Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
05/1999
05/20/1999CA2309331A1 Agent acting on retinoid receptor
05/20/1999CA2309319A1 Benzothiazole protein tyrosine kinase inhibitors
05/20/1999CA2309177A1 Pyrimidinone compounds and pharmaceutical compositions containing them
05/20/1999CA2308716A1 Urea derivatives and their use as integrin inhibitors
05/19/1999EP0916668A1 Chemokine receptor antagonists
05/19/1999EP0916667A1 Optically active 1,4-dihydropyridine derivatives and process for the preparation thereof
05/19/1999EP0916666A1 3-alkyloxy-,aryloxy-, or arylalkyloxy-benzo[b]thiophene-2-carboxamides as inhibitors of cell adhesion
05/19/1999EP0915868A1 Carbanilides used as pesticides
05/19/1999EP0915858A1 Intermediates for the preparation of 2-imidazoline-5-ones
05/19/1999EP0915847A1 Substituted sulfonamides as selective beta3 agonists for the treatment of diabetes and obesity
05/19/1999EP0915846A2 2- and 2,5-substituted phenylketoenols
05/19/1999CN1216991A Mesylate dihydrate salts of 5-(2-(4-(1,2-benzi sothiazol-3-yl)-1-piperazinyl)-ethyl)-6-chloro-1,3-dihydro-2(1H)-indol-2-one
05/19/1999CN1216990A Mesylate trihydrate salt of 5-(2-(4-(1,2-benzi isothiazol-3-yl)-1-piperazinyl) ethyl)-6-chloro-1,3-dihydro-2(1H)-indol-2-one
05/19/1999CN1216986A Isoxazole derivatives
05/19/1999CN1216982A Nitrogenous tricycle compounds and drugs comprising same
05/19/1999CN1216923A Inclusion complexes of aryl-heterocyclic salts
05/19/1999CN1216762A 2-(arylphenyl) amino-imidazoline derivatives
05/18/1999US5905077 Inhibitors of HIV protease useful for the treatment of AIDS
05/18/1999CA2158952C 2-substituted morpholine and thiomorpholine derivatives as gaba-b antagonists
05/14/1999WO1999023095A1 Process for the preparation of thiazolidinedione derivatives
05/14/1999WO1999023092A2 3-aminoalkylamino-2h-1,4-benzoxa(thia-)zines and pharmaceutical compositions containing them
05/14/1999WO1999023083A1 Novel alkylamino derivatives
05/14/1999WO1999023082A1 AMINOTHIAZOLE DERIVATIVES USEFUL IN THE PREPARATION OF β-LACTAM ANTIBIOTICS
05/14/1999WO1999023079A1 Carbamoylphenylsulfonyl ureas, method for their production and their application as herbicides and plant growth regulators
05/14/1999WO1999022738A1 Compositions of lipid lowering agents
05/14/1999WO1999007692A3 New epothilone derivatives, method for producing same and their pharmaceutical use
05/14/1999WO1999001124A9 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
05/14/1999CA2309461A1 Process for the preparation of thiazolidinedione derivatives
05/14/1999CA2309438A1 Carbamoylphenylsulfonylureas, processes for their preparation and their use as herbicides and plant growth regulators
05/14/1999CA2307905A1 3-aminoalkylamino-2h-1,4-benzoxazines and 3-aminoalkylamino- 2h-1,4-benzothiazines: dopamine receptor subtype specific ligands
05/14/1999CA2307097A1 Compositions of lipid lowering agents
05/12/1999EP0915090A1 Compounds useful as hypoglycemic agents and for treating Alzheimer's disease
05/12/1999EP0915088A1 D-Proline derivatives
05/12/1999EP0914605A1 Molecular model for vla-4 inhibitors
05/12/1999EP0914322A1 New indolyl and benzofuranyl carboxamides as inhibitors of nitric oxide production
05/12/1999EP0914319A1 Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists
05/12/1999EP0914158A2 Pharmaceutical combination containing a compound having angiotensin ii and antagonistic activity
05/12/1999EP0914125A1 Hiv protease inhibitors useful for the treatment of aids
05/12/1999CN1216541A N-3 substituted pyrimidin-4-ones with all antagonistic activity
05/12/1999CN1216540A 2,1,3-benzothia (oxa) diazole derivatives having an endothelin receptor antagonistic effect
05/12/1999CN1216530A Ethylene derivatives and pest controlling agents
05/11/1999US5902813 Modulators of the benzodiaxepine receptor ot the gamma-butyric acid(a) receptor complex; anxiolytic, antiepileptic and -convulsant agents; sleep and memory disorders
05/11/1999CA1340541C Analgesic carboxylic acid amide derivatives
05/06/1999WO1999021845A2 4-aminothiazole derivatives, their preparation and their use as inhibitors of cyclin-dependent kinases
05/06/1999WO1999021844A1 Antirheumatic
05/06/1999WO1999021835A1 QUINOLINE DERIVATIVES AS H+-ATPase INHIBITORS AND AS BONE RESORPTION INHIBITORS
05/06/1999WO1999021834A1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors
05/06/1999EP0913396A2 Sulphonamide substituted benzopyran derivatives, process of preparation, their use as medicines and pharmaceutical compositions containing them
05/06/1999EP0913392A1 Ethylene derivatives and pest controlling agents
05/06/1999EP0912655A1 Liquid crystalline saccharose derivatives
05/06/1999EP0912560A1 Indole derivatives for the treatment of osteoporosis
05/06/1999EP0912553A1 BENZO[g]QUINOLINE DERIVATIVES
05/06/1999EP0912549A1 Compounds and methods for providing pharmacologically active preparations and uses thereof
05/06/1999EP0912547A2 New substituted pyridyl keto enols
05/06/1999EP0912542A1 Oxocoumarin and barbituric acid derivates, their preparation and their use as ligand inhibitors of a corticotropin-releasing factor (crf) and/or a crf-binding protein complex
05/06/1999EP0912519A1 Quinoline sulfonamides as tnf inhibitors and as pde-iv inhibitors
05/06/1999EP0912514A1 Novel sterically hindered piperidine derivatives acting as light stabilisers for polymers
05/06/1999EP0912512A1 Sulphonamide derivatives and their use in the treatment of cns disorders
05/06/1999EP0912504A1 Process to prepare taxol
05/06/1999EP0626068B1 Luminescent lanthanide chelates
05/06/1999DE19749717A1 New epothilone derivatives
05/06/1999DE19748470A1 Carbamoylphenylsulfonylharnstoffe, Verfahren zu ihrer Herstellung und ihre Verwendung als Herbizide und Pflanzenwachstumsregulatoren Carbamoylphenylsulfonylharnstoffe, processes for their preparation and their use as herbicides and plant growth regulators
05/06/1999CA2306914A1 Antirheumatic
05/06/1999CA2306082A1 Substituted 4-amino-thiazol-2-y compounds as cdks inhibitors
05/05/1999CN1216045A N-(2,1,3-benzothia (oxa) diazolyl)-sulphonamides having endothelin receptor antagonistic effect
05/05/1999CN1216043A Substd. benzenesulfonamide derivs as prodrugs of COX-2 inhibitors
05/05/1999CN1216039A Process to prepare taxol
05/04/1999US5900486 Fungicides
05/04/1999US5900427 N-heteroarenesulfonyl-protected amino acid reagents for peptide synthesis
05/03/1999CA2252733A1 Sulfonamide-substituted benzopyran derivatives, processes for their preparation, their use as a medicament, and pharmaceutical preparations comprising them
04/1999
04/29/1999WO1999020618A1 Thiadiazoles amides useful as antiinflammatory agents
04/29/1999WO1999020617A1 Antiinflammatory thiadiazolyl ureas which act as lfa-1 and mac-1 inhibitors
04/29/1999WO1999020616A1 2-substituted 1,2-benzisothiazole derivatives and their use as serotonin antagonists (5-ht1a, 5-ht1b and 5-ht1d)
04/29/1999WO1999020611A1 Imidazole derivatives and their use as farnesyl protein transferase inhibitors
04/29/1999WO1999020110A1 Combination therapy for reducing the risks associated with cardio- and cerebrovascular disease
04/29/1999DE19748928A1 New epothilone derivatives
04/29/1999DE19746612A1 New 2-substituted 1,2-benzisothiazole derivatives
04/29/1999CA2307199A1 2-substituted 1,2-benzisothiazole derivatives and their use as serotonin antagonists (5-ht1a, 5-ht1b and 5-ht1d)
04/29/1999CA2306646A1 Combination therapy for reducing the risks associated with cardio- and cerebrovascular disease
04/28/1999EP0911331A2 Substituted dibenzoxazepine compounds, pharmaceutical compositions and methods of use
04/28/1999EP0911329A1 3-Substituted arylpyrazole derivatives
04/28/1999EP0910566A1 Heterocyclic compounds and their preparation and use
04/28/1999EP0556381B1 N-(4-pyridyl or 4-quinolinyl) arylacetamide pesticides
04/28/1999CN1215401A 4-(benzo-1,3-dioxolyl)-pyrrolidine-3-carboxylic acid derivatives endothelin antagonists
04/28/1999CN1215391A 6-phenylpyridyl-2-amine derivatives
04/28/1999CN1215338A Pharmaceutical combination containing a compound having angiotensin II and antagonisti activity
04/22/1999WO1999019313A1 Novel tricyclic compounds and their use in medicine; process for their preparation and pharmaceutical compositions containing them
04/22/1999WO1999019303A1 Pyrazole derivatives
04/22/1999WO1999019301A1 Piperazine compounds and medicinal use thereof
04/22/1999WO1999019300A1 Prostaglandin agonists and their use to treat bone disorders
04/22/1999WO1999019299A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
04/22/1999WO1999018960A1 Novel combination
04/22/1999WO1999018944A1 Use of thiazolidinediones for the treatment of hyperglycaemia
04/22/1999WO1999018943A1 Use of thiazolidinediones for the treatment of hyperglycaemia
04/22/1999WO1999005114A3 1h-4(5)-substituted imidazole derivatives, their preparation and their use as histamine h3 receptor ligands
04/22/1999WO1999002146A8 Amino acid derivatives
04/22/1999CA2306811A1 Piperazine compounds and medicinal use thereof
04/22/1999CA2306086A1 Use of thiazolidinediones for the treatment of hyperglycaemia
04/22/1999CA2305353A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
04/22/1999CA2305289A1 Use of thiazolidinediones for the treatment of hyperglycaemia