Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
01/1996
01/24/1996CN1030765C 2-aryl-5-trifluoromethyl-2-pyrroline compounds and process for manufacture of insecticidal, 2-aryl-1(alkoxymethyl)-4-halo-5-(trifluoromethyl)
01/23/1996US5486623 Cysteine protease inhibitors containing heterocyclic leaving groups
01/23/1996US5486620 Intermediates for the synthesis of kainic acid
01/23/1996US5486528 Antiulcer agents, anxiolytic agents
01/23/1996US5486527 Anticholinergic agents
01/23/1996US5486275 Decarbonylation an acyl bromide derivative with exposure to ultraviolet light
01/18/1996WO1996001253A2 Pla2 inhibitors and their use for inhibition of intestinal cholesterol absorption
01/18/1996DE4425781A1 Technetium-Sulfonamid-Komplexe, deren Verwendung, diese enthaltende pharmazeutische Mittel, sowie Verfahren zur Herstellung der Komplexe und Mittel Technetium-sulfonamide complexes, their use, pharmaceutical compositions containing them, and processes for producing the complexes and agents
01/18/1996CA2191775A1 Pla2 inhibitors and their use for inhibition of intestinal cholesterol absorption
01/17/1996EP0692471A1 Process for the preparation of optically active 3-hydroxypyrrolidine derivatives with high optical purity
01/17/1996EP0692470A1 Process for the preparation of optically active 1-substituted-2-(aminomethyl)pyrrolidine derivatives
01/17/1996EP0692011A1 Fuel compositions
01/17/1996EP0691962A1 1-amino-3-phenoxy propane derivatives as modulators of multi-drug resistance
01/17/1996EP0691954A1 Asymmetrical polypyrrolidonyl compounds having a wide liquid range
01/17/1996EP0691953A1 1-amidinophenyl-pyrrolidones piperidinones azetinones as platelet aggregation inhibitors
01/17/1996EP0691950A1 Imino-substituted phenylacetic acid amides, their preparation and fungicides containing them
01/17/1996EP0691845A1 Use of cis- or transurocamic acid for the treatment of photodermatoses and immunogenic skin diseases
01/17/1996EP0602028B1 Aromatic sulfonamide derivatives, their use as enzyme inhibitors and pharmaceutical compositions containing them
01/17/1996EP0537313B1 Arylalkyl esters of 4,5-dihydroxy-9,10-dihydro-9,10-dioxo-2-anthracenecarboxylic acid having therapeutical activity
01/17/1996CN1030702C 芪衍生物 Stilbene derivatives
01/17/1996CN1030699C Process for preparation of insecticidal acaricidal and nematicial 2-aryl-5-(triflumethyl) pyrrole compounds
01/16/1996US5484948 Bismaleimide compounds
01/16/1996US5484946 Cyclization and dehydration a methionine derivative
01/16/1996US5484926 HIV protease inhibitors
01/16/1996US5484925 Synthesis of (-)-swainsonine and intermediate compounds employed in such synthesis
01/16/1996US5484807 Haloalkylthio, -sulfinyl and -sulfonyl arylpyrrole insecticidal and acaricidal agents
01/16/1996US5484797 Naphthly compounds, intermediates, processes, compositions, and method for inhibiting endometrosis
01/16/1996US5484796 Naphthyl compounds, intermediates, processes, compositions, and method of inhibiting aortal smooth muscle cell proliferation
01/16/1996US5484795 Naphthyl compounds, intermediates, processes, compositions, and method of inhibiting restenosis
01/16/1996US5484763 Substituted benzisoxazole and benzisothiazole herbicidal agents
01/16/1996US5484722 Biopolymer and effector substance conjugates, process for the preparation thereof and their use
01/16/1996CA1337938C Hydrophilic modifier monomers
01/11/1996WO1996000720A1 Aryl and heteroaryl alkoxynaphthalene derivatives
01/11/1996DE4424294A1 Prodn. of poly:ene-carbonyl cpds. with high all-E content
01/11/1996DE4423603A1 N-alkyl lactam prodn. from lactam
01/10/1996EP0691330A1 Ester compounds and noxious life-controlling agents containing the same as an active ingredient
01/10/1996EP0691129A2 Thiazolidone and pyrrolidinone compounds for inhibiting bone loss
01/10/1996EP0691128A1 Methods of administering CRF antagonists
01/10/1996EP0690851A1 Guanidine derivatives useful in therapy
01/10/1996EP0690840A1 Novel distamycin analogues
01/10/1996EP0600949B1 New 3,5-di-tert.butyl-4-hydroxyphenyl derivatives, methods of preparing them and drugs containing them
01/09/1996US5482957 Azole derivatives, process for their preparation and their use
01/09/1996US5482938 Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment
01/09/1996US5482921 Herbicides
01/07/1996CA2153213A1 Methods of inhibiting bone loss
01/04/1996WO1996000214A1 Arylsulfonamido-substituted hydroxamic acids as matrix metalloproteinase inhibitors
01/03/1996EP0689536A1 Naphthalene derivatives
01/03/1996EP0553130B1 Pyrrolidine dione derivatives
01/02/1996US5481036 Renin inhibitors, hypotensive agents
01/02/1996US5480998 Oxime derivative
01/02/1996US5480720 Adhesive composition
01/02/1996US5480631 Images using iodinated benzamides for contrast
01/02/1996CA1337869C Transvinylation reaction
12/1995
12/28/1995WO1995035310A1 Pyrrolidine derivatives for the treatment of cholecystokinine and gastrine-related disorders
12/28/1995WO1995035309A1 New thrombin inhibitors, their preparation and use
12/28/1995WO1995035280A1 Methods of synthesis of peptidyl argininals
12/28/1995WO1995035278A1 Methods for synthesizing diverse collections of pyrrolidine compounds
12/28/1995CA2193133A1 Novel thrombin inhibitors, the preparation and use thereof
12/28/1995CA2192697A1 Methods of synthesis of peptidyl argininals
12/27/1995EP0688765A1 Cyanoketone derivative and herbicide containing it as an active component
12/27/1995EP0688316A1 Coupling method using selective amination of maleimide
12/27/1995EP0688315A1 New heterocyclic compounds, their preparation and their use
12/27/1995EP0688314A1 Prodrug derivatives of enzyme inhibitors with hydroxyl groups, methods of preparing them and their use
12/27/1995EP0688211A1 Methods and compositions for inhibition of angiogenesis
12/26/1995US5478950 Reacting dicarboxylic acid(or anhyudride) with hydrogen in first catalytic bed, then reaction with primary amine or ammonia in second downstream catalytic bed
12/26/1995US5478820 Antibiotic compounds
12/24/1995CA2126620A1 Cyanoketone derivative and herbicide containing it as an active component
12/21/1995WO1995034813A1 Resins for solid state synthesis
12/21/1995WO1995034577A1 Template directed cyclization
12/21/1995WO1995034538A2 Purification of serine proteases and synthetic inhibitors thereof
12/21/1995WO1995034530A1 2-acylaminopropanol compound and medicinal composition
12/20/1995EP0687250A1 1-vinyl-3(e)-ethylidene pyrrolidone
12/20/1995EP0687249A1 Balanoids
12/20/1995EP0462258B1 Ureido derivatives of poly-4-amino-2-carboxy-1-methyl compounds
12/19/1995US5476934 Oxidation a nitrogen-containing perfluoroacyl halide
12/19/1995US5476865 Methods of inhibiting bone loss
12/19/1995US5476791 Process for producing optically active carboxylic acid amide
12/19/1995CA2077542C Chiral catalysts for enantioselective synthesis
12/19/1995CA1337771C Unsaturated .beta.-keto-ester acetals and their uses
12/19/1995CA1337770C Hydrocarbon substituted pyrrolidinones
12/19/1995CA1337765C Titanocenes, the use thereof, and n-substituted pyrroles
12/18/1995CA2150501A1 Ester compounds and noxious life-controlling agents containing the same as an active ingredient
12/14/1995WO1995033731A1 Hydroxamic acid derivatives
12/14/1995WO1995033719A1 Substituted pyrrolidone, thiazolidones or oxazolidones as herbicides
12/14/1995WO1995033718A1 Novel pyrrolidine-2-thione derivatives as herbicides
12/14/1995WO1995033717A2 Heterocyclic imino derivatives
12/14/1995WO1995033462A1 Anti-inflammatory compounds
12/14/1995CA2190979A1 Substituted pyrrolidone, thiazolidones or oxazolidones as herbicides
12/13/1995EP0686642A2 Modified guanidino and amidino thrombin inhibitors
12/13/1995EP0686627A2 Substituted perfluoroalkylguanidines, process for their preparation, their use as medicine or diagnostic as well as medicines containing them
12/13/1995EP0686152A1 Ortho-substituted 2-methoxyiminophenylacetic acid methylamides
12/13/1995EP0686147A1 Novel 2,2'-bi-1h-pyrrole derivatives with immunosuppressant activity
12/13/1995EP0513149B1 Pyridylphenyl nitrogen heterocycle-substituted carbinols and derivatives thereof with anti-inflammatory activity
12/13/1995CN1113233A A method for producing a pyrrolidire derivative
12/12/1995US5475138 Method preparing amino acid-derived diaminopropanols
12/12/1995US5475132 Fungicide intermediates
12/12/1995US5475119 Diallylammonium compounds, processes for their preparation and their use
12/12/1995US5475118 1-phenylpyrrolidone derivatives having optical activity, intermediate for the preparation thereof and processes for their preparation
12/12/1995US5475117 Process for optically active 2-alkyl-2,5-diazabicyclo[2.2.1]heptanes
12/12/1995US5475105 N-substituted azabicycloheptane derivatives