Patents
Patents for A61P 21 - Drugs for disorders of the muscular or neuromuscular system (23,287)
09/1989
09/27/1989CN1035823A 1,4-disubstituted-piperidnyl compounds
09/12/1989US4866077 Treatment of nervous system disorders such as alzheimer*s disease
09/12/1989US4866057 4-substituted 10-cyanomethylenepyrrolo[4,3-e]-benzazepines
08/1989
08/23/1989CN1034926A Process for preparing dioxazocine derivatives
08/22/1989US4859685 Anesthetic composition and method of using the same
08/08/1989US4855297 Tricyclic pyridone derivatives
07/1989
07/26/1989EP0325268A1 1,4-Disubstituted-piperidinyl compounds
07/18/1989US4849431 Piperidine derivative and pharmaceutical composition
06/1989
06/28/1989EP0322251A2 Benzothiopyran derivatives
06/13/1989US4839380 Antihypoxic agents
06/07/1989EP0318682A2 Tricyclic thiazole derivatives
05/1989
05/24/1989CN1033000A Magnesium additive for nutrients, feed and medicaments
05/16/1989US4831155 Physostigmine derivatives with acetylcholinesterase inhibition properties, and manufacture
05/10/1989EP0315433A2 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics
05/05/1989WO1989003837A1 Acylated uridine and cytidine and uses thereof
05/02/1989US4826866 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics
04/1989
04/19/1989CN1032440A 4-aminopyridine derivatives
04/18/1989US4822629 Azumolene dosage form
04/12/1989EP0311303A2 4-aminopyridine derivatives
04/11/1989CA1252462A1 Imidazodiazepine derivatives
04/04/1989CA1252092A1 1,3-oxazolidine-2-one derivatives and processes for their preparation
03/1989
03/29/1989EP0309422A2 New amidino tricycle derivatives
03/22/1989EP0307904A1 Covered sustained-release forms
02/1989
02/22/1989EP0304223A2 Beta-carbolines as cholecy-stokinin and gastrin antagonist
02/01/1989EP0301371A2 Benzofuran carboxamides with basic substituents, process for their preparation and therapeutical compositions containing them
01/1989
01/11/1989EP0298202A1 Organic salts of physostigmine derivatives
01/10/1989CA1248454A1 Cytidyl diphosphocholine-drug composition and process
01/03/1989CA1248108A1 Benzo¬c|-1,5-naphthyridines, a process and intermediates for their preparation and their use as medicaments
12/1988
12/28/1988EP0296721A2 Heterocyclic compounds
12/28/1988CN88103535A Tricyclic pyridone derivatives
12/21/1988EP0295411A1 Pharmaceutical preparation for percutaneous administration containing eperisone or tolperisone or a salt thereof
12/20/1988CA1247105A1 Tetrahydroisoxazolo 4,5-c pyridine derivatives, pharmaceutical compositions and method of treatment
12/14/1988EP0294599A2 Tricyclic pyridone derivatives
11/1988
11/23/1988EP0291888A2 4-Substituted 1-cyanomethylene pyrrolo[4,3-e]-benzo-azepins
11/23/1988EP0291862A1 5-Substituted 10-cyanmethylene-thieno[3,4-b]benzoazepines
11/17/1988DE3814521A1 Neue anwendung von dopaminrezeptor-agonisten New application of dopamine receptor agonists
11/15/1988US4785089 Hypotensive agents
11/02/1988CN88100346A 3-aryl-5-alkylthio-4h-1,2,4-triazoles
11/01/1988US4782052 Antiulcer
11/01/1988CA1244030A1 1,2,4-triazolo-carbamate and the acid addition salts thereof, processes for preparing them and pharmaceutical compositions
10/1988
10/26/1988EP0288102A1 Novel 2 beta, 16beta-diamino-androstanes
10/19/1988EP0287150A1 Novel 2 beta-morpholino-androstane derivatives and processes for their preparation
10/04/1988US4775671 Imidazodiazepines
09/1988
09/21/1988EP0282502A1 Imidazole derivatives.
09/21/1988CN87108354A 6-benzoxazinyl-and 6-benzothiazinyl-2,3,4,5-tetrahydropyridazin-3-ones
09/20/1988US4772738 Muscle relaxants, analgesics, anticonvulsants, antidepressant
08/1988
08/17/1988EP0278002A1 1-thiocarbamoylmethylpyrrolidine-2-thione and method of obtaining it
08/16/1988US4764518 Antibacterial agents containing oxo-4-pyridine carboxylic acid derivatives
08/03/1988EP0276793A2 3-Aryl-5-alkylthio-4H-1,2,4-triazoles
08/02/1988US4761418 Novel compounds
07/1988
07/20/1988EP0274930A1 Pyrrole derivatives, their preparation and pharmaceutical compositions containing them
07/20/1988EP0274929A1 Pyrrole derivatives, their preparation and pharmaceutical compositions containing them
07/06/1988EP0273262A2 Chroman derivatives
06/1988
06/28/1988US4753941 Hypnotics, muscle relaxants
06/28/1988US4753933 Anxiolytic amides derived from certain 1,8-naphthyridine-2-amines
06/15/1988EP0271404A2 Pyrrole derivatives, their preparation and pharmaceutical compositions containing them
06/15/1988EP0271151A2 Azumolene dosage form
06/01/1988EP0269220A2 Derivatives of alpha-hANP and their production
05/1988
05/31/1988CA1237436A1 4-oxothiazolidin-2-ylidene-acetamide derivatives, processes for their preparation and their use in the combating of diseases of the central nervous system
04/1988
04/05/1988US4735940 Tricyclic pyridine derivatives and pharmaceutical compositions
03/1988
03/23/1988EP0260467A2 Quinoxaline compounds and their preparation and use
03/22/1988US4732900 Treatment of senility, alzheimer*s disease
03/10/1988WO1988001620A1 1-thiocarbamoylmethylpyrrolidine-2-thione and method of obtaining it
02/1988
02/25/1988WO1988001268A1 Imidazole derivatives
02/24/1988EP0256798A1 Anaesthetic composition
02/23/1988CA1233174A1 Aryl and heteroaryl¬7-(aryl and heteroaryl)- pyrazolo-¬1,5-a|-pyrimidin-3-yl|methanones
01/1988
01/26/1988US4721784 6-benzoxazinyl-2,3,4,5-tetrahydropyridazin-3-ones
10/1987
10/07/1987CN87101762A Process for the preparation of novel alkylenediamine derivatives
09/1987
09/09/1987EP0235942A1 Alkylenediamine derivatives
09/09/1987EP0235408A1 Pharmaceutical composition and treatment
09/02/1987EP0234971A1 Substituted amides, their preparation and pharmaceutical compositions containing them
08/1987
08/26/1987EP0233801A1 Substituted amides, their preparation and pharmaceutical compositions containing them
07/1987
07/28/1987CA1224787A1 Subtituted amids, preparation and pharmaceutical compositions containing same
07/22/1987EP0229391A1 Piperidine derivate, its use and pharmaceutical composition containing it
07/08/1987CN86108467A Trycyclic pyridazopyridone derivatives
06/1987
06/30/1987US4677101 Substituted dihydroazepines useful as calcium channel blockers
06/24/1987EP0226196A2 Tricyclic pyridone derivatives
06/16/1987US4673674 Diazepinoindoles useful for treating depression, schizophrenia, social withdrawal or anxiety and pharmaceutical compositions containing them
06/03/1987EP0223974A1 N-Substituted-N-[3-(1,2,4-triazolo[4,3-b]pyridazin-6-yl)-phenyl]alkanamides, carbamates and ureas
05/1987
05/19/1987CA1221969A1 3-methylflavone-8-carboxylic acid esters
04/1987
04/07/1987US4656298 Muscle relaxants, stimulants, analgesics, anticonvulsants, antidepressants
03/1987
03/31/1987US4654343 N-substituted-N[3-(1,2,4-triazolo[4,3-b]pyridazin-6-yl)phenyl]alkanamides, carbamates and ureas
03/26/1987WO1987001589A1 Method of treating catabolic dysfunction
03/24/1987US4652567 Benzo(c)-1,5-naphthyridines useful for treating a patient having drug induced memory impairment in need of memory enhancement
02/1987
02/17/1987US4644063 1,3-oxazolidine-2-one derivatives
02/10/1987US4642308 Anticonvulsants, anxiolytic agents, antiepileptic agents, hypnotics, muscle relaxants
01/1987
01/14/1987EP0208497A2 Diamino-androstane derivatives
01/07/1987EP0207845A1 Bactericides containing 4-oxopyridocarboxylic acid derivatives and process for their preparation
12/1986
12/30/1986EP0206993A1 Sulphonic-acid esters
12/09/1986US4628056 Novel oxopyrimidine derivatives, pharmaceutical compositions containing them and their use as anticonvulsant, antianxiety and muscle relaxant agents
11/1986
11/19/1986CN86102329A Process for preparing a new derivatives of an aminoketone
11/12/1986EP0200942A2 New derivatives of an aminoketone
11/05/1986CN85108120A Process for the preparation of tricyclische pyridinderivate and their use
10/1986
10/15/1986EP0197318A1 Benzo[C]-1,5-naphthyridines, a process and intermediates for their preparation and their use as medicaments
10/08/1986CN85109716A Process for the preparation of octahydroindolo/2,3-a/-quinolizin-1-yl-alkanecarboxylic acid amides and acid addition salts and pharmeutical composition thereof
09/1986
09/30/1986US4614740 Nervous system disorders
08/1986
08/26/1986US4608378 Tetrahydroisoxazolo[4,5-c]pyridine derivatives useful in the treatment of malfunctions of the acetylcholine or muscarinic systems
08/05/1986US4604392 2-substituted benzofuran derivatives useful in treating cardiac arrhythmic, histaminic and tussive conditions
06/1986
06/11/1986EP0183994A1 Tricyclic pyridone derivatives
06/10/1986US4594190 Quaternary salts of dibenzo[1,4]diazepinones, pyrido-[1,4]benzodiazepinones, pyrido[1,5]benzodiazepinones with antiulcer, antisecretory, spasmolytic and antimusarinic activities