Patents
Patents for C07D 473 - Heterocyclic compounds containing purine ring systems (11,932)
04/1996
04/18/1996CA2202368A1 Lta4 hydrolase inhibitor pharmaceutical compositions and methods of use
04/18/1996CA2201773A1 Purine and guanine compounds as inhibitors of pnp
04/16/1996US5508277 Administering to suppress tumor cell resistance to antineoplastic drugs
04/11/1996WO1996010568A1 Substituted aryl piperazines as neurokinin antagonists
04/11/1996CA2199621A1 Substituted aryl piperazines as neurokinin antagonists
04/10/1996EP0705265A1 Novel chemical compounds having pde-iv inhibition activity
04/10/1996EP0705264A1 Carbo-acyclic nucleoside derivatives as antiviral and antineoplastic agents
04/10/1996CN1120044A Preparation of N-9 substituted guanine compounds
04/10/1996CN1120043A Method of extracting natural caffeine from tea
04/09/1996US5506349 Reacting 5'-silylated-2',3'-deoxyuridine with 2,3,4-triazole, phosphorus oxychloride and ammonia; cleaving silyl group with ion exchange resin
04/09/1996US5506347 Lyxofuranosyl analogues of adenosine
04/09/1996US5506337 Morpholino-subunit combinatorial library and method
04/09/1996US5506243 Sulfonamide derivatives
04/03/1996EP0704445A1 Preparation of N-9 substituted guanine compounds
03/1996
03/28/1996DE4434049A1 Heterocyclic cpds. used in aq. soln. for compacting anodised layers
03/27/1996EP0702683A1 06-substituted guanine derivatives, a process for their preparation and their use in treating tumour cells
03/27/1996EP0702682A1 Amino acid ester of nucleoside analogues
03/27/1996EP0548250B1 Substituted bicyclic aryl compounds exhibiting selective leukotriene b4 antagonist activity
03/27/1996CN1031404C Process for production of substituted azole
03/27/1996CN1031403C Process for preparation of hydroxyalkylfuranyl derivatives
03/19/1996US5500428 Furyl-substituted purines and adenosine antagonists
03/13/1996EP0700908A1 1-Arylpyrimidine derivatives and pharmaceutical use thereof
03/13/1996CN1118600A 2-benzyl-polycyclic guanine derivatives and process for preparing them
03/13/1996CN1118599A Xanthine derivatives as adenosine A1 receptor antagonists
03/07/1996WO1996006845A1 Substituted 9-alkyladenines
03/07/1996WO1996006844A1 4-(2-amino-6-(cyclopropylamino)-9h-purin-9-yl)-2-cyclopentene-1-methanol succinate as antiviral agent
03/07/1996WO1996006833A1 Novel nucleotide analogs
03/07/1996WO1996006614A1 Novel antibiotic compounds and methods to treat gram-positive bacterial and mycoplasmal infections
03/07/1996CA2198739A1 Novel antibiotic compounds and methods to treat gram-positive bacterial and mycoplasmal infections
03/06/1996EP0699208A1 Novel peptide nucleic acids
03/05/1996US5496945 Reaction of guanimine with hexamethyldisilazane with aprotic solvent and ammonium sulfate, reaction with acyloxyethoxy methyl halide then hydrolyzed with aqueous sodium acetate
03/05/1996US5496823 Administering propentofylline or a salt thereof to a patient
03/05/1996CA2085733C Polycyclic guanine derivatives
02/1996
02/28/1996EP0698607A1 Xanthine derivative
02/28/1996EP0697873A1 Olefin-substituted long chain compounds
02/28/1996CN1031132C Process for preparation of carbocyclic adenosine analogs useful as immunosuppressants
02/27/1996US5495023 Nitro compounds, process for preparation thereof and use thereof
02/21/1996EP0697020A1 8-substituted xanthines as selective adenosine receptor agents
02/21/1996CN1031056C Process for preparing 6-substituted purinyl piperazine derivatives
02/21/1996CN1031055C Process for preparing dideoxycarbocyclic nucleosides
02/21/1996CN1031054C Process for production of bis-(hydroxymethyl)-cyclobutyl-purines and pyrimidines
02/15/1996WO1996004281A1 Substituted o6-benzylguanines and 6(4)-benzyloxypyrimidines
02/15/1996WO1996004280A1 Phenyl xanthine derivatives
02/15/1996CA2632452A1 Substituted o6-benzylguanines and use thereof
02/14/1996CN1116625A Method for preparing anti-asthmatic and antitussive medicine
02/13/1996US5491146 Adenosin deaminase inhibitors
02/08/1996WO1996003125A1 Carbon monoxide dependent guanylyl cyclase modifiers
02/08/1996CA2195302A1 Carbon monoxide dependent guanylyl cyclase modifiers
02/07/1996CN1116204A Processes for the diastereoselective synthesis of nucleosides
02/07/1996CN1030916C Process for preparing hydroxymethyl (methylenecyclopentyl) purines and pyrimidines
02/01/1996WO1996002543A1 2,3-dihydroxy cyclopentane derivatives of purines
02/01/1996DE19526163A1 New ganciclovir mono:esters and intermediates
01/1996
01/31/1996EP0694547A2 2-(2-amino-1,6-dihydro-6-oxo-purin-9-yl)methoxy-1,3-propanediol derivative
01/27/1996CA2152863A1 Preparation of acyclovir
01/25/1996WO1995028402A3 Preparation of purines
01/24/1996EP0693498A1 Antiviral compounds
01/24/1996EP0693071A1 New carboxylic-acid esters of 2-amino-7-(1,3-dihydroxy-2-propoxymethyl)purine, the preparation of such esters and their use
01/23/1996US5486520 1,3-oxathiolanes useful in the treatment of hepatitis
01/20/1996CA2154293A1 1-arylpyrimidine derivatives and pharmaceutical use thereof
01/17/1996CN1114880A Novel treatment
01/16/1996US5484920 Therapeutic agent for Parkinson's disease
01/10/1996EP0690861A1 Substituted heteroannulated imidazoles and their use as herbicides
01/03/1996EP0690056A2 Process for the preparation of purins
01/03/1996EP0689460A1 Cyclobutyl antisense oligonucleotides, methods of making and use thereof
01/03/1996CN1114318A Novel purine derivatives and pharmaceutically acceptable salts thereof
01/03/1996CN1114317A Cyclopropane derivatives and method of preparing the same
12/1995
12/29/1995CA2152722A1 Process for the production of purines
12/28/1995WO1995035304A1 Hydroxyalkylammonium-pyrimidines or purines and nucleoside derivatives, useful as inhibitors of inflammatory cytokines
12/28/1995WO1995035297A1 Novel substituted purinyl derivatives with immunomodulating activity
12/28/1995CA2193645A1 Hydroxyalkylammonium-pyrimidines or purines and nucleoside derivatives, useful as inhibitors of inflammatory cytokines
12/28/1995CA2165956A1 Novel substituted purinyl derivatives with immunomodulating activity
12/27/1995EP0688784A2 3'-Modified oligonucleotide derivatives
12/26/1995US5478928 2',3'-dideoxy-4'-thioribonucleosides and synthetic precursors thereof
12/26/1995US5478831 R-(-)1-(5-hydroxyhexyl)-3-methyl-7-propylxanthine, a process for its preparation and pharmaceuticals containing this compound
12/26/1995US5477857 Measuring myocardial function in mammals
12/19/1995US5476938 Reacting protected purine or pyrimidine base with oxiranyl compound,reacting the intermediate with a phosphonate, removing protecting groups
12/19/1995US5476931 Reacting with a base in a mixed solvent containing alcohol
12/14/1995WO1995033750A1 Corticotropin releasing factor antagonists
12/13/1995EP0686157A1 2-benzyl-polycyclic guanine derivatives and process for preparing them
12/13/1995EP0686155A1 Xanthine derivatives as adenosine a1 receptor antagonists
12/13/1995EP0311694B1 Nucleoside derivatives and process for their preparation
12/12/1995US5475107 Alkylation in the presence of quaternary ammonium and/or phosphonium compounds and ethers in a two-phase mixture
12/12/1995US5475002 Use of 1-(5-oxohexyl)-3-methyl-7-n-propylxanthine in vascular surgery
12/06/1995EP0684953A1 Adenosine kinase inhibitors comprising lyxofuranosyl derivatives
12/05/1995US5473070 Substituted long chain alcohol xanthine compounds
12/05/1995US5473063 Reacting 2,3-epoxy-butanediol/1,4-/(having protected hydroxyl groups) with an alpha allylic nucleophile yields 2-hydroxy-3-allyl-1,4-butanediol, then oxidatively cleaving the double bond, cyclization, halogenation, acetylation or oxyalkylation
12/05/1995US5472873 Rhodotorula rubra useful in a process for the preparation of (ω-1)-hydroxyalkylxanthines
11/1995
11/29/1995EP0684243A1 Process for preparing 2-amino-6-chloropurine and 2-acylamino-6-chloropurine
11/29/1995EP0586523A4 Determination of prodrugs metabolizable by the liver and therapeutic use thereof
11/28/1995US5470878 Cell signaling inhibitors
11/28/1995US5470867 Imidazoles and their salts having antagonistic activity to angiotesin II recetors
11/28/1995US5470858 Derivatives of (hetero)aromatic ethers and thioethers having antihyperlipidemic activity, process for their preparation and pharmaceutical compositions containing them
11/28/1995US5470837 Autoimmune disease
11/28/1995US5470579 Xanthines, optionally incorporated in liposomes, for promoting skin or hair pigmentation
11/23/1995WO1995031774A1 Graphical user interfaces having animated control elements
11/23/1995WO1995031460A1 Process for producing xanthine derivative
11/23/1995WO1995031459A1 Morpholino-subunit combinatorial library and method
11/23/1995WO1995031450A1 Asymmetric synthesis of chiral secondary alcohols
11/23/1995CA2190511A1 Asymmetric synthesis of chiral secondary alcohols
11/23/1995CA2167314A1 Process for producing xanthine derivative