Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
05/2005
05/19/2005CA2541212A1 Fused phenylalanine derivatives as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes
05/18/2005EP1530564A2 Compounds derived from aryl carbamates, preparation thereof and uses of same
05/18/2005EP1263724B1 Novel compounds
05/18/2005EP1176139B1 Medicinal compositions with 2.2.1] and 3.1.1] bicycloskeleton antagonistic to both of pgd 2?/txa 2? receptors
05/18/2005CN1617881A Chemical process
05/18/2005CN1617852A Alpha-(n-sulphonamido)acetamide derivatives as beta-amyloid inhibitors
05/18/2005CN1617744A Combined therapy against tumors comprising substituted acryloyl distamycin derivatives and protein kinase (serine/threonine kinase) inhibitors
05/18/2005CN1617718A N-aryl-N'-arylcycloalkyl-urea derivatives as MCH antagonists for the treatment of obesity
05/18/2005CN1616452A 维生素d类似物 Vitamin d analogues
05/18/2005CN1616432A Compound, its use and pharmaceutical compositions comprising same
05/18/2005CN1616424A Novel ceramide compound with cell fading inducing activity and its preparing method
05/18/2005CN1202113C Ru-polypyridine complex and its synthesizing process and use
05/18/2005CN1202052C Enantioselective reduction of ketones with silane agent/metal compound/chiral ligand system
05/18/2005CN1201735C Mycobacterial inhibitors
05/17/2005US6894185 Substituted chiral allosteric hemoglobin modifiers
05/17/2005US6894072 Compounds as NS3-serine protease inhibitors of hepatitis C virus
05/17/2005US6894005 Heterocyclic compound containing phenyl groups; postemergence herbicides
05/17/2005US6893650 Fungicides; locus infestation; such as N,N-dimethyl-N'-(4-(3-trifluoromethylbenzylthio)-2,5-xylyl)formamidine
05/17/2005CA2103845C 9-[(substituted glycyl)-amido]-6-demethyl-6-deoxytetracyclines
05/12/2005WO2005042516A2 Ligands of melanocortin receptors and compositions and methods related thereto
05/12/2005WO2005042489A1 N-substituted benzene sulfonamides
05/12/2005WO2005042484A1 Preparation of 4,5-dialkyl-3-acyl-pyrrole-2-carboxylic acid derivatives by fischer-fink type synthesis and subsequent acylation
05/12/2005WO2005042483A1 [r-(r*,r*)]-2-(4-fluorophenyl)-beta, delta-dihydroxy-5-((1-methylethyl) -3-phenyl-4-[(phenylamino) carbonyl]- 1h-pyrrole-1-heptanoic acid iron salt
05/12/2005WO2005042482A1 Vitamin d3 lactam derivative
05/12/2005WO2005042466A1 Quaternary ammonium salt, electrolyte, electrolyte solution and electrochemical device
05/12/2005WO2005023765A8 Method for catalyzing amidation reactions by the presence of co2
05/12/2005WO2005018635A3 Ion channel modulating activity i
05/12/2005WO2005014539A3 Pyrrole-based hmg-coa reductase inhibitors
05/12/2005WO2003006454A8 Heterocyclic carboxamides and their use as fungicides
05/12/2005US20050101783 N-(heterocycle-methyl)alkylamine derivative, process for producing the same, and bactericide
05/12/2005US20050101760 reacting polyhydroxypropionate isolated from plant biomass with ammonia to form alkenoic amide (acrylamide, methacrylamide); depolymerization
05/12/2005US20050101671 Compounds and compositions for delivering active agents
05/12/2005US20050101663 Synthetic lactone formulations and method of use
05/12/2005US20050101657 Pyrrole derivatives for preventing or treating cancer sensitive to hormones; administered with luteininzing hormone releasing hormone derivative
05/12/2005US20050101651 Viricides; protease inbhibitors; useful for inhibiting the activity of picornaviral 3C proteases; for example, 6-carbamoyl-4S-{2S-[(5-naphthalen-1-yl-1H-pyrrole-2-carbonyl)-amino-3-phenyl-propionylamino}-hex-2(trans)-enoic acid ethyl ester
05/12/2005US20050101644 Benzylether amine compounds useful as CCR-5 antagonists
05/12/2005US20050101567 Using a sulfonamide containing compound
05/12/2005CA2544725A1 Vitamin d3 lactam derivative
05/12/2005CA2544350A1 N-substituted benzene sulfonamides
05/11/2005EP1529529A1 Medicament containing an effector of the glutathione metabolism together with $g(a)-lipoic acid for immunomodulation, immunostimulation and/or antiphlogistic treatment
05/11/2005EP1529042A1 Arylamides
05/11/2005EP1337532B1 Compound for chelating a metal, radiopharmaceutical, manufacturing process therefor, and diagnostic kit
05/11/2005EP1057485B1 Potassium channel activators
05/11/2005CN1615311A 3-biphenyl-substituted-3-substituted-4-ketolactam and ketolactone and their utilization as pesticide
05/11/2005CN1615153A Drug for preventing vascular restenosis and instrument to be embedded in vessel coated with the drug
05/11/2005CN1613857A Dipyrromethene metal chelate compounds
05/11/2005CN1613853A PDF enzyme inhibitor-hydroxamic acid serial compounds synthetic method and use thereof
05/11/2005CN1200930C New crystalline polymorphic form of 1-methyl-5-P-toluoylpyrroel-2-ac-etamidoacetic acid guaiacyl ester (MED 15)
05/10/2005US6891071 Halogenated styrene compounds and very low-loss polymers made therefrom
05/10/2005US6891047 Process for the preparation of amorphous atorvastatin
05/10/2005US6891046 Solution and solid phase synthesis of pyrrolinones and polypyrrolinones
05/10/2005US6890939 Aminopyrrolidine sulfonamides as serine protease inhibitors
05/10/2005US6890932 Anthranilic acid derivative
05/10/2005US6890921 Selectively inhibit binding to alpha-1a adrenergic receptor; 1-(2-phthalimidoethyl)-4-(2-isopropyloxyphenyl)piperazine; N-(Ethyl-2-(2-iso-propyloxyphenyl)piperazin-4-yl))-(1'-(2-oxy -piperdinyl))acetamidemide
05/10/2005US6890362 Oxidation base chosen from certain para-phenylenediamine derivatives and their addition salts with an acid and at least one suitably selected coupler
05/06/2005WO2005040355A2 Tao kinase modulators and methods of use
05/06/2005WO2005040128A1 Heterocyclyl compounds
05/06/2005WO2005040110A1 Pyrrole and pyrazole derivatives as potentiators of glutamate receptors
05/06/2005WO2005040109A1 Ligands of melanocortin receptors and compositions and methods related thereto
05/06/2005WO2005040108A1 Prolinamide derivatives as sodium and/or calcium channel blockers or selective mao-b inhibitors
05/06/2005WO2005040101A1 Acylurea connected and sulfonylurea connected hydroxamates
05/06/2005WO2005019240A3 Melanin concentrating hormone receptor antagonists
05/06/2005WO2005012249A3 Adamantyglycine- based inhibitors of dipeptidyl peptidase iv for the treatment of diabetes
05/06/2005WO2004113394A3 Living radical polymerization initiator comprising a functional group capable of reacting with polypeptides or the like, comb polymer obtained therewith, polypeptide conjugates and drugs obtained therefrom
05/06/2005WO2004092116A8 Bicyclic compounds having bradykinin receptors affinity and pharmaceutical compositions thereof
05/06/2005CA2543570A1 Acylurea connected and sulfonylurea connected hydroxamates
05/06/2005CA2542064A1 Tao kinase modulators and methods of use
05/05/2005US20050096478 Derivatives of fluoro(hydro)carbons attached to an -alkylene-oxy-carbonyl-leaving group; reactive with amine-containing compounds to form a fluoro-substituted carbamyl protective group useful for the efficient separation, recovery and purification of synthsized organic compounds; libraries
05/05/2005US20050096468 Inhibitors of histone deacetylase
05/05/2005US20050096466 Process for the preparation of tetrazol-derived compounds as growth hormone secretagogues
05/05/2005US20050096358 Treating rheumatoid arthritis, psoriasis, reperfusion injury, cardiovascular , autoimmune, inflammatory disorders and bronchial asthma
05/05/2005US20050096357 Antibiotics; therapy for infections which is caused by drug-resistant Streptococcus, or bacteria infections
05/05/2005US20050096348 non-insulin dependent diabetes mellitus, and impaired glucose tolerance; dipeptidyl peptidase IV (DPP-IV) inhibitors eg (2S)-1-{[(1S)-2-(5-cyano-2-methyl-indol-1-yl)-1-methyl-ethylamino]-acetyl}-pyrrolidine-2-carbonitrile
05/05/2005US20050096325 use of specified inhibitors of chemokine receptors to treat inflammatory diseases such as asthma, allergic rhinitis, atopic dermatitis, inflammatory bowel diseases, idiopathic pulmonary fibrosis, bullous pemphigoid, allergic colitis, eczema, conjunctivitis, familial eosinophilia
05/05/2005US20050096312 Antiserotonine agents; antidepressants; eating disorders; anxiolytic agents; sleep disorders; gastrointestinal disorders; cardiovascular disorders; muscular disorders; endocrine system diseases; muscular disorders; psychological disorders
05/05/2005US20050096309 For use as anticoagulant agents for therapy of thromboembolic disorders
05/04/2005EP1528055A2 Sulphonamide Derivatives
05/04/2005EP1527207A1 Pyrrolyl complexes of copper for copper metal deposition
05/04/2005EP1442022A4 Polyamide modulators of cox2 transcription
05/04/2005CN1612887A Phosphino-aminophosphines
05/04/2005CN1612859A Crystalline (r-(r*, r*))-2-(4-fluorophenyl)-beta, delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-((phenylamino)carbonyl)-1h-pyrrole-heptanoic acid calcium salt (2:1)
05/04/2005CN1612856A 1, 3-diarylprop-2-en-1-ones, compositions containing same and use thereof
05/04/2005CN1612732A Analgesics and methods of use
05/04/2005CN1611524A Polyethylene glycol amino acid N-internal ring carbonyl anhydride active derivatives, and medicinal bonding compound and gel thereof
05/04/2005CN1199945C Method for producing cyclic lactams
05/03/2005US6888032 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
05/03/2005US6888006 Method for processing pyrollidone and n-vinyl pyrollidone residues
05/03/2005US6887952 For use as cross-linking agents
05/03/2005US6887893 Methods and compositions for treatment and prevention of tumors, tumor-related disorders and cachexia
05/03/2005US6887887 Asymmetric synthesis of (S,S,R)-(-)-actinonin and its analogs and uses therefor
05/03/2005US6887877 Viricide for hepatitis virus
05/03/2005US6887872 Propenecarboxylic acid amidoxime derivatives, a process for the preparation thereof, and pharmaceutical compositions containing the same
05/03/2005US6887871 Use of phenylheteroakylamine derivatives
05/03/2005US6887863 Such as (2RS,3R)-3-amino-4-cyclohexyl-2-hydroxy-N-phenoxybutanamide; methionine aminopeptidase type 2 inhibitors
04/2005
04/28/2005WO2005037826A1 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases
04/28/2005WO2005037810A2 Cyclopropyl methanone derivatives, the preparation and the therapeutic use thereof
04/28/2005WO2005037809A1 Substituted aryl cycloalkanol derivatives and methods of their use
04/28/2005WO2005037786A1 Heterocyclyl compounds
04/28/2005WO2005037785A2 Derivatives of n-[phenyl(pyrrolidine-2-yl)methyl]benzamide and n-[(azepan-2-yl)phenylmethyl]benzamide, preparation method thereof and application of same in therapeutics
04/28/2005WO2005037772A2 Novel ligand activating receptors rars used for human medicine and cosmetics