Patents
Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041)
02/2005
02/02/2005EP1501838A1 A process for the preparation of clopidogrel
02/02/2005EP1501832A1 Triazolopyrimidines
02/02/2005EP1501507A2 Tetrahydropyranyl cyclopentyl tetrahydropyridopyridine modulators of chemokine receptor activity
02/02/2005EP1235574B1 Methods for making sustained-release pharmaceutical compositions of ergot alkaloids having improved bioavailability and compositions thereof
02/02/2005CN1187354C Adenosine receptor antagonists and methods of making and using the same
01/2005
01/27/2005WO2004092181A9 Heterocyclic mchr1 antagonists
01/27/2005WO2004064972A3 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions
01/27/2005US20050020598 Antiserotonine agents; central nervous system disorders; anxiolytic agents; cognition activators; schizophrenia ; antidepressants; Alzheimer's disease; Parkinson's disease
01/27/2005US20050020574 dipeptidylpeptidase-IV inhibitors; treatment of diabetes and obesity
01/26/2005EP1499622A1 Heterotricyclyl 6-alkylidene-penems as beta-lactamase inhibitors
01/26/2005EP1499621A1 Bicyclic 6-alkylidene-penems as beta-lactamases inhibitors
01/26/2005EP1499620A1 Process for preparing 6-alkylidene penem derivatives
01/26/2005EP1499308A2 Tri-substituted heteroaryls and methods of making and using the same
01/26/2005CN1571788A Photoactivable nitrogen bases
01/20/2005WO2005005432A1 Novel 2,7-dioxo-bicyclo[4.3.0]non-5-yl-urea derivatives
01/20/2005WO2003076443A9 Spiro compounds with npy antagonistic activity
01/20/2005US20050014761 Antitumor agents; antiancer agents; antiinflammatory agents; autoimmune disease
01/20/2005US20050014760 Methods of treating diseases or conditions using dihydropteridinone compounds
01/20/2005US20050014700 Cbi analogues of cc-1065 and the duocarmycins
01/19/2005EP1497287A1 Quinolinone derivatives
01/19/2005EP1496903A1 Anhydrovinblastine for the treatment of cancer
01/19/2005EP1496896A1 Inhibitors of akt activity
01/13/2005US20050009849 Pyridopyrimidine kinase inhibitors
01/12/2005EP1495022A1 Diazabicyclo alkane derivatives with nk1 antagonistic activity
01/12/2005EP1494676A1 Fused quinoxaline derivatives as inhibitors of akt activity
01/11/2005US6841677 For use as semiconductors or charge transport materials in optical, electrooptical or electronic devices including field effect transistors, electroluminescent, photovoltaics, sensors and electrophotographic recording devices
01/11/2005US6841567 Cyclic substituted fused pyrrolocarbazoles and isoindolones
01/06/2005WO2005000852A2 Product containing at least one phosphatase cdc25 inhibitor combined with at least one other anticancer agent
01/06/2005WO2005000814A1 Polymethine ethers
01/06/2005WO2004096800A3 Quinuclidine derivatives binding to mucarinic m3 receptors
01/06/2005US20050004153 inhibitors of Lymphocyte Function-associated Antigen 1 (LFA-1)/intercellular adhesion molecule (ICAM); use treating transplant rejection, rheumatoid arthritis, diabetes, inflammatory bowel disease, and chronic obstructive pulmonary disease; 2,4-dioxo-1,3,7-triazaspiro[4.4]nonanes
01/06/2005US20050004142 furo(2,3-d)pyrimidine and thieno(2,3-d)pyrimidine compounds for treating cancer and hyperproliferative diseases; receptor tyrosine kinase inhibitors
01/06/2005US20050004128 4-(6-chloro-, methyl- or thien-3-yl-oxazolo[4,5-b]pyrid-2-yl)-1,4-diazabicyclo[3.2.2]nonane or salts; nicotinic receptor associated disorders; cholinergic agents
01/06/2005US20050004026 Induction of capacse cascade ; administering apoptosis inducing protein; drug screening; anticancer agents
01/06/2005CA2530668A1 Product containing at least one phosphatase cdc25 inhibitor combined with at least one other anticancer agent
01/05/2005EP1493057A1 Colour photographic recording material
01/05/2005EP1492803A1 New analogs of nitrobenzylthioinosine
01/05/2005EP1492789A1 Tropane derivatives as ccr5 modulators
01/05/2005EP1492571A2 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
01/05/2005DE10327439A1 Neue Imidazopyridazinon- und Imidazopyridonderivate, deren Herstellung und deren Verwendung als Arzneimittel New Imidazopyridazinon- and Imidazopyridonderivate, their preparation and their use as medicaments
01/05/2005CN1560060A Synthesis for compound of diamine bridge linking ortho phenanthroline hydrous lanthanum (III) and anti-cancer activity thereof
01/05/2005CN1183129C Condensed azepines as vasporession agonists
01/04/2005US6838459 7-alkyl-and cycloalkyl-substituted imidazotriazinones
12/2004
12/30/2004US20040266860 Dihydroartemisinin and dihydroartemisitene dimers as anti-cancer and anti-infective agents
12/30/2004US20040266666 Cross-linked glycopeptide-cephalosporin antibiotics
12/29/2004WO2004113350A1 Cross-linked glycopeptide - cephalosporin antibiotics
12/29/2004EP1490374A2 Dithiolopyrrolone derivatives useful in the treatment of proliferative diseases
12/29/2004EP1490344A2 Anxiolytic agents with reduced sedative and ataxic effects
12/28/2004CA2105923C 7-isoindolinyl-quinolone derivatives and 7-isoindolinyl-naphthyridone derivatives
12/23/2004WO2004111054A1 Pyridinylpyrazolopyrimidinone derivatives as pde 7 inhibitors
12/23/2004WO2004111051A1 Imidazo-pyridazinone derivatives and imidazo-pyridone derivatives, production thereof, and use thereof as medicaments
12/23/2004WO2004110990A2 Imidazothiazoles and imidazoxazole derivatives as inhibitors of p38
12/23/2004WO2004091482A3 M3 muscarinic acetylcholine receptor antagonists
12/23/2004US20040259907 4-oxo-4,7-dihydrofuro[2,3-b]pyridine-5-carboxamide antiviral agents
12/23/2004US20040259897 transplant rejection, rheumatoid arthritis, osteoarthritis, diabetes, asthma, inflammatory bowel disease, and chronic obstructive pulmonary disease; inhibitors of Lymphocyte Function-associated Antigen 1 (LFA-1)/intercellular adhesion molecule (ICAM); 2,4-dioxo-1,3,7-triazaspiro[4.4]nonanes
12/23/2004US20040259888 Antiischemic agents; cardiovascular disorders; analgesics; neurodegenerative disease
12/23/2004CA2529729A1 New imidazopyridazinone and imidazopyridone derivatives, the preparation thereof and their use as pharmaceutical compositions
12/23/2004CA2526285A1 Inhibitors of p38 and methods of using the same
12/22/2004EP1489084A1 Broad-spectrum cephem compounds
12/22/2004CN1181075C Pyrimidine-4-keto compound, its preparation method and medicine composition containing them
12/22/2004CN1181050C Noval substituted dimeric compounds, its preparing process and medicinal composition containing same
12/21/2004US6833455 Coloring plastics
12/16/2004WO2004108728A1 Cannabinoid receptor ligands and uses thereof
12/16/2004WO2004107863A1 Sustituted imidazolopyrazine and triazolopyrazine derivatives: gabaa receptor ligands
12/16/2004US20040254198 Respiratory system disorders; asthma; chronic obstructive pulmonary disease
12/16/2004CA2525752A1 Cannabinoid receptor ligands and uses thereof
12/16/2004CA2524376A1 Substituted imidazolopyrazine and triazolopyrazyne derivatives: gabaa receptor ligands
12/15/2004EP1485389A1 Antiparasitic artemisinin derivatives (endoperoxides)
12/15/2004EP1485387A1 Carbamates as hiv protease inhibitors
12/15/2004CN1554656A Yunnan tolal biological coronaridine and its salts and preparing method and use
12/14/2004US6831075 Heterocyclic substituted pyrazolones
12/14/2004US6830836 Heterocyclic compounds, materials for light emitting devices and light emitting devices using the same
12/09/2004WO2004092173A3 A2a adenosine receptor antagonists
12/09/2004US20040249152 Activation of the carboxyl function of a CNA monomer building block, subsequent esterification of this monomer building block with a free hydroxyl function,thereafter assembly of the oligomer by repetitive cycles starting from elimination of the protective group
12/09/2004US20040248920 Spiro-hydantoin compounds useful as anti-inflammatory agents
12/09/2004US20040248907 reacting 4,6-dichloro-5-nitropyrimidine with acyclic carboxy amines, then cyclization of the intermediates to form cellular adhesion inhibitors
12/09/2004US20040248881 such as 1-[2-(2-chloro-phenyl)-3-(4-fluoro-phenyl)-2H-pyrazolo[3,4-d]pyridazin-7-yl]-4-isopropylamino-piperidine-4-carboxylic acid amide; for treatment of eating disorders and psychological disorders
12/08/2004EP1483270A1 Heterocyclic amide derivatives as inhibitors of glycogen phosphorylase
12/08/2004EP1483266A1 Spiro compounds with npy antagonistic activity
12/08/2004EP1483265A1 Purine derivatives as kinase inhibitors
12/08/2004EP1483264A2 1-allyl ergot alkaloid derivatives, method for producing the same and the use thereof for preventing and treating migraine
12/08/2004EP1483257A1 Quinazoline compounds useful in therapy
12/08/2004EP1482971A1 Strategy for retroviral immunotherapy
12/08/2004EP1482933A2 Potent, simplified derivatives of immunosuppressive agents
12/08/2004CN1552716A Synthesis of vinorelbine
12/08/2004CN1552715A Preparation of dehydrate catharahhine from intermediate of vinorelbine synthesis
12/07/2004US6828330 Quinuclidine-substituted hetero-bicyclic aromatic compounds for the treatment of disease
12/07/2004CA2272136C Pyrazole derivatives having crf antagonist activity
12/07/2004CA2147755C 6-(substituted methylene) penems and intermediates
12/02/2004WO2004104008A1 PROCESS FOR SYNTHESIZING β-LACTAMASE INHIBITOR INTERMEDIATES
12/02/2004WO2004104004A2 Triaza-spiro compounds as nociceptin analogues and uses thereof
12/02/2004WO2004104001A2 Pyrrolopyridine-2-carboxylic acid amide inhibitors of glycogen phoshorylase
12/02/2004US20040242884 3-Substituted-7-oxo-4,7-dihydro-thieno(3,2-b)pyridine-6-carboxylic acid benzylamide derivatives; for herpes viruses
12/02/2004US20040242867 Photoinitiators; basic catalyst; absorption of light
12/02/2004CA2532059A1 Triaza-spiro compounds as nociceptin analogues and uses thereof
12/02/2004CA2525507A1 Process for synthesizing .beta.-lactamase inhibitor intermediates
12/02/2004CA2525504A1 Process for synthesizing .beta.-lactamase inhibitor in intermediates
12/01/2004EP1481077A2 Mitotic kinesin inhibitors
12/01/2004EP1480983A1 Heteroaryl substituted 2-pyridinyl and 2-pyrimidinyl-6,7,8,9-tetrahydropydimido[1,2-a]pyrimidin-4-one derivatives
12/01/2004EP1480979A2 Gadolinium chelate oligomers, their use as contrast products in magnetic resonance imaging and their synthesis intermediates
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