Patents
Patents for A61P 21 - Drugs for disorders of the muscular or neuromuscular system (23,287)
03/1981
03/04/1981EP0024272A1 1,4-Benzodiazepines and their salts, process for their preparation and pharmaceutical compositions containing them
02/1981
02/24/1981US4252810 9,10-Dihydro-4H-benzo[4,5]cyclohepta [1,2-b]thiophen-4,9-imines
01/1981
01/06/1981US4243589 Sedatives, muscle relaxants, anticonvulsants
01/06/1981CA1093073A1 Benzodiazepine derivatives
12/1980
12/23/1980CA1092105A1 Pyrrolo(2,1-b) (3)benzazepines
11/1980
11/25/1980US4236012 5-Phenethyl-2-oxazolidone derivatives and a process for producing the same
11/25/1980US4235897 Benzodiazepine derivatives and pharmaceutical compositions thereof
11/25/1980CA1090333A1 Process for the manufacture of diazepine derivatives
11/04/1980US4231930 1-Substituted thiomethyltriazolobenzodiazepines
10/1980
10/21/1980US4229453 Substituted 5,6-dimethylpyrrolo[2,3-d]pyrimidine compounds, their production and their medicinal use
10/15/1980EP0017523A1 Dithiepinno (1,4)(2,3-c) pyrrol derivatives, their preparation and pharmaceutical compositions containing them
10/07/1980US4226768 From 2-substituted 1,4-benzodiazepines, anesthetics
09/1980
09/17/1980EP0015615A1 Phenyl piperazine derivatives, their preparation and antiagressive medicines containing them
08/1980
08/26/1980CA1084510A1 1- 5-(substituted phenyl)-2-oxazolyl -methylene - amino -2,4-imidazolidinediones
08/26/1980CA1084484A1 Triamino-androstanes and a process for the preparation of the said compounds
08/19/1980CA1084044A1 Diamino-androstanes and a process for the preparation of the said compounds
08/05/1980CA1083148A1 Method for the preparation of new heterocyclic derivatives
08/05/1980CA1083146A1 Process for the preparation of new benzodiazepine derivatives
07/1980
07/29/1980CA1082714A1 Indazole derivatives
06/1980
06/17/1980US4208408 Muscle relaxants
06/10/1980CA1079279A1 Triazolylphenyl ketone derivatives and production thereof
05/1980
05/28/1980EP0011206A1 9,10-Dihydro-4H-benzo(4,5)cyclohepta(1,2-b)thiophen-4,9 imines, process for their preparation and pharmaceutical compositions containing them
04/1980
04/30/1980EP0010119A1 Isoquinoline derivatives, their preparation and pharmaceutical compositions containing these compounds
04/29/1980US4200636 Muscle relaxant
04/29/1980CA1076572A1 Diazepine derivatives
04/16/1980EP0010030A1 Derivatives of 2'-(ortho-chloro-benzoyl),4'-chloro-glycin anilide, their preparation and their use in medicines
04/16/1980EP0009808A1 Composition having skeletal muscle relaxant activity
04/08/1980CA1075241A1 Quaternary isoquinoline derivatives
02/1980
02/26/1980CA1072557A1 Dithiepinno (1,4)(2,3-c) pyrrol; methods of preparation, compositions thereof
02/19/1980CA1072095A1 Phenyl piperazine olefins
01/1980
01/08/1980CA1069497A1 Diepoxy-androstanes and a process for the preparation thereof
01/08/1980CA1069441A1 Pharmaceutical composition containing 2,1,3-benzothiazole
12/1979
12/18/1979US4179507 Quarternary ammonium compounds
12/18/1979CA1068276A1 1-aminomethyl-6,7-dihydroxy-1,2,3,4-tetrahydroisoquinoline compounds
12/04/1979CA1067491A1 Diazepine derivatives
11/1979
11/20/1979US4175079 Cyclization, formation/c-n/, dehydration
11/14/1979EP0005205A1 Substituted 5.6-dimethylpyrrolo(2,3-d)pyrimidines, methods for their preparation and medicines containing them
10/1979
10/16/1979US4171306 Diepoxy-androstanes and a process for the preparation thereof
10/16/1979CA1064489A1 Process for the preparation of new benzenesulfonamides
10/09/1979US4170649 1,4-Benzodiazepine derivatives, pharmaceutical compositions thereof, and process for their preparation
10/03/1979EP0004320A1 1-Substituted-thiomethyltriazolobenzodiazepines, preparation thereof, their use, and a pharmaceutical composition
09/1979
09/19/1979EP0004018A1 1-Oxa-4-aza-2,6-disilacyclohexanes, their production and use as muscle relaxants and pharmaceutical compositions containing them
08/1979
08/14/1979CA1060452A1 3-(aminoacyl)-1-((5-(substituted phenyl) furfurylidene)amino) hydantoins
06/1979
06/27/1979EP0002512A1 Imino-bridged benzocycloheptapyridines, process for their preparation and pharmaceutical composition thereof
06/26/1979US4159374 Anticonvulsants, muscle relaxants, anxiolytic agents, hypnotics
04/1979
04/18/1979EP0001401A1 Thienobenzazepine derivatives, processes for their production and pharmaceutical compositions containing them
04/03/1979US4147875 Imidazo[1,5-α][1,4]benzodiazepines
03/1979
03/27/1979US4146722 Sedatives, muscle relaxants, anticonvulsants
03/27/1979US4146537 Process for preparing imidazo[1,5-a][1,5]benzodiazepines
03/20/1979US4145550 Chemical intermediates for b-adrenergic blocking agents
03/20/1979US4145421 Aminoimidazoline-substituted quinoxalines
02/1979
02/21/1979EP0000770A2 1-Methylisoguanosin, processes and intermediates for its preparation, its pharmaceutical compositions and their preparation
01/1979
01/30/1979US4137402 Quaternary ammonium salts of dantrolene and clodanolene
01/30/1979US4137229 Process for preparing imidazo[1,5-A][1,5]benzodiazepines
01/02/1979US4132791 Use of etoperidone in parkinsonism and in other extrapyramidal syndromes characterized by tremors
12/1978
12/20/1978EP0000089A1 Imidazole-2-carbamates and process for their production and pharmaceutical compositions containing them.
12/19/1978US4130646 1,2,3,4-Tetrahydro-2-((4-(phenyl)-1-piperazinyl)methyl)-1-naphthalenols and derivatives and analogs thereof
12/05/1978CA1043783A1 Triazolobenzodiazepine derivatives
11/1978
11/21/1978US4126676 Modified neurotoxin derived from naja genus snake venom
11/14/1978US4125726 Sedatives, muscle relaxants, anxiolytics, anticonvulsants
11/07/1978US4124711 Derivatives of dithiepino[1,4][2,3-C]pyrrole
10/1978
10/03/1978US4118499 Anti-anxiety and anti-parkinsonian 1-aminoalkyl-2-endo-chloro-7,7-dimethylnorbornanes
10/03/1978US4118386 Synthesis of imidazo[1,5-a]diazepine-3-carboxylates
09/1978
09/05/1978US4111931 Anxiolytics, anticonvulsant, muscle relaxant, sedative
08/1978
08/29/1978US4110463 Muscle relaxant
07/1978
07/18/1978US4101545 Neuromuscular blocking agents
07/11/1978US4100286 Anticonvulsant, cns depressant
06/1978
06/27/1978US4097528 Muscle relaxants, vasodilation
06/20/1978US4096263 Smooth muscle relaxants
05/1978
05/09/1978US4088771 1-Lower alkyl-4,5-dihydro-5-phenyl-2-lower alkoxy carbonylaminoimidazoles and substituted phenyl derivatives thereof
04/1978
04/25/1978US4086353 Certain azolinylamino (azolidinylimino) indazoles
03/1978
03/21/1978US4080323 Anxiolytics, anticonvulsants, muscle relaxants, sedatives
02/1978
02/28/1978US4076939 2-(4-Substituted-1,2,5-thiadiazole-3-yloxy)-acetaldehydes
02/28/1978US4076823 Triazolo-2,4-benzodiazepines
01/1978
01/31/1978US4071515 Triamino-androstanes and a process for the preparation of the said compounds
10/1977
10/11/1977US4053617 Antispasmodic agents, muscle relaxants
09/1977
09/20/1977US4049812 Benzodiazepine carboxamides and pharmaceutical compositions with central nervous system activity
09/20/1977US4049650 Muscle relaxants
09/13/1977US4048313 Stimulating gastric evaculation
09/06/1977US4046772 Benzodiazepine derivative and process for producing the same
08/1977
08/23/1977US4044129 Central nervous system, muscle relaxants, sedatives
06/1977
06/07/1977US4028356 Cyclization, sedatives, tranquilizers, muscle relaxants
04/1977
04/12/1977US4017492 As-triazinobenzodiazepin-1-ones
04/05/1977US4016165 Triazino benzodiazepines
01/1977
01/04/1977US4001222 3-(Aminoacyl)-1-{[5-(substituted phenyl)furfurylidene]amino}hydantoins and process for their preparation thereof
07/1976
07/06/1976US3968236 2-Aminomethyl-5-hydroxy-4H-pyran-4-one and derivatives thereof
03/1976
03/30/1976US3947417 Tranquilizers, muscle relaxants, sedatives, anticonvulsants, sleep inducers