Patents
Patents for C07D 521 - Heterocyclic compounds containing unspecified hetero rings (16,203)
01/2003
01/22/2003EP1276725A2 5-substituted tetralones as inhibitors of ras farnesyl transferase
01/22/2003EP1034159B1 Process for the preparation of acylated cyclic 1,3-dicarbonyl compounds
01/22/2003CN1099407C Novel amino acid derivatives with improved multi-drug resistance activity
01/21/2003US6509379 Variables are as disclosed herein, their salts, processes and intermediates for their preparation, and their use for controlling harmful fungi and animal pests.
01/16/2003WO2003004512A1 Activators for oligonucleotide synthesis
01/16/2003WO2003004493A1 Novel compounds, their preparation and use
01/16/2003WO2003004467A2 Thiazole benzamide derivatives and pharmaceutical compositions for inhibiting cell proliferation, and methods for their use
01/16/2003WO2003004027A1 Substituted anilinic piperidines as mch selective antagonists
01/16/2003WO2003004023A1 1-alkyl-2-aryl-benzimidazole derivatives, their use for producing medicaments and pharmaceutical preparations containing said derivatives
01/16/2003US20030013715 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases
01/16/2003US20030013708 Therapeutic heterocyclic compounds
01/16/2003US20030013704 Adamantane derivatives
01/16/2003CA2454613A1 Substituted anilinic piperidines as mch selective antagonists
01/16/2003CA2452609A1 Thiazole benzamide derivatives and pharmaceutical compositions for inhibiting cell proliferation, and methods for their use
01/16/2003CA2448913A1 Sulfone containing bicyclic aromatic ring compounds, their preparation and use as nicotinic acetyl-chloine receptors
01/15/2003EP0974584B1 Fused ring compounds, process for producing the same and use thereof
01/15/2003CN1391555A Benzamides and related inhibitors of factor Xa
01/15/2003CN1391469A Npyy5拮抗剂 Npyy5 antagonist
01/14/2003US6506901 1-(9H-Carbazol-4-yloxy)-3-((1-(7-trifluoromethyl-quinolin-4-yl) -piperidin-4-lmethyl)-amino)-propan-2-ol, for example; treating diabetes, urinary continence, atherosclerosis, gastrointestinal disorders, glaucoma
01/14/2003CA2217516C Triazole antifungal agent
01/13/2003WO2002006237A1 Medicine comprising dicyanopyridine derivative
01/13/2003CA2415899A1 Medicine comprising dicyanopyridine derivative
01/09/2003WO2003002542A1 N-heterocyclic inhibitors of tnf-alpha expression
01/09/2003WO2003002519A1 Phenol derivatives and their use in medicaments
01/09/2003WO2003002518A1 Novel 2,4-difluorobenzamide derivatives as antiviral agents
01/09/2003WO2003002498A1 Intermediate halophenyl derivatives and their use in a process for preparing azole derivatives
01/09/2003WO2002059111A3 Pyrazole compounds useful as protein kinase inhibitors
01/09/2003WO2001072728B1 Novel piperazine derivatives
01/09/2003US20030008881 Substituted phenylcyclohexanecarboxamides and their use
01/09/2003US20030008879 For therapy of symptoms caused by withdrawal or partial withdrawal from the use of tobacco or of nicotine; for therapy of anxiety
01/09/2003US20030008832 Method of inhibiting neoplastic cells with benzimidazole derivatives
01/08/2003EP1272485A1 Novel 1,2,3,4-tetrahydrosioquinoline, their preparation method and their use as fungicides
01/08/2003EP1272472A1 1h-pyrazole derivatives, method for the production thereof and their use for inhibiting and controlling nitrification
01/08/2003CN1390206A Inhibitors of factor Xa
01/08/2003CN1098264C Substituted 4-(1H-benzimidzol-2-yl-amino) piepridines useful for the treatment of allergic diseases
01/07/2003US6504033 Nitrogen compounds formed from stoichiometric amounts of formic acid and hydrazine; by product inhibition; purity
01/07/2003US6503898 Administering 4,7-dibenzyl-5,6-dihydroxy-N,N*-di(m-aminobenzyl)--1,3-diazepin-2-one or salt to treat human immunodeficiency virus infection
01/03/2003WO2003000664A1 Uracil derivatives and the use thereof for treating bacterial diseases
01/03/2003WO2003000653A1 Substituted n-acyl aniline derivatives, production and use thereof as medicaments
01/03/2003WO2003000180A2 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/03/2003WO2002046170A8 Anilinopyrimidine derivatives as jnk pathway inhibitors and compositions and methods related thereto
01/03/2003CA2451625A1 Substituted n-acyl-aniline derivatives, the preparation thereof and the use thereof as pharmaceutical compositions
01/03/2003CA2450579A1 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/02/2003US20030004351 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
01/02/2003US20030004164 Anticancer agents; autoimmune diseases
01/02/2003US20030004161 Anticancer agents; autoimmune diseases
01/02/2003US20030004137 Muscle relaxants, controlling immunology, strokes, antidiabetic agents
01/02/2003EP1270571A1 Heterocyclic compounds, their production and use
01/02/2003EP1270561A1 Brassinosteroid biosynthesis inhibitor
01/02/2003EP1268471A1 N-heterocyclic derivatives as nos inhibitors
01/02/2003EP1268455A2 Piperazine derivatives
01/02/2003EP1268445A1 4-amino-5-cyano-2-anilino-pyrimidine derivatives and their use as inhibitors of cell-cycle kinases
01/02/2003EP1268444A1 2,4-di(hetero-)arylamino(-oxy)-5-substituted pyrmidines as antineoplastic agents
01/02/2003EP1268440A1 Imidazole carbenes
01/02/2003EP1268437A1 Inhibitors of protein kinases
01/02/2003EP1268412A1 Sulphonamido-substituted bridged bicycloalkyl derivatives
01/02/2003EP1268396A1 Diphenyl ether compounds useful in therapy
01/01/2003CN1388804A Amino acid-N-carboxy anhydrides having substitent at nitrogen
01/01/2003CN1097592C Slfonic acid amide derivatives with herbicides activity
12/2002
12/31/2002US6500952 Processes for preparing aminophenylsulfonylureas, and intermediates therefor
12/31/2002US6500817 Thiazolyl urea derivatives and their utilization as antiviral agents
12/31/2002CA2094917C Herbicidal n-[(1,3,5-triazin-2-yl)-aminocarbonyl]-benzenesulfonamides
12/27/2002WO2002074753A3 5-phenylpyrimidine, methods and intermediate products for the production thereof and use of the same for controlling pathogenic fungi
12/27/2002WO2002070473A3 Carboxamide derivatives as therapeutic agents
12/26/2002US20020198378 For therapy of retroviral infection, e.g., an HIV infection
12/26/2002US20020198216 Novel farnesyl protein transferase inhibitors as antitumor agents
12/25/2002CN1387529A N-substd. carbamoyloxyalkyl-azolium derivs.
12/25/2002CN1387528A Heterocyclic substd, pyrazolones
12/25/2002CN1387514A Aromatic sulfone hydroxamic acid metalloprotease inhibitor
12/25/2002CN1097052C Process for production of amidinoindole derivs, and salts thereof
12/24/2002US6498253 Acylated aminophenylsulfonylureas, processes for their preparation and their use as herbicides and plant growth regulators
12/24/2002US6498190 Bicyclic amino derivatives and PGD2 antagonist containing the same
12/24/2002US6498159 Such as 4-((3-chloro-4-methoxybenzyl)amino)-1-((4-hydroxy-4 -hydroxymethyl)piperidino)-6-phthalazine carbonitrile
12/24/2002US6497905 Aqueous solubility pharmaceutical formulations
12/24/2002CA2252402C Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment
12/24/2002CA2150812C Catechol diethers as selective pde iv inhibitors
12/19/2002WO2002100813A2 Modulators of peroxisome proliferator activated receptors
12/19/2002WO2002059080A3 Trisubstituted carbocyclic cyclophilin binding compounds and their use
12/19/2002WO2002042248A3 Naphthalene derivatives
12/19/2002US20020193614 Treatment of cardiovascular disorders
12/19/2002US20020193596 Inhibitors of protein isoprenyl transferases
12/19/2002US20020193578 Compounds having activity as inhibitors of cytochrome P450RAI
12/19/2002US20020193432 Useful as modulators of the interaction between the receptor for advanced glycated end product and its ligands
12/19/2002US20020193414 Adamantane derivatives
12/19/2002US20020193411 Pesticidal 1-polyarylpyrazoles
12/19/2002US20020193405 For prophylaxis and therapy of diseases, such as cell proliferation or apoptosis mediated diseases
12/19/2002US20020193398 For therapy and prophylaxis of blood coagulation and cardiovascular disorders
12/19/2002US20020193382 Sulfonamide derivatives, their production and use
12/19/2002DE10121003A1 Anthranilsäureamide, Verfahren zur Herstellung, ihrer Verwendung als Medikament sowie sie enthaltende pharmazeutische Zubereitungen Anthranilic acid amides, processes for preparing, their use as a medicament as well as pharmaceutical compositions containing them
12/19/2002CA2449256A1 Modulators of peroxisome proliferator activated receptors
12/18/2002EP1064273B1 1,3,4-thiadiazoles useful for the treatment of cmv infections
12/17/2002US6495699 Antiarthritic agents; osteoporosis
12/17/2002US6495564 Such as 3-(6-((4-chloro-phenyl)-hydroxy-(3-methyl-3h-imidazol-4-yl)-methyl)-1-methyl-2-oxo-1,2-dihydro-quinolin-4-yl)-benzaldehyde o-methyl-oxime; inhibiting abnormal cell growth
12/17/2002US6495552 Treatment or prevention of the diseases and conditions which respond to treatment by retinoids and or which in healthy mammals, including humans, are controlled by natural retinoic acid.
12/17/2002US6495550 Substituted benzamido-pyridine derivatives for treatment of disorders mediated by potassium channels
12/17/2002US6495542 Such as 2-methoxy-n-(2-methyl-1h-benzimidazol-4-yl)-4-(2,3,4,5-tetrahydro-5-oxo-1h-1-benzazepin-1-yl)carbonyl-benzam ide; hypertension, heart failure, renal insufficiency, edema, ascites, vasopressin parasecretion syndrome
12/17/2002US6495270 Addition product of a heterocyclic amidine and a quinone is accelerator; encapsulation of electronic component parts; rapid curability, curability after moisture absorption under moist condition, pot life and flow properties
12/12/2002WO2002098852A2 Novel benzothienyl or indole derivatives, and use thereof as inhibitors of prenyl transferase proteins
12/12/2002WO2002098849A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer’s disease and similar diseases
12/12/2002WO2002098848A1 Benzoylsulfonamides and sulfonylbenzamidines for use as antitumour agents
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