric oxide NO-synthase enzymes inhibitor; selective or non selective traps for reactive oxygen species; antiproliferative, antiinflammatory agent
01/06/2009US7473703 e.g. N-(4-{1-Hydroxy-1-[1-(2-methoxyethyl)-1H-pyrrol-2-yl]-ethyl}-phenyl)-N-methyl-benzenesulfonamide; liver X receptor (LXR) agonist; antidiabetic, antiproliferative agent; lipid, metabolic disorders, obesity, diabetes, hypercholesterolemia, atherosclerosis, hyperlipoproteinemia
01/06/2009CA2421008C Substituted heterocyclic compounds for treating multidrug resistance
01/06/2009CA2414095C Novel compounds
01/06/2009CA2391357C A process for producing crystalline atorvastatin calcium
01/06/2009CA2295446C Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same
01/06/2009CA2169219C Substituted benzenesulfonylureas and -thioureas, processes for their preparation, their use for the production of pharmaceutical preparations, and pharmaceutical preparations containing them
01/01/2009US20090005577 Method of producing 1-substituted 3-pyrrolates
01/01/2009US20090005576 Production Method of Optically Active Cyclohexane Ether Compounds
01/01/2009US20090005574 reacting a 9-hydroxymethyl-2-amino fluorene with a silyl protecting reagent e.g. tert-butyldimethylsilyl chloride to form tert-butyldimethylsiloxy-9-methyl-2-aminofluorene, reacting intermediate with 3-maleimidopropionic acid; protecting; chemical intermediates for protein and peptide drugs
01/01/2009US20090005542 Hydrolysable polymeric FMOC- linker
01/01/2009US20090005410 N-(4-Chloro-2-[1,2,3]triazolo[4,5-b]pyridin-1-yl-phenyl)-4-(1-hydroxy-1-methyl-ethyl)-benzene-sulfonamide sodium salt, used as chemokine receptors antagonists, useful for treating inflammation
01/01/2009US20090004641 Site-specific labeling of affinity peptides in fusion proteins
01/01/2009US20090004140 4-substituted pyrrolidine as anti-infectives
12/2008
12/31/2008WO2009002203A1 Polyfunctional fullerene c60 aminoacid derivatives
12/31/2008WO2009001127A1 Cyanocyclopropylcarboxamides as cathepsin inhibitors
12/31/2008WO2009000878A1 Kallikrein 7 modulators
12/31/2008WO2009000523A1 Method for preparing fmoc-based hydrolysable linkers
12/31/2008WO2009000049A1 Intrinsically conducting polymers
12/31/2008WO2008132139A3 New heterocyclic derivatives useful for the treatment of cns disorders
12/31/2008WO2008053221A3 Process for preparing indol- 5 -oxy- quinazoline derivatives and intermediates
12/31/2008WO2008014381A3 Modulators of chemokine receptor activity, crystalline forms and process
12/31/2008WO2008014360A3 Modulators of chemokine receptor activity, crystalline forms and process
12/31/2008EP2009010A1 Cocrystal of c-glycoside derivative and l-proline
12/31/2008EP2008999A1 N-tert-butoxycarbonyl-2-pyrrolidinones and process for producing the same
12/31/2008EP2008997A1 Process for production of ethylenediamine derivative having halogenated carbamate group and acyl group, and intermediated for production of the derivative
12/31/2008EP2007749A2 Tetralines antagonists of the h-3 receptor
12/31/2008EP2007745A2 Fungicide n-cyclopropyl-sulfonylamide derivatives
12/31/2008EP2007720A1 Benzamide derivatives as inhibitors of histone deacetylase
12/31/2008EP2007719A2 Inhibitors of the 11-beta-hydroxysteroid dehydrogenase type 1 enzyme
12/31/2008EP2007705A1 Nitric oxide enhancing prostaglandin compounds, compositions and methods of use
12/31/2008EP2007383A2 Inhibitors of protein prenyltransferases
12/31/2008EP1851198B1 Substituted pyrroles, compositions containing same, method for making same and use thereof
12/31/2008EP1051397B1 Method for preparing an n- (aliphatic or aromatic)carbonyl -2-aminoacetamide compound and a cyclyzed compound
12/31/2008CN101336229A 改性的拟赖氨酸化合物 Proposed modification of lysine compound