Patents
Patents for C07D 521 - Heterocyclic compounds containing unspecified hetero rings (16,203)
02/2004
02/11/2004CN1474816A 4-amino-quinazolines
02/11/2004CN1474803A Novel amide derivatives and medicinal use thereof
02/11/2004CN1137888C Inhibitor of cysteninyl aspartic acid proteinase
02/10/2004CA2291975C Quaternary ammonium compounds
02/05/2004WO2004011460A2 Pyrazolylbenzothiazole derivatives and their use as therapeutic agents
02/05/2004WO2004011437A1 Novel imidazole alcohol compound, process for producing the same, and surface-treating agent comprising the same
02/05/2004WO2004011436A1 Quinoline derivatives and their use as mycobacterial inhibitors
02/05/2004WO2004011410A1 Chemical compounds
02/05/2004WO2004011399A1 Ionic liquid osmium oxide
02/05/2004US20040024215 Such as 4'-trifluoromethyl-biphenyl-2-carboxylic acid(4-(4-(alpha-methyl-benzyl)-piperazin-1-yl)-phenyl)-amide; apoprotein B-100 (apoB-100) and microsomal triglyceride transfer protein (MTP)
02/05/2004US20040024205 Monomethylation of nitrogeneous heterocycles
02/05/2004DE10231627A1 New 1-benzoyl-3-(heterocyclyl-phenyl)-urea derivatives, are glycogen phosphorylase a inhibitors useful e.g. for treating type II diabetes, dyslipidemia or arteriosclerosis
02/05/2004CA2494668A1 Chemical compounds
02/04/2004EP1386916A1 Process for the monomethylation of nitrogen containing heterocycles
02/04/2004EP1386912A1 Cyclic amidine derivative
02/04/2004EP1385820A1 Anthranilic acid amides, method for the production thereof, their use as antiarrhythmia agents, and pharmaceutical preparations thereof
02/04/2004EP0813526B1 Process for preparing n-substituted pyrazoles
02/04/2004EP0813525B9 Benzamidine derivatives their preparation and their use as anti-coagulants
02/04/2004CN1473161A Pyrazole compounds as protein kinase inhibitors
02/04/2004CN1473160A Indole derivatives as medicinal compositions for antifungal and/or antiparasitic agents
02/04/2004CN1473155A Pyrimidine derivatives and herbicides containing the same
02/04/2004CN1137119C Substituted thineyl (amino) sulfonylureas
02/04/2004CN1137118C Water soluble azoles as broad-spectrun antifungals
02/04/2004CN1137102C Substituted propyl triazole as antifungal compound and its salts and their prepn
02/04/2004CN1137084C Aryne intermediates and process for preparation thereof
02/03/2004US6686368 Inhibitors of factor Xa
02/01/2004CA2434481A1 Process for the methylation of nitrogenated heterocyclics
01/2004
01/29/2004WO2003000180A3 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/29/2004US20040019216 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
01/29/2004US20040019045 Pyrazole compounds as anti-inflammatory and analgesic agents
01/29/2004US20040019016 Polycyclic compounds containing a central trivalent atom to which is attached either direct or indirectly via a linker a two or three ring system and a ring system contining sulphamate group as substituent; steroid sulfatase inhibitor
01/28/2004EP1384712A1 Derivatives of N-((quinolinyl)oxy)-phenyl)-urea and N-((quinazolinyl)oxy)-phenyl)-urea with antitumor activity
01/28/2004EP1383731A1 Biaryl compounds as serine protease inhibitors
01/28/2004EP0794947B1 N-substituted hydrazinophenylsulphonyl ureas used as herbicides and plant-growth regulators
01/28/2004CN1471524A Novel farnesyl protein transferase inhibitors as antitumor
01/28/2004CN1471522A Cholesterol lowering benzo [b] thiophenes and benzo[d] isothiazoles
01/28/2004CN1471506A Method for preparing carbonyl alpha-substituted nitrogen compounds
01/28/2004CN1136213C New benzothiophene, benzofuran and indole compounds, preparation method there for and medicine composition containing them
01/28/2004CN1136203C Benzoxazine and penzothiazine derivatives and their use in pharmaceuticals
01/27/2004US6683215 N-(4-carbamimidoyl-phenyl)-glycine derivatives
01/27/2004US6683097 Imidazole derivatives
01/27/2004US6683093 Enzyme inhibitors; cardiovascular disorders; antiinflammatory agents; autoimmune disease
01/27/2004US6683091 Heterocyclic sulfanamides; alzheimer's disease; preventing deposition of amyloid protein
01/27/2004CA2089464C N-heteroaryl-n'-(pyrid-2-yl-sulfonyl)ureas, processes for their preparation, and their use as herbicides and plant growth regulators
01/27/2004CA2062387C Process for the preparation of sulfonylureas
01/22/2004WO2004007469A1 New alkynylated quinazolin compounds as mmp-13 inhibitors
01/22/2004WO2004007455A1 Heterocyclically substituted benzoylureas, method for their production and their use as medicaments
01/22/2004US20040014967 Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound
01/22/2004CA2493374A1 Heterocyclically substituted benzoylureas, method for their production and their use as medicaments
01/21/2004EP1381598A1 Novel tyrosine kinase inhibitors
01/21/2004CN1469876A Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
01/21/2004CN1469875A Pyrazole compounds useful as protein kinase inhibitors
01/21/2004CN1469874A Pyrazole compounds useful as protein kinase inhibitors
01/21/2004CN1135229C Water soluble azoles as broad-spectrum antifungals
01/20/2004US6680315 Compounds that down-regulate interleukin-12 production used for treating inflammatory diseases: rheumatoid arthritis, sepsis, chrohn's disease, multiple sclerosis, psoriasis or insulin-dependent diabetes
01/20/2004US6680312 Sulfonamide derivatives, their production and use
01/20/2004CA2174104C Tricyclic amide and urea compounds useful for inhibition of g-protein function and for treatment of proliferative diseases
01/15/2004WO2004005249A1 Pyrrolidine derivatives as oxytocin antagonists
01/15/2004US20040010143 Viricides
01/15/2004US20040009992 Azolylalkylazole derivatives, their preparation, and their use as pesticides
01/15/2004US20040009526 Common ligand mimics: thiazolidinediones and rhodanines
01/14/2004EP1379525A2 Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
01/14/2004EP1379510A1 Aryl and heteroaryl urea chk1 inhibitors for use as radiosensitizers and chamosensitizers
01/14/2004EP1379498A1 Sulphones which modulate the action of gamma secretase
01/14/2004EP1379496A1 Sulphones which modulate the action of gamma secretase
01/14/2004EP1379493A2 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
01/14/2004CN1468227A Non-imidazole aryloxyalkylamines
01/14/2004CN1468221A Non-imidazole aryloxypiperidines
01/14/2004CN1468207A New retinoids for the treatment of emphysema
01/14/2004CN1134421C Antifungal and its preparation method and intermediate
01/14/2004CN1134411C Bicyclic amino derivatives and PGD2 antagonist containing same
01/14/2004CN1134410C Amine derivative, process for producing same, and use thereof as antiarrhythmic medicine
01/13/2004US6677452 Pyridine carboxamide or sulfonamide derivatives and combinatorial libraries thereof
01/08/2004WO2004002985A1 Peptidic thrombin inhibitor compound
01/08/2004US20040006238 As chemical intermediates for production of pharmacologically useful oxazolidinones
01/08/2004US20040006105 Thrombin receptor antagonists
01/08/2004US20040006076 Thiazolyl amide derivatives
01/08/2004US20040006068 Pyrimidine derivatives
01/07/2004EP1378507A2 Process for producing optically active imidazole compounds, intermediates for synthesizing the same, and process for producing the same
01/07/2004EP1377582A1 Novel 3-c(o)r substituted 10-cyclohexylbenzoyl pyrrolobenzodiazepines; tocolytic oxytocin receptor antagonists
01/07/2004EP1377556A1 Pyrazole derivatives for treating hiv
01/07/2004EP1377295A2 Carboxamide derivatives as therapeutic agents
01/07/2004CN1133623C Process for producing optically active imidazole compound, intermediates for synthesizing samke and mfg method
01/07/2004CN1133372C Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl] piperidines
01/06/2004US6673931 (4-(4-(3-(2-methoxy-benzyloxy)-propoxy)-phenyl)-5-(4-methoxy -naphthalen-2-ylmethoxy)-piperidin-3-yl)-methanol for example; use treating restenosis, glaucoma, cardiac and kidney insufficiency
01/06/2004CA2285891C Triazole antifungal agents
01/02/2004EP1373228A1 Substituted fluoroalcoxyphenylsulfonylurea
01/02/2004EP1373222A2 5-phenylpyrimidine, methods and intermediate products for the production thereof and use of the same for controlling pathogenic fungi
01/02/2004EP1373203A1 Cyclopropylindole derivatives as selective serotonin reuptake inhibitors
01/02/2004EP1372615A1 Compounds and compositions for delivering active agents
01/01/2004US20040002542 Succinoylamino hydroxyethylamino sulfonyl urea derivatives useful as retroviral protease inhibitors
01/01/2004US20040002523 Aryl substituted pyrazoles, triazoles and tetrazoles, and the use thereof
01/01/2004US20040002506 Antiproliferative agents; antitumor agents
01/01/2004US20040002496 Compositions useful as inhibitors of protein kinases
01/01/2004US20040002491 Melatonergic receptors
01/01/2004US20040002490 Melatonergic receptors
12/2003
12/31/2003WO2004000835A1 Method for the production of 1,2,4-triazolylmethyl-oxiranes
12/31/2003WO2004000826A1 Processes for producing epoxytriazole derivative and intermediate therefor
12/31/2003WO2004000808A2 N-substituted piperidine derivatives as serotonin receptor agents
12/31/2003WO2004000214A2 Use of compounds having an amine nucleus in manufacture of a medicament useful for treating factor viia-associated conditions
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