Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304) |
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07/10/2008 | US20080167462 2-substituted phenyl-5, 7-dehydrocarbyl-3, 7-dihydropyrrolo [2, 3-d] pyrimidin-4-one derivatives, the preparation and the pharmaceutical use thereof |
07/10/2008 | US20080167368 4-{4-[3-(2-fluoro-5-trifluoromethylphenyl)ureido]phenyl}-1H-pyrrole-3-carboxamide; anticarcinogenic agents; FAK, KDR and Tie2 kinase inhibitors |
07/10/2008 | US20080167366 Use of 2-oxo-1-pyrrolidine derivatives for the preparation of a drug |
07/10/2008 | US20080167361 Piperazinyl-substituted quinolinone compounds ;to treat nervous system diseases, neurodegenerative diseases; gastrointestinal tract disorders; cognition enhancers; 3-[4-(3-Ethylsulfanyl-benzenesulfonyl)-2-methoxy-phenyl]-pyrrolidine and 5-(3-Ethylsulfanyl-benzenesulfonyl)-2-pyrrolidin-3-yl-phenol |
07/10/2008 | US20080167318 Pharmaceutically active pyrrolidine derivatives |
07/10/2008 | US20080167306 Novel Heteroaryl Derivative |
07/10/2008 | US20080167288 Substituted cyclic hydroxamates as lnhibitors of matrix metalloproteinases |
07/09/2008 | EP1940813A1 Heterocyclic amide derivatives useful as microbiocides |
07/09/2008 | EP1940805A1 Benzodiazepine and benzopiperazine analog inhibitors of histone deacetylase |
07/09/2008 | EP1940782A1 N-phenyl phenylacetamide non-nucleoside reverse transcriptase inihibitors |
07/09/2008 | EP1940390A2 Antibacterial pyrrols |
07/09/2008 | EP1940387A1 Process for the stereoselective preparation of (-)-halofenate and intermediates thereof |
07/09/2008 | EP1720825B1 Anthranilic acid derivatives, methods for their preparation and use as dhodh inhibitors |
07/09/2008 | EP1673084B1 1-2' (1,4'-biperidin-1'-yl)-1-(phenyl)-ethylcyclohexanol derivatives as monoamine reuptake modulators for the treatment of vasomotor symptoms |
07/09/2008 | CN101218240A Process for preparing bicyclic compounds |
07/09/2008 | CN101218239A Process for preparing bicyclic compounds |
07/09/2008 | CN101215285A Polyhydroxy substituted octahydroindolizidine and synthesis method thereof |
07/09/2008 | CN101215255A Method for preparing N-(2-methylphenyl)maleimide |
07/09/2008 | CN101215254A Method for purifying N-(3-methylphenyl)maleimide |
07/09/2008 | CN101215253A Crystalline forms of atorvastatin |
07/09/2008 | CN101215252A Method for preparing N-Boc or N-Cbz derivatives of chiral alpha,alpha'-disubstituted pyrrolidines containing olefinic bond and acetylene bond |
07/09/2008 | CN100400509C Pyrrolidone derivatives as MAOB inhibitors |
07/09/2008 | CN100400487C Glucocorticoid receptor modulators |
07/08/2008 | US7396851 Heterocyclic and benzoheterocyclic polyamides structurally related to the natural antibiotic distamycin A for the treatment of β-thalassaemia |
07/08/2008 | US7396846 Growth hormone secretagogues |
07/08/2008 | US7396844 3-(4-amidinobenzoylamino)-4-[5-amidino-2-(2-carboxy-2-oxoethyl)phenoxy]butanoic acid; anticoagulant; blood coagulation factor X and thrombin inhibitor; cerebral infarction, thrombosis, embolism, transient ischemic attack (TIA) and subarachnoidal hemorrhage (vasospasm); ischemic heart diseases |
07/08/2008 | US7396828 PI-3 kinase inhibitor prodrugs |
07/03/2008 | WO2008079266A2 Synthesis of pyrrolidine compounds |
07/03/2008 | WO2008078762A1 Novel n-(2-aminophenyl)benzamide derivative having an urea structure |
07/03/2008 | WO2008078341A2 Stable pharmaceutical formulations of atorvastatin magnesium salt |
07/03/2008 | WO2008077897A1 New products for the treatment of the iron chlorosis |
07/03/2008 | WO2007123686A3 Dpp inhibitors and uses thereof |
07/03/2008 | WO2007107276A3 Process for preparing c7 intermediates and their use in the preparation of n-substituted pyrrole derivatives |
07/03/2008 | US20080161577 Muscarinic receptor antagonists; longer duration of action; side effect reduction; high potency; chronic obstructive pulmonary disease; asthma; inhalation; 2-[(S)-1-(8-Methylaminooctyl)pyrrolidin-3-yl]-2,2-diphenylacetamide |
07/03/2008 | US20080161325 e.g. N1-[3-amino-4-(3,5-difluorophenyl)-2-hydroxybutyl]-3-(butylsulfonyl)-N1-(3-ethylbenzyl)-D-alaninamide dihydrochloride; inhibitors of amyloid beta-secretase enzyme; neurodegenerative diseases: Alzheimer's, Parkinson's diseases, Down's syndrome |
07/03/2008 | US20080161310 (2S)-4,4-difluoro-1-(2-{[1-(2-pyrazinyl)piperidin-4-yl]amino}acetyl)-2-pyrrolidine carbonitrile; enzyme inhibitors; diabetes |
07/03/2008 | US20080161306 Pyrrole Derivatives as Dna Gyrase and Topoisomerase Inhibitors |
07/03/2008 | US20080161281 Amino-Substituted Tricyclic Derivatives and Methods of Use |
07/03/2008 | US20080160017 Cross-Linked Antibodies |
07/03/2008 | CA2674548A1 Novel n-(2-aminophenyl) benzamide derivative having urea structure |
07/03/2008 | CA2673466A1 Substituted tetracycline compounds |
07/03/2008 | CA2672727A1 Sphingosine-1-phosphate receptor agonist and antagonist compounds |
07/02/2008 | EP1939625A2 Methods for ligand discovery |
07/02/2008 | EP1939175A1 Sulfonamide derivative having pgd2 receptor antagonistic activity |
07/02/2008 | EP1939157A1 New products for the treatment of the iron chlorosis |
07/02/2008 | EP1937664A1 Hydrazide compound and pesticidal use of the same |
07/02/2008 | EP1937637A1 New n-alkyl-heterocyclyl carboxamide derivatives |
07/02/2008 | EP1937634A1 Cathepsin cysteine protease inhibitors |
07/02/2008 | EP1937632A1 Novel compounds |
07/02/2008 | EP1937252A2 Methods and compositions for stimulating neurogenesis and inhibiting neuronal degeneration |
07/02/2008 | EP1937242A2 Methods and compositions for the treatment of neuropsychiatric and addictive disorders |
07/02/2008 | EP1830841B1 Cycloalkyl lactam derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1 |
07/02/2008 | EP1729773B1 8-hydroxy-5- [(-hydroxy-2- [[ (1r)-2-(4-methoxyphenyl)-1-methylethyl] amino ][ethyl -2(1h)-quinolinone monohydrochloride in crystalline form and the process for its preparation |
07/02/2008 | EP1648858B1 Method for production of alpha, beta-unsaturated amide compounds |
07/02/2008 | EP1646626B1 Pyrrole-2, 5-dione derivatives as liver x receptor modulators |
07/02/2008 | EP1646625B1 Pyrrole-2, 5-dithione derivatives as liver x receptor modulators |
07/02/2008 | EP1633702B1 Protease inhibitors |
07/02/2008 | EP1496838A4 Substituted amides |
07/02/2008 | EP1487791B1 A novel antifungal molecule 2-(3,4-dimethyl-2,5-dihydro-1h-pyrrol-2-yl)- methylethyl pentanoate |
07/02/2008 | CN101213171A New crystalline atorvastatin hemicalcium salt polymorph form |
07/02/2008 | CN101209987A Thermosetting resin composition containing maleimide and/or vinyl compound |
07/02/2008 | CN100398517C substituted pyrrolidone synthesized ion liquid and its synthesis method |
07/01/2008 | US7393873 Arylsulfonamide derivatives |
06/26/2008 | WO2008077035A2 Processes for the preparation of levetiracetam |
06/26/2008 | WO2008076754A2 Compounds and compositions as inhibitors of cannabinoid receptor 1 activity |
06/26/2008 | WO2008075353A1 Sulfonamide derivatives with therapeutic indications |
06/26/2008 | WO2008075165A1 Novel process for the synthesis of [r-(r*, r*)]-2-(4-fluorophenyl)-beta, delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoic acid or a pharmaceutically acceptable salt thereof |
06/26/2008 | WO2008074703A1 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives |
06/26/2008 | WO2008014311A3 Inhibitors of undecaprenyl pyrophosphate synthase |
06/26/2008 | WO2008002820A3 Substituted benzyl amine compounds |
06/26/2008 | US20080153896 Polymorphic Forms of an HMG-CoA Reductase Inhibitor and Uses Thereof |
06/26/2008 | US20080153892 1-(Urea-, thiourea- and cyanoguanidine-methylene)benzyl)imidaoles, treatment of neuronal disorders, especially Alzheimer's disease, Down Syndrome, Parkinson's disease and Huntington's disease |
06/26/2008 | US20080153836 1H-Quinazoline-2,4-Diones |
06/26/2008 | US20080153826 substituted aryl cycloalkanoyl derivatives, compositions containing these derivatives, and methods of their use for the prevention and treatment of conditions ameliorated by monoamine reuptake including, inter alia, vasomotor symptoms (VMS), sexual dysfunction, gastrointestinal and genitourinary disorder |
06/26/2008 | US20080153821 Nitrogen-containing 5-membered ring compound |
06/26/2008 | US20080152619 Hepatitis C virus inhibitors |
06/26/2008 | US20080152588 Metal Chelators and Methods of Their Use |
06/26/2008 | CA2695613A1 Sulfonamide derivatives with therapeutic indications |
06/26/2008 | CA2672271A1 Compounds and compositions as inhibitors of cannabinoid receptor 1 activity |
06/26/2008 | CA2671378A1 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives |
06/25/2008 | EP1935881A1 Aryl-substituted nitrogen-containing heterocyclic compound |
06/25/2008 | EP1935879A1 Substituted cycloalkene derivative |
06/25/2008 | EP1935869A1 Retinoids for the treatment of emphysema |
06/25/2008 | EP1934177A1 Prolinamide derivatives as sodium channel modulators |
06/25/2008 | EP1934176A1 Quaternary alpha-aminocarboxamide derivatives as modulators of voltage-gated sodium channels |
06/25/2008 | EP1193253B1 Process for producing optically active azetidine-2-carboxylic acids |
06/25/2008 | EP0986382B1 Raf kinase inhibitors |
06/25/2008 | CN101208334A Novel cyclic amines |
06/25/2008 | CN101208300A Derivatives of 4,5-diarylpyrrole, preparation method thereof and use of same in therapeutics |
06/25/2008 | CN101205209A Method for refining atorvastatin intermediate |
06/25/2008 | CN100396756C Material for light-oriented film, light-oriented film and its manufacture method |
06/25/2008 | CN100396679C Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase |
06/25/2008 | CN100396668C Non-imidazole aryloxypiperidines |
06/25/2008 | CN100396667C Unsaturated five heterocycle compound for up-regulating bone formation protein BMP-2 expression activity |
06/25/2008 | CN100396666C (4S)-1-tert butoxy carbonyl-4-amino-L-ethyl prolinate and its synthesis technology |
06/25/2008 | CN100396665C Pyrrolidine derivative, preparation method thereof and pharmaceutical composition containing the compound |
06/24/2008 | US7390910 Antitumor, anticancer agents; for drug resistant tumors, cancers |
06/24/2008 | US7390890 1,4-Dideoxy-1-C-(4-hydroxypyrrolo[3,2-d]pyrimidin-7-yl)-1,4-imino-D-ribitol derivatives or salts; parasite purine nucleoside, -hydrolase, -phosphorylase and/or phosphoribosyl transferase inhibitors; antiprotozoa, anticarcinogenic, antiinflammatory, and immunosuppressant agents; autoimmune diseases |
06/24/2008 | US7390835 Aralkyl amines as cannabinoid receptor modulators |
06/24/2008 | US7390830 MIP-1 alpha and/or MCP-1 antagonists; rheumatoid arthritis; nephritis; multiple sclerosis; nephropathy |