Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
05/1996
05/30/1996WO1996015792A1 Methods for treating or preventing alzheimer's disease using substituted 1-aryl-3-piperazin-1'-yl propanones
05/30/1996DE4441984A1 New tri:fluoromethyl-pyrrolidinone derivs.
05/30/1996CA2205586A1 Certain substituted 1-aryl-3-piperazin-1'-yl propanones
05/30/1996CA2205504A1 Certain substituted 1-aryl-3-piperazin-1'-yl propanones
05/30/1996CA2205412A1 Bleaching compositions and bleach-additives comprising bleach activators effective at low perhydroxyl concentrations
05/29/1996EP0713868A1 Process for the manufacture of insecticidal arylpyrroles via oxazole amine intermediates
05/29/1996EP0713866A1 Process for preparing 4-mercaptopyrrolidine compound
05/29/1996EP0713864A1 Substituted benzoylguanidines, process for their preparation, their use as medicament of diagnostic agent as well as medicaments containing them
05/29/1996EP0713483A1 Amidine derivatives with nitric oxide synthetase activities
05/29/1996EP0311632B1 Surface active lactams
05/29/1996CN1123545A Guanidine derivatives as inhibitors of Na+/H+ exchange in cells
05/29/1996CN1123544A Optically active 3-(1-(alkylamino)) alkyl pyrrolidines
05/29/1996CN1031880C Process for preparing novel analogs of peptidase substrates
05/28/1996US5521290 Reaction of maleimide groups of bifunctional linking compounds with molecules to be linked, then reacting remaining aldehyde and hydrazide groups of linking compounds
05/28/1996US5521211 Insecticides, nematocides
05/28/1996US5521206 Hypotensive agents, treatment of atherosclerosis
05/28/1996US5521182 1,2,3,4 tetrahydropteridinone cyclic amide derivatives
05/25/1996CA2163598A1 Substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
05/23/1996WO1996015108A1 Pyrrolidinyl di-carboxylic acid derivatives as metabotropic glutamate receptor agonists
05/23/1996WO1996015104A2 Methods and compositions for treating phytopathogenic fungi infections
05/23/1996WO1996015096A1 Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitiors
05/23/1996WO1996014856A1 Cancer inhibitory peptides
05/23/1996WO1996014844A1 Cyclic amidine analogs as inhibitors of nitric oxide synthase
05/23/1996CA2204767A1 Pyrrolidinyl di-carboxylic acid derivatives as metabotropic glutamate receptor agonists
05/23/1996CA2203681A1 Cyclic amidine analogs as inhibitors of nitric oxide synthase
05/23/1996CA2163327A1 Process for the manufacture of insecticidal arylpyrroles via oxazole amine intermediates
05/23/1996CA2162786A1 Heterocyclic tachykinin receptor antagonists
05/22/1996EP0712387A1 2-aminoindans as selective dopamine d3 ligands
05/21/1996US5519142 Homobidental, trifunctional linkers, method for their preparation and use in immunologically active conjugates
05/21/1996US5519134 Pyrrolidine-containing monomers and oligomers
05/21/1996US5519052 Insecticides using phenolic furanone derivatives
05/21/1996US5518650 Imidocarboxylic acid activators and sulfimidocarboxylic acid activators, processes for their preparation and their use
05/17/1996WO1996014296A1 Novel pyrrolinone-based compounds
05/17/1996CA2204014A1 Process for the production of acyl lactams
05/15/1996EP0711755A1 Pyrrolidinyl di-carboxylic acid derivatives as metabotropic glutamate receptor antagonists
05/15/1996EP0711554A1 Antidepressant
05/15/1996EP0711279A1 2-phenylpyrrole derivatives as dopamine d3 receptor antagonists
05/15/1996EP0711278A1 2-(2-hydroxyphenyl)-5-(n-phenylmethyl-aminomethyl)-pyrroles as antipsychotic agents
05/15/1996EP0711177A1 Improvements relating to prodrugs
05/15/1996CN1122600A Second messenger cell signaling inhibitors
05/15/1996CN1122594A Deallylation reagent and deallylation method using said reagent
05/14/1996US5516931 Release tag compounds producing ketone signal groups
05/14/1996US5516797 Suppressing graft rejection
05/14/1996US5516783 Platelet activating factor
05/09/1996WO1996013502A1 Phenyloxazolidinone antimicrobials
05/09/1996WO1996013491A1 Bisarylcarbinol cinnamic acids as inhibitors of leukotriene biosynthesis
05/09/1996WO1996013266A1 Boronic ester and acid compounds, synthesis and uses
05/08/1996EP0710109A1 Compounds
05/08/1996CN1121917A Derivative of 3-benzol pyrrole alkyl
05/08/1996CN1121806A Pharmaceutical agents for treatment of emesis
05/08/1996CN1031752C Process for preparing pyrolidine carboxylic acid derivatives
05/07/1996US5514815 Succinimide derivatives and process for preparing the same
05/07/1996US5514814 Pyrrolinone-based compounds
05/07/1996US5514777 Methods of synthesis of peptidyl argininals
05/07/1996US5514702 Arylamidoalkyl-N-hydroxyurea compounds having lipoxygenase inhibitory activity
05/07/1996US5514701 Thromboxane a2 antagonist
05/07/1996US5514683 Bicyclo 2,2,2!octane derivatives
05/07/1996US5514678 Arthropodicidal 1,2,4-triazinyl amides
05/07/1996US5514677 Hydroxamic acid based collagenase inhibitors
05/02/1996WO1996012697A2 Calcium receptor-active compounds
05/02/1996WO1996012499A1 Amidino and guanidino substituted inhibitors of trypsin-like enzymes
05/02/1996DE4438083A1 New aminoalkylphenyl substd. acyl-pyrrolidine or piperidine derivs.
05/02/1996DE4437999A1 New N,N-di:substd. aryl-cycloalkyl-amine derivs.
05/01/1996EP0709373A1 Novel pyrrolidine derivative
05/01/1996EP0709372A1 N-arylthiohydrazone derivatives as insecticidal and acaricidal agents
05/01/1996EP0708765A1 Substituted piperazinylcamphor derivatives as oxytocin antagonists
05/01/1996CN1121716A 3-halo-3-heteroaryl carboxylic acid derivatives, methods of preparing them and intermediates used in their preparation
05/01/1996CN1121511A Ester compounds and noxious life-controlling agents containing the same as an active ingredient
04/1996
04/30/1996US5512667 Trifunctional intermediates for preparing 3'-tailed oligonucleotides
04/30/1996US5512579 Aminobenzoic acid derivatives
04/30/1996US5512560 Conformationally restricted HIV-1 protease inhibitors
04/30/1996US5512553 Preventing or treating bacterial infections
04/30/1996US5512450 Test device for determining the presence of leukocyte cells, esterase or protease in a test sample
04/30/1996US5512290 Powder-form on support
04/30/1996US5512204 Curing, crosslinking agent; fireproofing
04/28/1996CA2161375A1 N-arylthiohydrazone derivatives as insecticidal and acaricidal agents
04/25/1996WO1996011902A1 Pharmaceutically active substituted aromatic compounds
04/25/1996WO1996011697A1 Thrombin inhibitors
04/24/1996EP0708090A1 Intermediates useful for the synthesis of pesticides
04/24/1996EP0708085A2 Antiviral ethers of aspartate protease substrate isosteres
04/24/1996EP0707586A1 Positive inotropic and lusitropic pyrroloquinolinone derivatives
04/24/1996EP0707584A1 Novel (1-heteroazolyl-1-heterocyclyl)alkane derivatives and their use as neuroprotective agents
04/24/1996EP0707576A1 Substituted aryl-keto-enolic heterocycles
04/24/1996EP0691954A4 Asymmetrical polypyrrolidonyl compounds having a wide liquid range
04/24/1996EP0625142B1 Process for producing pyrrolidone and n-alkyl pyrrolidones
04/24/1996CN1121068A Prolineamide derivatives
04/23/1996US5510488 Chemical intermeidates
04/23/1996US5510477 Process for the acylation of lactams
04/23/1996US5510369 Pyrrolidine thrombin inhibitors
04/23/1996US5510344 Acrylate fungicides
04/20/1996CA2160763A1 Antiviral ethers of aspartate protease substrate isosteres
04/18/1996WO1996011192A1 Lta4 hydrolase inhibitors
04/18/1996WO1996011183A1 N-(ortho-substituted benzyloxy)imine derivatives and their use as fungicides, acaricides or insecticides
04/18/1996WO1996010999A2 Lta4 hydrolase inhibitor pharmaceutical compositions and methods of use
04/18/1996CA2202371A1 Lta4 hydrolase inhibitors
04/18/1996CA2202368A1 Lta4 hydrolase inhibitor pharmaceutical compositions and methods of use
04/18/1996CA2200590A1 N-(ortho-substituted benzyloxy)imine derivatives and their use as fungicides, acaricides or insecticides
04/17/1996EP0706999A1 Novel dipiperidine derivative
04/17/1996EP0600952B1 Azacyclic compounds, processes for their preparation and pharmaceutical compositions containing them
04/17/1996EP0558656B1 New methods for the catalytic reduction of organic substrates