Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
01/1999
01/19/1999US5861427 Substituted 4-biarylbutyric acid derivatives as matrix metalloprotease inhibitors
01/19/1999US5861421 Useful for treating allergic and inflammatory diseases
01/19/1999US5861413 2-oxo- and 2-thio-1,2-dihydroquinolinyl-oxazolidinones
01/19/1999US5861392 Therapeutic heterocycles
01/19/1999US5861380 Oxadiazole, thiadiazole and triazole peptoids as inhibitors of human neutrophil elastase; adult respiratory distress syndrome; antiarthritic,-inflammatory,-ischemic,-tumor and -carcinogenic agents and other hne-mediated conditions
01/19/1999CA2166902C 3-amidopyrazole derivatives, process for preparing these and pharmaceutical compositions containing them
01/19/1999CA2061607C 1-biphenylimidazole derivatives, their preparation and their therapeutic use
01/14/1999WO1999001444A1 Polymorphic form of the tachykinin receptor antagonist 2-(r)-(1-(r) -(3,5-bis(trifluoromethyl) phenyl)ethoxy)-3-(s)-(4-fluoro) phenyl-4-(3-5 (-oxo-1h,4h-1,2,4,-triazolo) methylmorpholine
01/14/1999WO1999001443A1 2-(2-methylphenyl)-oxazolines
01/14/1999WO1999001441A1 Quinazoline analogs and related compounds and methods for treating inflammatory conditions
01/14/1999WO1999001128A1 Certain diarylimidazole derivatives; a new class of npy specific ligands
01/14/1999WO1999001127A1 Compounds and methods
01/14/1999WO1999001124A1 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
01/14/1999WO1998051311A3 Dihydropyrimidines and uses thereof
01/14/1999WO1998045276A3 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinones useful as hiv reverse transcriptase inhibitors
01/14/1999DE19728996A1 Triazolverbindungen und deren Verwendung Triazole compounds and the use thereof
01/14/1999CA2294898A1 Certain diarylimidazole derivatives; a new class of npy specific ligands
01/14/1999CA2294770A1 Compounds and methods
01/13/1999EP0889889A1 Piperazine and piperidine compounds
01/13/1999EP0889887A1 Novel treatment for cns injuries
01/13/1999EP0889885A1 Method for selective protection of baccatin derivatives and its application to taxane synthesis
01/13/1999CN1041629C Pyrrole thioformylamine insecticidal and acaricidel
01/12/1999US5859261 Synthesis of indolylmaleimides
01/12/1999US5859257 Isoxazole compounds as cyclooxygenase inhibitors
01/12/1999US5859254 Process to chloroketones using oxazolines
01/12/1999US5859248 Process for the production of a β-amino alcohol
01/12/1999US5859244 1,4-dihydropyridine derivatives and methods of producing the same
01/12/1999US5859047 Antiarthritic agents, nervous system disorders
01/12/1999US5859035 Arylheteroaryl inhibitors of farnesyl-protein transferase
01/12/1999US5859030 Substituted arylalkylthioalkylthiopyridines for use in the control of helicobacter bacteria
01/12/1999US5859014 Pyrimidinedione, pyrimidinetrione, triazinedione and tetrahydroquinazolinedione derivatives as α1 -adrenergic receptor antagonists
01/12/1999US5859008 Arylalkyl diazinones
01/12/1999US5859007 Treatment of diabetes, obesity
01/12/1999US5858995 Administering to humans and animals in the treatment of diseases caused by abnormal bone metabolism
01/12/1999CA2151890C Quinoline carboxylic acid derivatives having 7-(4-aminomethyl-3-oxime)pyrrolidine substituent and processes for preparing thereof
01/07/1999WO1999000384A1 New quinoxaline dione derivatives, the production thereof and use of the same in medicaments
01/07/1999WO1999000132A1 Use of phospholamban inhibitors for increasing coronary flow
01/07/1999EP0889043A1 5,11-DIHYDRODIBENZ b,e] 1,4]OXAZEPINE DERIVATIVES AND DRUG COMPOSITIONS CONTAING THE DERIVATIVES
01/07/1999EP0889034A1 Aminopyridine derivatives
01/07/1999EP0889033A1 Alpha-substituted benzyl heterocyclic derivatives, intermediates for producing the same, and pesticides containing the same as active ingredient
01/07/1999EP0888344A1 Spirocycle integrin inhibitors
01/07/1999EP0888340A1 4-(benzo-1,3-dioxolyl)-pyrrolidine-3-carboxylic acid derivatives as endothelin antagonists
01/07/1999EP0888339A1 Synthesis of indolylmaleimides
01/07/1999EP0888317A1 Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma
01/07/1999EP0888310A1 Cinnoline derivatives and use as medicine
01/07/1999EP0888307A1 1,3,5-trisubstituted indazole derivatives with an anti-asthmatic, anti-allergic, anti-inflammatory and immunomodulating action
01/07/1999DE19728326A1 Neue Chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln New quinoxalinedione derivatives, their preparation and use in medicaments
01/07/1999DE19727889A1 2-(2-Methylphenyl)-oxazoline 2- (2-methylphenyl) -oxazolines
01/07/1999CA2294550A1 Use of phospholamban inhibitors for increasing coronary flow
01/06/1999CN1204330A Heterocyclic fungicides
01/06/1999CN1204328A 1,3-oxazin-4-one derivatives as herbicides
01/06/1999CN1204327A Pharmaceutically active quinazoline compounds
01/06/1999CN1204323A Use of tricyclic 1,4-dihydro-1,4-dioxo-1 H-naphthalene derivatives, resulting novel compounds and therapeutical use thereof
01/05/1999US5856514 Arylpyrazole fungicides
01/05/1999US5856478 Anellated (oxa)hydantoins and their use as herbicides
01/05/1999US5856353 Sulfonamide inhibitors of aspartyl protease
01/05/1999US5856324 Use of dioxomorpholines for combat endoparasites, dioxomorpholines and process for their production
01/05/1999CA2046956C O-methyl derivatives of azithromycin a, process and intermediate for their preparation, and use thereof in the preparation of pharmaceuticals
12/1998
12/30/1998WO1998058934A1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and compositions containing same
12/30/1998WO1998058905A1 Novel amidrazone derivatives having antifungal activity
12/30/1998WO1998058646A1 Use of somatostatin agonists and antagonists for treating diseases related to the eye
12/30/1998EP0887346A2 Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists
12/30/1998EP0886637A1 Inhibitors of microsomal triglyceride transfer protein and method
12/30/1998CN1203599A Substitued pyrrolidinone, thiazolidinone or oxazolidinone as herbicides
12/30/1998CN1203598A Farnesyl protein transferase inhibiting (imidazol-5-yl) methyl-2-quinolinone derivatives
12/30/1998CN1203590A Substituted imidazoles having anti-cancer and cytokine inhibitory activity
12/30/1998CN1203228A Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives
12/29/1998US5854277 Thiophenebutanoic acid derivatives as matrix metalloprotease inhibitors
12/29/1998US5854274 Tricyclic heterocyclic sulfonamide and sulfonic ester derivatives
12/29/1998US5854265 Biheteroaryl inhibitors of farnesyl-protein transferase
12/29/1998US5854263 1- (1,4-benzodioxanyl)alkyl!-3-(heteroaryl) pyrrolidines and related compounds and their therapeutic utility
12/29/1998US5854262 Aminomethylene substituted non-aromatic heterocycles and use as substance P antagonists
12/29/1998US5854261 Prokinetic compounds
12/29/1998US5854247 Piperazine, piperidine and tetrahydropyridine derivatives useful as 5-HT1 recepter agonists
12/29/1998US5854243 3-heteroaryl-1-pyrrolidinealkylthiols and derivatives thereof and their therapeutic utility
12/29/1998US5854242 Benzoxazine antimicrobial agents
12/29/1998US5854232 Acyclic anc cyclic amides as neurotransmitter release enhancers
12/29/1998US5853930 Electrophotographic photoconductors using bisazo compounds
12/23/1998WO1998057970A1 Benzo(5,6)cycloheptapyridine compounds useful as farnesyl protein transferase inhibitors
12/23/1998WO1998057969A1 4-haloalkyl-3- heterocyclylpyridines and 4-haloalkyl -5-heterocyclylpyridines, method for the production thereof, agents containing the same and their use as pesticides
12/23/1998WO1998057955A1 Compounds useful for inhibition of farnesyl protein transferase
12/23/1998WO1998057954A1 Aroyl-piperazine derivatives, their preparation and their use as tachykinin antagonists
12/23/1998WO1998057951A1 NOVEL GUANIDINE MIMICS AS FACTOR Xa INHIBITORS
12/23/1998WO1998057949A1 Novel tricyclic sulfonamide inhibitors of farnesyl-protein transferase
12/23/1998WO1998057944A1 Benzo(5,6)cyclohepta(1,2b)pyridine derivatives useful for inhibition of farnesyl protein transferase
12/23/1998WO1998057940A1 Heterocyclic substituted piperidines and uses thereof
12/23/1998WO1998057937A2 Inhibitors of factor xa with a neutral p1 specificity group
12/23/1998WO1998057642A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998WO1998057641A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998WO1998057640A1 Alpha 1a adrenergic receptor antagonists
12/23/1998WO1998057639A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998WO1998057638A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998WO1998057632A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998EP0885891A1 Isoxazole derivatives
12/23/1998EP0885887A2 Sulfonamide inhibitors of HIV-Aspartyl protease
12/23/1998EP0885883A1 Fused heterocyclic compounds and pharmaceutical applications thereof
12/23/1998EP0885263A1 Benzophenoxazine dyes
12/23/1998EP0885218A1 Oxa- and thia-diazole muscarinic receptor antagonists
12/23/1998EP0885217A1 Endothelin receptor antagonists
12/23/1998EP0885215A1 Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists