Patents
Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041)
11/2000
11/02/2000CA2371274A1 Selective npy (y5) antagonists
11/02/2000CA2369109A1 Thrombin inhibitors
10/2000
10/31/2000CA2149514C Novel cephem derivatives
10/26/2000WO2000063215A2 Indazole derivatives, preparation and therapeutic application thereof
10/26/2000WO2000035919A3 Quinoline derivatives
10/26/2000WO2000035886A3 (hetero)aryl-bicyclic heteroaryl derivatives, their preparation and their use as protease inhibitors
10/19/2000WO2000061583A1 Xanthine derivatives and analogs as cell signaling inhibitors
10/19/2000WO2000012507A8 Pyrrolobenzodiazepines
10/19/2000CA2369981A1 Therapeutic compounds for inhibiting interleukin-12 signaling and methods for using same
10/18/2000EP1043988A1 C-10 carbon-substituted artemisinin-like trioxane compounds having antimalarial, antiproliferative and antitumour activities
10/18/2000EP0633886B1 Pharmaceutically active bicyclic-heterocyclic amines
10/18/2000CN1270519A Anti-first-pass effect compounds
10/17/2000US6133260 Use of 7-(2-oxa-5,8-diazabicyclo[4.3.0]non-8-yl)-quinolone carboxylic acid and naphthyridon carboxylic acid derivatives for the treatment of Helicobacter pylori infections and associated gastroduodenal diseases
10/17/2000CA2001205C Antimicrobial quinolonyl lactams
10/11/2000CN1269800A Tetrahydro Gamma-carbolines
10/04/2000EP1041074A1 Light-sensitive 4-cyanocoumarin derivatives
10/04/2000EP1040112A1 Imidazonaphthyridines and their use in inducing cytokine biosynthesis
10/04/2000EP1040111A1 Integrin receptor antagonists
10/04/2000EP1040098A1 Integrin receptor antagonists
10/04/2000EP1039906A1 Novel metal complexes
10/04/2000CN1057091C Novel carbapenem derivatives
10/03/2000US6127377 Chlorinated vinblastine as anticancer chemotherapy drug
09/2000
09/28/2000WO2000056734A1 Bicyclic heterocycles, method for producing them and their use as herbicides and pharmaceutical agents
09/28/2000WO2000056719A1 FUSED PYRIDOPYRIDAZINE INHIBITORS OF cGMP PHOSPHODIESTERASE
09/28/2000WO2000056304A2 Anti-inflammatory uses of manzamines
09/28/2000WO2000044727B1 Inhibitors for the biosynthesis of vitamin b2 and method for producing same
09/28/2000CA2368023A1 Fused pyridopyridazine inhibitors of cgmp phosphodiesterase
09/27/2000EP1038863A2 Substituted dimeric compounds, process for their preparation and pharmaceutical compositions thereof
09/27/2000EP1038027A1 Decreasing cell proliferation by decreasing levels of pp5
09/27/2000EP1037865A1 Synthesis of cc-1065/duocarmycin analogs
09/27/2000CN1056832C Fused dihydropyridine derivate, its producing process, and its pharmaceutical composition
09/26/2000US6124293 Semi-synthetic ecteinascidins
09/21/2000WO2000054768A1 Anti-first-pass effect compounds
09/21/2000WO2000012508A3 Pyrrolbenzodiazepines
09/21/2000DE19912636A1 Bicyclische Heterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Herbizide und pharmazeutische Mittel Bicyclic heterocycles, process for their preparation and their use as herbicides and pharmaceutical compositions
09/20/2000EP1036821A1 Process for the preparation of thiazine-indigo compounds and of new intermediates therefor
09/20/2000EP1036076A1 Novel compounds
09/14/2000WO2000053602A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone
09/14/2000WO2000053185A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone
09/14/2000WO2000053181A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone
09/14/2000WO2000053180A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone
09/14/2000WO1999063999A8 H1-histamine receptor antagonists
09/14/2000CA2367130A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone
09/14/2000CA2367126A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone
09/14/2000CA2367121A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone
09/14/2000CA2366615A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone
09/13/2000EP0983248A4 Analogs of duocarmycin and cc-1065
09/06/2000EP1032384A1 Carbapenem antibacterial compounds, compositions and methods of treatment
09/06/2000EP1032383A1 Antibacterial carbapenems, compositions and methods of treatmemt
09/06/2000EP0593766B1 Pyridonecarboxylic acid derivative
09/06/2000CN1265671A Alatrofloxacin parenteral compositions
09/05/2000US6114351 N-oxides as antibacterial agents
08/2000
08/31/2000WO2000012507A3 Pyrrolobenzodiazepines
08/30/2000EP0770083B1 PYRIDO[3,2,1-i,j][3,1]BENZOXAZINE DERIVATIVES
08/29/2000US6110931 For pregnancy prophylaxis and treatment of glandular disorders, hormone deficiency disorders, gastrointestinal disorders, growth disorders
08/24/2000WO2000037470A8 Antihistaminic spiro compounds
08/23/2000EP1028962A1 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment
08/17/2000WO2000047583A1 Cyclic substituted fused pyrrolocarbazoles and isoindolones
08/17/2000WO2000047571A1 Piperidine and piperazine derivatives as inhibitors of the abeta fibril formation
08/17/2000CA2362389A1 Piperidine and piperazine derivatives as inhibitors of the abeta fibril formation
08/16/2000CN1263531A Azadirachtin extraction process
08/16/2000CN1055474C Noval crystal type anhydrous 7-([1 alpha, 5 alpha, 6 alpha]=6-amino-3-azabicyclo [3,1,0] hexyl-3-group)-6-fluorine-1-(2,4-difluorophenyl
08/15/2000US6103751 Injecting a carotene conjugate of a photosensitizer selected from porphyrins, chlorins and bacteriochlorins into an animal at a desired dosage and detecting loactions of the concentrated uptake of the compound by spectroscopy
08/10/2000WO1999063936A9 Novel therapeutic agents that modulate endothelin receptors
08/09/2000EP1025109A1 Benzoxazine derivatives, preparation and application in therapy
08/09/2000EP1025099A1 Bis-quaternary ammonium derivatives as neuromuscular relaxants
08/08/2000US6100392 Electron-deficient porphyrins and processes and intermediates for preparing same
08/08/2000US6100252 Specified compounds including methyl 2-butyl-1-((2'-(2-oxo-3h-1,2,3,5-oxathiadiazol-4-yl)biphenyl) methyl)-benzimidazole-7-carboxylate; use to treat circulatory diseases such as hypertensive diseases and heart diseases
08/03/2000WO2000045165A1 Methods of identifying therapeutically effective antineoplastic agents with cultured cells having intact cell membranes and corresponding products
08/03/2000WO2000044755A1 Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands
08/03/2000WO2000044727A1 Inhibitors for the biosynthesis of vitamin b2 and method for producing same
08/03/2000WO2000044377A1 Mono-acyloxy aralkyl neuromuscular relaxants
08/03/2000WO2000044216A2 Gambogic acid, analogs and derivatives as activators of caspases and inducers of apoptosis
08/03/2000WO2000020421A3 TRICYCLIC Δ3-PIPERIDINES AS α2-ANTAGONISTS
08/03/2000WO2000006582A9 Trimeric and polymeric alkaloids
08/03/2000DE19903736A1 Inhibitoren der Biosynthese von Vitamin B2 und Verfahren zu ihrer Herstellung Inhibitors of the biosynthesis of vitamin B2 and process for their preparation
08/03/2000CA2396005A1 Gambogic acid, analogs and derivatives as activators of caspases and inducers of apoptosis
08/03/2000CA2360790A1 Mono-acyloxy aralkyl neuromuscular relaxants
08/02/2000EP1023302A1 Binuclear complex
08/02/2000EP1023293A1 Aryloxymethyl carbapenem antibacterials
08/02/2000EP1023062A1 Antibacterial carbapenems, compositions and methods of treatment
08/02/2000EP1022951A1 Compositions and methods for the treatment of primary and metastatic neoplastic diseases using arsenic compounds
08/02/2000EP0527889B1 Quinolizinone type compounds
07/2000
07/27/2000WO2000042989A2 Novel hydrogel isolated cochleate formulations, process of preparation and their use for the delivery of biologically relevant molecules
07/27/2000WO1999066944A9 Methods for identifying novel multimeric agents that modulate receptors
07/27/2000WO1999064033A9 Phosphodiesterase-v modulator drugs and their uses
07/27/2000WO1999063994A9 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE
07/26/2000EP1022279A1 New carbapenem derivatives
07/26/2000EP1021451A1 Asymmetric synthesis and catalysis with chiral heterocyclic compounds
07/26/2000EP1021445A1 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment
07/26/2000EP1021438A1 Trioxane dimer compounds having antiproliferative and antitumor activities
07/25/2000US6093717 Imidazopyridine thrombin inhibitors
07/25/2000US6093714 An antiallergens for treatment and prevention of bronchial asthma, eczema, hives, allergic gastrointestinal troubles, allergic rhinitis, allergic conjunctivitis
07/20/2000WO2000042046A1 Artemisinin analogs having antimalarial, antiproliferative, and antitumor activities and chemoselective methods of making the same
07/20/2000WO2000042040A1 Tricyclic inhibitors of poly(adp-ribose) polymerases
07/20/2000WO1999064048A9 Inhibitors of hiv reverse transcriptase
07/20/2000CA2360383A1 Artemisinin analogs having antimalarial, antiproliferative, and antitumor activities and chemoselective methods of making the same
07/19/2000EP1020446A1 Naphthalimidobenzamide derivatives
07/19/2000EP1019426A1 Novel a 1? adenosine receptor agonists and antagonists
07/19/2000EP1019408A1 1,2,3,4-TETRAHYDRO-BENZOFURO 3,2-c]PYRIDINE DERIVATIVES--
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