Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
04/1999
04/22/1999CA2305141A1 Novel combination
04/22/1999CA2304979A1 Pyrazole derivatives having a calcium release-activated calcium channel inhibitory effect
04/21/1999EP0633261B1 Quinoline-3-acetic acid derivative, process for producing the same, and use thereof
04/21/1999CN1214685A Inhibitors of farnesyl protein transferase
04/21/1999CN1214339A Pyrazole derivatives, their preparation and their use in pharmaceuticals
04/21/1999CN1043041C Ethers derivatives containing heterocyclic radical and insecticide using the same as active composition
04/15/1999WO1999018102A1 Fungicidal and arthropodicidal cyclic amides
04/15/1999WO1999018099A1 Aryl thiophene derivatives as pde iv inhibitors
04/15/1999WO1999018095A1 Aryl furan derivatives as pde iv inhibitors
04/15/1999WO1999018091A1 Novel compounds useful as neuro-protective agents
04/15/1999WO1999018081A1 Substituted fused heterocyclic compounds
04/15/1999WO1999018077A1 Fused pyridine derivatives
04/15/1999WO1999018074A1 Novel lactam metalloprotease inhibitors
04/15/1999WO1999018073A1 Azetidinone derivatives for the treatment of hcmv infections
04/15/1999WO1999018072A1 Azetidinone derivatives for the treatment of hcmv infections
04/15/1999WO1999017775A1 QUINOLINE-CONTAINING α-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS
04/15/1999WO1999009025A3 2-(4-aryl or heteroaryl-piperazin-1-ylmethyl)-1h-indole derivatives interacting with the dopamine d4 receptor
04/15/1999WO1999000399A9 Method of producing tiazofurin and other c-nucleosides
04/15/1999CA2305679A1 Novel lactam metalloprotease inhibitors
04/15/1999CA2305538A1 Novel compounds useful as neuro-protective agents
04/15/1999CA2305414A1 Aryl thiophene derivatives as pde iv inhibitors
04/15/1999CA2305413A1 Aryl furan derivatives as pde iv inhibitors
04/14/1999EP0908457A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents
04/14/1999EP0908456A1 Pyrazole derivatives, their preparation and their use in drugs
04/14/1999EP0908454A2 Oxazoles, thiazoles, oxazolines, oxadiazoles and benzoxazoles useful as neuro-protective agents
04/14/1999EP0908453A1 Water-soluble tetrazolium salt compounds
04/14/1999EP0907650A1 N- 4-(heteroarylmethyl)phenyl]-heteroarylamines
04/14/1999EP0907640A1 Substituted n-(4-pyridyl)-thioamides with pesticide activity
04/14/1999EP0810991B1 1-aryl-2-acylamino-ethane compounds and their use as neurokinin especially neurokinin 1 antagonists
04/14/1999CN1214041A Sulfonated amino acid derivatives and metalloproteinase inhibitors contg. same
04/14/1999CN1214039A Carbamoyloxy derivatives of mutiline and their use as antibacterials
04/14/1999CN1042936C Substituted aminoquinolone compound, its application and medicinal compsns. containing same
04/13/1999CA2155236C Gas phase polymerization process
04/13/1999CA2045553C Process for the preparation of vinyl ethers
04/13/1999CA1340499C Thiazolyl derivatives useful as interediates for the preparation of cephem or cepham compounds
04/08/1999WO1999016755A1 Novel angiogenesis inhibitors
04/08/1999WO1999003823A3 Novel polyamine analogues as therapeutic and diagnostic agents
04/08/1999WO1998054161A9 Oxazolidinone antibacterial agents having a thiocarbonyl functionality
04/08/1999CA2303830A1 Novel angiogenesis inhibitors
04/07/1999EP0906370A1 Pyridone colorants
04/07/1999EP0906297A1 1,2,4-benzothiadiazine derivatives, their preparation and use
04/07/1999EP0906296A1 Process for the preparation of chiral keto-heterocycles of basic amino acids
04/07/1999EP0906294A1 Benzoxazinone dopamine d4 receptor antagonists
04/07/1999EP0906094A1 Substituted n- (aminoiminomethyl or aminomethyl)phenyl]propyl amides
04/07/1999EP0877026A4 Substituted 6-r-1,3,4-thiadiazine-2-amines, the use thereof as anaesthetising, cardiovascular and hypometabolic agents, and a pharmaceutical composition containing them
04/07/1999EP0683776B1 Substituted heteroarylalkylthiopyridines for controlling helicobacter bacteria
04/07/1999EP0659181B1 Sulfonamide inhibitors of hiv-aspartyl protease
04/07/1999EP0607374B1 Novel cyclic lipid derivatives as potent paf antagonists
04/07/1999CN1213369A Quinoxalinediones
04/07/1999CN1212964A Sulfonic acid amide substituted benzodihydropyrane processes for their preparation, their use as medicament and pharmaceutical preparations comprising them
04/06/1999US5892052 Process for making retroviral protease inhibiting compounds
04/06/1999US5892046 Methine and azamethine dyes based on trifluoromethylpyridones
04/06/1999US5892039 Piperazino derivatives as neurokinin antagonists
04/06/1999US5891897 Oxopropionitrile derivative and vermin controlling agent
04/06/1999US5891894 2-amino oxazole derivatives; antagonists of platelet activating factor useful in treatment of asthma, inflammation, cardiovascular disorders, renal diseases, or as contraceptives
04/06/1999US5891893 5-amino-1,2,4-oxa(or thia)diazoles; antagonists of platelet activating factor useful in treatment of asthma, allergies, inflammation, cardiovascular diseases, renal diseases, or as contraceptives
04/06/1999US5891892 Small molecule biaryl compounds as inhibitors of endothelin converting enzyme
04/06/1999US5891852 Serine protease inhibitors-cycloheptane derivatives
04/06/1999US5891626 Enzyme-linked analysis; using surfactant
04/01/1999WO1999015525A1 Carboxamidothiazole derivatives, preparation, pharmaceutical compositions containing them
04/01/1999WO1999015524A1 Thiazole derivatives
04/01/1999WO1999015523A1 Bisethers of 1-oxa, aza and thianaphthalen-2-ones as phospholamban inhibitors
04/01/1999WO1999015504A1 4-phenyltetrahydrochinoline utilized as an inhibitor of the cholesterol ester transfer protein
04/01/1999WO1999015500A1 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
04/01/1999WO1999014998A2 Method for preventing and treating hearing loss using sensorineurotrophic compounds
04/01/1999WO1998056812A3 Estrogen receptor crystals and ligands
04/01/1999CA2304849A1 Bisethers of 1-oxa, aza and thianaphthalen-2-ones as phospholamban inhibitors
04/01/1999CA2304647A1 Method for preventing and treating hearing loss using sensorineurotophic compounds
04/01/1999CA2304397A1 Carboxamidothiazole derivatives, preparation, pharmaceutical compositions containing them
04/01/1999CA2302572A1 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
03/1999
03/31/1999EP0905255A2 Process for the preparation of pharmaceutically active thiazolidine or oxazolidine compounds by a yeast reductase
03/31/1999EP0905134A1 Piperidine derivatives as LTD4 and H1 antagonists
03/31/1999EP0905131A1 Sulfonamid-substituted chromans, process for their preparation, their use as medicine, and pharmaceutical preparation containing them
03/31/1999EP0904273A1 Mesylate trihydrate salt of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)ethyl)-6-chloro-1,3-dihydro-2(1h)-indol-2-one (=ziprasidone), its preparation and its use as dopamine d2 antagonist
03/31/1999EP0904269A1 3,4-diaryl-2-hydroxy-2,5-dihydrofurans as prodrugs to cox-2 inhibitors
03/31/1999EP0904262A1 Conformationally restricted aromatic inhibitors of microsomal triglyceride transfer protein and method
03/31/1999EP0904076A1 Inhibitors of farnesyl-protein transferase
03/31/1999EP0637298B1 Substituted cyclohexene-1,2-bicarboxylic acid derivatives and raw materials for producing them
03/31/1999CN1212705A Serine protease inhibitors
03/31/1999CN1212692A Substituted A2a-and diazacycloheptane and cyclooctane compounds and their use
03/30/1999US5889163 Method for producing azo dye compounds
03/30/1999US5889036 Prophylactic or therapeutic drug for renal diseases
03/30/1999US5889035 1-(Arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-3-(heteroaryl) pyrrolidines and related compounds useful as antipsychotics and analgesics
03/30/1999US5889032 Heterocyclic compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them
03/30/1999US5889025 Antidiabetic compounds having hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them
03/30/1999US5889009 Method of inhibiting cell adhesion
03/30/1999US5889004 4-heteroaryl-1-piperazinealkylthiols and derivatives thereof and their therapeutic utility
03/30/1999US5888998 Increase effectiveness of b-lactam antibiotics
03/30/1999US5888941 Carbozamides with antifungal activity
03/30/1999US5888940 Desiccating plants
03/30/1999US5888422 Fluorinated phenanthrene derivatives and their use in liquid-crystal mixtures
03/26/1999CA2249074A1 Sulfonamide-substituted chromans, processes for their preparation, their use as a medicament, and pharmaceutical preparations comprising them
03/25/1999WO1999014216A1 Substituted 3(-1,2-benzisothiazol or isoxazol-5 yl)-substituted pyrimidine as herbicides
03/25/1999WO1999014210A1 Process for the preparation of substituted 5,6-dihydro-2h-pyran-2-ones
03/25/1999WO1998051665A3 Novel macrocyclic compounds as metalloprotease inhibitors
03/25/1999DE19741399A1 New tetrahydroquinoline derivatives useful in treatment of elevated lipid levels and arteriosclerosis
03/24/1999EP0903348A1 Epothilone derivatives, preparation and utilization
03/24/1999EP0903346A1 Sydnone imine derivatives
03/24/1999EP0667855B1 Substituted arylalkynyl- and heteroarylalkynyl-n-hydroxyurea inhibitors of leukotriene biosynthesis
03/24/1999EP0640595B1 Substituted tertiary amino compound or salt thereof