Patents
Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041)
12/2002
12/12/2002WO2002098427A2 Sustained-release analgesic compounds
12/12/2002US20020188124 Novel spiro compounds
12/12/2002US20020187999 Anti-inflammatory uses of manzamines
12/12/2002US20020187983 Process for the synthesis of derivatives of 2, 3-dihydro-1, 4-dioxino- [2, 3-f] quinoline
12/12/2002CA2448665A1 Sustained-release analgesic compounds
12/12/2002CA2445460A1 Carboline derivatives as pde-5 inhibitors
12/11/2002EP1263762A1 Anti-infective ectatm
12/11/2002EP1263759A2 Azaindoles
12/11/2002CN1384833A Synthesis and methods of use of 9-substituted guanine derivatives
12/10/2002US6492408 Peptidomimetic inhibitors of intercellular adhesion molecules binding to leukointegrins, such as lfa-1 and mac-1
12/10/2002CA2092431C 3,9-diazabicyclo (3.3.1) nonan-7-yl derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them
12/05/2002WO2002096907A1 Bicyclic nitrogen-containing heterocyclic derivatives for use as antibacterials
12/05/2002WO2002096426A1 Hydantion derivatives as inhibitors of matrix metalloproteinases
12/05/2002US20020183385 Administering a therapeutically effective amount of arsenic compounds to a mammal for treating solid tumor
12/05/2002US20020183354 For therapy of depression and other diseases such as obsessive compulsive disorder, panic attacks, generalized anxiety disorder, social anxiety disorder, sexual dysfunction, eating disorders, obesity, addictive disorders
12/05/2002US20020183353 For therapy of depression, obsessive compulsive disorder, panic attacks, generalized anxiety disorder, social anxiety disorder, sexual dysfunction, eating disorders, obesity, addictive disorders caused by ethanol or cocaine abuse
12/05/2002US20020183352 Antidepressant indoletetrahydropyridine derivatives of 2,3-dihydro-7H-[1,4]dioxino[2,3-e]indole
12/05/2002US20020183351 For therapy of depression, obsessive compulsive disorder, panic attacks, generalized anxiety disorder, social anxiety disorder, sexual dysfunction, eating disorders, obesity, addictive disorders caused by ethanol or cocaine abuse
12/05/2002US20020183341 Antidepressant azaheterocyclylmethyl derivatives of 2,3-dihydro-1,4-dioxino[2,3-f]quinazoline
12/05/2002US20020183336 Azabicyclylmethyl derivatives of 7,8-dihydro-1,6,9-trioxa-3-aza-cyclopenta[a]naphthalene as 5-ht1a antagonists
12/05/2002US20020183330 For therapy of schizophrenia, schizoaffective disorder, bipolar disorder, Parkinson's disease, L-DOPA induced psychoses or dyskinesias, Tourette's syndrome, hyperprolactinemia, or addiction to ethanol, nicotine, cocaine
12/05/2002US20020183329 Antidepressant azaheterocyclylmethyl derivatives of 2,3-dihydro-1,4-dioxino[2,3-f]quinoxaline
12/05/2002US20020183322 Azabicyclylmethyl derivatives of 2,3-dihydro-1,4-dioxino[2,3-f]quinoline as 5-HT1A antagonists
12/05/2002US20020182151 Aids therapy
12/05/2002CA2447475A1 Hydantion derivatives as inhibitors of matrix metalloproteinases
12/04/2002EP1262477A1 Anti-acid-fast bacterial agents containing pyridonecarboxylic acids as the active ingredient
12/04/2002EP1261607A1 2,4-disubstituted thiazolyl derivatives
12/03/2002US6489477 Nmda nr2b antagonists. accordingly, another aspect of the invention is the treatment of pain, migraine, depression, anxiety, schizophrenia, parkinson's disease, or stroke--maladies that are amenable to amelioration through
12/03/2002US6489471 A process of synthesizing a carbapenem compound of formula (6) is disclosed, wherein r represents h or methyl, p and p* independently represent h or protecting groups and each r.sup.1 is independently selected from: h, halo, oh, op
11/2002
11/28/2002US20020177609 Fatty alcohol drug conjugates
11/28/2002US20020177600 Two or more ligand moieties covalently linked together by one or more linking groups enabling binding to multiple binding sites; increased efficacy, selectivity and duration; anti-proliferative and anticarcinogenic
11/28/2002US20020177591 Central nervous system (CNS); diazabicyclo compounds such as 1,4-Diaza-bicyclo(3.2.2)nonane-4-carboxylic acid, 4-cyclohexyl-phenyl ester; CNS-penetrant alpha 7 nicotinic receptor agonist
11/28/2002US20020177559 Inhibitors of cellular efflux pumps of microbes
11/27/2002EP1259514A2 3-(pyrolyllactone)-2-indolinone compounds as kinase inhibitors
11/27/2002EP1259236A1 Tyrosine kinase inhibitors
11/27/2002CN1381456A Pyrimidine-4-keto compound, its preparation method and medicine composition containing them
11/26/2002CA2102889C Imidazo[1,2-a](pyrrolo, thieno or furano)[3,2-d]azepine derivatives, compositions and methods of use
11/26/2002CA2076465C Cell binding agent conjugates of analogues and derivatives of cc-1065
11/21/2002WO2002092602A2 PROCESSES FOR THE SYNTHESIS OF DERIVATIVES OF 2,3-DIHYDRO-1,4-DIOXINO-[2,3-f] QUINOLINE
11/21/2002WO2002022598A8 Quinolinone derivatives as tyrosine kinase inhibitors
11/21/2002US20020173654 Imidazonaphthyridine and tetrahydroimidazonaphthyridine compounds induce the biosynthesis of cytokines such as interferon and tumor necrosis factor, and useful as viricides and antitumor agents
11/21/2002US20020173445 Selective androgen receptor modulators and methods for their identification, design and use
11/21/2002CA2447150A1 Processes for the synthesis of derivatives of 2,3-dihydro-1,4-dioxino-[2,3-f] quinoline
11/20/2002EP0656360B1 Trifluoromethylpyrroloindole carboxylic ester derivative and process for producing the same
11/19/2002US6482845 Method for inhibiting interleukin-2 production using tricyclo compounds
11/14/2002WO2002090362A1 Azaheterocyclylmethyl derivatives of 7,8-dihydro-1,6,9-trioxa-3-aza-cyclopenta[a]naphthalene as 5-ht1a antagonists
11/14/2002WO2002090357A1 Disubstituted 1,7-guanines
11/14/2002WO2002089806A1 Heterobicycles fkbp-ligands
11/14/2002WO2002076399A3 YOHIMBINE DIMERS EXHIBITING BINDING SELECTIVITES FOR α2 ADRENERGIC RECEPTORS
11/14/2002US20020169178 Benzothieno[3,2-c]pyridines as alpha2 antagonists
11/14/2002US20020169155 A nitrogen-ring containing triheterocyclic compound is useful for treating a disease associated with aberrant leukocyte recruitment and/or activation
11/14/2002CA2446795A1 Sulfamide, sulfamate, sulfonamide, urea, amide, alpha, alpha-difluoro amide oxalyl diamide, and heterobicycles fkbp-binding ligands
11/13/2002EP1256583A1 Pyrimidine-4-one derivatives, process for their preparation and pharmaceutical compositions containing them
11/13/2002EP1256582A1 1h-imidazopyridine derivatives
11/13/2002EP1256581A1 Preventive or therapeutic agents for gastric or esophageal regurgitation
11/13/2002EP1255739A1 3-aminoquinazolin-2,4-dione antibacterial agents
11/13/2002EP1090006A4 Alkyl ether analogs of chlorins having an n-substituted imide ring
11/13/2002EP0846119B1 Thienopyrimidine derivatives, their production and use as endothelin antagonists
11/13/2002CN1379777A Amino-triazolopyridine derivatives
11/12/2002CA2103242C Imidazo[2,1-b][3]benzazepine derivatives, compositions and method of use
11/07/2002WO2002088274A1 Double-spiro organic compounds and electroluminescent devices
11/07/2002WO2002088147A1 Sulfate of cephem compound
11/07/2002WO2002088146A2 ANTIDEPRESSANT INDOLETETRAHYDROPYRIDINE DERIVATIVES OF 2,3-DIHYDRO-7H-[1,4]DIOXINO[2,3-e]INDOLE
11/07/2002WO2002088145A1 AZABICYCLYLMETHYL DERIVATIVES OF 7,8-DIHYDRO-1,6,9-TRIOXA-3-AZACYCLOPENTA[a]NAPHTHALENE AS 5-HT1A ANTAGONISTS
11/07/2002WO2002088144A2 ANTIDEPRESSANT AZAHETEROCYCLYLMETHYL DERIVATIVES OF 2,3-DIHYDRO-1,4-DIOXINO[2,3-f]QUINOXALINE
11/07/2002WO2002088143A2 Dihydroimidazo[4,5-e]indole and 7h-pyrrolo[3,2-f]quinoxaline derivatives as nicotinic acetylcholine receptor ligands and/or serotonergic ligands
11/07/2002WO2002088140A1 Antidepressant azaheterocyclylmethyl derivatives of 7,8-dihydro-1,6,9-trioxa-3-aza-cyclopenta[a]naphthalene
11/07/2002WO2002088139A1 6h-oxazolo[4,5-e]indole derivatives as nicotinic acetylcholine receptor ligands and/or serotonergic ligands
11/07/2002WO2002088135A1 Antidepressant azaheterocyclylmethyl derivatives of oxaheterocycle-fused-[1,4]-benzodioxans
11/07/2002WO2002088132A1 Azaheterocyclylmethyl derivatives of 2,3-dihydro-1,4-dioxino[2,3-f]quinoline as 5-ht1aantagonists
11/07/2002WO2002088131A1 Antidepressant (sssri) azaheterocyclymethyl derivatives of 7,8-dihydro-3h-t,9-dioxa-1,3-diazacyclopenta[a]naphthalene
11/07/2002WO2002088130A1 Azabicyclylmethyl derivatives of 2,3-dihydro-1,4-dioxino-[2,3-f]quinoline as 5-ht1a antagonists
11/07/2002WO2002088129A1 Antidepressant azaheterocyclylmethyl derivatives of 2,3-dihydro-1,4-dioxino[2,3-f]quinazoline
11/07/2002WO2001042243A3 Protein kinase inhibitors
11/07/2002US20020165391 Novel spiro compounds
11/07/2002US20020165365 Synthetic catalyst for selective cleavage of protein and method for selective cleavage of protein using the same
11/07/2002US20020165245 Antidepressant azaheterocyclymethyl derivatives of 2,3-dihydro-1,4-dioxino[2,3-f]quinoline
11/07/2002US20020165241 Such as 4-((methyl-pyrimidin-2-ylamino)-methyl)-piperidine-1-carboxylic acid benzyl ester; useful for pain relief; treating migraine, depression, anxiety, schizophrenia, Parkinson's disease, and stroke; N-methyl-D-aspartate (NMDA)
11/07/2002CA2445859A1 Antidepressant azaheterocyclylmethyl derivatives of 7,8-dihydro-1,6,9-trioxa-3-aza-cyclopenta[a]naphthalene
11/07/2002CA2445583A1 Antidepressant indoletetrahydropyridine derivatives of 2,3-dihydro-7h-[1,4]dioxino[2,3-e]indole
11/07/2002CA2445581A1 Antidepressant azaheterocyclylmethyl derivatives of 2,3-dihydro-1,4-dioxino[2,3-f]quinoxaline
11/07/2002CA2445552A1 Antidepressant (sssri) azaheterocyclymethyl derivatives of 7,8-dihydro-3h-t,9-dioxa-1,3-diazacyclopenta[a]naphthalene
11/07/2002CA2445543A1 Antidepressant azaheterocyclylmethyl derivatives of oxaheterocycle-fused-¬1,4|-benzodioxans
11/07/2002CA2444897A1 Sulfate of cephem compound
11/06/2002EP1254908A1 Preparation of a camptothecin derivative by intramolecular cyclisation
11/06/2002EP0758335B1 Preparation of a camptothecin derivative by intramolecular cyclisation
11/05/2002US6476066 Anti-first-pass effect compounds
11/05/2002US6476029 7-alkyl- and cycloalkyl-substituted imidazotriazinones
10/2002
10/31/2002WO2002085912A1 ANTIPSYCHOTIC AMINOMETHYL DERIVATIVES OF 7,8-DIHYDRO-3H-6,9-DIOXA-1,3-DIAZA-CYCLOPENTA[a]NAPHTHALENE
10/31/2002WO2002085886A2 Chiral, broad-spectrum antibacterial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation and compositions
10/31/2002WO2002085413A1 Synthetic catalyst for selective cleavage of protein and method for selective cleavage of protein using the same
10/31/2002US20020161001 Heterocyclic compounds, which are inhibitors of the enzyme DPP-IV
10/31/2002DE10121217A1 6H-Oxazolo[4,5-e]indol-Derivate als nikotinische Acetylcholinrezeptor Liganden und/oder serotonerge Liganden 6H-oxazolo [4,5-e] indole derivatives as nicotinic acetylcholine receptor ligands and / or serotonergic ligands
10/31/2002DE10121215A1 Dihydro-imidazo[4,5-e]indol- und 7H-Pyrrolo[3,2-f]chinoxalin Derivate als nikotinische Acetylcholinrezeptor Liganden und/oder serotonerge Liganden Dihydro-imidazo [4,5-e] indole and 7H-pyrrolo [3,2-f] quinoxaline derivatives as nicotinic acetylcholine receptor ligands and / or serotonergic ligands
10/31/2002CA2445888A1 Chiral, broad-spectrum antibacterial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation and compositions
10/29/2002US6472527 New heterocyclic compounds are disclosed which are used as intermediates for the preparation of trans-thiazine-indigo pigments which are in part new compounds and can be used for the mass pigmentation of organic substrates.
10/24/2002WO2002083678A1 Tricyclic diazepines as tocolytic oxytocin receptor antagonists
10/24/2002WO2002030931A3 Aza- and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors
10/24/2002US20020156081 Pyrazolopyrimidines as therapeutic agents
10/24/2002US20020155484 Oligonucleotide for use as tool in the detection of preferential compounds in solution
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