Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304) |
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12/06/2005 | CA2096528C Retroviral protease inhibitors |
12/01/2005 | WO2005113605A1 Cross-linked antibodies |
12/01/2005 | WO2005113558A2 Simple stereocontrolled synthesis of salinosporamide a |
12/01/2005 | WO2005113534A2 Cxcr1 and cxcr2 chemokine antagonists |
12/01/2005 | WO2005113525A1 N, n’-substituted-1,3-diamino-2-oxopropane derivatives, their pharmaceutical compositions and use |
12/01/2005 | WO2005113503A2 Metabolites of (+)-(2s, 3s)-3-(2-methoxy-5-trifluoromethoxybenzylamino)-2-phenyl-piperidine |
12/01/2005 | WO2005113498A1 Adrenergic receptor antagonists |
12/01/2005 | WO2005113497A1 Substituted 5-aminomethyl-1h-pyrrol-2-carbxylic acid amides |
12/01/2005 | WO2005113011A2 Prodrugs of ion channel modulating compounds and uses thereof |
12/01/2005 | WO2005090301B1 Crystalline form of atorvastatin hemi calcium |
12/01/2005 | WO2005082848A3 Method for preparing pyrrolidine oximes |
12/01/2005 | WO2005077899A3 Amino-substituted tricyclic derivatives and methods of use |
12/01/2005 | WO2005042516A3 Ligands of melanocortin receptors and compositions and methods related thereto |
12/01/2005 | WO2004089894A8 Process for preparing 5-(4-fluorophenyl)-1-[2-((2r,4r)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)ethyl]-2-isopropyl-4-phenyl-1h-pyrrole-3-carboxylic acid phenylamide |
12/01/2005 | US20050267198 Novel processes for preparing amorphous atorvastatin hemi-calcium |
12/01/2005 | US20050267169 Watersoluble prodrugs of propofol |
12/01/2005 | US20050267152 Gly1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders |
12/01/2005 | US20050267126 Compounds derived from aryl carbamates, preparation thereof and uses of same |
12/01/2005 | US20050267123 6-Membered heterocyclic compounds useful for selective inhibition of the coagulation cascade |
12/01/2005 | US20050267118 Inhibitors of factor Xa and other serine proteases involved in the coagulation cascade |
12/01/2005 | US20050267043 Novel inhibitors of hepatitis C virus NS3 protease |
12/01/2005 | US20050266567 Methods for generating high titer helper-free preparations of released recombinant AAV vectors |
12/01/2005 | US20050265961 Biodegradable poly(beta-amino esters) and uses thereof |
12/01/2005 | CA2566920A1 Metabolites of (+)-(2s, 3s)-3-(2-methoxy-5-trifluoromethoxybenzylamino)-2-phenyl-piperidine |
12/01/2005 | CA2566892A1 Substituted 5-aminomethyl-1h-pyrrol-2-carbxylic acid amides |
12/01/2005 | CA2565519A1 Cxcr1 and cxcr2 chemokine antagonists |
12/01/2005 | CA2562701A1 Cross-linked antibodies |
12/01/2005 | CA2561819A1 Prodrugs of ion channel modulating compounds and uses thereof |
11/30/2005 | EP1600437A1 Acid generators, sulfonic acids, sulfonyl halides, and radiation-sensitive resin compositions |
11/30/2005 | EP1599445A1 Compounds having activity at 5ht2c receptor and uses thereof |
11/30/2005 | EP1509500B1 Process for the preparation of the amorphous form of atorvastatin calcium salt |
11/30/2005 | EP1091943B1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases |
11/30/2005 | EP0963200B9 Compositions for inhibition of angiogenesis comprising thalodomide and a nsaid |
11/30/2005 | CN1703410A Isoquinoline compounds and medicinal use thereof |
11/30/2005 | CN1703399A Pharmaceutical compositions as inhibitors of dipeptidyl peptidase-IV (DPP-IV) |
11/30/2005 | CN1703397A Sulfonylamino-acetic acid derivatives and their use as orexin receptor antagonists |
11/30/2005 | CN1703395A Aryl and heteroaryl compounds and methods to modulate coagulation |
11/30/2005 | CN1229377C Spiro [Piperidine-4,1'-pyrrolo[3,4-c] pyrrole] |
11/30/2005 | CN1229348C Method for preparing amlodipine |
11/30/2005 | CN1229344C Farnesyl transferase inhibitors |
11/30/2005 | CN1229343C Chemotactic factor receptor active regulator |
11/30/2005 | CN1229323C Dialkoyl-halogen phenyl substituted keto-enol |
11/30/2005 | CN1229100C Primary intermediates for oxidative coloration of hair |
11/29/2005 | US6969770 reacting an alpha-keto carboxy acid ester or derivative with a pyrrolidinone to form an intermediate, subjecting the intermediate to asymmetric hydrogenation using a chiral catalyst to form the end product |
11/29/2005 | US6969744 Living and quasiliving cationic telechelic polymers quenched by N-substituted pyrrole and methods for their preparation |
11/29/2005 | US6969715 6-membered heterocyclic compounds useful for selective inhibition of the coagulation cascade |
11/29/2005 | CA2288445C 5-oxo-pyrrolidine-2-carboxylic acid hydroxamide derivatives |
11/29/2005 | CA2194189C Process for producing cyclic lactames |
11/24/2005 | WO2005111116A1 Biological molecule-reactive hydrophilic silicone surface |
11/24/2005 | WO2005110992A1 Amido compounds and their use as pharmaceuticals |
11/24/2005 | WO2005110984A1 Process for producing cyclic n-hydroxyimide compound |
11/24/2005 | WO2005087722A9 Diphenylmethyl compounds useful as muscarinic receptor antagonists |
11/24/2005 | WO2004113297A9 Aza-ring derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
11/24/2005 | US20050261504 Process for preparing intermediates |
11/24/2005 | US20050261501 e.g. 1-({[9-(hydroxymethyl)-3-oxaspiro[5.5]undec-9-yl]amino}acetyl)-2-pyrrolidinecarbonitrile; dipeptidyl-peptidase IV inhibitor; antidiabetic, hypoglycemic agent; non-insulin dependent diabetes, obesity |
11/24/2005 | US20050261361 Novel crystal forms of atorvastatin hemi-calcium and processes for their preparation as well as novel processes for preparing other forms |
11/24/2005 | US20050261360 Dissolving the crystalline form in acetone, allowing to convert to amorphous form and then precipitating it out |
11/24/2005 | US20050261359 Novel processes for preparing amorphous atorvastatin hemi-calcium |
11/24/2005 | US20050261342 Metabolites of (+)-(2S,3S)-3(2-methoxy-5- trifluoromethoxybenzylamino)-2-phenyl-piperidine |
11/24/2005 | US20050261291 1-Cyclopropylmethyl-4-[2-(3,3,5,5-tetramethylcyclohexyl)phenyl]piperazine or a salt or hydrate; exhibit excellent cell adhesion inhibitory action or cell infiltration inhibitory action; for treating inflammatory diseases and autoimmune diseases such as inflammatory bowel diseases and rheumatoid arthritis |
11/24/2005 | US20050261290 Novel compounds of proline and morpholine derivatives |
11/24/2005 | US20050261273 Substituted urea and carbamate, phenacyl-2-hydroxy-3-diaminoalkane, and benzamide-2-hydroxy-3-diaminoalkane aspartyl-protease inhibitors |
11/24/2005 | US20050261161 Stable crystals of pyrrole compound |
11/24/2005 | US20050260126 Diagnostic probes and remedies for diseases with accumulation of prion protein, and stains for prion protein |
11/24/2005 | CA2567630A1 Biological molecule-reactive hydrophilic silicone surface |
11/24/2005 | CA2565238A1 Amido compounds and their use as pharmaceuticals |
11/23/2005 | EP1598350A1 Pyrrolidines and thiazolidines derivatives, their preparation and their use in the treatment of hyperglycaemia and of type II Diabetis |
11/23/2005 | EP1598337A1 Method of obtaining an antiepileptic agent |
11/23/2005 | EP1598067A1 Carbamic acid compounds comprising an amide linkage as HDAC inhibitors |
11/23/2005 | EP1597262A2 Substituted heterocycles |
11/23/2005 | EP1597248A2 Sulfonamide derivatives as ppar modulators |
11/23/2005 | EP1597229A2 Pyrrolidine derivatives as oxytocin antagonists |
11/23/2005 | EP1597228A2 Substituted n-arylheterocycles, method for production and use thereof as medicaments |
11/23/2005 | EP1335898B1 Carbamic acid compounds comprising an amide linkage as hdac inhibitors |
11/23/2005 | EP1320522B1 Compositions and methods of the use thereof achiral analogues of cc-1065 and the duocarmycins |
11/23/2005 | EP0934263B1 Non-immunosuppressant fkbp rotamase inhibitors |
11/23/2005 | CN1701059A Chemotherapeutic agents |
11/23/2005 | CN1699545A Apparatus and method for controlling biofilms |
11/23/2005 | CN1699349A Method and reagents for N-alkylating ureides |
11/23/2005 | CN1228326C Method for producing N-alkenyl amides |
11/23/2005 | CN1228325C Biguanide derivatives |
11/22/2005 | US6967220 antibiotics; treating respiratory system disorders; n-hydroxy benzyl formamide derivatives |
11/22/2005 | US6967199 Substituted diamine derivatives useful as motilin antagonists |
11/22/2005 | US6967107 reacting with first one end and then the other of a polyoxyalkylene terminated on one end with a maleimidylarylaminocarbonyloxy group and on the other by a compound having a succinimidyloxycarbonyl group |
11/22/2005 | CA2162122C Use of glycine-n,n-diacetic acid derivatives as biodegradable complexing agents for alkaline earth and heavy metal ions, and method of preparing them |
11/17/2005 | WO2005109562A1 Material for electrolytic solution, ionic material-containing composition and use thereof |
11/17/2005 | WO2005108594A1 Enzymatic ammonolysis process for the preparation of intermediates for dpp iv inhibitors |
11/17/2005 | WO2005108393A1 Pyrrole or imidazole amides for treating obesity |
11/17/2005 | WO2005108391A1 Amides as bace inhibitors |
11/17/2005 | WO2005108384A1 3- or 4-monosubstituted phenol and thiophenol derivatives useful as h3 ligands |
11/17/2005 | WO2005108370A1 Benzene compounds |
11/17/2005 | WO2005108368A1 Adamantyl-acetamide derivatives as inhibitors of the 11-beta-hydroxysteroid dehydrogenase type 1 enzyme |
11/17/2005 | WO2005108361A1 Adamantyl pyrrolidin-2-one derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors |
11/17/2005 | WO2005108360A1 Pyrrolidin-2-one and piperidin-2-one derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors |
11/17/2005 | WO2005108359A1 Novel compounds of proline and morpholine derivatives |
11/17/2005 | WO2005108358A2 Pyrrolidine derivatives useful as bace inhibitors |
11/17/2005 | WO2005108351A1 Benzonitrile derivatives to treat musculoskeletal frailty |
11/17/2005 | WO2005107762A2 Certain chemical entities, compositions, and methods |
11/17/2005 | WO2005085177A3 Biaryl amino acids and their use in dna binding oligomers |
11/17/2005 | WO2005016264A3 Diamine derivatives of quinone and uses thereof |