Patents
Patents for C07J 43 - Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta[a]hydrophenanthrene skeleton (2,516)
11/1995
11/14/1995US5466815 Antilipemic agents
11/08/1995EP0680327A1 Therapeutic uses and delivery systems of dehydroepiandrosterone
11/02/1995WO1995029186A1 Compositions and methods for cell transformation
11/02/1995CA2188320A1 Compositions and methods for cell transformation
10/1995
10/31/1995US5462933 Modified bile acid conjugates, and their use as pharmaceuticals
10/26/1995WO1995028413A1 17β-SUBSTITUTED 3-CARBOXY STEROIDS THAT INHIBIT 5-α-REDUCTASE
10/19/1995WO1995027702A1 Novel functionalized hydrophilic acridinium esters
10/19/1995CA2186463A1 Novel functionalized hydrophilic acridinium esters
10/17/1995US5459255 For incorporation into oligonucleotides, cleaving RNA site specifically
10/11/1995EP0676410A2 Bile acids derivatives useful in the therapy of the biliary calculosis from cholesterol and of the pathologies caused by cholestasis
10/11/1995EP0676202A2 Use of aromatic steroids substituted in 3-position by a disubstituted aminoalkoxy chain for the manufacture of a medicament for the control of fertility, in particular male fertility
10/10/1995USRE35053 Intermediates for amino substituted steroids
10/10/1995US5457191 3-deazapurines
10/03/1995US5455335 Glycosylated steroids
09/1995
09/27/1995EP0673251A1 17 substituted acyl-3-carboxy 3,5-diene steroidals as 5-alpha-reductase inhibitors
09/25/1995CA2145469A1 Disubstituted aminoalkyloxy 3-substituted aromatic steroids used for the preparation of a drug to control fertility, especially male fertility; pharmaceutical compositions containing the same
09/20/1995CN1108661A Corticoid 17,21-dicarboxylic esters and corticosteroid 17-carboxylic ester 21-carbonic esters, processes for their preparation and pharmaceuticals containing these compounds
09/14/1995WO1995024415A1 Steroid derivatives, pharmaceutical compositions containing them, and their pharmaceutical uses
09/13/1995EP0529002A4 Fluorescent porphyrin, and fluorescent phthalocyanine - polyethylene glycol, polyol, and saccharide derivatives as fluorescent probes
09/12/1995US5449556 Chemiluminescent markers
09/10/1995CA2122639A1 Bile acids for biological and chemical applications and processes for the production thereof
09/06/1995EP0669932A1 17-alpha and 17-beta substituted acyl-3-carboxy-3,5-dienes and use in inhibiting 5-alpha-reductase
09/06/1995CN1029683C Process for preparing new steroids substituted at position 10 by a radical including a double or triple bond
08/1995
08/29/1995US5446036 13-alkyl-11beta-phenylgonanes
08/23/1995EP0110955B1 Brain-specific drug delivery
08/22/1995US5444055 17-hydroxyiminomethyl-5-β, 14 β-androstane derivatives active on the cardiovascular system, processes for their preparation and pharmaceutical compositions containing same
08/22/1995US5443758 A ketone cis- or trans-gonanes; nonlinear optical response
08/17/1995WO1995021617A1 Androstanes and pregnanes for allosteric modulation of gaba receptor
08/17/1995CA2183231A1 Androstanes and pregnanes for allosteric modulation of gaba receptor
08/10/1995WO1995021184A1 Substituted purines and oligonucleotide cross-linking
08/08/1995US5439913 Contraception method using competitive progesterone antagonists and novel compounds useful therein
08/03/1995WO1995020567A1 Codrugs as a method of controlled drug delivery
07/1995
07/25/1995US5436337 Anticarcinogenic agents
07/19/1995CN1105368A Corticosteroid 17-alkyl carbonate 21-|O¨-carboxylic and carbonic esters, processes for their preparation, and pharmaceuticals containing these compounds
07/11/1995US5432169 Cyclopentanperhydrophenanthren-17β-(3-furyl)-3-derivatives and pharmaceutical compositions comprising same for the treatment of cardiovascular disorders
07/06/1995WO1995018141A1 Medicinal composition for bone resorption inhibition and osteogenesis acceleration
07/05/1995EP0661270A1 Nucleophilic polysubstituted aryl acridinium esters, conjugates, production and uses thereof
07/04/1995US5430116 Polymers and oligomers of bile acid derivatives, process for their preparation and their use as pharmaceuticals
06/1995
06/28/1995EP0659763A2 Steroid derivatives
06/28/1995EP0659761A2 New 17-iminomethylalkenyl-5beta-14beta-androstane and 17-iminoalkyl-5beta-14beta-androstane derivatives active on the cardiovascular system, processes for their preparation and pharmaceutical compositions containing same
06/23/1995CA2136803A1 Steroid derivatives
06/20/1995US5426102 Antigestagenic, antiandrogenic, antiglucocorticoid, antimineralcorticoid properties
06/14/1995EP0656790A1 Compositions and methods for modulating rna
06/07/1995EP0656365A1 Substituted 2beta-morpholinoandrostane derivatives
06/03/1995CA2136915A1 Substituted 2.beta.- morpholino-androstane derivatives
06/01/1995WO1995014707A1 N-2 substituted purines
05/1995
05/30/1995US5420120 Anti-inflammatory glucocorticoid compounds for topical ophthalmic use
05/23/1995US5418226 Neuromuscular blocking agent anesthetic, fast-acting
05/16/1995US5416203 Steroid modified oligonucleotides
05/16/1995US5416079 21-chloro-pregnane derivative
05/04/1995WO1995011914A1 Δ16 unsaturated c¿17? heterocyclic steroids useful as steroid c17-20 lyase inhibitors
05/03/1995EP0650495A1 Improved antiandrogens
04/1995
04/26/1995EP0649431A1 17-AMINO SUBSTITUTED 4-AZASTEROID 5$g(a)-REDUCTASE INHIBITORS
04/26/1995CN1101916A Compounds
04/26/1995CN1101915A New 19-nor steroids having a phenoxyalkylsulphonamide or phenoxyalkylsulphonylurea chain in position llbeta, preparation process and intermediates, use as medicaments and pharmaceutical compositions..
04/26/1995CN1101914A Compounds
04/25/1995US5410040 Mono- and diquaternary 5-alpha-hydroxy-3,16-diaminoandrostane salts; curare-like muscle relaxant activity
04/11/1995US5405979 Stereoselectively reducing phenyl-substituted estradiene with electropositive metal in electron-solvating solvent, cleaving ketone protective group with acid
04/06/1995WO1995009178A1 Synthesis of 17-(3-pyridyl) steroids
04/06/1995WO1995009177A1 21-substituted steroid compound
04/06/1995CA2172983A1 21-substituted steroid compound
04/05/1995EP0646593A1 Corticoid-17,21-dicarboxylic acid ester and corticosteroid-17-carboxylic acid ester-21-carbonic, process for their production and medicaments containing them
04/05/1995EP0646126A1 Novel steroids with pregnane skeleton, pharmaceutical compositions containing them and process for preparing same
04/04/1995US5403928 Fluorescent marker components and fluorescent probes
03/1995
03/30/1995WO1995008559A1 Novel urethane-containing aminosteroid compounds
03/30/1995CA2172495A1 Novel urethane-containing aminosteroid compounds
03/29/1995EP0644882A1 Novel piperzinyl-bis(alkylamino)pyrimidine derivatives and process for preparing same
03/22/1995EP0643724A1 Process of preparing 3-carbonylandrostadiene 17-carboxamides
03/22/1995EP0643723A1 Halogenation using halo-vilsmeier reagent
03/21/1995CA1334844C 9-alpha-hydroxysteroids, process for their preparation, process for the preparation of the corresponding 9(11)-dehydro-derivatives and pharmaceutical preparations containing said steroids
03/15/1995EP0643071A1 Compound for inhibiting bone resorption and accelerating osteogenesis
03/15/1995EP0573604B1 Methods for the treatment of osteoporosis
03/15/1995EP0431151B1 Method for preparing 21-brom-4-pregnen-3,20-dione derivatives
03/09/1995WO1995006474A1 Thiol-derivatized nucleosides and oligonucleosides
03/08/1995EP0641355A1 Steroid sulphatase inhibitors
03/08/1995EP0641211A1 INHIBITORS OF TESTOSTERONE 5$g(a)-REDUCTASE ACTIVITY
03/07/1995CA1334668C 13-alkyl-11beta-phenylgonanes
03/01/1995EP0640616A2 17-Alkylcarbonate, 21-0-carbonic/carboxylic acid esters of corticosteroids, a method for their production and pharmaceutical compositions containing them
03/01/1995EP0639970A1 Contraception method using competitive progesterone antagonists and novel compounds useful therein
02/1995
02/21/1995US5391776 Steroid derivatives
02/15/1995EP0638090A1 17$g(a) AND 17$g(b)-SUBSTITUTED ESTRA-1,3,5(10)-TRIENE-3-CARBOXYLIC ACID
02/14/1995US5389623 Redox carriers for brain-specific drug delivery
01/1995
01/18/1995EP0633893A1 17-substituted steroids useful in cancer treatment
01/17/1995US5382661 Useful in treating spinal trauma, head injury, subarachnoid hemorrhage
01/10/1995US5380841 Pyridinylpiperazinyl steroids
01/10/1995US5380840 Triazinylpiperazinyl steroids
01/10/1995US5380839 Phenylpiperazinyl steroids
01/05/1995WO1995000147A1 4-AZA-PREGNANE 5α-REDUCTASE ISOZYME 1 INHIBITORS
01/05/1995CA2165077A1 4-aza-pregnane 5.alpha.-reductase isozyme 1 inhibitors
12/1994
12/28/1994EP0630249A1 Dual action 2',5'-oligoadenylate antiviral derivatives and uses thereof
12/21/1994EP0629635A1 New 19-nor 11-beta-phenoxysulfonamide or 11-beta-phenoxyalkylsulfonylurea steriod derivatives, a process and intermediates for their production and their use as medicaments and pharmaceuticals containing them
12/18/1994CA2126158A1 19-nor steroids phenoxyalkylsulfonamide or phenoxyalkylsulfonylurea chain on 11 beta position, process and intermediates for their preparation, application as medicaments and pharmaceutical compositions containing them
12/13/1994US5373095 Phospholipase inhibitor
12/08/1994WO1994027608A1 Methods and compositions for inducing sleep
12/07/1994EP0280741B1 Mitomycin derivatives
11/1994
11/24/1994WO1994026767A1 Improved antiandrogens
11/24/1994WO1994016709A3 Therapeutic uses and delivery systems of dehydroepiandrosterone
11/24/1994CA2136303A1 Improved antiandrogens
11/23/1994EP0532565B1 STARTING COMPOUNDS FOR THE PRODUCTION OF 10$g(b)-H STEROIDS AND PROCESS FOR PRODUCING SUCH STARTING COMPOUNDS
11/23/1994EP0532562B1 PROCESS FOR PRODUCING 10$g(b)-H-STEROIDS
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