Patents
Patents for C07J 21 - Normal steroids containing carbon, hydrogen, halogen, or oxygen, having an oxygen-containing hetero ring spiro-condensed with the cyclopenta[a]hydrophenanthrene skeleton (1,576)
10/1995
10/19/1995CA2186463A1 Novel functionalized hydrophilic acridinium esters
10/18/1995CN1030081C New 11-aryl sleroid derivs
10/12/1995WO1995026974A1 Novel progesterone compound and use thereof
10/10/1995USRE35053 Intermediates for amino substituted steroids
09/1995
09/12/1995US5449556 Chemiluminescent markers
09/06/1995CN1029683C Process for preparing new steroids substituted at position 10 by a radical including a double or triple bond
08/1995
08/31/1995WO1995018821A3 Novel antiandrogenic agents and related pharmaceutical compositions and methods of use
08/30/1995CN1107478A Steroalkenol polyfluohydrocarbyl sulfonate compound and its deriv., use and preparing process
08/29/1995US5446178 Process for preparing 19,11β-bridged steroids
08/29/1995US5446036 13-alkyl-11beta-phenylgonanes
08/03/1995WO1995020567A1 Codrugs as a method of controlled drug delivery
07/1995
07/13/1995WO1995018821A2 Novel antiandrogenic agents and related pharmaceutical compositions and methods of use
07/13/1995CA2180548A1 Novel antiandrogenic agents and related pharmaceutical compositions and methods of use
06/1995
06/29/1995WO1995017093A1 New cryptophycins
06/29/1995CA2179490A1 New cryptophycins
06/22/1995WO1995016699A1 Steroid derivative
06/22/1995CA2178900A1 Steroid derivative
06/20/1995US5426179 Substituted androstanes
06/20/1995US5426102 Antigestagenic, antiandrogenic, antiglucocorticoid, antimineralcorticoid properties
06/08/1995WO1995015166A1 Use of aldosterone antagonists to inhibit myocardial fibrosis
06/08/1995CA2177848A1 Use of aldosterone antagonists to inhibit myocardial fibrosis
05/1995
05/31/1995EP0655071A1 METHOD OF PREPARING 1-METHYL-3-KETO--g(D)?1,4 -STEROIDS.
05/03/1995EP0650495A1 Improved antiandrogens
04/1995
04/20/1995WO1995010527A1 3,17-dihydroxy-3,7,16 and/or 17-methyl-androst-5-ene compounds, derivatives thereof, and their use
04/18/1995US5407928 Progesterone antagonist suitable for inducing labor or an abortion
04/11/1995US5405979 Stereoselectively reducing phenyl-substituted estradiene with electropositive metal in electron-solvating solvent, cleaving ketone protective group with acid
03/1995
03/28/1995US5401864 Protecting 3-keto group with heterocyclic spiro ring
03/28/1995US5401840 Intermediate steroid compounds
03/21/1995US5399685 Process for the preparation of 20-keto-21 alpha-01-steroids
03/21/1995CA1334844C 9-alpha-hydroxysteroids, process for their preparation, process for the preparation of the corresponding 9(11)-dehydro-derivatives and pharmaceutical preparations containing said steroids
03/07/1995US5395842 Inhibitors of sex steroids
03/07/1995CA1334668C 13-alkyl-11beta-phenylgonanes
02/1995
02/28/1995US5393785 Therapeutic antiestrogens
01/1995
01/17/1995US5382661 Useful in treating spinal trauma, head injury, subarachnoid hemorrhage
01/12/1995DE4321937A1 Cardiac glycosides
01/10/1995US5380841 Pyridinylpiperazinyl steroids
01/10/1995US5380840 Triazinylpiperazinyl steroids
01/10/1995US5380839 Phenylpiperazinyl steroids
12/1994
12/28/1994CN1096790A New 17,20-epoxide derivatives of pregnane, their preparation, their use in the preparation of cortisome derivatives and intermediates
12/13/1994US5372996 Method of treatment of androgen-related diseases
11/1994
11/24/1994WO1994026767A1 Improved antiandrogens
11/24/1994CA2136303A1 Improved antiandrogens
11/23/1994EP0532565B1 STARTING COMPOUNDS FOR THE PRODUCTION OF 10$g(b)-H STEROIDS AND PROCESS FOR PRODUCING SUCH STARTING COMPOUNDS
11/23/1994EP0532562B1 PROCESS FOR PRODUCING 10$g(b)-H-STEROIDS
11/17/1994EP0624162A1 Novel steroid intermediates and processes for their preparation
11/15/1994US5364847 Inhibitors of sex steroid biosynthesis and methods for their production and use
11/10/1994WO1994025479A1 Spirostanyl glycosidal crystalline monohydrate
11/10/1994CA2161239A1 Spirostanyl glycosidal crystalline monohydrate
11/09/1994EP0623140A1 Novel 19-nor steroids having a thiocarbon-containing chain in the 11beta position, a method for preparing same and intermediates therefor, medicinal uses thereof and compositions containing said steroids
11/08/1994US5362721 Corticoid-17-alkyl-carbonates substituted in the 17-position, process for their preparation and pharmaceuticals containing them
10/1994
10/26/1994CN1026324C 11beta-(4-isopropenylbenzene)-4,9-estrobiene, preparation of same and pharmaceutical containing same
10/25/1994US5359071 15-substituted 4-azasteroids
10/25/1994US5359054 Initial compounds for the production of 10β-H-steroids and a process for the production of these initial compounds
10/19/1994CN1026236C Steroid 5-alpha-reductase inhibitors
10/11/1994CA1332409C 9-alpha-hydroxy-17-methylene steroids, process for their preparation and their use in the preparation of corticosteroids
10/04/1994US5352809 9-alpha-hydroxy steroids, process for their preparation, process for the preparation of the corresponding 9(11)-dehydro derivatives and pharmaceutical preparations containing such steroids
09/1994
09/21/1994EP0615448A1 Sex steroid activity inhibitors
09/15/1994WO1994020104A1 15-substituted 4-azasteroids
09/15/1994CA2157363A1 15-substituted 4-azasteroids
09/01/1994WO1994019366A1 Chemical synthesis of squalamine
08/1994
08/18/1994WO1994018224A1 Steroids for treating menopausal complaints
08/18/1994CA2155532A1 Steroids for treating menopausal complaints
08/16/1994CA1331457C Aromatic steroid 5-–-reductase inhibitors
08/09/1994US5336686 17 Methylene lactones of steroids
07/1994
07/20/1994EP0607088A1 New 17,20-epoxy pregnane derivatives, their use in the preparation of cortisone derivatives and intermediates therefor
06/1994
06/21/1994US5322943 Piperazine compounds which are substituted
06/07/1994US5319115 Chemoselective and diastereoselective process from pregnane-3,20-dione; no need to protect 20-keto group
05/1994
05/03/1994CA1329195C Steroids useful as anti-cancer and anti-obesity agents
04/1994
04/06/1994CN1084857A 17-spiromethylene steroids
03/1994
03/31/1994WO1994006819A1 Gestagen-effective 4,5;11,12-estradienes, process for their production, medicaments containing these estradienes and their use in producing medicaments
03/30/1994EP0589034A1 METHOD FOR MAKING 3$g(a)-HYDROXY,3$g(b)-SUBSTITUTED-PREGNANES
03/24/1994DE4232521A1 Gestagen wirksame 4,5;11,12-Estradiene, Verfahren zu ihrer Herstellung, diese Estradiene enthaltende Arzneimittel sowie deren Verwendung zur Herstellung von Arzneimitteln Progestin effective 4,5; 11,12-Estradiene, to processes for their preparation, pharmaceutical compositions containing Estradiene and their use for the preparation of medicaments
03/15/1994US5294704 4,9(11),17(20)-pregnatriene-3-ones
03/08/1994US5292878 17-spirofuran-3'-ylidene steroids
03/03/1994WO1994004553A1 Method of preparing 1-methyl-3-keto-δ1,4-steroids
03/01/1994CA1327352C Steroid 5-.alpha.-reductase inhibitors
02/1994
02/17/1994DE4227053A1 Verfahren zur Herstellung von 1-Methyl-3-keto-ï·1·,·4·-steroiden -steroiden Process for the preparation of 1-methyl-3-keto-i · 1 · · · 4
02/09/1994EP0582338A2 17-Spiromethylene steroids
02/09/1994CN1081682A 甾类衍生物 Steroid derivatives
02/03/1994WO1993010741A3 Sex steroid activity inhibitors
02/03/1994DE4221960A1 Cardiac glycoside(s) prepd. e.g. from canrenone - with a more potent positive inotropic effect than spironolactone or canrenone but without their undesirable side effects
01/1994
01/11/1994CA1326015C 19,11.beta.-bridged steroids, their manufacture and pharmaceutical preparations containing them
01/11/1994CA1326014C 11.beta.-alkynl-estrenes and -estradienes, their production, and pharma ceutial preparations containing them
12/1993
12/29/1993EP0377009B1 1$g(b),15$g(a)-DIHYDROXY-1$g(a)-METHYL-5$g(a)-ANDROSTAN-3,17-DIONE, ITS PREPARATION AND USE
12/28/1993US5273971 13-alkyl-11β-phenylgonanes
12/23/1993WO1993025569A1 Oestradiol prodrugs
12/22/1993CN1079747A Steroid 5-alpha-reductase inhibitors
12/21/1993US5272140 11-aryl steroid derivatives
12/15/1993EP0574317A1 A new process for the preparation of 20-keto, 21-alpha-hydroxy steroids and intermediates therefor
12/07/1993US5268477 Triazinylpiperazinyl amine intermediates
11/1993
11/25/1993WO1993015103A3 Novel steroid intermediates and processes for their preparation
11/09/1993US5260463 Process for the preparation of hydrocortisone
11/03/1993EP0567472A1 D-homo-(16-en)-11 beta-aryl-4-estrenes, process for producing them and their use as medicaments
10/1993
10/20/1993EP0565553A1 6,7-MODIFIED 11$g(b)-ARYL-4-ESTRENES
10/12/1993US5252565 Haloethyl-substituted steroid enzyme inhibitors
10/05/1993US5250712 1β,15α-dihydroxy-1α-methyl-5α-androstane-3,17-dione, its production and use
09/1993
09/29/1993EP0562849A2 Steroid derivatives
09/28/1993CA2092766A1 Steroid derivatives
09/16/1993WO1993018053A1 METHOD FOR MAKING 3α-HYDROXY,3β-SUBSTITUTED-PREGNANES
09/01/1993EP0558416A1 New 17-(methylene)-lactone spiro condensed steroids, method and intermediates for their production, their use as medicines and pharmaceutical compositions containing them
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