Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
12/1995
12/12/1995US5475021 Compounds and compositions for inhibition of cyclooxygenase activity
12/12/1995US5475017 Diaryl-substituted heterocyclic compounds, drugs and cosmetics obtained therefrom
12/12/1995US5475004 Angiotensin II receptor antagonists for the treatment and prophylaxis of coronary heart disease
12/12/1995US5474995 Phenyl heterocycles as cox-2 inhibitors
12/11/1995CA2151412A1 Modified guanidino and amidino thrombin inhibitors
12/07/1995WO1995032949A1 Gastrin and cck antagonists
12/07/1995WO1995032945A1 Compositions and methods for treating mast-cell mediated conditions
12/07/1995WO1995032937A1 TETRAHYDROINDENO[1,2-d][1,3,2]OXAZABOROLES AND THEIR USE AS ENANTIOSELECTIVE CATALYSTS
12/07/1995DE4419587A1 Heterocyclische Imino-Derivate Heterocyclic imino derivatives
12/06/1995EP0685457A1 Glycerol derivative, device and pharmaceutical composition
12/06/1995EP0685234A1 Drug composition containing nucleic acid copolymer
12/06/1995EP0684945A1 Heterocyclic-substituted alkyl amide acat inhibitors
12/06/1995EP0684830A1 Inhibitors of thrombosis
12/06/1995EP0588850B1 N-hydroxyurea derivatives which inhibit lipoxygenase
12/05/1995US5473081 Reacting proline with acylthiopropionic acid halide, deacylating product
12/05/1995US5473077 4-aminopyrrolidine-2,4-substitude independently with carboxylic acid or 5-tetrazolyl for treating nervous system disorders and psychological disorders
12/05/1995US5472984 1,2-ethanediol derivative and salt thereof and cerebral function-improving agent comprising the same
12/05/1995US5472978 Aromatic compounds, pharmaceutical compositions containing them and their use in therapy
12/05/1995US5472976 Poly 4-aminopyrrole-2-carboxyamide derivatives, and pharmaceutical compositions which contain them
12/05/1995US5472946 Transdermal penetration enhancers
12/05/1995US5472933 Plant growth regulators
12/05/1995CA1337698C Pyrethroids and their use for controlling pests
11/1995
11/30/1995DE4418304A1 Novel N-alkyl cyclohexyl maleimide, useful esp. for polymers prodn.
11/29/1995EP0684240A1 Hydroxamic acid derivatives with tricyclic substitution
11/29/1995EP0683770A1 Substituted tetrahydropyridazine carboxamides
11/29/1995EP0683767A1 Azacyclic compounds, compositions containing them and their use as tachykinin antagonists
11/29/1995CN1112548A Polyiodinated compounds, process for preparing them and diagnostic compositions
11/28/1995US5470981 Process for trans-6-[2-(substituted-pyrrol-1-yl)alkyl]pyran-2-one inhibitors of cholesterol synthesis
11/28/1995US5470878 Cell signaling inhibitors
11/28/1995US5470863 Oximic derivatives with a fungicide activity
11/28/1995US5470858 Derivatives of (hetero)aromatic ethers and thioethers having antihyperlipidemic activity, process for their preparation and pharmaceutical compositions containing them
11/28/1995US5470848 Penetration enhancers for transdermal delivery of systemic agents
11/28/1995CA2025959C Process for optically active 2-alkyl-2,5-diazabicyclo[2.2.1]heptanes
11/23/1995WO1995031433A1 Derivatives of aminosulfonic acids, utilization of the same in the synthesis of pseudopeptides and process for their preparation
11/23/1995WO1995031429A1 Photocleavable agents and conjugates for the detection and isolation of biomolecules
11/23/1995CA2189896A1 Derivatives of aminosulfonic acids, utilization of the same in the synthesis of pseudopeptides and process for their preparation
11/22/1995EP0682653A1 Process for the production of pure vinyl pyrrolidone
11/22/1995CN1112104A Acetic acid derivatives
11/22/1995CN1030353C Nonlinear optical materials
11/21/1995USRE35096 Antilipemic, anticholesterol, arteriosclerosis
11/21/1995US5468877 For protecting crops
11/21/1995US5468876 Intermediates for the stereoconservative synthesis of 1-substituted (S)-and (R)-2-aminomethylpyrrolidines
11/21/1995US5468857 Fungicides
11/21/1995US5468774 Antiinflammatory agents
11/21/1995US5468764 Administering to a mammal an azole derivative
11/21/1995US5468733 For treating cancer
11/21/1995US5468731 Peptide compounds, a process for preparation thereof and pharmaceutical composition comprising the same
11/21/1995US5468404 Lubricating oil additives, their preparation and use
11/16/1995WO1995030661A1 Substituted aromatic thiocarboxylic acid amides and their use as herbicides
11/16/1995WO1995030647A1 Cck and gastrin receptor ligands
11/16/1995WO1995030646A1 Compounds containing a michael-acceptor, especially maleimide or maleic acid derivatives, directly or indirectly linked to a chromophore and their use in long lasting sunscreen compositions
11/16/1995WO1995030644A1 Amide derivatives and their therapeutic use
11/16/1995WO1995030641A1 Nitro compounds and their compositions having anti-inflammatory, analgesic and anti-thrombotic acitivities
11/16/1995CA2189337A1 Compounds containing a michael-acceptor, especially maleimide or maleic acid derivatives, directly or indirectly linked to a chromophore and their use in long lasting sunscreen compositions
11/15/1995EP0682028A1 5,6-Dihydro-4H-thieno 3,4-C pyrroleerivatives, their preparation and their therapeutic use
11/15/1995EP0682027A1 Pyrrolopyrimidine derivatives with antiproliferative action
11/15/1995EP0682013A1 Novel process for the preparation of enantiomerically pure diarylprolinols
11/15/1995EP0681572A1 Cyclic imide thione activated polyalkylene oxides
11/14/1995US5466828 Chiral 3-cyano-1-substituted-pyrrolidines
11/14/1995US5466684 7-(substituted)-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
11/11/1995CA2148880A1 5,6-dihydro-4h-thieno[3,4-c]pyrrole derivatives; process for preparing the same and their use as therapeutic agents
11/09/1995WO1995029916A1 Electron-deficient porphyrins and processes and intermediates for preparing same
11/09/1995WO1995029892A1 Hydroxamic acid and amino acid derivatives and their use as anti-arthritic agents
11/09/1995WO1995029891A1 N-(3-pyrrolidinyl)benzamide derivative
11/09/1995DE19500439A1 Substituierte aromatische Thiocarbonsäureamide Substituted aromatic Thiocarbonsäureamide
11/09/1995CA2187949A1 Electron-deficient porphyrins and processes and intermediates for preparing same
11/09/1995CA2187429A1 N-(3-pyrrolidinyl)benzamide derivative
11/08/1995EP0680963A1 (Hydroxyphenylamino)carbonyl pyrroles
11/08/1995EP0680484A1 OPTICALLY ACTIVE $g(b)-AMINOALKOXYBORANE COMPLEX
11/08/1995EP0680320A1 Stable oral ci-981 formulation and process of preparing same
11/08/1995EP0434765B1 Targeting substance-diagnostic/therapeutic agent conjugates having schiff base linkages
11/08/1995CN1111457A Thermoplastic resin composition and process for molding the same
11/07/1995US5464809 Fungicidal 2-methoximinocarboxylic esters
11/07/1995US5464739 Urinalysis, hydrolysis of lactate ester
11/04/1995CA2148324A1 Pyrrolopyrimidine derivatives having pharmacological activity
11/02/1995WO1995029158A1 Heterocyclylbenzonitriles
11/02/1995WO1995029148A1 O-acyl-4-phenyl-cyclohexanols, their salts, medicaments containing such compounds and their use, as well as a method of preparing them
11/02/1995EP0679157A1 Novel 3,4-diaryl thiophenes and analogs thereof having use as antiinflammatory agents
11/02/1995EP0679084A1 Hydantoin and succinimide-substituted derivatives of spiroindanylcamphorsulfonyl oxytocin antagonists
11/02/1995DE4414568A1 Heterocyclylbenzonitrile Heterocyclylbenzonitriles
11/02/1995CA2188294A1 Synthesis of prototypes for renin inhibitors
10/1995
10/31/1995US5463122 Arylthio compounds
10/31/1995US5463083 2,5-diaryl tetrahydrothiophenes, tetrahydrofurans and 1,3-diaryl-cyclopentanes which act as platelet activating factor receptor antagonists and/or inhibitors of the enzyme 5-lipoxygenase
10/31/1995US5463080 Isotopic 5-((4-carboxy-1-oxobutyl)amino)-2,4,6-triiodo-1,3-benzenedicarboxylic acid, dimethyl ester for indirect radiohalogenation of proteins; non-deiodination in vivo
10/31/1995US5463079 Preparation of five-membered nitrogen heterocycles
10/31/1995US5463078 Anisomycin derivatives and anticancer agents, antifungal agents and antiprotozoan agents containing the same
10/31/1995US5463076 Crosslinking phenylimide end caps condensed onto aromatic hub through ether linkages
10/31/1995US5463064 Vasodilating and hypotensive activity
10/31/1995US5463062 Inhibitors of glucose-6-phosphatase system
10/31/1995US5463052 Method for producing benzylidene derivatives
10/31/1995US5462964 Dipeptide boronic acid inhibitors of trypsin-like enzymes
10/31/1995US5462947 Nervous system disorders
10/31/1995US5462946 Metal-independent nitroxide or oxazolidine-1-oxyl forming compound in biologically acceptable carrier to protect biological material from oxidative stress
10/31/1995CA2030421C Agent for treatment of cerebrovascular contraction
10/26/1995WO1995028286A1 Dye diffusion thermal transfer printing
10/26/1995WO1995028177A1 Medicinal composition for treating tardive dyskinesia and utilization thereof
10/26/1995CA2187086A1 A pharmaceutical composition for therapeutically treating tardive dyskinesia and uses therof
10/25/1995EP0678507A1 Method for preparing homochiral maleimide intermediates, via silylation techniques, used in the enantioselective preparation of anti-thrombotic and anti-vasospastic compounds
10/25/1995EP0678503A1 Delta-amino-gamma-hydroxy-omega-aryl alkanoic acid amides with enzyme especially renin inhibiting activities
10/25/1995EP0678089A1 N-acyl pyrrolidines and drugs for the treatment or prevention of cholecystokinin and gastrin-related disorders.