Patents
Patents for C07J 21 - Normal steroids containing carbon, hydrogen, halogen, or oxygen, having an oxygen-containing hetero ring spiro-condensed with the cyclopenta[a]hydrophenanthrene skeleton (1,576)
06/2002
06/13/2002US20020072624 As antiestrogenic and anti-proliferative agent
05/2002
05/30/2002US20020065257 17beta-amino and hydroxylamino-11beta-arylsteroids and their derivatives having agonist or antagonist hormonal properties
05/23/2002WO2001087284A3 Aldosterone antagonist composition for release during aldosterone acrophase
05/16/2002WO2002038582A2 Method for the production of 4-(17alpha substituted 3-oxoestra-4,9-dien-11-yl)benzaldehyd-(1e or 1z)-oximes
05/16/2002WO2002038581A2 Method for the production of 4-(17alpha-methyl substituted 3-oxoestra-4,9-dien-11beta-yl)benzaldehyd-(1e or 1z)-oximes
05/16/2002DE10056676A1 Preparation of estradienyl-benzaldoxime derivative preparation in high yield, for use e.g. in treating endometriosis, from epoxy-estrenone by multi-stage process including selective Grignard reaction
05/16/2002DE10056675A1 Preparation of estradienyl-benzaldoxime derivative preparation in high yield, for use e.g. in treating endometriosis, from estradienone by multi-stage process including selective Grignard reaction
05/10/2002WO2002036606A1 Selective glucocorticoid receptor agonists
05/02/2002EP0615448B1 Sex steroid activity inhibitors
04/2002
04/18/2002US20020045746 Form L crystalline eplerenone having a monoclinic crystal system and an X-ray powder diffraction pattern with a peak at 8. 0+-0.2 degrees 2 theta .
04/11/2002US20020042507 Process for preparation of 9,11-epoxy steroids and intermediates useful therein
03/2002
03/28/2002WO2002024715A2 Gamma-hydroxybutyrate compositions containing carbohydrate, lipid or amino acid carriers
03/28/2002US20020038021 Eplerenone crystalline form exhibiting enhanced dissolution rate
03/20/2002EP0730458B1 Use of aldosterone antagonists to inhibit myocardial fibrosis
03/07/2002WO2002017895A2 Use of an aldosterone receptor antagonist to improve cognitive function
03/07/2002CA2419256A1 Use of an aldosterone receptor antagonist to improve cognitive function
03/06/2002CN1080267C Preparation of intermediat of 19, 11 beta-bridge steroid
03/05/2002US6352697 Immunostimulating complex matrices; quil a fractions
02/2002
02/28/2002US20020025951 Urogenital disorders
02/14/2002US20020019522 Steroids
02/07/2002WO2002009760A2 Epoxy-steroidal aldosterone antagonist and beta-adrenergic antagonist combination therapy for treatment of congestive heart failure
02/07/2002WO2002009759A2 Aldosterone antagonist and cyclooxygenase-2 inhibitor combination therapy to prevent or treat inflammation-related cardiovascular disorders
02/07/2002WO2002009683A2 Aldosterone blocker therapy to prevent or treat inflammation-related disorders
02/07/2002US20020016455 Epoxidation of cyclopenta(a)phenanthrene derivatives
02/07/2002CA2416152A1 Aldosterone blocker therapy to prevent or treat inflammation-related disorders
02/07/2002CA2415789A1 Epoxy-steroidal aldosterone antagonist and beta-adrenergic antagonist combination therapy for treatment of congestive heart failure
02/07/2002CA2415078A1 Aldosterone antagonist and cyclooxygenase-2 inhibitor combination therapy to prevent or treat inflammation-related cardiovascular disorders
01/2002
01/09/2002EP1170299A2 Processes for preparation of 9,11-epoxy steroids and intermediates useful therein
01/02/2002EP1167381A2 Process for preparation of 7 alpha-carboxyl 9,11-epoxy steroids and Intermediates useful therein
01/02/2002EP1167380A2 11.alpha.-hydroxy-steroid-4,6-dien-3-one compounds and a process for their preparation
01/02/2002EP1167364A1 Benzopyran-containing compounds and prodrug forms thereof
01/01/2002US6335441 5β-cyano-substituted steroid compounds
12/2001
12/18/2001US6331622 Processes for preparation of 9, 11-epoxy steroids and intermediates useful therein
12/18/2001US6331534 Steroids as neurochemical stimulators of the VNO to alleviate pain
12/12/2001EP0785802B1 Saponin preparations and use thereof in iscoms
12/12/2001CN1326461A Meiosis regulating compounds
11/2001
11/22/2001WO2001087284A2 Aldosterone antagonist composition for release during aldosterone acrophase
11/22/2001CA2409437A1 Aldosterone antagonist composition for release during aldosterone acrophase
11/14/2001CN1322130A Inhibitors of type 3 3a -hydrosteroid dehydrogenase
10/2001
10/25/2001WO2001079255A1 A process for the preparation of 7.alpha.-hydroxy 3-aminosubstituted sterols using intermediates with an unprotected 7.alpha.-hydroxy group
10/24/2001EP1148061A2 Process for preparation of 9, 11- epoxy steroids and intermediates useful therein
10/11/2001WO2001074839A2 Methods of making the 4-n-butylcyclohexanoic and the undecanoic acid esters of (7 alpha, 11 beta)-dimethyl-17 beta-hydroxy-4-estren-3-one and their medical use
10/04/2001WO2001072293A2 Antiprogestins with partial agonist activity
10/04/2001CA2404172A1 Antiprogestins with partial agonist activity
09/2001
09/12/2001EP1131336A1 Estrogenic estra-1,3,5(10)-trienes with differential effects on the alpha and beta estrogen receptors, having a linear hydrocarbon chain of from 5-9 carbon atoms in position 11
08/2001
08/28/2001US6281204 19-nor steroids having a thiocarbonated chain in position 11beta, their preparation process and the intermediates of this process, and the intermediates of this process, their use as medicaments and compositions
07/2001
07/17/2001US6262042 17β-amino and hydroxylamino-11β-arylsteroids and their derivatives having agonist or antagonist hormonal properties
07/11/2001EP0735819B1 Cryptophycins
07/11/2001CN1303391A 17 Beta-amino and hydroxylamino-11 beta-arylsteroids and their derivatives having agonist or antagonist hormonal properties
07/10/2001US6258946 Chemical intermediate for diuretic
07/10/2001US6258803 11-ethyl-17-hydroxy-19-norpregn-4-en-20-yn-3-one for menopause treatment
07/05/2001WO2001047945A1 Process for preparing 17alpha-acetoxy-11beta-[4-n,n-(dimethylamino)phenyl]-21-methoxy-19-norpregna-4,9-diene-3,20-dione, intermediates useful in the process, and processes for preparing such intermediates
06/2001
06/14/2001US20010003782 Novel sterol derivatives used for regulating the meiosis in oocytes and in male germ cells
05/2001
05/30/2001EP1102582A2 Inhibitors of type 3 3alpha-hydroxysteroid dehydrogenase
05/02/2001EP1094798A2 INHIBITORS OF TYPE 5 AND TYPE 3 17beta-HYDROXYSTEROID DEHYDROGENASE AND METHODS FOR THEIR USE
03/2001
03/21/2001EP0738275B9 Novel antiandrogenic agents and related pharmaceutical compositions and methods of use
03/14/2001EP1082337A1 17 beta-amino and hydroxylamino-11 beta-arylsteroids and their derivatives having agonist or antagonist hormonal properties
03/07/2001CN1286694A Novel 19-norsteroids substd in position 11 'beta', preparation method and intermediates, application as medicines and pharmaceutical compositions contg. them
02/2001
02/28/2001EP1077992A1 Meiosis regulating compounds
02/22/2001WO1999046279A3 INHIBITORS OF TYPE 5 AND TYPE 3 17β-HYDROXYSTEROID DEHYDROGENASE AND METHODS FOR THEIR USE
02/14/2001CN1061983C 4-trifluoromethyl-3-ketosteroid compound and synthesizing method thereof
01/2001
01/30/2001US6180803 Steroid drugs
01/30/2001US6180780 Processes for preparation of 9,11-epoxy steroids and intermediates useful therein
01/24/2001CN1061052C 11 Beta-aromatic group-4-estraene and acid additive salt application in medicine
01/23/2001US6177418 Epoxidized and/or hydroxylated prostane derivatives derived from a fusidium coccineum fungus metabolite isolated from metabolite mixture of fusidic acid
12/2000
12/05/2000CA2027627C Process for preparing 21-desoxyprednisolone 17-esters
11/2000
11/21/2000US6150336 Steroidal glycosides
11/08/2000EP0738275B1 Novel antiandrogenic agents and related pharmaceutical compositions and methods of use
11/08/2000EP0650495B1 Improved antiandrogens
10/2000
10/25/2000CN1057770C Application of 19,11 beta-bridged sterodal compound in pharmaceutical working
10/11/2000CN1057304C 17,20-epoxide derivatives of pregnance, their preparation, their use in preparation of cortisome derivatives and intermediates
10/11/2000CN1057303C Preparation process for 16 beta-methyl steroid and new intermediates thereof
09/2000
09/12/2000US6117994 Intermediates for 16β-methyl steroids
09/12/2000US6117860 Nasally administering steroid which binds to a specific neuroepithelial receptor for alleviating premenstrual tension and anxiety
09/06/2000EP1032584A1 Novel 19-nor steroids substituted in position 11beta, preparation method and intermediates, application as medicines and pharmaceutical compositions containing them
08/2000
08/30/2000CN1055930C Steroalkenol polyfluohydrocarbyl sulfonate compound and its deriv., use and preparing process
08/29/2000US6110906 Androgen derivatives for use in the inhibition of sex steroid activity
08/22/2000US6107036 Heterocyclic dioxethane substrates, process for their preparation and their use
07/2000
07/11/2000CA2016780C Dihydrospirorenone as an antiandrogen
07/05/2000EP0900234B1 21-substituted progesterone derivatives as new antiprogestational agents
07/05/2000EP0554436B1 Gaba receptor modulators
07/05/2000CN1259137A Estra-5(10), 7-dienes with estrogenic activity
07/05/2000CN1054133C 17-spiromethylene steroids
07/04/2000US6083940 Method and composition for effecting contraception in a mammalian male
06/2000
06/13/2000CA2000979C Specific ligands of receptors of oestrogen and progesterone steroidal hormones, use and synthetic intermediates
06/06/2000US6072068 Treating glucocorticoid-dependent diseases or symptoms
06/02/2000WO2000031112A1 Estrogenic estra-1,3,5(10)-trienes with differential effects on the alpha and beta estrogen receptors, having a linear hydrocarbon chain of from 5-9 carbon atoms in position 11
05/2000
05/17/2000CN1253564A Processes for preparation of 9,11-epoxy steroids and intermediates useful therein
05/10/2000CN1052237C Steroids with 17-spiromethylene lactone or ortho -hydroxyl inner ether base
05/09/2000US6060503 Antiestrogenic, anticarcinogenic stereospecific benzopyran derivative; breast cancer
05/02/2000US6057439 Epoxysteroids
04/2000
04/04/2000US6046185 6,7-oxygenated steroids and uses related thereto
03/2000
03/30/2000WO2000007576A3 INHIBITORS OF TYPE 3 3α-HYDROSTEROID DEHYDROGENASE
03/22/2000CN1248262A 16-hydroxy-11-(substituted phenyl)-estra-4,9-diene derivatives
03/14/2000US6037339 C-11 substituted steroids for treating menopausal complaints
03/01/2000EP0982298A1 Novel functionalized hydrophilic acridinium esters
02/2000
02/17/2000WO2000007576A2 INHIBITORS OF TYPE 3 3α-HYDROSTEROID DEHYDROGENASE
02/17/2000CA2339368A1 Inhibitors of type 3 3.alpha.-hydroxysteroid dehydrogenase
01/2000
01/26/2000EP0973792A1 16-hydroxy-11-(substituted phenyl)-estra-4,9-diene derivatives
01/26/2000EP0973791A2 Process for preparation of 7 alpha-carboxyl 9, 11-epoxy steroids and intermediates useful therein and a general process for the epoxidation of olifinic double bonds
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