Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
03/1999
03/03/1999EP0745080B1 Novel mercaptoacetylamide disulfide derivatives useful as inhibitors of enkephalinase and ace
03/02/1999US5877178 Aids therapy
03/02/1999US5877172 Process for isolating galanthamine
03/02/1999US5877120 Nicotinic acid derivatives and herbicides
03/02/1999US5876984 Sequiterpene derivatives having antiviral activity
02/1999
02/25/1999WO1999009006A1 SYNTHESIS OF CLASTO-LACTACYSTIN β-LACTONE AND ANALOGS THEREOF
02/25/1999WO1999008528A1 Noscapine derivatives, useful as anticancer agents
02/25/1999CA2301054A1 Synthesis of clasto-lactacystin .beta.-lactone and analogs thereof
02/24/1999EP0897924A1 Process for the preparation of tetrahydro-indolizines
02/24/1999EP0897387A1 New benzazepine derivatives, medicaments containing the same and their use to prepare medicaments
02/24/1999CN1042228C Antiallergic imidazoazepines
02/23/1999US5874587 Imidazolium cations, processes for their preparation, and uses therefor
02/23/1999US5874473 Substituted cycloalkanecarboxylic acid derivatives as matrix metalloprotease inhibitors
02/23/1999US5874441 Carbocyclic and hetertocyclic fused-ring quinolinecarboxylic acids useful as immunosuppressive agents
02/23/1999US5874426 Cyclic amine derivatives of substituted quinoxaline 2,3-diones as glutamate receptor antagonists
02/18/1999WO1999007709A1 Methods of preparing and purifying 9-nitro-20-camptothecin
02/18/1999WO1999007708A1 1,3-dioxolo/4,5-h//2,3/benzodiazepine derivatives as ampa/kainate receptor inhibitors
02/18/1999WO1999007707A1 8-SUBSTITUTED-9H-1,3-DIOXOLO/4,5-h//2,3/BENZODIAZEPINE DERIVATIVES, AS AMPA/KAINATE RECEPTOR INHIBITORS
02/18/1999WO1999007378A1 Nicotine antagonists for nicotine-responsive neuropsychiatric disorders
02/18/1999WO1999007359A1 Use of cholinesterase inhibitors for treating attention deficit disorders
02/18/1999CA2300302A1 8-substituted-9h-1,3-dioxolo/4,5-h//2,3/benzodiazepine derivatives, as ampa/kainate receptor inhibitors
02/18/1999CA2300142A1 1,3-dioxolo/4,5-h//2,3/benzodiazepine derivatives as ampa/kainate receptor inhibitors
02/16/1999US5872251 Process for preparing intermediates of inhibitors of enkephalinase and angiotensin converting enzyme and intermediates thereof
02/16/1999US5872130 Quinoline type mevalonoactones
02/11/1999WO1999006410A1 Hydroxamic acid substituted fused heterocyclic metalloproteinase inhibitors
02/11/1999WO1999006402A1 N-acylamino acid amide compounds and intermediates for preparation thereof
02/11/1999WO1999006397A2 Pyrrolidine-3-carboxylic acid derivatives and their use as endothelin antagonists
02/11/1999WO1999006374A1 Condensed pyrazole compounds
02/11/1999WO1999006041A1 SUBSTITUTED ALKANOHYDROXAMIC ACIDS AND METHOD OF REDUCING TNFα LEVELS
02/11/1999WO1998042693A3 NEUTRAL COLOURING PHOTOCHROMIC 2H-NAPHTHO[1,2-b]PYRANS AND HETEROCYCLIC PYRANS
02/11/1999DE19733779A1 New pyrano-pyridine compounds are potassium channel blockers
02/11/1999CA2297988A1 Hydroxamic acid substituted fused heterocyclic metalloproteinase inhibitors
02/11/1999CA2297894A1 Pyrrolidine-3-carboxylic acid derivatives and their use as endothelin antagonists
02/11/1999CA2297815A1 N-acylamino acid amide compounds and intermediates for preparation thereof
02/11/1999CA2297096A1 Condensed heterocyclic compounds
02/11/1999CA2295295A1 Substituted alkanohydroxamic acids and method of reducing tnf.alpha. levels
02/10/1999EP0895999A1 C-4" substituted macrolide antibiotics
02/10/1999EP0895994A2 Sulphonamide-substituted Pyranopyridines, process for their production and their use as a drug or diagnostics as well as medicaments containing them
02/10/1999CN1207741A Synthetic metal-substituted bacteriochlorophyll derivs. and use thereof
02/10/1999CN1207732A Process for preparation of phenylimidazolidine derivs.
02/10/1999CN1207391A Sulfonamide-substituted compounds, processes for their preparation, their use and medicament comprising them
02/09/1999US5869686 Substituted pyrazole derivatives, processes for their preparation and their use as herbicides
02/09/1999US5869518 Azacycloalkane derivatives, their preparation and their application in therapy
02/09/1999US5869496 Treating asthma, emesis
02/09/1999US5869490 Adminstering to treat brain dopamine dysregulation; schizophrenia
02/09/1999US5869484 Treating diseases derived by acetylcholine deficiency; alzheimer*s disease
02/05/1999CA2244577A1 Sulfonamide-substituted compounds, processes for their preparation, their use as a medicament or diagnostic, and medicament comprising them
02/04/1999WO1999005521A2 Conjugate for differentiating between healthy and unhealthy tissue
02/04/1999WO1999005138A1 Heterocyclic compounds and antitumor agent containing the same as active ingredient
02/04/1999WO1999005116A1 Nitrophenyl-sulfonyl-imidazoles and use thereof for controlling vegetable and animal pests
02/04/1999WO1999005113A1 Substituted 6-phenylphenanthridines
02/04/1999WO1999005112A1 Substituted 6-alkylphenanthridines
02/04/1999WO1999005111A1 Novel tetrazole derivatives
02/04/1999WO1999005103A2 2o(s)-7-ethyl-9-(n-methyl-n-phenyl)amidino-camptothecin, its preparation and its use as antitumor agent
02/04/1999CA2297923A1 Novel tetrazole-substituted 6-phenyl-pheanathridines as pde inhibitors
02/04/1999CA2266891A1 Amidino-camptothecin derivatives
02/03/1999EP0894799A1 Indolomorphinane derivatives and remedies/preventives for cerebral disorders
02/03/1999EP0623619B1 PREPARATION METHOD OF ARENO[e]INDOLS
02/03/1999CN1207091A 1-arylsulphonyl, aryl(thio) carbonyl pyridazino derivatives and methods of preparation
02/03/1999CN1206713A Process for preparing 2-chloro-benzimidazole derivatives
02/02/1999US5866589 Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds
02/02/1999US5866587 Hydroxamide derivatives of fused piperidine derivatives
02/02/1999US5866579 Imidazole and imidazoline derivatives and uses thereof
01/1999
01/28/1999WO1999003859A1 Novel spiroazabicyclic heterocyclic compounds
01/28/1999WO1999003846A1 Tricyclically substituted oxazolidinones
01/28/1999DE19829740A1 Nitrophenyl-sulfonyl-imidazole Nitrophenyl-sulfonyl-imidazole
01/28/1999DE19731741A1 Konjugat zur Unterscheidung von krankhaftem und gesundem Gewebe Conjugate to distinguish between diseased and healthy tissue
01/28/1999DE19730847A1 Tricyclisch substituierte Oxazolidinone Tricyclic substituted oxazolidinones
01/27/1999EP0893445A1 Process for the preparation of 2-chlorobenzimidazole derivatives
01/27/1999EP0892800A1 3- (1,2,3,4-tetrahydroisoquinoline-2-yl)methyl]-8-azabicyclo 3.2.1]octane derivatives, their preparation and their application in therapeutics
01/27/1999EP0892797A1 Inhibitors of farnesyl protein transferase
01/27/1999EP0892793A1 Substituted tetracyclic tetrahydrofuran derivatives
01/27/1999EP0892787A1 NOVEL $g(a)-HYDROXYLIC ACID DERIVATIVES, THEIR PRODUCTION AND USE
01/27/1999EP0892786A1 New carboxylic acid derivatives, their production and use
01/27/1999EP0892780A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS
01/27/1999CN1206406A 1-(1,2-disubstituted piperidinyl)-4-substituted piperidine derivatives as tachykinin receptor antagonists
01/27/1999CN1206009A Extraction of anhydro tetraodotoxin
01/26/1999US5864035 Used for photodynamic thearpy
01/26/1999US5863933 Substituted benzimidazoles
01/26/1999US5863920 Anticarcinogenic agents and bactericides
01/21/1999WO1999002530A1 A process of manufacturing camptothecin derivatives
01/21/1999WO1999002514A2 Epothilone derivatives
01/21/1999WO1999002154A1 Highly selective butyrylcholinesterase inhibitors for the treatment and diagnosis of alzheimer's disease and dementias
01/20/1999EP0891330A1 Substituted phenyl keto enols as pesticides and herbicides
01/20/1999EP0719259B1 Substituted pyridines and pyrimidines, process for producing them and their use as pesticides and fungicides
01/20/1999EP0630242B1 Further indole derivatives with antiviral activity
01/20/1999CN1205335A Tricyclic diazepine vasopression antagonists
01/20/1999CN1041730C Method for preparing tetrahydrothienopyridine derivatives
01/19/1999US5861510 Antiarthritic agents, antiulcer agents, restenosis, oral diseases
01/19/1999US5861428 Alleviation of osteoarthritis, rheumatoid arthritis, septic arthritis, periodontal disease, corneal ulceration, proteinuria, aneurysmal aortic disease, dystrophobic epidermolysis bullosa, inflammation, osteopenias, tempero
01/19/1999US5861427 Substituted 4-biarylbutyric acid derivatives as matrix metalloprotease inhibitors
01/19/1999US5861426 Nitro esters of aromatic compounds with amide or ester groups
01/19/1999US5861418 Aminobenzoic acid derivatives
01/19/1999US5861412 Dihydro-isoquinoline compounds and their use as pharmaceuticals
01/19/1999US5861411 Treating disturbances of memory such as senile dementia and alzheimer's disease
01/19/1999US5861407 Tetrahydropyridine derivatives as dopamine receptor subtype ligands
01/19/1999CA2028960C Novel isoindole derivatives and salts thereof, processes for producing the same and antitumor agent comprising the same
01/14/1999WO1999001456A1 Synthesis of and intermediates for camptothecins
01/14/1999WO1999001127A1 Compounds and methods
01/14/1999WO1998051311A3 Dihydropyrimidines and uses thereof