Patents
Patents for C07D 455 - Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine (2,122)
05/2001
05/16/2001EP1098896A1 5-bicycloindole compounds
05/16/2001EP1098650A1 Benzoquinolizidine and benzoindolizidine derivatives and therapeutic uses thereof
05/16/2001EP1098644A1 Substituted benzimidazole antiviral agents
05/16/2001CN1295573A Pharmaceutically available protoberberine salt derivatives, and protoberberine derivatives and salt thereof
05/09/2001EP1097138A1 Pharmaceutical compositions comprising 2-quinolones
04/2001
04/26/2001WO2001029035A1 4-oxoquinolizine antimicrobials having 2-pyridone skeletons as the partial structure
04/26/2001WO2000008020A8 Tricyclic carboxamides
04/17/2001US6218426 For therapy of mammalian reproductive disorders and steroid hormone-dependent tumors as well as for regulating fertility, where suppression of gonadotropin release is indicated
04/11/2001EP1089993A1 5-ht 1f? agonists
03/2001
03/22/2001WO2000068229A3 (s)-benzoquinolizine carboxylic acids and their use as antibacterial agents
02/2001
02/28/2001CN1285354A Thalictrum acutifolium thalicrine having anti-tumour phological activity and extration method thereof
02/21/2001CN1284954A Benzo[c]quinolizine derivatives and their use as 5 alpha-reductases inhibitors
02/13/2001US6187786 Antitumor and anticarcinogenic agents
02/13/2001CA2001203C Novel antimicrobial dithiocarbamoyl quinolones
02/07/2001EP1073655A1 Pharmaceutically available protoberberine salts derivatives, and protoberberine derivatives and salts thereof
02/07/2001CN1283197A Pleuromutilin derivatives as antimicrobials
01/2001
01/24/2001EP1070711A2 Heteroaryl-substituted pyrrole derivatives, their preparation and their therapeutic uses
01/21/2001CA2314373A1 Heteroaryl-substituted pyrrole derivatives, their preparation and their thereapeutic uses
01/17/2001EP1068178A1 NON-PEPTIDE GnRH AGENTS
01/10/2001EP1066284A1 Benzo c]quinolizine derivatives and their use as 5 alpha-reductases inhibitors
01/03/2001EP1065203A2 Heterocyclic compounds as retinoic acid receptor antagonists
01/03/2001EP1064284A1 Hypnotic beta-carboline derivatives, process for their preparation and their use as medicinal products
01/02/2001CA1341161C Quinolone- and naphthyridone carboxylic acid derivatives, process for their production, antibacterial compositions and feed additives containing them
12/2000
12/27/2000CN1278260A Aminomethyl-benzo [a] quinolizidine derivatives, prepns. and therapeutic applications for neurodegenrative diseases
12/19/2000CA2001225C Antimicrobial lactam-quinolones
12/13/2000CN1276370A Process for preparing anticancer compound, and intermediate
12/13/2000CN1059442C Use of 1,2-bridged 1,4-dihydropyridines as medicaments
11/2000
11/16/2000WO2000068229A2 (s)-benzoquinolizine carboxylic acids and their use as antibacterial agents
11/14/2000US6147087 Use of 1,2-Bridged 1,4-dihydropyridines as medicaments
11/09/2000WO2000066522A1 Glucocorticoid receptor modulators
11/09/2000WO2000042045A3 Functionalized heterocycles as chemokine receptor modulators
11/09/2000CA2372173A1 Glucocorticoid receptor modulators
11/02/2000EP1047690A1 Heterocyclic ether and thioether compounds useful in controlling chemical synaptic transmission
11/01/2000CN1058009C 8-oxy-5,8-dihydro-6H-dibenzo [a,g] quinolizine -13-propionic acid derivant, its preparation method and medicinal use thereof
10/2000
10/24/2000US6136806 Remedy for rosacea
10/18/2000EP1044969A2 Processes and intermediates for preparing anti-cancer compounds
10/17/2000US6133290 Derivatives of 3-piperidin-4-yl-1h-indazolines; inhibit peptide extravasation due to stimulation of the trigeminal ganglia; treatment of migraines and associated disorders
10/17/2000US6133283 Mono- or polyenic carboxylic acid derivatives
09/2000
09/19/2000US6121281 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
08/2000
08/23/2000EP1028961A1 Pleuromutilin derivatives as antimicrobials
08/16/2000EP1027350A1 Aminomethyl-benzo a]quinolizidine derivatives, preparation and therapeutic applications for neurodegenrative diseases
08/10/2000WO2000046223A1 Tricyclic quinolonecarboxylic acid derivatives or salts thereof
08/02/2000EP0527889B1 Quinolizinone type compounds
08/01/2000US6096246 Photochromic naphthopyrans, compositions and articles containing them
07/2000
07/20/2000WO2000042045A2 Functionalized heterocycles as chemokine receptor modulators
07/20/2000CA2372197A1 Functionalized heterocycles as chemokine receptor modulators
07/13/2000WO2000008020A3 Tricyclic carboxamides
06/2000
06/29/2000WO2000037468A1 DIBENZO[a,g]QUINOLIZINIUM DERIVATIVES AND THE SALTS THEREOF
06/29/2000CA2355469A1 Dibenzo[a,g]quinolizinium derivatives and the salts thereof
06/07/2000CN1053188C Quinolizinone type compounds
05/2000
05/31/2000EP1003735A1 Quinolizine carboxylic acid derivatives
05/17/2000EP0999747A1 Use of benzo c]quinolizine derivatives as plant growth regulators
05/03/2000EP0997466A1 Novel antimicrobial lactam-quinolones
04/2000
04/06/2000WO2000006173A8 5-ht1f agonists
04/05/2000CN1249753A Farnesyl transferase inhibiting 1,8-annelated quinolinone derivs. substd. with N- or C-linked imidazoles
04/04/2000CA2107432C Quaternary basic amides, method of preparing them and pharmaceutical compositions in which they are present
03/2000
03/30/2000WO2000017197A1 Quinolizinones as integrin inhibitors
03/22/2000CN1248256A Process for preparation of 4H-4-oxo-quinolizine-3-carboxylic acid derivatives
02/2000
02/29/2000US6030984 7-(4-phenoxyphenyl)-6-oxoquinolizines and derivatives of tricyclic ring analogues, particularly 7-oxothieno-(2,3-a)quinolizine; inhibiting beta-amyloid peptide activity
02/29/2000US6030979 Pharmaceutical composition comprising 5,6-dihydrodibenzo[A,G] Quinolizinium derivatives and the salts thereof
02/29/2000US6030978 Exhibit fungicidal effect or growth-inhibitory effect against fungi including cutaneous filamentous fungus, such as epidermophyton, microsporum, trichophyton, sporothrix schenckii, aspergillus or candida; nontoxicity;
02/29/2000US6030964 Binds to retinoic acid receptors and useful for treating psoriasis, autoimmune diseases, tumors, rheumatoid arthritis and for inducing immunosuppression in organ transplantation
02/22/2000US6028197 Dibenzo[a,g]quinolizinium derivatives and the salts thereof
02/17/2000WO2000008022A1 Urea derivatives
02/17/2000WO2000008020A2 Tricyclic carboxamides
02/17/2000WO2000008019A1 Process for the synthesis of (1h)-benzo[c]quinolizin-3-ones derivatives
02/17/2000CA2339362A1 Tricyclic carboxamides
02/10/2000WO2000006572A1 Bensoquinolizine derivatives and process for producing the same
02/10/2000WO2000006173A1 5-ht1f agonists
02/09/2000EP0978514A1 Indazole derivatives as 5-HT1F agonists
02/03/2000WO2000004905A1 Benzoquinolizidine and benzoindolizidine derivatives and therapeutic uses thereof
02/03/2000WO2000004900A1 Substituted benzimidazole antiviral agents
02/03/2000CA2338222A1 Benzoquinolizidine and benzoindolizidine derivatives and therapeutic uses thereof
02/03/2000CA2338147A1 Substituted benzimidazole antiviral agents
02/01/2000US6020368 Microbiocides
01/2000
01/27/2000WO2000004019A1 5-bicycloindole compounds
01/27/2000WO2000003990A1 Pharmaceutical compositions comprising 2-quinolones
01/27/2000CA2343748A1 5-bicycloindole compounds
01/27/2000CA2337115A1 Pharmaceutical compositions comprising 2-quinolones
01/19/2000EP0971919A1 Process for preparation of 4h-4-oxo-quinolizine-3-carboxylic acid derivatives
01/19/2000CN1242011A Tricyclic amine derivatives
01/06/2000WO2000000487A1 5-ht1f agonists
01/06/2000CA2336254A1 5-ht1f agonists
12/1999
12/28/1999US6008356 Pharmaceutically available protoberberine salts derivatives, and protoberberine salts derivatives, and protoberberine derivatives and salts thereof
11/1999
11/23/1999US5990121 Use of 1,2-bridged 1,4-dihydropyridines as medicaments
11/04/1999WO1999055704A1 Pharmaceutically available protoberberine salts derivatives, and protoberberine derivatives and salts thereof
11/04/1999CA2329434A1 Pharmaceutically available protoberberine salts derivatives, and protoberberine derivatives and salts thereof
11/02/1999US5977125 Mono-or polyenic carboxylic acid derivatives
10/1999
10/13/1999CN1231665A Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
10/06/1999EP0947513A1 Tricyclic amine derivatives
09/1999
09/23/1999WO1999047521A1 HYPNOTIC β-CARBOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINAL PRODUCTS
09/23/1999CA2324270A1 Hypnotic .beta.-carboline derivatives, process for their preparation and their use as medicinal products
09/21/1999US5955470 Derivatives of amide analogs of certain methano bridged quinolizines
09/15/1999EP0641339B1 Azaspiro quinolone antibacterial agents
09/10/1999WO1999044987A1 NON-PEPTIDE GnRH AGENTS
09/10/1999CA2322444A1 Non-peptide gnrh agents
08/1999
08/25/1999EP0937044A1 Cftr channel activator compounds and pharmaceutical compositions containing same
08/25/1999EP0920645A4 Naphthopyrans, compositions and articles containing them
08/24/1999US5942532 Inhibitors of histidine protein kinase; bacteria resistant to other antibiotics
08/11/1999EP0934316A1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
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