Patents
Patents for C07D 473 - Heterocyclic compounds containing purine ring systems (11,932)
02/1992
02/19/1992EP0471383A2 Use of 5'-vinylhalo-aristeromycin/adenosine analogs as immunosuppressants
02/19/1992EP0471057A1 Methods and compositions for the prophylaxis and treatment of cytomegalovirus infections
02/18/1992US5089618 Process for the purification of adenine
02/18/1992US5089500 Viricides; hepatitis, aids
02/18/1992CA1296001C 1-hydroxyalkylxanthines, processes for their preparation and medicaments containing them
02/13/1992DE4025358A1 New bi:phenyl:methyl-substd. imidazole derivs.
02/12/1992EP0470543A1 Heterocyclic imidazoles, remedies containing them and processes for their preparation
02/12/1992EP0470317A1 Use of a derivative of 1,3,7-trimethylxanthine for the treatment of memory disorders, senile intellectual disorders and Alzheimer's disease
02/11/1992US5087697 Therapeutic nucleosides
02/11/1992CA2048809A1 Heterocyclic imidazoles, pharmaceutical compositions containing these compounds and processes for preparing them
02/06/1992WO1992001697A1 Novel substituted thiazolyl and substituted pyridinyl derivatives
02/06/1992CA2086546A1 Novel substituted thiazolyl and substituted pyridinyl derivatives
02/05/1992CN1058406A Substituted azole, process for production and use thereof
02/04/1992US5086056 Treating allergic diseases
01/1992
01/29/1992EP0468866A1 Novel carbocyclic analogs of certain nucleosides
01/29/1992EP0468372A2 Substituted azoles, process for their preparation and their use
01/29/1992EP0468352A2 Novel nucleic acid derivatives
01/29/1992EP0468119A1 Novel carbocyclic analogs of certain nucleosides
01/29/1992EP0467895A1 Dihydropyridine antiallergy agents
01/29/1992CN1058216A Substituted thiazolyl and substituted pyridinyl derivatives
01/29/1992CN1058215A Oxazolyl derivatives
01/25/1992CA2047644A1 Nucleic acid derivatives
01/25/1992CA2047390A1 Carbocyclic analogs of certain nucleosides
01/23/1992WO1992000742A1 Penciclovir and famciclovir and related guanine derivatives for the treatment of the hiv-1 infections
01/23/1992DE4023215A1 New substd. azole derivs. angiotensin II antagonists - for treating hypertension, coronary insufficiency, myocardial infarct, coronary hypertrophy, arteriosclerosis etc.
01/22/1992EP0467207A2 Purinderivate
01/22/1992CA2047467A1 Substituted azoles, a process for their preparation, and their use
01/21/1992US5082845 Gastrointestinal
01/20/1992WO1992002511A1 Novel process for the preparation of nucleotides
01/20/1992WO1992001698A1 Antiviral phosphono-alken derivatives of purines
01/20/1992WO1992001687A1 Novel oxazolyl derivatives
01/20/1992CA2087446A1 Antiviral phosphono-alken derivatives of purines
01/20/1992CA2086545A1 Oxazolyl derivatives
01/19/1992CA2044806A1 Purine derivatives
01/15/1992EP0466164A2 Process for the preparation of 2-chloro-1,7-dihydropurin-6-one and process for the purification of the same
01/15/1992EP0344288A4 Method of inhibiting the activity of leukocyte derived cytokines
01/14/1992CA2046846A1 Process for preparing 2-chloro-1,7-dihydropurin-6-one and a process for its purification
01/09/1992WO1992000315A1 Oligonucleotide functionalization method
01/09/1992WO1992000297A1 New xanthine derivatives
01/09/1992CA2064742A1 Xanthine derivatives
01/08/1992EP0464769A2 Purinyl and pyrimidinyl tetrahydrofurans
01/08/1992EP0464511A2 Process for the preparation of acyclic, substituted nucleosides and its intermediates
01/08/1992EP0464137A1 Inhibition of hiv using synergistic combinations of nucleoside derivatives
01/08/1992EP0464112A1 A process for the preparation of 9-substituted guanine derivatives and intermediates for use in the process.
01/08/1992CN1057652A Process for preparing substituted acyclic nucleosides and intermediates occurring therein
01/07/1992US5079252 Valeryl ester of acyclovir improves bioavailability of acylclovir, viricides, treatment of herpes
01/02/1992DE4019892A1 New xanthine derivs. are selective A1 adenosine antagonists - useful for treating CNS disorders (e.g. senile dementia) and heart and circulation disorders
01/01/1992CN1057463A 6-substituted purinyl piperazine derivatives
12/1991
12/28/1991CA2045730A1 Process for the preparation of substituted acyclic nucleosides, and intermediates occurring therein
12/25/1991CN1057257A Imidazole derivatives, their preparation process, intermediates obtained, their use as medicaments and pharmaceutical compositions containing them
12/24/1991US5075445 Viricides
12/22/1991WO1991019717A1 Polycyclic guanine derivatives
12/18/1991EP0461407A1 Improved process for the preparation of 2-amino(2,3,5-tri-O-benzyl-beta-D-arabinofuranosyl)adenine
12/18/1991CA2019145A1 U.s.p. caffeine extraction and purification
12/17/1991US5073559 2-Substituted purinone having phosphodiesterase inhibitory activity
12/12/1991WO1991018969A1 Fluorinated bis(hydroxymethyl)cyclobutyl purines and pyrimidines
12/12/1991WO1991018898A1 Nucleic acid homolog
12/11/1991EP0461040A1 Imidazol derivatives, their process for production, intermediates, their application as medicaments and the pharmaceutical compositions containing them
12/10/1991US5071846 Anti-hystaminic [(bicyclic heterocyclyl) methyl and --hetero] substituted hexahydro-1H-azepines and pyrrolidines
12/09/1991CA2044087A1 Imidazole derivatives, process for their preparation, novel intermediate products, their applications as pharmaceuticals and pharmaceutical compositions holding same
12/04/1991CN1056692A Method of extracting natural caffeine from tea
12/03/1991US5070205 Alkyl 2-benzylidene-4-(benzimidazol-1-yl) benzoylacetate esters as intermediates
11/1991
11/27/1991EP0458618A1 6-Substituted purinyl piperazine derivatives
11/27/1991EP0458459A2 Substituted benzhydryl 2-hydroxypropyl piperazine derivatives
11/27/1991EP0458363A1 Fluorinated bis(hydroxymethyl) cyclobutyl purines and pyrimidines
11/27/1991EP0458312A1 Novel cyclobutane derivatives
11/27/1991EP0457773A1 N?6 -substituted 9-methyladenines: a new class of adenosine receptor antagonists
11/26/1991US5068320 2-amino-6-(cyclopropylamino)purine-9-β-D-2',3'-dideoxyribofuranoside and its pharmaceutically acceptable salts
11/26/1991US5068236 Xanthine derivatives
11/25/1991WO1991017993A1 1-7 substituted xanthine derivatives having antiasthmatic activity, their salts physiologically acceptable, pharmaceutical composition containing them and process for their preparation
11/25/1991CA2083257A1 1-7 substituted xanthine derivatives having antiasthmatic activity, their salts physiologically acceptable, pharmaceutical composition containing them and process for their preparation
11/25/1991CA2043099A1 Cyclobutane derivatives
11/25/1991CA2042931A1 Fluorinated bis (hydroxymethyl) cyclobutyl purines and pyrimidines
11/24/1991CA2042944A1 6-substituted purinyl piperazine derivatives
11/19/1991US5066805 Catalytic hydrogenation of 2-amino-6-chloropurine
11/19/1991US5066655 Inhibiting adenylate cyclase
11/19/1991US5066652 Antiulcer agents
11/19/1991US5066426 Fluorescence polarization immunoassay utilizing substituted carboxyfluoresceins
11/13/1991EP0456514A1 2-Fluoroneplanocin A and its production
11/12/1991US5064961 Process for preparing an optically active cyclobutane nucleoside
11/06/1991EP0454773A1 Novel prodrug derivatives of biologically active agents containing hydroxyl groups or nh-acidic groups
11/06/1991CN1055930A Process for preparing optically active isomers of 6-substituted purinyl piperazine derivatives
11/05/1991US5063237 Antiallergens and antiinflammatory agents
11/05/1991US5063233 Cardiovascular disorders
10/1991
10/30/1991EP0454385A1 Process for preparing optically active isomers of 6-substituted purinyl piperazine derivatives
10/29/1991US5061708 Treatment of infection by herpes or cytomegalo virus
10/24/1991CA2040886A1 Process for preparing optically active isomers of 6-substituted purinyl piperazine derivatives
10/24/1991CA2040885A1 Substituted benzhydryl 2-hydroxypropyl piperazine derivatives
10/23/1991EP0452729A1 Process for preparing substituted cyclobutanes
10/23/1991EP0452680A1 Substituted purines, process for their preparation and their use as antiviral agents
10/22/1991US5059690 Purinyl tetrahydrofurans
10/22/1991US5059604 2-amino purine derivatives
10/21/1991WO1991016333A1 2',3'-dideoxy-4'-thioribonucleosides as antiviral agents
10/21/1991CA2080916A1 2',3'-dideoxy-4'-thioribonucleosides as antiviral agents
10/17/1991WO1991015490A1 Synthesis of purine substituted cyclopentene derivatives
10/17/1991WO1991015489A1 Process for the synthesis of cyclopentene derivatives
10/17/1991WO1991015447A1 Synthesis of cyclopentene derivatives
10/17/1991CA2040485A1 Process for preparing substituted cyclobutanes
10/15/1991US5057630 Reacting 4-nitromethyl-2-cyclopentene-1-ol with strong base, ozone, alkali or alkaline earth metal hydride yields 4-hydroxymethyl-2-cyclopentene-1-ol
10/15/1991US5057518 Pharmaceutical preparations