Patents
Patents for C07D 487 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups (57,272)
08/2008
08/06/2008EP1432714B1 Chemical compounds
08/06/2008EP1385518B1 Benzimidazolone compounds
08/06/2008CN101238131A Bridged piperazine and piperidine derivatives as CCR1 antagonists
08/06/2008CN101238130A Preparation of a 7H-pyrrolo[2,3-D]pyrimidine derivative
08/06/2008CN101238129A Compounds that maintain pluripotency of embryonic stem cells
08/06/2008CN101238128A Azabicyclic heterocycles as cannabinoid receptor modulators
08/06/2008CN101238127A Pyrimidine or triazine fused bicyclic metalloprotease inhibitors
08/06/2008CN101238126A Pyrrolobenzodiazepines and heteroaryl, aryl and cycloalkylamino ketone derivatives as follicle stimulating hormone receptor -(FSH-R) antagonists
08/06/2008CN101235037A Method for synthesizing alkoxyporphyrin
08/06/2008CN101235036A Porphyrin derivative and application for the same as small molecule antioxidant
08/06/2008CN101235035A Method for preparing tetramethoxymethylglycoluril
08/06/2008CN100408643C Use of marine fungus originated compounds as antifouling agents
08/06/2008CN100408581C 3-(1-alkoxy ethyl)-8-ethyl-2,7,12,15,18-pentamethyl-13-carboxylic acid-17-propionic acid, its synthetic method and light power therapeutic medicine
08/06/2008CN100408573C Pyrazole compounds useful as protein kinase inhibitors
08/06/2008CN100408564C Pyrazole derivatives for treating HIV
08/06/2008CN100408038C Use of a vitamin combination for the treatment of primary headaches
08/05/2008US7408065 P2X7 receptor antagonists and their use
08/05/2008US7408063 1,8-annelated quinoline derivatives substituted with carbon-linked triazoles as farnesyl transferase inhibitors
08/05/2008US7408061 Rylene dyes
08/05/2008US7408058 Regioisomerically pure oxochlorins and methods of synthesis
08/05/2008US7407974 e.g. 4-Methoxy-pyrrolidine-1,2-dicarboxylic acid 1-[(4-chloro-phenyl)-amide] 2-{[2-fluoro-4-(2-oxo-2H-pyridin-1-yl)-phenyl]-amide}; anticoagulant, thrombolytic agent; thrombus formation within blood vessels; cardiovascular disease
08/05/2008US7407971 Substituted pyrrolo-pyrazole derivatives as kinase inhibitors
08/05/2008US7407964 Stable; potent; penetrates cell membranes; effectively hinders cellular apoptosis; Antiinflammatory agents, Ischemic agents, cancer, autoimmune diseases and nervous system disorders.
08/05/2008US7407962 Heteroaryl compounds useful as inhibitors or protein kinases
08/05/2008US7407952 substance P, integrin receptor antagonist; mimic the secondary structure of reverse-turn regions of biologically active peptides and proteins; antiinflammatory agent; cell adhesion-mediated disease and central nervous system disorders
08/05/2008US7407951 Pyrrolobenzodiazepines
08/05/2008US7407949 4-(2-Cyclopropyl-ethyl)-piperazine-1-carboxylic acid 2-methyl-4-(3-methyl-4,10-dihydro-3H-2,3,4,9-tetraaza-benzo[f]azulene-9-carbonyl)-benzylamide; inter alia, primary dysmenorrhoea, male erectile dysfunction
08/05/2008US7407938 1,4-Diphenyl-3-(3-hydroxy-3-phenylpropyl)-2-azetidinones, e.g., 2,3,4,5,6-Pentahydroxyhexylamide of 4-(4-{4-[3-[3-(4-fluorophenyl)-3-hydroxypropyl]-2-(4-methoxyphenyl)-4-oxoazetidin-1-y]lbenzylcarbamoyl}phenoxy)benzoic acid; antilipemic agents that have intestinal absorption of less than 10%,
08/05/2008CA2388476C Bicyclic imidazo-5-yl-amine derivatives
08/05/2008CA2224435C Pyrrolopyrimidines and processes for the preparation thereof
07/2008
07/31/2008WO2008090379A1 Pyrazoloquinazolinones as inhibitors of poly(adp-ribose)polymerase (parp)
07/31/2008WO2008073687A3 Compounds and compositions as protein kinase inhibitors
07/31/2008WO2008065444A3 Substituted quinazolines
07/31/2008WO2008063232A3 Substituted pyrazolopyrimidines
07/31/2008WO2008045267A3 Pyrazolopyrimidines as cyclin dependent kinase inhibitors
07/31/2008WO2008011557A3 Heteroaryl inhibitors of rho kinase
07/31/2008WO2008005456A3 Fused heterocyclic inhibitors of d-amino acid oxidase
07/31/2008US20080182881 TNF-alpha production inhibitors
07/31/2008US20080182861 Inhibitors of diacylglycerol o-acyltransferase type 1 enzyme
07/31/2008US20080182849 Certain Heterocyclic Substituted Imidazo[1,2-A]Pyrazin-8-Ylamines And Methods Of Inhibition Of Bruton's Tyrosine Kinase By Such Compounds
07/31/2008US20080182848 anxiety; insomnia; high yielding; optically resolving eszopiclone using a multi-column continuous process or a simulated moving bed process; stationary phase used in chiral chromatography process is a derivative of tris(3,5-dimethylphenyl carbamate), or a derivative of tris- alpha -methylbenzylcarbamate
07/31/2008US20080182834 less toxic than the unassociated metal complex by hindering reactions in the blood stream; antitumor agents; platinum, palladium, gold amine inclusion compounds
07/31/2008US20080182302 Open reading frames which encode polypeptides sufficient to direct the biosynthesis synthesis of a safracin molecule having improved properties and that could be used in the hemi-synthesis of new ecteinascidins compounds; combinatorial chemistry; antitumor agents; broad-spectrum antibiotics; bactericides
07/30/2008EP1950213A2 Process for the synthesis of N-[3- (3-cyanopyrazolo [1,5a] pyrimidin-7-yl) -phnyl] -N-ethyl-acetamide
07/30/2008EP1950212A1 Polycyclic carbamoylpyridone derivative having inhibitory activity on hiv integrase
07/30/2008EP1950199A1 Proline derivatives and use thereof as drugs
07/30/2008EP1948664A2 Pyrrolotriazine kinase inhibitors
07/30/2008EP1948663A2 Pyrazolo-pyrimidines as casein kinase ii (ck2) modulators
07/30/2008EP1948662A2 Tricyclic compounds useful as oxytocin receptor agonists
07/30/2008EP1948661A1 Pyrazolo[4,3-d]pyrimidin-5-yl)derivative used as pde5 inhibitors
07/30/2008EP1948660A1 Tetracyclic indole derivatives as antiviral agents
07/30/2008EP1948659A1 Pyrrolopyrimidine derivatives as syk inhibitors
07/30/2008EP1948658A1 Pyrrolopyrimidine derivatives as syk inhibitors
07/30/2008EP1948656A2 Azaindole compounds and use thereof as phospholipase-a2 inhibitors
07/30/2008EP1948601A1 Fab i inhibitor and process for preparing same
07/30/2008EP1948242A2 Duocarmycin derivatives as novel cytotoxic compounds and conjugates
07/30/2008EP1948162A1 Pharmaceutical compositions containing erythrine mulungu derivatives and processes for their production
07/30/2008EP1725558A4 Method for preparing compounds comprising cucurbituril groups
07/30/2008EP1716152B1 Fused hetrocyclic compounds and their use as metabotropic receptor antagonists for the treatment of gastrointestinal disorders
07/30/2008EP1603918B1 Boronated metal-phthalocyanines, process for their preparation, pharmaceutical compositions comprising them and use thereof
07/30/2008EP1592684B1 Malonamide derivatives as gamma-secretase inhibitors
07/30/2008CN101233138A Pyrrolo[2,3-d]pyrimidine derivatives, their intermediates and synthesis
07/30/2008CN101233137A Macrocylic inhibitors of hepatitis c virus
07/30/2008CN101233136A Pyrrolotriazine compounds useful as kinase inhibitors and methods of treating kinase-associated conditions therewith
07/30/2008CN101233135A Diaryl-purine, azapurines and -deazapurines as non-nucleoside reverse transcriptase inhibitors for treatment of HIV
07/30/2008CN101233134A 制备泛昔洛韦和其它嘌呤衍生物 Preparation of famciclovir and other purine derivatives
07/30/2008CN101232885A Substituted pyridazinyl- and pyrimidinyl-quinolin-4-ylamine analogues
07/30/2008CN101230034A Nitrogen hetero-cycle compounds for use in the treatment of 5-hydroxide tryptamines related diseases
07/30/2008CN101229164A Composition and antiviral activity of substituted azaindoleoxoacetic piperazine derivatives
07/30/2008CN100406466C Nucleic acid hydrolysis cutting agent based on cucurbituril
07/30/2008CN100406459C 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino[4,5-b]indole-1-acetamide derivatives, preparation and use thereof in medicaments
07/30/2008CN100406454C Pyrazole compounds useful as protein kinase inhibitors.
07/30/2008CN100406010C Antitumor agents and process for producing the same
07/29/2008US7405306 3-(2-alkoxycarbonyl-3-indolyl)-3-oxo-propionic acid ester or propionamide intermediates: methyl 3-[6-fluoro-2-(methoxycarbonyl)-1-methyl-1H-indol-3-yl]-3-oxopropanoate; peripheral neuropathy, Parkinson's disease, Alzheimer's disease
07/29/2008US7405300 Central nervous system disorders; cardiovascular disorders; antiischemic agents; strokes; antiarthritic agents; anticancer agents; muscular disorders
07/29/2008US7405299 Compounds as pharmaceutical agents
07/29/2008US7405298 Process for making risperidone and intermediates therefor
07/29/2008US7405297 3-amino-2-ethoxycarbonylpyrrole; chemical intermediate in synthesis of 3H,5H-pyrrolo[3,2-d]pyrimidin-4-one; a convergent synthesis route rather than a linear one
07/29/2008US7405295 Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compounds
07/29/2008US7405221 2-(4-fluorobenzyloxy)-4-(2,4-dichlorophenyl)-5-(4-chlorophenyl)pyrimidine; antagonists or inverse agonists of the Cannabinoid-1 (CB1) receptor; antidepressant, neuroleptic, anxiolytic, antiinflammatory agent, cognition activator; psychosis, epilepsy, Parkinson's disease, and schizophrenia
07/29/2008US7405220 Pyrazolopyrimidines
07/29/2008US7405219 3-(4-amino-3-methylbenzyl)-7-(2-furyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidine-5-amine; adenosine receptor antagonist; antidepressant, neurodegenerative disorders, cognition activator, attention deficit disorder
07/29/2008US7405218 Isothiazole derivatives useful as anticancer agents
07/29/2008US7405213 such as 3-chloro-4-fluoro-N-(5-{[6-({3-[4-(hydroxymethyl)piperidin-1-yl]propyl}oxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl]amino}pyrimidin-2-yl)benzamide; serine/threonine Aurora kinase inhibitor; anticarcinogenic agent
07/29/2008US7405212 Helix mimetics and composition and methods related thereto
07/29/2008US7405041 Methods for regulating transcription by targeting quadruplex DNA
07/29/2008CA2515596C Cannabinoid receptor ligands and uses thereof
07/29/2008CA2432222C Pyrazole compounds useful as protein kinase inhibitors
07/29/2008CA2432132C Pyrazole compounds useful as protein kinase inhibitors
07/29/2008CA2409842C 1,4-diazepan-2,5-dione derivatives and their use as nk-1 receptor antagonists
07/29/2008CA2254070C Method for treating viral infections
07/29/2008CA2214086C Pyrazole derivatives and processes for the preparation thereof
07/24/2008WO2008089390A1 New classical antifolates
07/24/2008WO2008089027A1 Compounds for the treatment of hepatitis c
07/24/2008WO2008087936A1 Condensed tetrahydroquinoline derivative and use thereof for medical purposes
07/24/2008WO2008087529A1 Nicotinic acetylcholine receptor modulators
07/24/2008WO2008087278A2 5-alkyloxy-indolin-2-one derivatives, preparation thereof and application thereof in therapy as selective ligands of v2 vasopressin receptors
07/24/2008WO2008068424A3 Substituted 2,5-dihydro-3h-pyrazolo[4,3-c]pyridazin-3-one derivatives, preparation thereof and use of same as cannabinoid cb1 receptor ligands
07/24/2008WO2008068272A3 Antibacterial quinoline derivatives
07/24/2008WO2008051808A3 Bicyclic triazoles as protein kinase modulators