Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559) |
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09/21/2005 | EP1575493A2 Indole, azaindole and related heterocyclic sulfonylureido piperazine derivatives |
09/21/2005 | EP1575486A2 Method and compositions for identifying anti-hiv therapeutic compounds |
09/21/2005 | EP1299382B1 Composition and antiviral activity of substituted indoleoxoacetic piperazine derivatives |
09/21/2005 | EP1220857B1 Gonadotropin releasing hormone receptor antagonists and their related methods of use |
09/21/2005 | EP1140091B1 Formulations comprising imiquimod or other immune response modifiers for treating cervical dysplasia |
09/21/2005 | EP1137640B1 Cyclic hydrazine derivatives as tnf-alpha inhibitors |
09/21/2005 | CN1671711A Calcitonin gene related peptide receptor antagonists |
09/21/2005 | CN1671707A Novel process for producting imidazo[1, 2-b]pyridazine derivative |
09/21/2005 | CN1671706A Modified pictet-spengler reaction and products prepared therefrom |
09/21/2005 | CN1671705A Ligand and complex for catalytically bleaching a substrate |
09/21/2005 | CN1671704A A method of preparing enantiomers of indole-2, 3-dione-3-oxime derivatives |
09/21/2005 | CN1671700A Substituted alkylamine derivatives and methods of use |
09/21/2005 | CN1671697A Indole, azaindole and related heterocyclic 4-alkenyl piperidine amides |
09/21/2005 | CN1671696A 激酶抑制剂 Kinase inhibitors |
09/21/2005 | CN1671690A Antimicrobial aza-bicyclic derivates, their compositions and uses |
09/21/2005 | CN1671667A Quinoline derivatives and their use as mycobacterial inhibitors |
09/21/2005 | CN1671386A Substituted anilinic piperidines as MCH selective antagonists |
09/21/2005 | CN1219780C Heterocyclic compounds binding chemotactic factor receptor |
09/21/2005 | CN1219511C Method for curing sepsis |
09/20/2005 | US6946478 Compounds |
09/20/2005 | US6946473 4-((4-But-2-ynyloxy-benzenesulfonyl)-methyl-amino)-1,3-dimethy l-1H- pyrazolo(3,4-b)and dericatives; bioavailability; no pharmacokinetic problems; bioselectiveity; rheumatoid arthritis, osteoarthritis, sepsis, AIDS, ulcerative colitis |
09/20/2005 | US6946472 Polycyclic compounds exhibiting anti-tumor activities |
09/20/2005 | US6946463 1,2,5,10-tetrahydropyridazino[4,5-b]quinoline-1,10-diones and their use for the treatment of pain |
09/20/2005 | US6946116 Amyloid plaque aggregation inhibitors and diagnostic imaging agents |
09/20/2005 | CA2188796C Heterocyclylbenzonitriles |
09/20/2005 | CA2125978C Improvements in chemical compounds |
09/20/2005 | CA2119757C New fluoro quinoline carboxylic-3 acid derivatives and their preparation |
09/15/2005 | WO2005085249A1 Fused derivatives of pyrazole |
09/15/2005 | WO2005085248A1 Heteroaryl-fused pyrazolo derivatives |
09/15/2005 | WO2005085245A1 Pyrrolopyridine-2-carboxylic acid hydrazides |
09/15/2005 | WO2005085244A1 3,5-disubstituted 1h-pzrrolo [2,3-b] pyridines as jnk inhibitors |
09/15/2005 | WO2005085231A1 Novel 4-benzimidazol-2-ylpyridazin-3-one derivatives |
09/15/2005 | WO2005085230A1 4-benzimidazol-2-yl-pyridazine-3-one-derivatives, production and use thereof in medicaments |
09/15/2005 | WO2005085228A1 Cycloalkanopyridine derivative |
09/15/2005 | WO2005085225A1 Novel hydroxy-6-heteroarylphenanthridines and their use as pde4 inhibitors |
09/15/2005 | WO2005085214A1 Diaryl-substituted five-membered heterocycle derivative |
09/15/2005 | WO2005085209A1 Basic amine compound and use thereof |
09/15/2005 | WO2005085200A1 Pyridone derivative |
09/15/2005 | WO2005085196A2 Inhibitors of dna methylation in tumor cells |
09/15/2005 | WO2005085194A2 Indole-2-carboxylic acid hydrazides as glycogen phosphorylase inhibitors |
09/15/2005 | WO2005068433A9 Benzimidazole derivatives |
09/15/2005 | WO2005067502A3 Alkylamino, arylamino, and sulfonamido cyclopentyl amide modulators of chemokine receptor activity |
09/15/2005 | WO2005065416A3 Process for the preparation of pyridopyrimidones |
09/15/2005 | WO2005065050A3 Bicyclic compound |
09/15/2005 | WO2005051300A3 Bicyclic inhibitors of mek and methods of use thereof |
09/15/2005 | WO2005049589A3 Heterocyclic compounds for the treatment of hyperlipidemia, diabetes, obesity and similar diseases |
09/15/2005 | WO2005025504A3 Modulators of calcitonin and amylin activity |
09/15/2005 | WO2005009389A3 Anaplastic lymphoma kinase modulators and methods of use |
09/15/2005 | WO2005007672A3 Small molecule toll-like receptor (tlr) antagonists |
09/15/2005 | WO2004073615A8 Deazaflavin compounds and methods of use thereof |
09/15/2005 | WO2004018465A9 Benzonaphthyridines with pde 3/4 inhibiting activity |
09/15/2005 | US20050203300 6-Alkoxy-pyrido-pyrimidines |
09/15/2005 | US20050203156 Hydantoins having RNase modulatory activity |
09/15/2005 | US20050203146 P2Y1 Purinoreceptor; thromboembolic disorders; compounds are 2-((hetero)arylamino) benzimidazoles, benzoxazoles or benzothiazoles such as [2-(2-tert-butyl-phenoxy)-pyridin-3-yl]-(6-methyl-1H-benzoimidazol-2-yl)-amine |
09/15/2005 | US20050203128 Antiinflammatory agents; antiallergens; antiproliferative agents; 4-(5-Fluoro-2-hydroxy-phenyl)-2-hydroxy-4-methyl-2-trifluoromethyl-pentanoic acid (3,5-dichloro-phenyl)-amide |
09/15/2005 | US20050203126 Inhibitors of basic fibroblast growth factors (FGFs); treating cancer, rheumatoid arthritis, inflammatory bowel disease, cardiovascular disorders, diabetic retinopathy, achondroplasia, hypochondoplasia, or thanathophoric dysplasia |
09/15/2005 | US20050203124 Compounds for the sustained reduction of body weight |
09/15/2005 | US20050203119 Dihydropyridine compounds for treating or preventing metabolic disorders |
09/15/2005 | US20050203118 Rheumatic diseases; antiarthritic agents; multiple sclerosis; antidiabetic agents; asthma therapy; skin disorders |
09/15/2005 | US20050203110 KINESIN SPINDLE PROTEIN INHIBITOR; ANTIPROLIFERATIVE AGENTS; ANTICANCER AGENTS; 4-(2,5-DIFLUOROPHENYL)-n-3 -FLUOROPYRROLIDIN-3-YL-2-HYDROXYMETHYL-2-PHENYL-2,5-DIHYDRO-1n-PYRROL-1-CARBOXAMIDE |
09/15/2005 | US20050203109 Novel Compounds |
09/15/2005 | US20050203101 Benzimidazole quinolinones and uses thereof |
09/15/2005 | US20050203094 Thromboembolic disorders; anticoagulants; e.g. 2-[5'-fluoro-2,2'-dihydroxy-5-(2-oxo-tetrahydro-furan-3-yl)-biphenyl-3-yl]-1H-benzoimidazole-5-carboxamidine |
09/15/2005 | US20050203091 Heteroaryl-fused pyrazolo derivatives and methods for using the same |
09/15/2005 | US20050203084 Protease inhibitors |
09/15/2005 | US20050203080 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds |
09/15/2005 | US20050203078 Inhibitors of factor Xa or related serine proteases; thrombosis; benzamide derivatives with benzimidazole, indole or imidazo(1,2-a)pyridine rings; e.g. 4-(azepan-2-on-1-yl)-N-[(1R)-1-(5-chloro-1H-benzimidazol-2-yl)-2-methoxy-ethyl]-3-methyl-benzamide |
09/15/2005 | US20050202076 Stabilization, homogenizing, sterile filtration, dehydration, reconstitution, ultrafiltration; storage stability; taxanes |
09/15/2005 | DE102004010207A1 New 4-benzimidazolyl-3(2H)-pyridazinone derivatives are kinase inhibitors, especially useful for treatment of cancer |
09/15/2005 | DE102004004972B3 Heterocyclisch substituierte 7-Amino-4-chinolon-3-carbonsäure-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Heterocyclic-substituted 7-amino-4-quinolone-3-carboxylic acid derivatives, to processes for their preparation and their use as medicaments |
09/15/2005 | DE102004004971B3 Cycloalkyl substituierte 7-Amino-4-chinolon-3-carbonsäure-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arnzeimittel Cycloalkyl substituted 7-amino-4-quinolone-3-carboxylic acid derivatives, to processes for their preparation and their use as Arnzeimittel |
09/15/2005 | CA2820541A1 Caspase inhibitors and uses thereof |
09/15/2005 | CA2558600A1 A substituted-trialkyl amine compound with anti-viral activity based on antagonism against a chemokine receptor cxcr4 |
09/15/2005 | CA2558278A1 Diaryl-substituted five-membered heterocycle derivative |
09/15/2005 | CA2558274A1 Cycloalkanopyridine derivative |
09/15/2005 | CA2558109A1 Heteroaryl-fused pyrazolo derivatives |
09/15/2005 | CA2557581A1 Inhibitors of dna methylation in tumor cells |
09/15/2005 | CA2557575A1 Fused derivatives of pyrazole |
09/15/2005 | CA2555161A1 Novel 4-benzimidazol-2-yl-pyridazin-3-one derivatives |
09/14/2005 | EP1574499A1 Inhibitors of DNA methylation in tumor cells |
09/14/2005 | EP1572693A1 Mitogen activated protein kinase-activated protein kinase-2 inhibiting compounds |
09/14/2005 | EP1572692A1 Enantiomer (-) of tenatoprazole and the therapeutic use thereof |
09/14/2005 | EP1572691A1 Pyrazole compounds as integrin receptor antagonists derivatives |
09/14/2005 | EP1572690A1 Thiazole compounds as integrin receptor antagonists derivatives |
09/14/2005 | EP1572689A1 Tetracyclic immunomodulatory compounds |
09/14/2005 | EP1572682A2 Acyclic pyrazole compounds for the inhibition of mitogen activated protein kinase-activated protein kinase-2 |
09/14/2005 | EP1572678A2 Substituted n-phenyl sulfonamide bradykinin antagonists |
09/14/2005 | EP1572662A1 Pyrazole and imidazole compounds and uses thereof |
09/14/2005 | EP1572659A2 The use of 4-phenyl substituted tetrahydroisoquinolines in the treatment of pain, migraine and urinary incontinence |
09/14/2005 | EP1572657A1 Processes for preparing quinolonecarboxylate derivatives |
09/14/2005 | EP1572239A1 Method of using a cox-2 inhibitor and a topoisomerase ii inhibitor as a combination therapy in the treatment of neoplasia |
09/14/2005 | EP1572215A1 Benzo[d]azepine derivatives for the treatment of neurological disorders |
09/14/2005 | EP1572209A1 Novel quinoxalinone derivatives as bradykinin b1 antagonists |
09/14/2005 | EP1572113A2 Calcium receptor modulating compound and use thereof |
09/14/2005 | EP1341781B1 Antimicrobial quinolones |
09/14/2005 | EP1283825B1 N-substituted peptidyl nitriles as cysteine cathepsin inhibitors |
09/14/2005 | EP1259509B1 Process for the preparation of 6-methyl-2-(4-methyl-phenyl)-imidazo 1,2-a]pyridine-3-(n,n-dimethyl-acetamide) and intermediates |
09/14/2005 | EP1258250B1 Nerve protective drugs |
09/14/2005 | EP0804437B1 [a]-ANNELATED PYRROLE DERIVATIVES AND PHARMACEUTICAL USES THEREOF |
09/14/2005 | CN1668708A Oxidation process for preparing quinacridone pigments |