Patents for C07D 487 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups (57,272) |
---|
11/05/2008 | EP1987036A1 Hetero-bycyclic antiviral compounds |
11/05/2008 | EP1987035A1 Heterocyclic antiviral compounds |
11/05/2008 | EP1987020A1 Azacyclyl-substituted aryldihydroisoquinolinones, process for their preparation and their use as medicaments |
11/05/2008 | EP1987010A1 Tricyclic n-heteroaryl-carboxamide derivatives containing a benzimidazole unit, method for preparing same and their therapeutic use |
11/05/2008 | EP1986652A2 Aminotetrahydropyrans as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes |
11/05/2008 | EP1986645A1 Glucokinase activators |
11/05/2008 | EP1781659B1 Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors |
11/05/2008 | EP1608374B1 2-phenoxy- and 2-phenylsulfomamide derivatives with ccr3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders |
11/05/2008 | EP1218383B1 Bicyclic imidazo-5-yl-amine derivatives |
11/05/2008 | EP1216247B1 Imidazoimidazoles and triazoles as anti-inflammatory agents |
11/05/2008 | CN101300260A Method for synthesizing spiro quaternary ammonium systems |
11/05/2008 | CN101300259A Tricyclic spiro derivatives as CRTH2 modulators |
11/05/2008 | CN101300233A Azafused cyclin dependent kinase inhibitors |
11/05/2008 | CN101298433A 2-, 3-, 4-, or 5-substituted-n1-(benzensulfonyl)indoles and their use in therapy |
11/05/2008 | CN100430398C Diazabicyclic central nervous systems active agents |
11/05/2008 | CN100430397C Phosphoric acid salt of a dipeptidyl peptidase-iv inhibitor |
11/05/2008 | CN100430396C 2-phenyl-substituted imidazo-triazone used as phosphodiesterase inhibitor |
11/04/2008 | US7446210 Factor Xa compounds |
11/04/2008 | US7446209 Diazotizing a blocked 5-amino-1H-imidazole-4-carboxamide; hydrolysis; antitumor agents |
11/04/2008 | US7446199 Compositions useful as inhibitors of protein kinases |
11/04/2008 | US7446196 Leptomycin compounds |
11/04/2008 | US7446113 the prodrug forms of compounds have good absorption, pharmacokinetics, distribution and transport to the brain; 4-[8-Trifluoromethyl-6-(4-trifluoromethyl-phenyl)-imidazo[1,2-a]pyridin-3-ylethynyl]-benzenesulfonamide; nervous system disorders like psychosis, schizophrenia, Alzheimer's disease, depression |
11/04/2008 | US7446108 Tri-and tetraaza-acenaphthylen derivatives as CRF receptor antagonists |
11/04/2008 | US7445845 Synthesis, spectroscopy, photophysics of multi-chromophoric ZN(II) group 8 metal complexes |
11/04/2008 | US7445768 Delivery of sedative-hypnotics through an inhalation route |
11/04/2008 | CA2443449C Pyrazole derivatives for treating hiv |
10/30/2008 | WO2008131050A1 Pyrrolotriazine kinase inhibitors |
10/30/2008 | WO2008130951A1 Fused heterocyclic 11-beta-hydroxysteroid dehydrogenase type i inhibitors |
10/30/2008 | WO2008130581A1 Pyrimidinone derivatives and methods of use thereof |
10/30/2008 | WO2008130314A1 Xanthine compounds having a positive allosteric gabab receptor modulator effect |
10/30/2008 | WO2008128942A1 Tricyclic nitrogen containing compounds as antibacterial agents |
10/30/2008 | WO2008128921A1 Process for hcv protease inhibitor intermediate |
10/30/2008 | WO2008085942A3 Methods for preparing arene-bis(dicarboximide)-based semiconducting materials and related intermediates for preparing same |
10/30/2008 | WO2008074752A3 Indolylmaleimide derivatives as kinase inhibitors |
10/30/2008 | WO2008005471A3 Novel heterobicyclic compounds |
10/30/2008 | WO2007147104A3 Novel compounds |
10/30/2008 | WO2007114926A3 Kinase antagonists |
10/30/2008 | WO2007106439A3 Homotropanes with central nervous system activity |
10/30/2008 | US20080269499 Crystalline forms and process for preparing spiro-hydantoin compounds |
10/30/2008 | US20080269485 Fluorinated dyes and their use in electrophoretic display devices |
10/30/2008 | US20080269257 Use of Substituted 2-Pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-A] Pyrimidin-4-one and 7-Pyrimidinyl-2,3-dihydroimidazo[1,2-A] Pyrimidin-5(1H)one Derivatives |
10/30/2008 | US20080269230 Inhibitors of proton-gated cation channels and their use in the treatment of ischaemic disorders |
10/30/2008 | US20080269217 Melanocortin-4 receptor binding compounds and methods of use thereof |
10/30/2008 | US20080269184 Niosome Having Metal Porphyrin Complex Embedded Therein, Process For Producing The Same And Drug With The Use Thereof |
10/30/2008 | US20080269140 Conformationally Constrained Smac Mimetics and the Uses Thereof |
10/30/2008 | US20080269061 Substituted thiene-3-ylsulphonylamino(thio)carbonyltriazolin(ethi)ones |
10/30/2008 | US20080268044 Novel Process and Formulations |
10/30/2008 | US20080267942 7-hydroxy-6-{[1-methyl-3-(1,3-thiazol-5-yl)propyl]amino}-4,5,6,7-tetrahydroimidazo[4,5,1-jk][1]benzazepin-2(1H)-one; agonists at the beta-2 adrenoceptor; feed additives for livestock animals; improving meat yield or meat quality |
10/30/2008 | US20080267906 Novel Spirotropane Compounds and Methods for the Modulation of Chemokine Receptor Activity |
10/30/2008 | US20080267867 Imidazole, pyridine derivative silver complexes; nanofiber with radioactive transition metal, lanthanide, actinide; radiopharmaceutical peptide, polyamine, imaging and tumor treatment |
10/30/2008 | US20080267866 Cross-bridged tetraamine macrocycles complexed with transition metal ions, radioactive metal species, fluorescent tag; as CXCR4 co-receptor antagonist is a dosage form for treatment of HIV; radiopharmaceutical for imaging chemokine receptors; drug screening assays for chemokine receptor binding |
10/30/2008 | US20080264487 Photoelectric Conversion Devices |
10/30/2008 | CA2684659A1 Tricyclic nitrogen containing compounds as antibacterial agents |
10/30/2008 | CA2684633A1 Pyrimidinone derivatives and methods of use thereof |
10/30/2008 | CA2684086A1 Process for hcv protease inhibitor intermediate |
10/30/2008 | CA2682301A1 Xanthine compounds having a positive allosteric gabab receptor modulator effect |
10/29/2008 | EP1984454A1 Method of manufacturing phthalocyanine compound |
10/29/2008 | EP1984374A1 Use of spiro ý imidazolidine-4, 3'-indole¨2, 2', 5' (1h) triones for treatment of conditions associated with vanilloid receptor 1 |
10/29/2008 | EP1984373A1 6,7-dihydrobenzimidazo[1 ,2-c]quinazolin-6-one carboxylic acids, their esters, and methods of synthesis thereof |
10/29/2008 | EP1984372A1 Organic compound, anisotropic optical film and method of production thereof |
10/29/2008 | EP1984371A1 Zopiclone resolution using l-tartaric acid |
10/29/2008 | EP1984370A1 Imidazopyridine derivatives inhibiting protein kinase activity, method for the preparation thereof and pharmaceutical composition containing same |
10/29/2008 | EP1984369A2 Nitroimidazole compounds |
10/29/2008 | EP1984368A2 Improved process for the preparation of an optically active 5h-pyrrolo [3,4-b]pyrazine derivative |
10/29/2008 | EP1984353A1 Aurora kinase modulators and method of use |
10/29/2008 | EP1984331A1 Pyrrolidine derivatives as erk inhibitors |
10/29/2008 | EP1556055B1 Cyclic nucleotide phosphodiesterase inhibitors having a benzodiazepine structure and their use in therapy |
10/29/2008 | EP1531811B1 Derivatives of 3-hydroxy-4-(cyclyl-alkylaminoalkyl)-5-phenyl-1h-pyrazole as antagonists of the gonadotropin releasing hormone (gnrh) for use in the treatment of sex hormone related conditions, such as prostatic of uterine cancer |
10/29/2008 | EP1216228B1 BENZAMIDES AND RELATED INHIBITORS OF FACTOR Xa |
10/29/2008 | CN101296929A Tricyclic compounds useful as oxytocin receptor agonists |
10/29/2008 | CN101296928A Compounds and compositions as protein kinase inhibitors |
10/29/2008 | CN101296926A Heterocyclic aspartyl protease inhibitors |
10/29/2008 | CN101296902A Compounds comprising a lactam or a lactam derivative moiety, processes for making them, and their uses |
10/29/2008 | CN101296699A Pyrazolo[1,5-a]pyrimidine compounds |
10/29/2008 | CN101293854A Novel midbody of pemetrexed, preparing method and application thereof |
10/28/2008 | US7442804 heating under microwave irradiation (3-hydroxymethylene-4-carboxylic acid ester-2-one)pyrroline derivatives in presence of inert solvent to produce 3,6-diphenylfuro[3,4-c]pyrrole-1,4-diones (furopyrroles); intermediates in process for preparation of diketopyrrolopyrroles; high yield and purity |
10/28/2008 | US7442795 Triazole compounds useful in therapy |
10/28/2008 | US7442792 halogenation of pyrazolo[1,5-a][1,3,5]triazin-4-ol's, with phosphorus oxyhalides, then dehalogenation and amination to yield dimethylpyrazolo[1,5-a][1,3,5]triazin-4-amine's, used as corticotropin releasing factor (CRF) receptor antagonists; anxiolytic agents; antidepressants |
10/28/2008 | US7442710 Substituted phenyl methanones |
10/28/2008 | US7442700 N-[4-({4-[(5-methyl-1H-pyrazol-3-yl)amino]pyrrolo[2,1f][1,2,4]triazin-2-yl}sulfanyl)phenyl]cyclopropanecarboxamide; serine/threonine Aurora kinase inhibitor; anticarcinogenic agent; allergies and asthma, Alzheimer's disease, rheumatoid arthritis, autoimmune diseases, bone diseases, inflammation |
10/28/2008 | US7442694 Diazabicyclic compounds useful in the treatment of CNS and other disorders |
10/28/2008 | US7442558 Phthalamide-lanthanide complexes for use as luminescent markers |
10/28/2008 | US7442368 Rapidly producing peak plasma concentration; condensation aerosol containing ephedrine and/or fenfluramine; vaporization without degradation |
10/28/2008 | CA2472107C Dibenzodiazepine derivates, their preparation and use |
10/28/2008 | CA2448735C Novel substituted tetracyclic imidazole derivatives, processes for their preparation, pharmaceutical compositions comprising them and their use as a medicine |
10/28/2008 | CA2380452C Imidazo-triazine derivatives as ligands for gaba receptors |
10/28/2008 | CA2291160C Combination therapy for modulating the human sexual response |
10/23/2008 | WO2008128072A2 Axl kinase inhibitors useful for the treatment of cancer or hyperproliferative disorders |
10/23/2008 | WO2008127275A2 Pyrrolinone compounds as inhibitors of bacterial peptidyl trna hydrolase and uses thereof |
10/23/2008 | WO2008127060A1 Aspartate of 1-cyclopropyl-6-fluoro-7-(8-methoxyimino-2,6-diaza- spiro[3.4]oct-6-yl)-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid, method for preparing the same, and antimicrobial pharmaceutical composition comprising the same |
10/23/2008 | WO2008126920A1 Remedy for diabetes |
10/23/2008 | WO2008126105A2 Improved process for the preparation of zopiclone and it's enantiomerically enriched isomer |
10/23/2008 | WO2008125945A2 3-amido-pyrrolo [3, 4-c] pyrazole-5 (1h, 4h, 6h) carbaldehyde derivatives as inhibitors of protein kinase c |
10/23/2008 | WO2008125833A1 Pharmaceutical compounds |
10/23/2008 | WO2008125618A1 Folate-conjugates and corresponding metal-chelate complexes for use in diagnostic imaging and radiotherapy |
10/23/2008 | WO2008099210A3 Piperazine derivatives for treatment of ad and related conditions |
10/23/2008 | WO2008040995A8 Indazoles for use as dpp-iv inhibitors |
10/23/2008 | WO2007139946A3 Gpcr ligands identified by computational modeling |
10/23/2008 | US20080262243 Reacting a vinyl sulfone compound with imide compound in presence of catalyst |
10/23/2008 | US20080262205 Unphosphorylated glycogen synthase kinase-3-g-beta (GSK) from baculovirus overexpression system; competitive binding; diabetes, Alzheimer's disease |