Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
08/2005
08/03/2005EP1330455B1 Novel 7-azaindoles, use thereof as phosphodiesterase 4 inhibitors and method for producing the same
08/03/2005EP1228059B1 Novel cyclopropanes as cgrp antagonists, medicaments containing said compounds and method for the production thereof
08/03/2005EP1123293B1 Core-extended perylene bisimides
08/03/2005EP0946550B1 PREPARATION OF [1S-[1a,2b,3b,4a(S*)]]-4-[7-[[1-(3-CHLORO-2-THIENYL)METHYL]PROPYL]AMINO]-3H-IMIDAZO[4,5-b]PYRIDIN-3-yl]-N-ETHYL-2,3-DIHYDROXYCYCLOPENTANECARBOXAMIDE
08/03/2005CN1649886A Electroluminescent materials
08/03/2005CN1649885A Cellular accumulation of phosphonate analogs of HIV protease inhibitor compounds and the compounds as such
08/03/2005CN1649879A Non-steroidal progesterone receptor modulators
08/03/2005CN1649870A 7-aryl-3, 9-diazabicyclo(3.3.1)non-6-ene derivatives and their use as renin inhibitors in the treatment of hypertension, cardiovascular or renal diseases
08/03/2005CN1649869A Azaindoles as inhibitors of c-Jun N-terminal kinases
08/03/2005CN1649868A Process for preparing acid salts of gemifloxacin
08/03/2005CN1649867A Novel 1, 2, 3-substituted indolizine derivatives, inhibitors of FGFs, method for making same and pharmaceutical compositions containing same
08/03/2005CN1649864A Inhibitors of serine proteases, particularly HCV NS3-NS4A protease
08/03/2005CN1649848A Fused pyrimidines derivatives as antagonists of the corticotropin releasing factor (CRF)
08/03/2005CN1649591A Tricyclic compounds useful as HIV reverse transcriptase inhibitors
08/03/2005CN1648128A Aromatic heterocyclic carboxylic derivative, preparing method and use on medicine
08/03/2005CN1648127A Imide sulfo N-hydroxy maleopimarate as light acid producing agent and its synthetic method
08/03/2005CN1648126A Compound and its preparing method and use
08/03/2005CN1213144C Recombination nucleic acid molecule and application thereof
08/03/2005CN1213049C Alkylated imidazopyridine derivatives and medicine containing them and use
08/03/2005CN1213046C Tetrahydropyridine derivatives, their preparation and their use as cell proliferation inhibitors
08/03/2005CN1213044C Amine and amide derivatives as ligands for neuropeptide YY5 receptor useful in treatment of obesity and other disorders
08/03/2005CN1213038C Benzophenones as inhibitors of reverse transcriptase
08/03/2005CN1212839C Use of substituted pyrazoles in preparing medicine for treating allergies
08/02/2005US6924300 Oxyiminoalkanoic acid derivatives
08/02/2005US6924293 Sulfonamide and sulfamide substituted imidazoquinolines
08/02/2005US6924290 Antitumor agents; anticancer agents; sexual disorders; cardiovascular disorders
08/02/2005US6924287 Respiratory syncytial virus replication inhibitors
08/02/2005US6924284 PARP inhibitors
08/02/2005US6924282 5-(1,1-dioxido-1,2-thiazinan-2-yl)-n-(4-fluorobenzyl)-8-hydrox y-1,6-naphthyridine-7-carboxamide; preventing or treating hiv or aids
08/02/2005US6924280 Dipeptide derivatives
08/02/2005US6924251 herbicides.
08/02/2005CA2446939C Pyridylpyrimidine derivatives as effective compounds against prion diseases
08/02/2005CA2370376C Anhydrous mirtazapine crystals and process for the production thereof
08/02/2005CA2321639C Bicyclo[2.2.1]heptanes and related compounds
08/02/2005CA2243199C Novel 3,4-diaryl thiophenes and analogs thereof having use as antiinflammatory agents
07/2005
07/28/2005WO2005068464A2 Process for preparing tadalafil and its intermediates
07/28/2005WO2005068463A1 Diaza-spiropiperidine derivatives
07/28/2005WO2005068462A1 Diaza-spiropiperidine derivatives as inhibitors of transporter 1 and glycine transporter 2
07/28/2005WO2005068433A1 Benzimidazole derivatives
07/28/2005WO2005068432A1 Malononitrile compound as pesticides
07/28/2005WO2005067932A1 (3-oxo-3, 4-dihydro-quinoxalin-2-yl-amino) -benzamide derivatives and related compound as glycogen phosphorylase inhibitors for the treatment of diabetes and obesity
07/28/2005WO2005067900A2 Azabenzofuran substituted thioureas as inhibitors of viral replication
07/28/2005WO2005067502A2 Alkylamino, arylamino, and sulfonamido cyclopentyl amide modulators of chemokine receptor activity
07/28/2005WO2005054246A3 Amine derivatives having a tyrosine-kinase-inhibiting effect
07/28/2005WO2005054241A3 Phenanthridinium derivatives as dna binding agents
07/28/2005WO2005048948A3 Urea derivatives as kinase modulators
07/28/2005WO2005034866A3 Preparation of 1, 6, 7- trisubstituted azabenzimidazoles as kinase inhibitors
07/28/2005WO2005034838A3 Protease inhibitors
07/28/2005WO2005033102A3 Thiophene-based compounds exhibiting atp-utilizing enzyme inhibitory activity, and compositions, and uses thereof
07/28/2005WO2005033073A3 Spirocyclic heterocyclic derivatives and methods of their use
07/28/2005WO2005016875A3 Geometrically restricted 3-cyclopentylidene-1,3-dihydroindol-2-ones as potent protein kinase inhibitors
07/28/2005WO2004093828A3 Reverse-turn mimetics and method relating thereto
07/28/2005WO2004052891A8 Heterocyclic compounds, preparation method thereof and use of same as medicaments, such as anti-bacterial medicaments and beta-lactamase inhibitors
07/28/2005US20050165236 Process for the preparation of Imiquimod and intermediates thereof
07/28/2005US20050165232 Phenyl substituted imidaopyridines and phenyl substituted benzimidazoles
07/28/2005US20050165089 Compounds, compositions and methods
07/28/2005US20050165074 inhibitors of protein tyrosine kinases, for preventing of cancer, cardiovascular disease, inflammation or multiple sclerosis
07/28/2005US20050165058 Oxybenzamide derivatives useful for inhibiting factor Xa or Vlla
07/28/2005US20050165049 2-(2,2,2-Trifluoro-ethyl)-1,2,3,4-tetrahydro-isoquinoline-6-carboxylic acid quinolin-7-ylamides; treatment of acute, inflammatory and neuropathic pain, dental pain, general headache, migraine, cluster headache, mixed-vascular and non-vascular syndromes, arthritis, gastrointestinal disorders
07/28/2005US20050165048 For prophylaxis and therapy of adverse conditions of the central nervous system, including anxiety, convulsions and cognitive disorders
07/28/2005US20050165040 Beta-carboline hydroxamic acid substituted pyrido 3,4-B indole compounds; 9-(4-fluorobenzyl)-N-hydroxy-9H- beta -carboline-3-carboxamide
07/28/2005US20050165036 Substituted benzofurans and benzothiophenes, methods of making and methods of use as integrin antagonists
07/28/2005US20050165032 Vanilloid receptor ligands and their use in treatments
07/28/2005US20050165031 1-(4-(3-(Pyridin-4-yl)propoxy)phenyl)-3-(5-tert-butylisoxazol-3-yl)urea; inhibits protein tyrosine kinases or a specific kinase or kinase class; for for treating and preventing conditions and diseases such as cancer, hematologic malignancies, cardiovascular disease, inflammation or multiple sclerosis
07/28/2005US20050165024 Urea derivatives as kinase modulators
07/28/2005US20050165022 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses
07/28/2005US20050165016 Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase
07/28/2005US20050165007 Benzimidazoles and analogs thereof as antivirals
07/28/2005US20050165003 Treating Alzheimer's Disease; 4-Chloro-N-(4-hydroxy-3-methoxy-benzyl)-N-(2-oxo-azepan-3-yl)-benzenesulfonamide for example; gamma secretase inhibitors; inhibition of beta-amyloid synthesis with minimal inhibition of Notch Signaling
07/28/2005US20050165000 Pharmaceutical compositions containing an hiv integrase inhibitor and a nonionic surfactant
07/28/2005US20050164990 Piperidinyl prostaglandin e analogs
07/28/2005US20050164883 agronomically tolerable salts, isomers and enantiomers of those compounds, are suitable for use as herbicides
07/28/2005US20050161635 Cycloamide-transition metal complexes and bleach catalysts
07/28/2005DE10360792A1 Spirocyclische Cyclohexan-Derivate Spirocyclic cyclohexane derivatives
07/28/2005CA2553938A1 Diaza-spiropiperidine derivatives as inhibitors of glycine transporter 1 and glycine transporter 2
07/28/2005CA2552403A1 Benzimidazole derivatives
07/28/2005CA2552002A1 Azabenzofuran substituted thioureas as inhibitors of viral replication
07/28/2005CA2551869A1 Alkylamino, arylamino, and sulfonamido cyclopentyl amide modulators of chemokine receptor activity
07/28/2005CA2551639A1 (3-oxo-3, 4-dihydro-quinoxalin-2-yl-amino) -benzamide derivatives and related compound as glycogen phosphorylase inhibitors for the treatment of diabetes and obesity
07/27/2005EP1557416A1 Oxazolidinone-quinolone hybrid antibiotics
07/27/2005EP1557411A1 N-phenyl-(2r,5s)dimethylpiperadine derivative
07/27/2005EP1557410A2 Bacterial gyrase inhibitors and uses thereof
07/27/2005EP1556382A1 3-phenyl substituted pyridoindolone, preparation and therapeutic use thereof
07/27/2005EP1556381A1 Pyrazole amides for treating hiv infections
07/27/2005EP1556380A1 Pyridoindolone derivatives substituted in the 3-position by a heterocyclic group, preparation thereof and application of same in therapeutics
07/27/2005EP1556356A1 Tetrahydroquinoline derivatives as crth2 antagonists
07/27/2005EP1556053A1 Antiinflammation agents
07/27/2005EP1556047A2 Pgd2 receptor antagonists for the treatment of inflammatory diseases
07/27/2005EP1432709B1 1-glyoxlylamide indolizines for treating cancer
07/27/2005EP1379523B1 1,2,3,4-tetrahydroisoquinolines derivatives as urotensin ii receptor antagonists
07/27/2005EP1377573B1 Pyrazolopyridine derivatives
07/27/2005EP1343766B1 Cyclization process step in the making of quinolones and naphthyridines
07/27/2005EP1313736B1 Condensed pyrazindione derivatives as inhibitors of pde5
07/27/2005EP1287004B1 Synthetic process for the manufacture of an ecteinascidin compound
07/27/2005EP1277754B1 Imidazopyridine derivatives
07/27/2005EP1250335B1 Process and intermediates for the preparation of imidazopyridines
07/27/2005EP1107966B1 Oxo-pyridoimidazole-carboxamides: gaba brain receptor ligands
07/27/2005EP0929526B1 Qinoline derivatives inhibiting the effect of growth factors such as vegf
07/27/2005CN1646530A Nitrosated imidazopyridines
07/27/2005CN1646529A Imidazo fused compounds