Patents
Patents for C07D 463 - Heterocyclic compounds containing 1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula: , e.g. carbacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (613)
09/1996
09/06/1996CA2213812A1 A process for preparing loracarbef monohydrate
09/04/1996EP0730035A1 Improved enzymatic process for producing penicillins and cephalosporins
09/04/1996EP0729959A1 A process for preparing loracarbef monohydrate
09/03/1996CA1338571C 3-(substituted)-1-carba (dethia)-3-cephems and cephalosporins and a process for production therefor
08/1996
08/29/1996CA2167118A1 Enzymatic process for producing penicillins and cephalosporins
08/27/1996US5550231 Loracarbef hydrochloride C1-C3 alcohol solvates and uses thereof
07/1996
07/23/1996US5538964 3-thioheteroaryl 1-carba-1-dethiacephalosporin compounds, compositions and methods of use
06/1996
06/25/1996US5530116 Antimicrobial quinolonyl lactams
06/18/1996US5527792 7-substituted-amino-3-substituted-3-cephem-4-carboxylic acids
06/13/1996WO1996017847A1 Process for the preparation of cephalosporins and analogues
06/11/1996US5525599 7-substituted-amino-3-substituted-3-cephem-4-carboxylic acids
05/1996
05/28/1996US5521307 Methods and compounds for the preparation of carbacephems
03/1996
03/13/1996CN1118349A Oxime derivatives of cephalosporanic structure and compounds for their preparation
02/1996
02/27/1996US5494666 Beta-lactamase inhibitors, antibacterials
02/15/1996WO1996004286A1 Process for making quinolonyl lactam antimicrobials and novel intermediate compounds
02/15/1996WO1996004247A1 Process for making antimicrobial compounds
02/13/1996US5491139 Antimicrobial quinolonyl lactams
01/1996
01/10/1996CN1030657C Method for preparing autibacterial compounds
01/03/1996EP0689540A1 Carbacephalosporin compound, their preparation and use
01/02/1996US5480879 Quinolonecarboxylic acids
11/1995
11/07/1995US5464617 1H-2,6a-diazacyclobut(cd)indene-6-carboxylic acid derivatives, antibiotics
10/1995
10/18/1995EP0677523A1 3-(substituted)-1-carba(dethia)-3-cephems and cephalosporins and a process for production therefor
10/12/1995WO1995026966A1 Cephalosporin antibiotics
10/12/1995CA2186894A1 Cephalosporin antibiotics
10/11/1995CN1029966C Crystalline beta-lactan hydrate
09/1995
09/26/1995US5453504 Bicyclic β-lactams intermediates having a new amino protecting group
09/26/1995US5453503 Azetidinone intermediates to carbacephalosporins and process
09/26/1995US5453502 Intermediates for carbacephalosporins
09/20/1995EP0672656A1 1,3,4 substituted and bicyclic derivatives of 2-azetidinones and processes for preparation thereof
09/17/1995CA2144491A1 1,3,4 substituted and bicyclic derivatives of 2-azetidinones and processes for preparation thereof
09/13/1995EP0671401A1 Beta lactames
09/12/1995CA2143519A1 Beta-lactams
08/1995
08/09/1995CN1106410A Bicyclic beta-lactam/paraben complexes
07/1995
07/18/1995US5434147 Antimicrobial quinolonyl lactam esters
05/1995
05/30/1995US5420269 3-fluorosulfonyloxyceph-3-em compounds
05/10/1995EP0651755A1 Cephalosporins and 1-carba-1-dethia cephalosporins
05/09/1995US5414081 Treating a 1-aza-3-thiabicycloalkane with base and phosphine or phosphite desulfurizing agent, and reacting the product with an active esterifying agent
05/02/1995US5412094 Bicyclic beta-lactam/paraben complexes
04/1995
04/25/1995US5409919 Pharmaceutically acceptable salt of 7B-[2-(5-amino-1,2,4-thio-diazol-3-yl)-2(Z)-metho-xyiminoacetamido]-3-[(imidazo[1,2-b]pyridazinium-1-yl)methyl]-3-cephem-4-carboxylate and composition comprising same
04/12/1995EP0647230A1 Cephalosporins and 1-carba-1-dethia cephalosporins
03/1995
03/29/1995EP0644886A1 3-substituted carbacephems
03/28/1995CA1334971C Intermediate for 1-carba(dethia)cephalosporin
03/28/1995CA1334970C Crystalline .beta.-lactam hydrate
03/21/1995US5399686 Loracarbef isopropanolate and a process for converting loracarbef isopropanolate to loracarbef monohydrate
02/1995
02/28/1995US5393882 Bicyclic β-lactam antibiotics
02/28/1995CA1334590C Crystalline antibiotic intermediate
02/21/1995US5391728 Bicyclic B-lactams intermediates having a new amino protecting group
02/15/1995EP0638574A1 Oxime derivatives of cephalosporanic structure and compounds for their preparation
02/10/1995CA2128557A1 Oxime derivatives of cephalosporanic structure and compounds for their preparation
02/08/1995EP0637587A1 Bicyclic beta-lactam/paraben complexes
02/07/1995US5387748 Antimicrobial dithiocarbamoyl quinolones
01/1995
01/25/1995CN1097755A Process for preparing crystalline beta-lactam monohydrate
01/25/1995CN1097754A Process for converting loracarbef dihydrate to loracarbef monohydrate
12/1994
12/29/1994CA2126401A1 Bicyclic beta-lactam/paraben complexes
12/21/1994EP0629625A1 Loracarbef hydrochloride C1-C3 alcohol solvates and uses thereof
12/20/1994US5374719 Process for converting loracarbef dihydrate to loracarbef monohydrate
12/16/1994CA2466974A1 Loracarbef hydrochloride c1-c3 alcohol solvates and uses thereof
12/16/1994CA2466964A1 Loracarbef hydrochloride c1-c3 alcohol solvates and uses thereof
12/16/1994CA2125762A1 Loracarbef hydrochloride c1-c3 alcohol solvates and uses thereof
12/07/1994EP0627431A1 Process for preparing crystalline loracarbef monohydrate
12/07/1994EP0627430A1 Process for converting loracarbef dihydrate to loracarbef monohydrate
12/07/1994EP0627429A1 Loracarbef isopropanolate and a process for converting loracarbef isopropanolate to loracarbef monohydrate
12/05/1994CA2125000A1 Process for preparing crystalline beta-lactam monohydrate
11/1994
11/08/1994US5362724 Antibiotics as bactericides
10/1994
10/05/1994CN1093089A Cephalosporin salts and process for the preparation thereof
10/04/1994US5352782 By steaming
09/1994
09/29/1994WO1994021633A1 Carbacephalosporin compound, their preparation and use
09/20/1994US5348951 Cephalosporins
08/1994
08/10/1994CN1025620C Process for 1-carba(dethia) cephalosporins
08/03/1994CN1090285A Quinolonecarboxylic acids
07/1994
07/12/1994US5328908 Antimicrobial quinolone thioureas
07/06/1994CN1025333C Method for preparing solvates of beta-lactam antibiotic
06/1994
06/29/1994EP0603755A2 Cephalosporin salts and processes for their preparation
06/25/1994CA2112196A1 Cephalosporin salts and process for the preparation thereof
05/1994
05/03/1994CA1329198C .beta.-lactam antibiotics, processes for their preparation and their useas and in medicaments
04/1994
04/27/1994EP0593457A1 Antimicrobial quinolone thioureas
04/13/1994EP0591808A1 Quinolonecarboxylic acids
04/12/1994US5302711 Deesterification of the blocked 3- or 4-carboxylate derivative of cepham or penam with lithium iodide in a nonbasic solvent having a dielectric constant of between 0 and 15
04/10/1994CA2107812A1 Quinolone carboxylic acids
02/1994
02/03/1994WO1994002489A1 Cephalosporins and 1-carba-1-dethia cephalosporins
02/01/1994US5283329 Chemical intermediate for biosynthesis of antibiotics
01/1994
01/25/1994US5281703 Process for making antimicrobial quinolonyl lactams
01/06/1994WO1994000457A1 Alphalosporins and 1-carba-1-dethia cephalosporins
01/04/1994US5275816 Cephalosporin derivatives
12/1993
12/28/1993US5273973 Antimicrobial quinolonyl esters
12/23/1993WO1993025551A1 3-substituted carbacephems
12/22/1993EP0574940A1 Method for removing the protecting group for carboxyl group
12/21/1993US5272265 3-(substituted or unsubstituted) thiazolo-1-carba (1-dethia)cephems
11/1993
11/09/1993US5260438 With fluorine compound
11/03/1993EP0567949A1 Method for removing the protecting group for hydroxy group
10/1993
10/19/1993US5254679 Containing a quaternized nitrogen
10/06/1993EP0564129A2 Process for the preparation of 3-substituted-2-azetidinones
10/05/1993US5250676 Reacting a 1-protected azetidione with a salt having a nucleophilic base and a conjugate acid with a specific dissociation constant; stereoselective
09/1993
09/24/1993CA2091977A1 Process for the preparation of 3-substituted-2-azetidinones
09/21/1993US5246926 Cephalosporin derivatives
09/21/1993CA1322368C Fused heteroalkylene quinolinamines, a process and intermediates for their preparation and their use as medicaments
09/14/1993US5245027 Antibiotics
09/08/1993EP0559533A1 Process for preparing beta-lactam derivative and synthetic intermediate thereof
09/07/1993CA2085540A1 Process for preparing beta-lactam derivative and synthetic intermediate the reof
09/01/1993EP0558215A1 Novel methods and compounds for the preparation of carbacephems
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