Patents
Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041)
03/2005
03/24/2005WO2005026168A1 Method for preparing cucurbiturils
03/24/2005WO2004110990A3 Imidazothiazoles and imidazoxazole derivatives as inhibitors of p38
03/24/2005WO2004085421A3 Bioreductively-activated prodrugs
03/24/2005US20050065341 Substituted 8-heteroaryl xanthines
03/24/2005US20050065164 Generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments
03/24/2005CA2537843A1 Method for preparing cucurbiturils
03/23/2005EP1515727A2 (halo-benzo carbonyl)heterobicyclic p38 kinase inhibiting agents
03/23/2005EP1381392A4 Synthetic catalyst for selective cleavage of protein and method for selective cleavage of protein using the same
03/23/2005CN1193788C Beta 2-adrenergic receptor agonist
03/22/2005CA2125189C Pyropheophorbides and their use in photodynamic therapy
03/17/2005WO2005023819A1 Thienopyrroles as antiviral agents
03/17/2005WO2005023816A2 Synthetic binding pairs comprising cucurbituril derivatives and polyammonium compouds and uses thereof
03/17/2005WO2005023806A2 Heteroaryl fused pyridines, pyrazines and pyrimidines as crf1 receptor ligands
03/17/2005WO2005023255A2 Use of indole-derived compounds for the preparation of a medicament that can be used to treat diseases related to the splicing process
03/17/2005US20050059628 Modulation of beta-catenin/TCF-activated transcription
03/17/2005CA2537829A1 Heteroaryl fused pyridines, pyrazines and pyrimidines as crf1 receptor ligands
03/17/2005CA2537752A1 Use of indole-derived compounds for the preparation of a medicament that can be used to treat diseases related to the splicing process
03/17/2005CA2537736A1 Synthetic binding pairs comprising cucurbituril derivatives and polyammonium compounds and uses thereof
03/17/2005CA2537545A1 Thienopyrroles as antiviral agents
03/16/2005EP1513848A2 Method of treating ischemia reperfusion injury using adenosine receptor antagonists
03/16/2005EP1513516A1 SUBSTITUTED 3-AMINO-THIENO(2,3-b) PYRIDINE-2-CARBOXYLIC ACID AMIDE COMPOUNDS ANDPROCESSES FOR PREPARING AND THEIR USES
03/16/2005EP1425283B1 Novel 4-aminofuropyrimidines and the use thereof
03/16/2005EP1392699B1 6h-oxazolo 4,5-e]indole derivatives as nicotinic acetylcholine receptor ligands and/or serotonergic ligands
03/16/2005EP0808164B1 Use of prolactin modulators and diet for the manufacture of a medicament for the treatment of obesity
03/16/2005CN1596253A Spiro-hydantoin compounds useful as anti-inflammatory agents
03/15/2005US6867300 Methods for the preparation of pyrrolotriazine compounds useful as kinase inhibitors
03/15/2005US6867200 Anticancer agents; anticoagulants
03/15/2005CA2146852C New substituted pyrazole derivatives, processes for their preparation and their use as herbicides
03/15/2005CA2086914C Quinolone-and naphthyridone-carboxylic acid derivatives
03/10/2005WO2005021548A2 Substituted 8-heteroaryl xanthines
03/10/2005WO2005021025A2 MODULATION OF β-CATENIN/TCF ACTIVATED TRANSCRIPTION
03/10/2005WO2005020987A1 Heterocyclic amide derivatives which posses glycogen phosphorylase inhibitory activity
03/10/2005WO2005020894A2 Rifamycin analogs and uses thereof
03/10/2005US20050054851 Pyrrolo pyrimidines as agents for the inhibition of cystein proteases
03/10/2005US20050054672 Quinolinone derivatives
03/10/2005CA2537099A1 Modulation of .beta.-catenin/tcf activated transcription
03/10/2005CA2536553A1 Substituted 8-heteroaryl xanthines
03/10/2005CA2536378A1 Rifamycin analogs and uses thereof
03/09/2005EP1512688A1 Use of K-252a derivatives for the treatment of Parkinson's disease
03/09/2005EP1512403A1 Methods for making sustained-release pharmaceutical compositions of ergot alkaloids having improved bioavailability and compositions thereof
03/09/2005EP1511744A2 Bis-benzimidazoles and related compounds as potassium channel modulators
03/09/2005EP1511492A2 Protease inhibitors
03/09/2005CN1592747A Diazabicyclo alkane derivatives with NK1 antagonistic activity
03/09/2005CN1592624A Substituted-triazolopyrimidines as anticancer agents
03/08/2005CA2153239C 5-alkoxy[1,2,4]triazolo[1,5-c]pyrimidine-2(3h)-thione compounds and their use in the preparation of 2,2'-dithiobis(5-alkoxy[1,2,4]triazolo[1,5-c]-pyrimidine) and 2-chlorosulfonyl-5-alkoxy[1,2,4]triazolo[1,5-c]pyrimidine compounds
03/03/2005WO2004104004A3 Triaza-spiro compounds as nociceptin analogues and uses thereof
03/03/2005WO2004104001A3 Pyrrolopyridine-2-carboxylic acid amide inhibitors of glycogen phoshorylase
03/03/2005WO2003031405A3 Methods for the synthesis of substituted purines
03/03/2005US20050049260 2-phenyl-4-pyridinyl- or -pyrimidinyl derivatives, e.g., N-Cyclopentyl-3-[2-(cyclopentylamino)-4-pyrimidinyl]-2-(4-methoxyphenyl)-pyrazolo[1,5-a]pyridin-7-amine and; especially for treatment of herpes simplex virus 1 and 2
03/03/2005US20050049250 7-Aikyl and cycloalkyl-substituted imidazotriazinones
03/02/2005EP1509522A1 1-(aminoalkyl)-3-sulfonylazaindoles as 5-hydroxytryptamine-6 ligands
03/02/2005EP1165563B1 Bicyclic heterocycles, method for producing them and their use as herbicides and pharmaceutical agents
03/02/2005EP1073661B1 Dioxazine derivatives and their use as dyestuffs
03/02/2005CN1589273A The use of anti-histaminics for acute reduction of elevated intracranial pressure
03/02/2005CN1589271A Fused heterocyclic succinimide compounds and analogs thereof as modulators of nuclear hormone receptor function
03/02/2005CN1589145A αv整联蛋白受体拮抗剂 αv integrin receptor antagonists
03/01/2005US6861430 β-carboline derivatives and its pharmaceutical use against depression and anxiety
03/01/2005US6861427 For therapy of cognitive deficits due to aging, stroke, head trauma, Alzheimer's disease or other neurodegenerative diseases, or schizophrenia, anxiety, aggression and stress, eating disorder, sleep disorder, sexual dysfunction
03/01/2005US6861422 Dihydropteridinones, processes for preparing them and their use as pharmaceutical compositions
02/2005
02/24/2005US20050043323 Pyrimidylpyrrole derivatives active as kinase inhibitors
02/24/2005US20050043298 Useful for treating or preventing a variety of antibiotic resistant microbial infections; for example, 3'-hydroxy-5'-(4-ethylcarbamyl-1-piperidinyl)benzoxazinorifamycin
02/24/2005US20050043242 Using dietary restriction to lower serum insulin levels and function along with troglitazone in treatment and prevention of alzheimer's diseases
02/24/2005US20050042771 Identifying non-drug targets; use in drug design for improving knowledge of drug-target and drug-non-target interactions, so that drug adverse reactions can be reduced or eliminated in drugs such as troglitazone, rosiglitazone, pioglitazone, methotrexate, atorvastatin, celecoxib, rofecoxib, cerivastatin
02/24/2005US20050041494 High density non-volatile memory device
02/23/2005EP1507778A1 Anti-tumour polycyclic carboxamides
02/23/2005CN1585772A Chemokine receptor antagonists and methods of use thereof
02/23/2005CN1583759A Preparing method for nanometer powder of synthetic metal ET salt
02/23/2005CN1583758A Use of Maituolaicin
02/23/2005CN1190440C Triazolo-epothilones
02/22/2005US6858613 Central nervous system disorders
02/17/2005WO2005014600A1 Antagonists of mcp-1 function and methods of use thereof
02/17/2005WO2005014599A1 Imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of bruton’s tyrosine kinase by such compounds
02/17/2005WO2005014581A2 Lanthanide complexes preparation and uses thereof
02/17/2005WO2005014572A1 Pyrimidylpyrrole derivatives active as kinase inhibitors
02/17/2005WO2004096982A3 Antibacterial agents
02/17/2005US20050038088 N-sulfonylheterocyclopyrrolyl-alkylamine compounds as 5-hydroxytryptamine-6 ligands
02/17/2005CA2535125A1 Pyridylpyrrole derivatives active as kinase inhibitors
02/17/2005CA2534496A1 Pyrimidylpyrrole derivatives active as kinase inhibitors
02/17/2005CA2533698A1 Lanthanide complexes preparation and uses thereof
02/16/2005EP1506192A1 Substituted pyrroline kinase inhibitors
02/16/2005EP1506174A2 Opioid and opioid-like compounds and uses thereof
02/16/2005CN1580055A Quinolone carboxylic acid derivatives and their salts
02/15/2005US6855724 Tropane derivatives useful in therapy
02/10/2005WO2005012311A1 N-sulfonylheterocyclopyrrolylalkylamine compounds as 5-hydroxytryptamine-6 ligands
02/10/2005US20050033048 Spiro[isobenzofuran-1,4'-piperidin]-3-ones and 3h-spiroisobenzofuran-1,4'-piperidines
02/10/2005US20050032860 CBI analogs of CC-1065 and the duocarmycins
02/10/2005US20050032820 Novel spiro compounds
02/10/2005US20050032817 Kinesin spindle protein (KSP) inhibitors, e.g., 3-benzyl-2-(1-{(4-bromobenzyl)[2-(dimethylamino)ethyl]amino}propyl)furo[2,3-d]pyrimidin-4(3H)-one; antiproliferative and -carcinogenic agents; side effects reduction; cancers of the brain, genitourinary tract, lymphatic system, stomach, larynx and lung
02/10/2005CA2532382A1 N-sulfonylheterocyclopyrrolylalkylamine compounds as 5-hydroxytryptamine-6 ligands
02/09/2005EP1505068A1 PYRAZOLO (1,5-a) PYRIMIDINE DERIVATIVE AND NAD(P)H OXIDASE INHIBITOR CONTAINING THE SAME
02/09/2005EP1504010A1 Vitamin-mitomycin conjugates
02/09/2005EP1503760A1 Camptothecin derivatives and polymeric conjugates thereof
02/09/2005EP1280805B1 Novel imidazotriazinones and the use thereof
02/08/2005US6852731 3-Substituted-7-oxo-4,7-dihydro-thieno(3,2-b)pyridine-6-carboxylic acid benzylamide derivatives; for herpes viruses
02/03/2005WO2005010006A1 Substituted furochromene compounds of antiinflammatory action
02/03/2005WO2004083175A3 Methods for identifying enzyme inhibitors and protein kinases
02/03/2005US20050026941 preferential inhibitors of cyclic guanosine 3',5'-monophosphate specific phosphodiesterase used for prophylaxis of erectile dysfunction and cardiovascular disorders
02/03/2005US20050026921 New imidazopyridazinone and imidazopyridone derivatives, the preparation thereof and their use as pharmaceutical compositions
02/03/2005US20050026901 Antihistaminic spiro compounds
02/03/2005CA2533584A1 Substituted furochromene compounds of antiinflammatory action
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