Patents
Patents for C07D 473 - Heterocyclic compounds containing purine ring systems (11,932)
04/2003
04/15/2003US6548486 New viricide compounds of the general formula: Nu-O-Fa, wherein O represents an oxygen, Nu is a nucleoside or nucleoside analogue, and Fa is an acyl group of mono-unsaturated c18-c20 fatty acid
04/10/2003WO2003028721A2 Substituted benzimidazole compounds and their use for the treatment of cancer
04/10/2003US20030069423 Novel processes for the preparation of adenosine compounds and intermediates thereto
04/10/2003US20030069259 Acyl and sulfonyl derivatives of 6,9-disubstituted 2-(trans-1,4-diaminocyclohexyl)-purines and their use as antiproliferative agents
04/10/2003US20030069257 Benzimidazole and pyridylimidazole derivatives
04/09/2003EP1300147A1 Purine compounds and adenosine A2 receptor antagonist as preventive or therapeutic agent for diabetes mellitus
04/09/2003CN1105109C Chloropyrimide intermediates
04/08/2003US6545002 Treating asthma, diarrhea, insulin resistance, diabetes, ischemia/reprefusion injuries, diabetic retinopathy or hyperbaric oxygen-induced retinopathy
04/08/2003US6545001 Antiviral nucleoside analogues
04/08/2003CA2086756C Penciclovir and famciclovir and related guanine derivatives for the treatment of the hiv-1 infections
04/03/2003WO2003026589A2 Methods and compositions for treating hepatitis c virus using 4'-modified nucleosides
04/03/2003WO2002102313A3 Pyrimidine inhibitors of phosphodiesterase (pde) 7
04/03/2003WO2002076460A3 Use of propentofylline to control intraocular pressure
04/03/2003US20030065187 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
04/03/2003US20030065146 Compound for use in the treatment of rheumatoid arthritis, osteoarthritis, inflammatory bowel disease and sepsis
04/03/2003US20030065023 Anticancer agents, viricides, psychological disorders
04/03/2003US20030064999 Therapy for asthma, diarrhea
04/03/2003US20030064982 Pyrazole compounds useful as protein kinase inhibitors
04/03/2003US20030064981 Anticancer agents; antidiabetic agents; Alzheimer's disease
04/03/2003US20030064374 Detecting neuronal stress in humans; obtain sample, measure phosphodiesterase concentration, evaluate for neuronal stress
04/02/2003EP1298348A1 Bush, group of bush, suspension cross-member, vehicle, method for mounting a bush and method for mounting a group of bushes
04/02/2003EP1298125A1 Substituted benzimidazole compounds and their use for the treatment of cancer
04/02/2003EP1296681A2 Use of microsomal triglyceride transfer protein (mtp) inhibitors for reducing the number of postprandial triglyceride-rich lipoprotein particles (pptrl)
04/02/2003EP1208100B1 Selective antagonists of a2b adenosine receptors
04/02/2003EP0874846B1 Purine derivatives and processes for their preparation
04/02/2003CN1406946A Technology for producing AR with IR as initiation material by liquid ammonia process
04/01/2003US6541625 Stereoselectively hydrolyzing an anomeric mixture of 2-benzoyloxydioxolanecarboxylate with an enzyme; separating product; replacing carboxylate by reaction with a purine or pyrimidinyl derivative
04/01/2003US6541482 Autoimmune disease
04/01/2003US6541477 Inhibitors of p38-a kinase
03/2003
03/27/2003WO2003025017A1 Cytokine receptor
03/27/2003WO2003024965A2 Heterocyclic compounds that are inhibitors of the enzyme dpp-iv
03/27/2003WO2003024962A1 Piperidine derivatives and their use as modulators of chemokine (especially ccr3) activity
03/27/2003WO2003024448A2 Inhibitors of histone deacetylase
03/27/2003US20030060627 8-Phenyl-6, 9-dihydro-[1,2,4] triazolo[3,4-i]purin-5-one derivatives
03/27/2003US20030060476 Method and compositions for the synthesis of dioxolane nucleosides with beta-configuration
03/27/2003US20030056712 Production method of famciclovir and production and crystallization method of intermediate therefor
03/27/2003CA2465978A1 Inhibitors of histone deacetylase
03/27/2003CA2460151A1 Cytokine receptor
03/26/2003EP1294722A2 Methods of synthesis for 9-substituted hypoxanthine derivatives
03/26/2003EP1294707A2 Thiophene derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
03/26/2003EP1294362A1 Novel process for preparing crystalline particles
03/26/2003EP0606248B1 Heteroaryl amines as novel acetyl cholinesterase inhibitors
03/26/2003CN1103593C Synergistic composition
03/20/2003WO2003022845A1 Pyrazolo-pyridines for the treatment of herpes infections
03/20/2003WO2003022805A2 Heterocycle substituted purines as antiproliferative agents
03/20/2003WO2003022284A1 Methods of treating pulmonary disease
03/20/2003WO2003022274A2 2-aroylimidazole compounds for treating cancer
03/20/2003WO2003022219A2 Biarylamino purine antiproliferative agents
03/20/2003WO2003022216A2 Biaryl substituted purine derivatives as potent antiproliferative agents
03/20/2003WO2003022214A2 Piperazine and homopiperazine compounds
03/20/2003WO2003022209A2 Crystalline forms of valacyclovir hydrochloride
03/20/2003US20030055068 Pyrazole compounds useful as protein kinase inhibitors
03/20/2003US20030055044 Administering pyrazole derivative for inhibiting GSK-3 or Aurora activity in a patient
03/20/2003US20030055021 Compounds for the treatment of ischemia
03/20/2003US20030054028 Sustained releasing drug in situ
03/20/2003CA2460345A1 2-aroylimidazole compounds for treating cancer
03/20/2003CA2459533A1 Methods of treating pulmonary disease
03/20/2003CA2457835A1 Crystalline forms of valacyclovir hydrochloride
03/19/2003EP1292606A2 Positively-charged peptide nucleic acid analogs with improved properties
03/19/2003EP1292603A2 Methods and compositions for treating hepatitis c virus
03/19/2003EP0874847B1 Novel purine derivatives having, in particular, antiproliferative properties, and biological uses thereof
03/19/2003CN1403457A Prepn process of 2,6-dichloropurine
03/18/2003US6534651 Substituted isoindolinone derivatives
03/18/2003US6534521 Useful in the treatment of inflammation, atherosclerosis, restenosis, and immune disorders such as arthritis and transplant rejection
03/18/2003US6534512 Dideoxycarbocyclic nucleosides
03/18/2003US6534511 The use of certain 6-arylpyrazolo(3,4-d)pyrimidin-4-ones, 2 arylquinazolin-4-ones, 2-arylpurin-6-ones and 2-arylpyrido(3,2- d)pyrimidin-4-ones, or a pharmaceutically acceptable salt thereof, forsexual disorders
03/13/2003WO2003020721A1 Pyrrolo pyrimidines as agents for the inhibition of cystein proteases
03/13/2003WO2003020281A1 Use of compounds for treating conditions resulting from injury to the corneal nerve after lasik and other ocular surgeries or trauma
03/13/2003WO2002094740A3 Hydrogenation processes performed in ionic liquids
03/13/2003WO2002088080A3 Dual inhibitors of pde 7 and pde 4
03/13/2003WO2002087513A3 Fused heterocyclic inhibitors of phosphodiesterase (pde) 7
03/13/2003WO2002040481A3 Adenine based inhibitors of adenylyl cyclase, pharmaceutical compositions and method of use thereof
03/13/2003US20030050275 Partial and full agonists of A1 adenosine receptors
03/13/2003US20030050229 Treatment with a 1' 2' and/or 3' nucleoside or a pharmaceutically acceptable salt or prodrug; nontoxic
03/13/2003CA2455896A1 Use of compounds for treating conditions resulting from injury to the corneal nerve after lasik and other ocular surgeries or trauma
03/12/2003EP1289958A2 BENZOPHENONES AS INHIBITORS OF IL-1$g(b) AND TNF-$g(a)
03/12/2003EP1289561A2 Ligand conjugates and methods for preparing same
03/12/2003EP1036058B1 Adamantane derivatives
03/12/2003EP1019426B1 Novel a1 adenosine receptor agonists and antagonists
03/12/2003CN1402729A Polycycloalkylpurines as adenosine receptor antagonists
03/12/2003CN1402724A Thiazolidinedione derivs. as antidiabetic agents
03/11/2003US6531600 Treatment and compounds
03/06/2003WO2003018745A2 Method of screening for drug hypersensitivity reaction
03/06/2003US20030045533 Phosphodiesterase 4 inhibitors
03/05/2003EP1288215A1 Production method of famciclovir and production and crystallization method of intermediate therefor
03/05/2003EP1287532A2 Method for producing ?18 f]fluoride ion
03/05/2003EP1115719B1 Novel amidine derivatives, their preparation and application as medicines and pharmaceutical compositions containing same
03/05/2003CN1400975A 嘌呤衍生物 Purine derivatives
03/05/2003CN1102593C N-[4(heteroarylmethyl)phenyl]-heteroarylamines compound
03/04/2003US6528515 Beta-2-hydroxymethyl-5-(5-fluorocytosin-1-yl)-1,3-oxathiolane (beta -FTC) and penciclovir
03/04/2003US6528494 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives
02/2003
02/27/2003WO2003016563A2 Novel molecular target for neurotoxicity
02/27/2003WO2003016561A2 Method for the production of cna
02/27/2003WO2003001881A3 Cell-based high-throughput screening methods
02/27/2003US20030040523 Pyrimidine compounds and their use as modulators of chemokine receptor activity
02/27/2003CA2457611A1 Novel molecular target for neurotoxicity
02/26/2003EP1284730A1 Aralkyl ester soft drugs
02/26/2003CN1399636A Adenosine receptor antagonists and methods of making and using the same
02/26/2003CN1399561A Conjugate having cleavable linkage for use in liposome
02/25/2003US6525070 Bipiperidine derivatives as modulators of CCR3 activity and as H1 antagonists
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