Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
10/1998
10/14/1998EP0869967A2 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME
10/14/1998EP0869966A1 Prodrugs of thrombin inhibitors
10/14/1998EP0869942A1 4-((heterocycloalkyl or heteroaromatic)-substituted phenyl]-2-azetidinones useful as hypolipidemic agents
10/14/1998CN1196052A Benzoxazepine compounds, their production method and use
10/14/1998CN1196050A Cyclic nitrones and pharmaceutical compositions containing them
10/14/1998CN1040213C Diaryl 5,6-fusedheterocylic acids as leukotriene antagonists
10/13/1998US5821365 Compounds as enzyme inhibitors for kinases formed by reaction of amine with anhydride group to form indolmaleimide macrocycles
10/13/1998US5821248 Substance p antagonists
10/13/1998US5821130 Chemical intermediates
10/08/1998WO1998043977A1 Quinolinomorphinane derivatives and medicinal use thereof
10/08/1998WO1998043969A1 Indazoles of cyclic ureas useful as hiv protease inhibitors
10/08/1998WO1998043960A1 Substituted 3-cyano quinolines
10/08/1998WO1998043956A1 1,4-substituted cyclic amine derivatives
10/08/1998CA2285241A1 Substituted 3-cyano quinolines
10/08/1998CA2282593A1 Indazoles of cyclic ureas useful as hiv protease inhibitors
10/07/1998EP0807115A4 High molecular weight polymer-based prodrugs
10/07/1998CN1194983A New 2-amino-1,2-indene compounds, process for their preparation and pharmaceutical compositions containing them
10/06/1998US5817679 Analgesics, antiinflammatory agents
10/06/1998US5817653 Endothelin receptor antagonists
10/01/1998WO1998042715A1 Spiro compounds and the use thereof
10/01/1998WO1998042714A1 New sesquiterpene derivatives
10/01/1998WO1998042713A1 2,3-DIHYDROFURO[3,2-b]PYRIDIN, PREPARATION AND APPLICATION THEREOF IN THERAPY
10/01/1998WO1998042712A1 Quinoline-2(1h)-one and dihydroquinoline-2(1h)-one derivatives as ligands of 5-ht, 5-ht2 and 5-ht1-like receptors
10/01/1998WO1998042709A1 Endothelin-receptor antagonists
10/01/1998WO1998042695A1 INTENSE COLOURING PHOTOCHROMIC 2H-NAPHTHO[1,2-b]PYRANS AND HETEROCYCLIC PYRANS
10/01/1998WO1998042694A1 Benzoxanthene derivatives exhibiting antiviral activity
10/01/1998WO1998042693A2 NEUTRAL COLOURING PHOTOCHROMIC 2H-NAPHTHO[1,2-b]PYRANS AND HETEROCYCLIC PYRANS
10/01/1998WO1998042675A1 Substituted isoquinolines as ultra short acting neuromuscular blockers
10/01/1998WO1998042674A1 Substituted isoquinolines as ultra short acting neuromuscular blockers
10/01/1998DE19711568A1 Spiroverbindungen und deren Verwendung Spiro compounds and their use
10/01/1998CA2282320A1 2,3-dihydrofuro¬3,2-b|pyridin, preparation and application thereof in therapy
09/1998
09/30/1998EP0866708A1 Dihydropyrimidines and uses thereof
09/30/1998CN1194648A Spiro (2H-1-benzopyran-2,4'-piperidine)-4-(3H)-one derivatives, acid addition salts thereof and pharmaceutical compositions containing them
09/24/1998WO1998041205A1 Cytochalasin and isoindolinone derivatives as inhibitors of angiogenesis
09/24/1998DE19711785A1 Endothelin-Rezeptor-Antagonisten Endothelin receptor antagonists
09/23/1998CN1193979A Macrolides
09/23/1998CN1193968A 2,3-dioxo-1,2,3,4-tetrahydro-quinoyxalinyl derivatives
09/23/1998CN1193960A Dialkyl phenyl halide-substituted keto-enols for use as herbicides and pesticides
09/23/1998CN1039911C Galanthamine derivatives, a process for their preparation and use as medicaments
09/23/1998CN1039910C Galanthamine derivatives, a process for their preparation and use as medicaments
09/23/1998CN1039908C Tricyclic diazepine vasopressin antagonists
09/22/1998US5811576 1-carboxy-2-loweralkyl-3,4,6-tri(halo)benzenes; grampositive and-negative bacteria; infections; sterilization of medical equipment
09/22/1998US5811558 Process for the resolution of etodolac using glucamine derivatives
09/22/1998US5811551 Palladium catalyzed indolization
09/22/1998US5811427 Heterocyclic N-acetonylbenzamides
09/22/1998CA2086434C Quinuclidine derivatives
09/17/1998WO1998040386A1 Dioxino derivatives and their use as therapeutic agents
09/17/1998WO1998040383A1 Farnesyl transferase inhibiting 1,8-annelated quinolinone derivatives substituted with n- or c-linked imidazoles
09/17/1998WO1998040373A1 Ring opening metathesis of alkenes
09/17/1998WO1998040068A1 Heterocyclic agents
09/17/1998WO1998040066A1 Metabolically stabilized oxyalkylene esters and uses thereof
09/17/1998CA2283182A1 Ring opening metathesis of alkenes
09/17/1998CA2283127A1 Heterocyclic agents
09/16/1998EP0864572A1 Crystal of hydrate and process for preparation thereof
09/16/1998EP0864087A1 Combinatorial dihydrobenzopyran library
09/16/1998EP0863906A2 Heterocyclic dioxethane substrates, process for their preparation and their use
09/16/1998EP0863904A2 Novel spiro 2h-1-benzopyran-2,4'-piperidine]- 4(3h)-one derivatives, acid addition salts thereof and pharmaceutical compositions containing them
09/16/1998EP0863903A1 Synthetic metal-substituted bacteriochlorophyll derivatives and use thereof
09/16/1998EP0863891A1 (methylsulfonyl)phenyl-2-(5h)-furanones as cox-2 inhibitors
09/16/1998EP0863878A1 Cyclic nitrones and pharmaceutical compositions containing them
09/16/1998CN1193321A Microbiocidal benzotriazoles compounds
09/16/1998CN1193019A Effective components of wild opium poppy and extracting process and product thereof
09/15/1998US5808093 L-tartaric acid salt of a (1R) diastereomer of a 2-azadihydroxybicyclo 2.2.1!heptane compound and the preparation of 2-azabicyclo 2.2.1!heptane compounds
09/15/1998US5807882 Anthracene compounds useful in treating certain cancers
09/15/1998US5807871 Psychological disorders, alzheimer or parkinson disease
09/15/1998US5807841 HIV protease inhibitors useful for the treatment of AIDS
09/15/1998CA2006269C 1,4-dideoxy-1,4-imino-l-allitol and its n-substituted alkyl and benzyl derivatives
09/11/1998WO1998039333A1 Crown ether-derivatised perylenes
09/11/1998WO1998039300A1 CYCLOALKA[b]PYRIDINE-3-CARBONYLGUANIDINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND DRUGS CONTAINING THE SAME
09/11/1998WO1998039010A1 Tricyclic and tetracyclic pyrones
09/11/1998WO1998038859A1 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
09/11/1998CA2283404A1 Cycloalka¬b|pyridine-3-carbonylguanidine derivatives, process for producing the same, and drugs containing the same
09/11/1998CA2283275A1 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
09/11/1998CA2283272A1 Aromatic sulfonyl alpha-cycloamino hydroxamic acid compounds
09/11/1998CA2283145A1 Aromatic sulfonyl alpha-hydroxy hydroxamic acid compounds
09/11/1998CA2282318A1 N-hydroxy 4-sulfonyl butanamide compounds
09/09/1998EP0862565A1 Tricyclic spiro compounds as 5ht 1d? receptor antagonists
09/09/1998EP0862562A1 Benzoxazepine compounds, their production and use as lipid lowering agents
09/09/1998CN1192740A Novel camptothecin analogues, prepn. method therefor, use thereof, and pharmaceutical compositions contg. same
09/09/1998CN1192732A CB2 receptor agonist compounds
09/09/1998CN1192682A Compositions for use against parasitic protozoa
09/08/1998US5804585 Thieno-pyridine sulfonamides derivatives thereof and related compounds that modulate the activity of endothelin
09/03/1998WO1998038189A1 Oxazolidines as 5-ht2a-antagonists
09/03/1998WO1998038187A1 Atropisomers of 3-heteroaryl-4(3h)-quinazolinones for the treatment of neurodegenerative and cns-trauma related conditions
09/03/1998WO1998038168A1 Isoquinolinone derivatives, process for preparing the same, and their use as phosphodiesterase inhibitors
09/02/1998EP0861842A1 Novel water-soluble fluoroethylcamptothecin derivative and process for production thereof
09/02/1998EP0861837A1 2-Aminoindane derivatives, process for their preparation and pharmaceutical compositions containing them
09/02/1998EP0861257A1 Spiro piperidine derivatives as 5mt receptor antagonists
09/02/1998EP0861253A1 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
09/02/1998EP0861249A1 Substituted sulfonylalkanoylamino hydroxyethylamino sulfonamide retroviral protease inhibitors
09/02/1998EP0861236A1 Cyclic and heterocyclic n-substituted alpha-iminohydroxamic and carboxylic acids
09/02/1998EP0593511B1 Piperidine derivates having anxiolytic effect
09/02/1998CN1192209A Method for preparing N-monosubstituted and N,N'-disubstituted unsymmetrical cyclic ureas
09/02/1998CN1192154A Combinatorial libraries of substrate-bound cyclic organic compounds
09/01/1998US5801242 Process for making quinolonyl lactam antimicrobials and novel intermediate compounds
09/01/1998US5801190 Fused pyrrolo 2,3-C! carbazole-6-ones
09/01/1998US5801180 Antiischemic agents and cardiovascular disorders
09/01/1998US5801175 Antitumor/anticarcinogenic agents
09/01/1998US5801167 Camptothecin derivatives and process for their preparation
09/01/1998US5800996 Energy transfer dyes with enchanced fluorescence