Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
08/2005
08/25/2005CA2552565A1 Aryloxyalkylcarbamate-type derivatives, preparation method thereof and use of same in therapeutics
08/24/2005EP1566385A1 Phosphorescent compound and electroluminescent element including the same
08/24/2005EP1566376A1 Preparation of amino acid amides
08/24/2005EP1565457A2 Process for synthesis bis-aryl diamidoxime compounds
08/24/2005EP1565437A1 Dipeptidyl peptidase iv inhibiting fluorinated cyclic amides
08/24/2005EP1565436A2 3-aminopyrrolidine derivatives as modulators of chemokine receptors
08/24/2005EP1565422A1 Vitamin d receptor modulators
08/24/2005EP1565192A2 Method and compositions for temporarily incapaciting subjets
08/24/2005EP1565190A2 Arylcyclopropylcarboxylic amides as potassium channel openers
08/24/2005EP1565178A2 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs
08/24/2005EP1334085B1 Sulfamides as gamma-secretase inhibitors
08/24/2005EP1163218B1 New salt of (2r,3r,4r)-3,4-dihydroxy-2-hydroxymethylpyrrolidine
08/24/2005EP1158980B1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
08/24/2005EP1019075B1 Beta 2-adrenergic receptor agonists
08/24/2005CN1659456A Filters for electronic displays
08/24/2005CN1659131A (2-((2-alkoxy) -phenyl) -cyclopent-1-enyl) aromatic carbo and heterocyclic acid and derivatives
08/24/2005CN1658867A Use of substituted cyanopyrrolidines and combination preparations containing them for treating hyperlipidemia and associated diseases
08/24/2005CN1216056C Sulfamato hydroxamic acid metalloprotease inhibitor
08/24/2005CN1216054C 1,4-dihydro pyridine-3,5-carboxylic-acid derivatives and preparation method thereof
08/24/2005CN1215835C Ketone derivatives and medical use thereof
08/23/2005US6933404 Methods of making intermediates from polyhydroxyalkanoates
08/23/2005US6933393 Reacting methyl cyanoacetate with morphiline to form 3-morpholin-4-yl-3-oxo- propionitrile; forming salt; reacting with phenylacetic acid and 2-(2-(4-fluorophenyl)-2-oxo-1-phenyl-ethyl)-4-
08/23/2005US6933390 Process for the arylation of aza-heterocycles with activated aromatics in presence of caesium carbonate
08/23/2005US6933351 Process for forming polyalkenyl acylating agents
08/23/2005US6933314 Integrin receptor inhibitors
08/23/2005US6933307 Fungicidal phenylimine derivatives
08/23/2005US6933261 2,4,5-Trisubstituted phenylketoenols
08/18/2005WO2005075978A2 Time-temperature indicator based on valence isomerizations
08/18/2005WO2005075973A2 Acousto-mechanical detection systems and methods of use
08/18/2005WO2005075477A1 Antibacterial compounds
08/18/2005WO2005075426A1 Novel dipeptidyl peptidase iv inhibitors; processes for their preparation and compositions thereof
08/18/2005WO2005075421A1 Bicycloester derivative
08/18/2005WO2005075420A2 Pyrrolidine derivatives acting as ccr3-receptor antagonists
08/18/2005WO2005075410A1 New compounds, methods for their preparation and use thereof
08/18/2005WO2005074919A1 Diurea derivatives
08/18/2005WO2005074686A1 N-(2-(hydroxymethyl) phenyl)-1h-pyrazole-4-carboxamide derivatives and related compounds as microbicidal active ingredients for phyto-protection and the protection of materials
08/18/2005WO2005074598A2 Nitroxyl progenitor compounds and methods of use
08/18/2005WO2005030794A3 Hemiasterlin derivatives and uses thereof
08/18/2005US20050182262 Reacting an amino acid or acid salt with a halogenating agent (thionyl chloride, phosphorous pentachloride or oxalyl chloride) , to form an intermediate, reacting the intermediate with ammonia; amidation; chemical intermediate to form Levetiracetam
08/18/2005US20050182260 Reacting substituted or unsubstituted aniline with maleic acid, succinic acid or glutaric acid in presence of polyphosporic acid; cyclization; imidation; chemical intermediates for drugs
08/18/2005US20050182235 Methods of making intermediates from polyhydroxyalkanoates
08/18/2005US20050182121 Thio semicarbazone and semicarbozone inhibitors of cysteine proteases and methods of their use
08/18/2005US20050182047 Treatment of demyelinating disorders
08/18/2005US20050182040 Benzamide derivatives
08/18/2005US20050182032 vitamin D3 antagonist activity; treating Paget's disease, bone diseases, hypercalcemia or osteoporosis; e.g. 1 alpha,25-dihydroxyvitamin D3-26 23-lactam, N-(p-methoxy)benzyl
08/18/2005US20050181455 aryl sulfonates and sulfates used for inhibiting bioadhesion to surfaces
08/18/2005US20050181416 N-aryl-carbamic acid ester-derived and valeric acid ester-derived cross-linkers and conjugates, and methods for their synthesis and use
08/18/2005DE102004001433A1 cis-Alkoxyspiro-substituierte Tetramsäure-Derivate cis-Alkoxyspiro-substituted tetramic acid derivatives
08/18/2005CA2555313A1 Heparanase inhibitors and uses thereof
08/18/2005CA2554771A1 Nitroxyl progenitor compounds and methods of use
08/18/2005CA2552942A1 New compounds, methods for their preparation and use thereof
08/18/2005CA2552928A1 Pyrrolidine derivatives acting as ccr3-receptor antagonists
08/18/2005CA2551957A1 Acousto-mechanical detection systems and methods of use
08/18/2005CA2551566A1 Diurea derivatives
08/18/2005CA2497062A1 Preparation of amino acid amides
08/17/2005EP1562949A2 Methods for the preparation of pyrrolotriazine compounds useful as kinase inhibitors
08/17/2005EP1562930A2 Synthetic lactone formulations and method of use
08/17/2005EP1562925A1 Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
08/17/2005EP1562916A1 Methods for preparing n-arylated oxazolidinones via a copper catalyzed cross coupling reaction
08/17/2005EP1562897A1 Phenylcarboxamide beta-secretase inhibitors for the treatment of alzheimer s disease
08/17/2005EP1562895A1 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
08/17/2005EP1562583A1 Atorvastatin calcium form vi or hydrates thereof
08/17/2005EP1181274A4 Iminocyclitol inhibitors of hexoaminidase and glycosidase
08/17/2005EP1161240B1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
08/17/2005EP0894085B1 Benzyl(idene)-lactam derivatives, their preparation and their use as selective (ant)agonists of 5-ht1a- and/or 5-ht1d receptors
08/17/2005CN1656077A Process for preparing chiral diol sulfones and dihydroxy acid HMG CoA reductase inhibitors
08/17/2005CN1656066A Pharmaceutical combination
08/17/2005CN1215055C Arylsulfonamido-substituted hydroxamic acid derivatives
08/16/2005US6930200 Mono-and di-substituted alpha-amino acid derivatives useful as raw materials for pharmaceutical and agro-chemical products
08/16/2005US6930185 Anorectic agents; obesity; such as 4'-chloro-N-(6-((N,N-dimethylamino)methyl)-2-naphthyl)(1,1'-biphenyl)-4 -carbox-amide
08/16/2005US6930126 Reacting oxo, esters with nitriles in the presence of hydrogen and reduction catalysts, to form heterocyclic amides, used as mixtures in drugs, cosmetics, inks, protective coatings, agriculture, stripping and cleaning compounds
08/16/2005US6930113 For therapy and prophylaxis of sexual dysfunctios; hypertension, pulmonary hypertension, congestive heart failure, renal failure, myocardial infraction, stable, unstable and variant (Prinzmetal) angina, atherosclerosis
08/16/2005US6930106 Inhibitors of HCV NS5B polymerase
08/16/2005CA2342974C Methods and compositions for inhibition of angiogenesis
08/11/2005WO2005073216A2 Hcv ns-3 serine protease inhibitors
08/11/2005WO2005073195A2 Hcv ns-3 serine protease inhibitors
08/11/2005WO2005073188A1 Aspartates useful as components in coating compositions and their preparation
08/11/2005WO2005073187A1 Improved process for the preparation of amorphous atorvastatin calcium
08/11/2005WO2005073165A1 Amide derivatives, process for production of the same, and method for application thereof as insecticide
08/11/2005WO2005066121A3 Multifunctional amine capture agents
08/11/2005WO2005065370A3 Soluble polymers as amine capture agents and methods
08/11/2005WO2005053663A3 Norepinephrine reuptake inhibitors useful for treatment of cognitive failure
08/11/2005WO2005051914A8 Benzylether and benzylamino beta-secretase inhibitors for the treatment of alzheimer's disease
08/11/2005WO2005044791A3 2-halogen-6-alkyl-phenyl-substituted tetramic acid derivatives
08/11/2005WO2005020897A3 Compositions and methods for the treatment of disease associated with trp-p8 expression
08/11/2005US20050176961 Reacting compounds such as 7-chloro-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid with 4-Aminomethyl-3-methoxyimino-pyrrolidinium dimethanesulfonate in presence of triethylamine or a tetraC1-6alkylammonium hydroxide, and an aqueous solvent
08/11/2005US20050176806 Use of 1-[3-hydroxy-1-adamantylamino]acetyl-2-cyano-pyrrolidine, for example with other anticholesterol drugs such as statins
08/11/2005US20050176802 Pyrrole substituted 2-indolinone protein kinase inhibitors
08/11/2005US20050176800 Preterm labor, dysmenorrhea, asthma, hypertension, fertility disorder, sexual dysfunction, undesired blood clotting, bone disorders, preeclampsia or eclampsia, or an eosinophil disorder; use with phosphodiesterase inhibitors; e.g. 7-[(2R,3R)-3-Chloro-1-(4-hydroxynonyl)-pyrrolidin-2-yl]-hept-5-enoic acid
08/11/2005US20050176771 4-fluoro-1-({[1-(methanesulfonyl)piperidin-4-yl]amino}acetyl)pyrrolidine-2-carbonitrile; insulin-dependent diabetes (type 1 diabetes), non insulin-dependent diabetes (type 2 diabetes), insulin-resistant disorders, obesity; dipeptidyl peptidase IV-inhibiting activity
08/11/2005US20050176766 2,3-Oxidosqualene-lanosterol cyclase inhibitors
08/11/2005US20050176760 and tumors; imino-, thiocarbonyl- or hydroxyimino-substituted N-heterocyclic amide compounds such as 2-(3-aminomethylphenylamino)-N-[3-chloro-4-(2-hydroxyiminopyrrolidin-1-yl)phenyl]-2-phenylacetamide
08/11/2005US20050176758 2-(hydroxy or methoxymethoxy)-4-(carboxy or alkoxycarbonyl)-5-(fluoro or hydrogen)-7-oxabicyclo(4.1.0)hept-3-ene chemical intermediates to neuraminidase inhibitors
08/11/2005US20050176731 N-[5-({(2S)-3-[(4-{4-[(4-benzylpiperidin-1-yl)carbonyl]phenyl}cyclohexyl)amino]-2-hydroxypropyl}oxy)-2-hydroxyphenyl]methanesulfonamide; beta 3 receptors agonist; gastrointestinal diseases; antiobesity, antidiabetic, cicatrizing agents, tocolytics, dysmenorrhea, antiglaucomatous; amidation
08/11/2005US20050176727 Male erectile dysfunction; 1-(3-chlorophenyl)-3-(4-pyridin-2-yl-piperazin-1-yl)propan-1-one O-methyloxime
08/11/2005CA2552317A1 Hcv ns-3 serine protease inhibitors
08/10/2005EP1560939A2 Immobilization of biological molecules onto surfaces coated with monolayers
08/10/2005EP1560812A1 Aminocyclohexyl ether compounds and uses thereof
08/10/2005EP1560811A2 Pharmaceutical compositions as inhibitors of dipeptidyl peptidase-iv (dpp-iv)
08/10/2005EP1560810A1 Bifunctional phenyliso(thio)cyanates; method and intermediate products for the production thereof