Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
10/2008
10/15/2008EP1142872B1 Aromatic heterocycle compounds having hiv integrase inhibiting activities
10/15/2008EP0923544B1 Method for the synthesis of amines and amino acids with organoboron derivatives
10/15/2008CN101287721A 酰肼化合物和其杀虫用途 Hydrazide compounds and their insecticidal use
10/15/2008CN101287706A Sulphonylpyrrole hydrochloride salts as histone deacetylases inhibitors
10/15/2008CN101287702A N-phenyl phenylacetamide non-nucleoside reverse transcriptase inhibitors
10/15/2008CN101287461A Use of 5-amido-1h-pyrrole-2-nitrile derivative as progesterone receptor modulators
10/15/2008CN101284865A New compound and its medicine use
10/15/2008CN101284810A Cyano-pyrrolidine and cyano-tetrahydrothiazole derivates
10/14/2008US7435833 Inhibitors of the 11-beta-hydroxysteroid dehydrogenase Type 1 enzyme
10/14/2008US7435815 Sulfonylamino-acetic acid derivatives
10/14/2008US7435745 Methods and compositions for inhibition of angiogenesis
10/14/2008CA2309328C Cyclic amine derivatives and their use as drugs
10/09/2008WO2008121877A2 Cftr inhibitor compounds and uses thereof
10/09/2008WO2008120759A1 Urea compound and use thereof
10/09/2008WO2008120725A1 Novel pyrrolinone derivative and medicinal composition containing the same
10/09/2008WO2008119804A1 New methods
10/09/2008WO2008119773A1 Amide derivatives as inhibitors of aspartyl proteases
10/09/2008WO2008077035A3 Processes for the preparation of levetiracetam
10/09/2008WO2008055236A3 Mapk/erk kinase inhibitors
10/09/2008WO2007092285A3 Treatment of synucleinopathies
10/09/2008US20080249315 Having an acylsulfonamide amine-reactive groups; crosslinker for amine containing material such as gel and hydrgels
10/09/2008US20080249158 Pyrrole derivatives as therapeutic compounds
10/09/2008US20080249157 Novel Inhibitors of the Lfa-1/Icam-1 Interaction and Uses Thereof
10/09/2008US20080249107 Comprising trihydroxy phenyl subunits; selectin inhibitors; side effect reduction; 3-{3-[3-(3,4,5-Trihydroxy-phenyl)-propionylamino]-phenylamino}-benzoic acid
10/09/2008US20080249071 inhibitory activity against the activation of inflammatory cytokines such as interleukin (IL)-1, IL-6, IL-8 and tumor necrosis factor (TNF- alpha ), NF- kappa K B; inflammatory disorders, autoimmune diseases; side effects reduction; immuno suressants; N-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxybenzamide
10/09/2008US20080249030 Age Inhibitors
10/09/2008US20080248584 Trityl derivatives for enhancing mass spectrometry
10/09/2008US20080248539 Ketoreductases of Saccharomyces cerevisiae; host cells
10/09/2008US20080248093 pH sensitive prodrugs of 2,6-diisopropylphenol
10/09/2008US20080247991 Solution Additives For the Attenuation of Protein Aggregation
10/09/2008CA2682473A1 Novel pyrrolinone derivative and pharmaceutical composition comprising the same
10/09/2008CA2681203A1 New methods
10/08/2008EP1978012A1 Alternative synthesis of renin inhibitors and intermediates thereof
10/08/2008EP1976830A1 Method of extracting domoic acid by selective adsorption using a halogenated carboxylic acid derivative
10/08/2008EP1976829A2 N-(6-membered aromatic ring)-amido anti-viral compounds
10/08/2008EP1976828A1 Diamine derivatives as inhibitors of leukotriene a4 hydrolase
10/08/2008EP1419144B1 Oxopyrrolidine compounds, preparation of said compounds and their use in the manufacturing of levetiracetam and analogues
10/08/2008EP1412078B1 Processes for the production of amino-protected derivatives of 4-aminomethylene-pyrrolidin-3-one, gemifloxacin or a salt thereof
10/08/2008EP1341785B1 Hydrolysis of r(r*,r*)-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4- [(phenylamino)carbonyl]-1h-pyrrole-1-heptanoic acid esters with calcium hydroxide
10/08/2008EP1064298B1 Inhibitors of caspases
10/08/2008CN101282937A Therapeutic agents
10/08/2008CN101282786A Catalyst with bimodal distribution of the particles of the catalytically active material, method for the production thereof and for the regeneration thereof and the use of the catalyst
10/08/2008CN101279969A Organic electroluminescent material and application thereof
10/07/2008US7432303 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states
10/07/2008US7432289 5-Acylamino-1,1′-biphenyl-4-carboxamide derivatives and their use as P38 kinase inhibitors
10/07/2008US7432288 Pyrrole-2,5-dione derivatives as Liver X receptor modulators
10/07/2008US7432285 Nitrosated and nitrosylated cyclooxygenase-2 inhibitors, compositions and methods of use
10/07/2008US7432281 4-(2,2-dichloro)-N-(quinolin-3-yl)benzamide; (1R,2R)2-methyl-N-(quinolin-3-yl)-4-(2-(trifluoromethyl)cyclopropyl)benzamide; inflammation-related conditions in mammals, arthritis, Parkinson's/Alzheimer's diseases, stroke, asthma; acute/chronic or neuropathic pain; VR1 agonist/antagonist
10/07/2008US7432225 Synergistic mixture containing cloquintocet-mexyl
10/07/2008CA2179955C Kappa-opiate agonists for inflammatory bowel disorders
10/02/2008WO2008117861A1 Intraocular pressure lowering agents containing phenylenediamine derivatives as the active ingredient
10/02/2008WO2008116814A1 Pyrrole and isoindole carboxamide derivatives as p2x7 modulators
10/02/2008WO2008116385A1 Caffeoyl quinic acid derivatives containing nitrogen, and preparation method, pharmaceutically composition and usage thereof
10/02/2008WO2007117591A9 Total synthesis of salinosporamide a and analogs thereof
10/02/2008US20080242861 Synthesis of amino-protected cyclohexane-1,4-diyldimethanamine and its derivatives
10/02/2008US20080242676 Drug resistant Mycobacterium tuberculosis
10/02/2008US20080242658 Inhibitors of Iap
10/02/2008US20080242656 N-Substituted-N-Sulfonylaminocyclopropane Compounds and Pharmaceutical Use Thereof
10/02/2008US20080242653 Cyclopropyl amine derivatives
10/02/2008US20080242651 3-(2-cyclopentyl-2-phenyl-2-hydroxyacetoxy)-1-(carboxymethyl)-1-methylpyrrolidinium inner salt; muscarinic receptor antagonist; chronic obstructive pulmonary disease or asthma; synergistic mixture with antiinflammatory corticosteroid, betamimetic agent or antiallergic agent
10/02/2008US20080241077 Benzoylguanidine salt and hydrates thereof
10/02/2008US20080235882 Wash, rub and perm fastness; hair, fur, feather and wool fiber coloration; vivid yellow tones; having 3-thienyl, 3-furyl or 3-pyrrolyl ring attached at 5 position
10/02/2008DE102007015034A1 Lactam-substituierte Dicarbonsäuren und ihre Verwendung Lactam substituted dicarboxylic acids and their use
10/01/2008EP1975243A1 A method of isolating stem cells
10/01/2008EP1975158A1 Novel pyrrole derivatives with histone deacetylase inhibitor activity
10/01/2008EP1975157A1 METHOD FOR PRODUCTION OF HETEROAROMATIC RING COMPOUND HAVING N-Rf GROUP
10/01/2008EP1975153A2 Protease inhibitors
10/01/2008EP1973875A1 Compounds and methods for inhibiting the interaction of bcl proteins with binding partners
10/01/2008EP1973656A1 Heterogeneous chiral catalyst
10/01/2008EP1973548A2 Soft protease inhibitors and pro-soft forms thereof
10/01/2008EP1372655B1 Cathepsin cysteine protease inhibitors
10/01/2008CN101277949A Dipeptidyl peptidase-iv inhibitors
10/01/2008CN101277932A Aryl-substituted nitrogen-containing heterocyclic compound
10/01/2008CN101277931A Synthetic processes for the preparation of aminocyclohexyl ether compounds
10/01/2008CN101274938A Preparation for (S) or (R)-2-methyl-CBS-chiral oxazaborolidine and toluene solution thereof
10/01/2008CN101274909A Brominated1-[3-(4-maleimido phenoxyl)propyl] trimethylamin, preparation and application thereof
10/01/2008CN101273987A Use of substituted cyanopyrrolidines and combination preparations containing them for treating hyperlipidemia and associated diseases
10/01/2008CN100422184C Preparation method of meluopeinan
10/01/2008CN100421665C Mitotic kinesin inhibitors
09/2008
09/30/2008US7429659 Isopropyl-piperazin-1-yl)-(5-piperidin-1-ylmethyl-furan-2-yl)-methanone; 5-(4-Fluoro-piperidin-1-ylmethyl)-furan-2-yl]-(4-isopropyl-piperazin-1-yl)-methanone, fumarate salt; insomnia, attention deficit hyperactivity disorders, learning disorders, cognitive dysfunction, eating disorders, obesity
09/30/2008US7429658 Synthesis of protected pyrrolobenzodiazepines
09/30/2008US7429614 Medicament containing an effector of the glutathione metabolism together with α-lipoic acid for treating diabetes mellitus
09/30/2008US7429613 Preparing 5-[2-(4-fluorophenyl)-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrol-1-yl]-3hydroxyl-1-pentanoic acid 7 by reacting aldehyde with 2-hydroxy-1,2,2-triphenylethyl acetate and a chelating cosolvent; hydrolysis; carboxylation by reaction with base; salt formation, purification
09/30/2008US7429603 C-fms kinase inhibitors
09/30/2008US7429587 e.g. 2-(4-Chlorophenyl)-N-{(3S)-1-[(1S)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}ethenesulfonamide; blood coagulation factor and trypsin-like serine protease inhibitor; anticoagulant, antiinflammatory agent; atherosclerotic plaque, myocardial infarction and unstable angina
09/30/2008US7429586 Non-imidazole aryloxyalkylamines
09/25/2008WO2008114857A1 Method for producing aminoacetylpyrrolidinecarbonitrile derivative
09/25/2008WO2008114067A1 Adamantane-dipyrromethane derivatives, method of preparation and applications in anion sensing
09/25/2008US20080234498 Dopamine transporters; therapy for attention deficit disorders; Alzheimer's disease; Parkinson's dosease; antidepressants
09/25/2008US20080234497 Reacting polyoxyethylene glycol with lysine ; enantiomorphic pure product
09/25/2008US20080234344 Amino Acid and Peptide Conjugates of Arylalkylic Acids for Cosmetic Use
09/25/2008US20080234292 Such as S)-(1-(1-Aminobicyclo[2.2.2]oct-4-yl)aminoacetyl)-2-cyanopyrrolidine; inhibitors of the enzyme dipeptidyl peptidase; antidiabetic agents
09/25/2008US20080234270 For modulating activity of one or more steroid nuclear receptors and for treatment, prevention, or amelioration of symptoms of disease or disorder related to the activity of receptors; 5-benzo[b]thiophen-2-yl-1,4-dimethyl-1H-pyrrole-3-carboxylic acid (4-methanesulfonyl-phenyl)-amide
09/25/2008US20080234247 Heterocyclic analgesic compounds and methods of use thereof
09/25/2008US20080234209 Derivatives of N-methyl-N-[(1S)-1-phenyl-2-((3S)-3-hydroxypyrrolidin-1-yl)ethyl]-2,2-diphenylacetamide; for preparation of drugs, gastrointestinal tract disease
09/25/2008US20080234202 Reacting carboxylic acid or amide derivative with amine compound to obtain amino acid analogs, peptides containing analogs of basic amino acids lysine and arginine; desamino amino acid compound, of the extended or truncated peptide; pain, psychosis, obesity; cosmetics
09/25/2008US20080230482 Optically active polymaleimide derivatives and process for their production
09/25/2008US20080230123 Photoelectric conversion element and solid-state imaging device
09/24/2008EP1971864A2 Kit comprising 2,4-dichlorophenoxyacetic acd derivatives and antibodies for highly sensitive detection assays
09/24/2008EP1163211B1 Method for acylating peptides and proteins