Patents
Patents for C07J 43 - Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta[a]hydrophenanthrene skeleton (2,516)
11/2002
11/21/2002WO2001042273A9 Asthma associated factors as targets for treating atopic allergies including asthma and related disorders
11/21/2002CA2447032A1 Kinetic assay
11/12/2002US6479476 Treating menopausal symptoms and osteoporosis in female warm-blooded animals
11/06/2002EP1254179A1 An in vivo screen using chemical inducers of dimerization
11/06/2002EP0639970B2 Contraception method using competitive progesterone antagonists and novel compounds useful therein
10/2002
10/31/2002US20020160972 Antisense compound with targeting and RNA cleaving moieties, preferably an imidazole functionality conjugated to the targeting oligonucleotide via linkers
10/16/2002CN1374968A 4-benzylaminoquinoline conjugates with bile acid and their heteroanalogues, method fo r producing the same, medicaments containing these compounds and their use
10/10/2002WO2002079220A2 Aminosterol compounds, their use in the preparation of meiosis-regulating medicaments and method for their preparation
10/10/2002CA2438210A1 Steroid compounds, use of these compounds for the preparation of meiosis-regulating medicaments and method for the preparation of these compounds
10/02/2002EP1245572A1 Aminosterol compounds, their use in the preparation of meiosis-regulating medicaments and method for their preparation
09/2002
09/24/2002US6455517 For therapy of conditions or diseases that are estrogen-dependent, i.e., are estrogen-induced or estrogen-stimulated
09/19/2002WO2002072598A1 Steroids as agonists for fxr
09/18/2002EP0630249B1 Dual action 2',5'-oligoadenylate antiviral derivatives and uses thereof
09/18/2002CN1370179A Aromatic and heterocyclic derivatives of phytosterols and/or phytosanols for use in treating or preventing cardiovascular disease
09/12/2002US20020128242 Novel cationic cholesteryl derivatives containing cyclic polar groups
09/11/2002EP1238285A1 Steroid compounds for steroid receptor binding assays
09/11/2002CN1368977A Unsaturated cholestane derivatives and their use for preparation of meiosis regulating medicaments
09/10/2002CA2132449C 17 - substituted steroids useful in cancer treatment
09/05/2002DE10109898A1 Lipide mit veränderlicher Ladung Lipids with variable charge
09/04/2002EP1236471A2 Angiostatic steroids
09/04/2002EP1236470A2 Angiostatic steroids
09/04/2002EP1236469A2 Angiostatic steroids
09/04/2002EP1235849A2 Asthma associated factors as targets for treating atopic allergies including asthma and related disorders
09/03/2002US6444683 17-azolyl steroids useful as androgen synthesis inhibitors
08/2002
08/29/2002WO2002066490A2 Cationic sterol derivatives, ph-sensitive liposomes comprising cationic sterol derivatives and method for loading liposomes with active substances
08/29/2002WO2002066489A2 Amphoteric sterols and the use thereof in the production of ph-sensitive liposomes
08/07/2002EP0885239B1 Novel steroid carbamates as potentiating agents
08/01/2002US20020103392 Corticoid-17,21-dicarboxylic esters and corticosteroid 17-carboxylic ester 21-carbonic esters, processes for their preparation and pharmaceuticals containing these compounds
07/2002
07/31/2002EP0799059B1 Cationic amphiphiles and plasmids for intracellular delivery of therapeutic molecules
07/24/2002CN1360591A 3 alpha-hydroxy-3 beta-methoxymethyl-21-heterocycle substd. steroids with anesthetic activity
07/23/2002US6423700 17-halogenated 19-nor steroids, method and intermediates for preparing same, use as medicines and pharmaceutical compositions containing same
07/18/2002WO2002055531A1 Conjugates of immune cell specific macrolide compounds with anti-inflammatory compounds for improved cellular targeting of anti-inflammatory therapy
07/11/2002US20020091278 Steroid derived antibiotics
07/03/2002EP1218401A1 4-benzylaminoquinoline conjugates with bile acid and their heteroanalogues, methods for producing the same, medicaments containing these compounds and their use
06/2002
06/20/2002WO2002026759A3 17α FLUOROALKYL STEROIDS, METHOD FOR PRODUCING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID COMPOUNDS
06/18/2002US6407086 Novel sterol derivatives used for regulating the meiosis in oocytes and in male germ cells
06/13/2002US20020072624 As antiestrogenic and anti-proliferative agent
06/13/2002US20020072510 3-nitrogen-6,7-dioxygen steroids and uses related thereto
06/04/2002US6399754 Sugar modified oligonucleotides
05/2002
05/30/2002WO2001042273A3 Asthma associated factors as targets for treating atopic allergies including asthma and related disorders
05/30/2002US20020065257 17beta-amino and hydroxylamino-11beta-arylsteroids and their derivatives having agonist or antagonist hormonal properties
05/29/2002EP1208113A2 17beta-acyl-alpha-propynyl-11beta-(cyclic amino)aryl steroids and their derivatives having antagonist hormonal properties
05/28/2002US6395713 Cationic lipidcationic lipid
05/28/2002US6395492 Derivatized oligonucleotides having improved uptake and other properties
05/23/2002US20020061868 Pharmaceutical preparations containing estra-1,3,5(10)-triene derivatives
05/16/2002WO2002000680A3 Cationic steroid derivatives for gene delivery
05/16/2002US20020058649 Administering during follicular phase of female menstrual cycle and in luteal phase, a competitive progesterone antagonist, which is less than an ovulation-inhibiting dose and less than an abortion-inductive dose
05/07/2002US6383814 Cationic amphiphiles for intracellular delivery of therapeutic molecules
05/02/2002WO2001074840A3 17-alpha-substituted-11-beta-substituted-4-aryl and 21-substituted 19-norpregna 21-substituted 19-norpregnadienedione as antiprogestational agents
04/2002
04/18/2002US20020045774 Antigestagenically active steroids with a fluorinated 17-alpha-alkyl chain
04/18/2002DE10049736A1 17alpha-Fluoralkylsteroide, Verfahren zu deren Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen 17alpha-Fluoroalkyl steroids, processes for their preparation and pharmaceutical compositions containing them
04/17/2002EP1196428A1 11$g(b)-ARYL-17,17-SPIROTHIOLANE-SUBSTITUTED STEROIDS
04/17/2002EP0970103B1 Antigestagenic steroids with a fluorinated 17alpha-alkyl chain
04/04/2002WO2002026759A2 17α FLUOROALKYL STEROIDS, METHOD FOR PRODUCING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID COMPOUNDS
04/04/2002CA2422056A1 17.alpha. fluoroalkyl steroids, method for producing the same and pharmaceutical compositions containing said compounds
04/02/2002US6365582 S-substitute 11β-benzaldoxime-estra-4, 9-diene-carbonic acid thiolesters, method for the production thereof and pharmaceutical preparations containing these compounds
03/2002
03/28/2002WO2002000679A3 9.alpha.-chloro-6.alpha.-fluoro-17.alpha.-hydroxy-16-methyl-17-beta-methoxycarbonyl-androst-1,4-dienes esterified in position 17.alpha. by a cyclic acyl group
03/27/2002EP1189923A1 Aromatic and heterocyclic derivatives of phytosterols and/or phytostanols for use in treating or preventing cardiovascular disease
03/20/2002EP1187846A2 11beta long-chain substituted estratrienes, method for their production, pharmaceutical preparations containing said 11beta long-chain substituted estratrienes, and their use for producing medicaments
03/19/2002US6358931 Oligonucletide conjugated to imidazole; intercalation and coordination compounds; medical diagnosis, gene therapy; antisense agents
03/14/2002US20020032181 For therapy of conditions or diseases that are estrogen-dependent, i.e., are estrogen-induced or estrogen-stimulated
03/14/2002US20020032180 For therapy of conditions or diseases that are estrogen-dependent, i.e., are estrogen-induced or estrogen-stimulated
03/12/2002US6355630 Estra-1,3,5(10)-triene-7α-thioethers
03/07/2002US20020028929 Estradiol derivative and immunoassay using the same
02/2002
02/14/2002WO2002012266A1 17.beta.-carbothioate 17.alpha.-arylcarbonyloxyloxy androstane derivative as anti-inflammatory agents
02/14/2002WO2002012265A1 6.ALPHA., 9.ALPHA.-DIFLUORO-17.ALPHA.-`(2-FURANYLCARBOXYL) OXY!-11.BETA.-HYDROXY-16.ALPHA.-METHYL-3-OXO-ANDROST-1,4,-DIENE-17-CARBOTHIOIC ACID S-FLUOROMETHYL ESTER AS AN ANTI-INFLAMMATORY AGENT
02/14/2002WO2001076531A3 Bile acid containing prodrugs with enhanced bioavailability
02/14/2002CA2634715A1 6.alpha.,9.alpha.-difluoro-17.alpha.-[(2-furanylcarboxyl)oxy}-11.beta.-hydroxy-16.alpha-methyl-3-oxo-androsta-1,4-diene-17.beta.carbothioic acids-fluoromethyl ester as an anti-inflammatory agent
02/14/2002CA2417826A1 17.beta.-carbothioate 17.alpha.-arylcarbonyloxyloxy androstane derivative as anti-inflammatory agents
02/06/2002EP1177206A1 3alpha-hydroxy-3beta methoxymethyl-21-heterocycle substituted steroids with anaesthetic activity
01/2002
01/31/2002US20020013282 Transfecting a cell comprising by contacting the cell with a biologically active nucleic acid molecule in the presence of a cationic lipid which can be protonated; cationic amphiphiles to transport drugs into cells; gene therapy
01/22/2002US6340688 Administering to female during menstrual cycle amount of competitive progesterone antagonist which is less than ovulation-inhibiting dose and less than abortion-inductive dose
01/16/2002EP1019095B1 Method for the preparation of facial metal tricarbonyl compounds and their use in the labelling of biologically active substrates
01/15/2002US6339077 Substituted 4-benzylaminoquinolines and their hetero analogs, process for their preparation, pharmaceuticals containing these compounds and use thereof
01/15/2002US6339066 Antisense oligonucleotides which have phosphorothioate linkages of high chiral purity and which modulate βI, βII, γ, δ, Ε, ζ and η isoforms of human protein kinase C
01/10/2002US20020004202 In vivo screen using chemical inducers of dimerization
01/03/2002WO2002000680A2 Cationic steroid derivatives for gene delivery
01/03/2002WO2002000679A2 9.alpha.-chloro-6.alpha.-fluoro-17.alpha.-hydroxy-16-methyl-17-beta-methoxycarbonyl-androst-1,4-dienes esterified in position 17.alpha. by a cyclic acyl group
12/2001
12/18/2001US6331524 Organ-specific targeting of cationic amphiphile / DNA complexes for gene therapy
12/13/2001DE10028193A1 New bile acid conjugates with benzylamino substituted aromatic and heteroaromatic compounds useful for prevention and treatment of gall stones
12/12/2001CN1326461A Meiosis regulating compounds
12/11/2001US6329354 Administering bone active phosphonate, administering estrogen hormone
12/05/2001EP0904282B1 Novel cationic cholesteryl derivatives containing cyclic polar groups
12/05/2001EP0749437B1 Pharmaceutical uses of steroid derivatives
12/05/2001CN1324802A Anti-pregnancy hormone active steroid with fluorated 17 alpha-alkyl-chain
11/2001
11/27/2001CA2025294C Bile acid derivatives, processes for their preparation, and use as pharmaceuticals
11/22/2001WO2001087299A1 Aralkyl ester soft drugs
11/22/2001CA2407099A1 Aralkyl ester soft drugs
11/13/2001US6316432 Antigestagenically active steroids with a flourinated 17 α-alkyl chain
11/08/2001WO2001083512A1 3-nitrogen-6,7-dioxygen steroids and uses related thereto
11/08/2001CA2418748A1 3-nitrogen-6,7-dioxygen steroids and uses related thereto
11/07/2001EP1150993A1 Unsaturated cholestane derivatives and their use for the preparation of meiosis regulating medicaments
11/07/2001CN1321166A Propanolamine derivs. linked with bile acid used for treating disorders of lipid metabolism
10/2001
10/30/2001US6310225 Useful as intermediates for producing vitamin d derivates
10/25/2001WO2001078606A1 Selective nuclear receptor-targeted systems for delivery of cytotoxins to cancer cells for targeted photodynamic therapy
10/18/2001WO2001076531A2 Bile acid containing prodrugs with enhanced bioavailability
10/18/2001CA2405151A1 Bile acid containing prodrugs with enhanced bioavailability
10/11/2001WO2001074840A2 17-alpha-substituted-11-beta-substituted-4-aryl and 21-substituted 19-norpregna 21-substituted 19-norpregnadienedione as antiprogestational agents
10/10/2001EP1140972A1 New 7-alpha, 17-alpha-bis-alkylated testosterone derivatives and their use in long-term therapy of androgen-dependent diseases
10/04/2001EP0529002B1 Fluorescent porphyrin, and fluorescent phthalocyanine - polyethylene glycol, polyol, and saccharide derivatives as fluorescent probes
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