Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
10/2004
10/21/2004US20040209875 Nonsteroidal antiinflammatory agents
10/21/2004US20040209863 5-chloro-N-(5-chloropyridin-2-yl)-2-[(4-{(Z)-(dimethylamino)[(methylsulfonyl)imino]methyl}benzoyl)amino]benzamide; treating thromboembolic disorders, optionally with other active agents
10/21/2004US20040209776 Azole derivatives useful as insecticide
10/21/2004DE10316081A1 Neue Verbindungen mit antibakterieller Aktivität New compounds with antibacterial activity
10/21/2004CA2521830A1 Heteroaromatic pentacyclic compound and medicinal use thereof
10/21/2004CA2521685A1 Antimicrobial [3.1.0] bicyclohexylphenyl-oxazolidinone derivatives and analogues
10/21/2004CA2521653A1 Aromatic sulfonamides as peroxynitrite-rearrangement catalysts
10/21/2004CA2521400A1 Piperazine derivative renin inhibitors
10/21/2004CA2521340A1 Aminopyrimidine derivatives and their medical use
10/21/2004CA2521227A1 Substituted pyrazole compounds
10/21/2004CA2521201A1 Substituted pyrazoles for use in the prophylaxis or treatment of a disease which can be influenced by the binding of the substitued pyrazoles to 5ht receptors
10/21/2004CA2518916A1 Pi-3 kinase inhibitor prodrugs
10/20/2004EP1468996A1 Indole derivatives for the treatment of CNS disorders
10/20/2004EP1467992A1 Antimicrobial dihydrothiazine and dihydrothiopyran oxazolidinones
10/20/2004EP1467986A1 Aza-cyclic compounds as modulators of acetylcholine receptors
10/20/2004EP1467981A1 4(hetero-) aryl substituted (thia-/oxa-/pyra) zoles for inhibition of tie-2
10/20/2004EP1467977A1 Novel antibacterial compounds:process for their preparation and pharmaceutical compositions containing them.
10/20/2004EP1467976A1 N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases
10/20/2004EP1467974A1 Benzimidazole derivatives and their use as gnrh antagonists
10/20/2004EP1467972A1 Indazole compounds useful as protein kinase inhibitors
10/20/2004EP1467971A1 Substituted pyrazolines for use as pesticides
10/20/2004EP1467734A1 Cotherapy with an oxazolidinone and a vitamin b
10/20/2004EP1467732A1 3-(imidazolyl)-2-aminopropanoic acids for use as tafi-a inhibitors for the treatment of thrombotic diseases
10/20/2004EP1467721A2 Substituted amine derivatives and their use for the treatment of angiogenesis
10/20/2004EP1467695A2 Hiv integrase inhibitors
10/20/2004EP1289964B1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists
10/20/2004EP0862555B1 Substituted aryl or heteroarylamides having retinoid-like biological activity
10/20/2004CN1538969A Novel benzothienyl or indole derivatives, preparation and use thereof as inhibitors of prenyl transferase proteins
10/20/2004CN1538968A Novel compounds
10/20/2004CN1538967A Heterocyclic compound and antitumour agent containing the same as active ingredient
10/20/2004CN1538955A Pyrrolidine derivatives as factor Xa inhibitors
10/20/2004CN1538848A Novel Benzo-fused heterocycles
10/20/2004CN1538845A Phenyl derivatives as factor Xa inhibitors
10/20/2004CN1538836A Substituted amine derivatives and method of use
10/20/2004CN1171887C Respiratory syncytial virus replication inhibitors
10/20/2004CN1171879C Herbicidal 3-aryl-1,2,4-triazole derivative
10/20/2004CN1171872C Compounds for modulation of PPAP gamma activity
10/20/2004CN1171582C Oral pharmaceutical extended release dosage form
10/19/2004US6806370 NK-1 receptor active amine oxide prodrugs
10/19/2004US6806287 2-oxo-1-pyrrolidine derivatives, process for preparing them and their uses
10/19/2004US6806286 Pyrrolecarboxamides and pyrrolethioamides as fungicides
10/19/2004US6806278 Amino-tetralin derivatives as muscarinic receptor antagonists
10/19/2004US6806269 Effective at lower concentrations; such as 6-(((1,1-dimethyl-ethoxy)carbonyl)amino)-5-methyl-2-(methyl(phenylmethyl) -amino)-4h-3,1-benzoxazin-4-one
10/19/2004US6806230 Pyrimidine derivatives and herbicides containing them
10/19/2004CA2296901C Piperidine derivates having anxiolytic effect
10/14/2004WO2004087880A2 Compounds and their use to treat diabetes and related disorders
10/14/2004WO2004087714A1 Indole acetamides as inhibitors of the hepatitis c virus ns5b polymerase
10/14/2004WO2004087697A1 N-aryl-2-oxazolidinone-5-carboxamides derivatives with antibacterial activity
10/14/2004WO2004087696A1 Pyrazolidine-1,2-dicarboxyldiphenylamide derivatives as coagulation factor xa inhibitors for the treatment of thromboses
10/14/2004WO2004087695A1 Method for the production of pyrrolidine-1,2-dicarboxylic acid-1-(phenyl(-amide))-2-(phenyl(-amide)) derivatives and 1-(phenylcarbamoyl)-pyrrolidine-2-carboxylic acid derivatives as intermediate products
10/14/2004WO2004087694A1 A heterocycle-substituted benzoxazine compounds having bioactivity
10/14/2004WO2004087690A2 Benzimidazole derivatives and their use for modulating the gaba-a receptor complex
10/14/2004WO2004087680A1 Novel quinazoline derivatives and methods of treatment related to the use thereof
10/14/2004WO2004087669A1 Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof
10/14/2004WO2004087647A2 4-substituted quinolein derivatives with antimicrobial activity
10/14/2004WO2004087646A2 Pyrrolidino-1,2-dicarboxy-1-(phenylamide)-2-(4-(3-oxo-morpholino-4-yl)-phenylamide) derivatives and related compounds for use as inhibitors of coagulation factor xa in the treatment of thrombo-embolic diseases
10/14/2004WO2004087641A1 Hydrazone derivative
10/14/2004WO2004087051A2 Ophthalmic compositions for treating ocular hypertension
10/14/2004WO2004078116A3 P38 inhibitors and methods of use thereof
10/14/2004WO2004056727A3 Process of making chalcone derivatives
10/14/2004WO2004050636A3 IMIDAZOLE-DERIVATIVES AS FACTOR Xa INHIBITORS
10/14/2004WO2004037176A3 Quinazolinones and derivatives thereof as factor xa inhibitors
10/14/2004WO2004024939A3 Ligands for the peroxisome proliferator-activated receptor, and methods of use thereof
10/14/2004WO2004004655A3 Substituted heterocyclic derivatives useful as antidiabetic and antiobesity agents and method
10/14/2004US20040204591 Reacting an amide compound containing hydroxy and a carboxyl group and having benzene ring, with a halogenated alkyl aminocarbonyl-pyrrolidine with 2-fluoro groups substituted at the ring carbon, by amindation of amine and carboxyl group
10/14/2004US20040204588 aryl hydrocarbon; oxidation of 4,5-dihydro-1,3-azoles to fully unsaturated ring; heterocyclic ketones
10/14/2004US20040204586 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
10/14/2004US20040204500 Preventives/remedies for organ functional disorders and organ dysfunction
10/14/2004US20040204498 Pyrimidine carboxamides; 5-hydroxy-2-(2-(1,1-Dioxo-6-[1,2]thiazinan-2-yl)-6-oxo-1,6-dihydropyrimidine-4-carboxamides; AIDS; AIDS related complex
10/14/2004US20040204477 For use as antiproliferative agents
10/14/2004US20040204463 Aantimicrobials with activity against human and veterinary pathogens: Gram-positive aerobic bacteria multiply-resistant staphylococci and streptococci, anaerobic organisms bacteroides and clostridia and acid-fast organisms such as Mycobacterium
10/14/2004US20040204462 E.g., l2-{3-[2-(4-Fluorophenyl)oxazol-4-ylmethoxy]cyclohexyloxy}-6-methylbenzoic acid; lipid- and/or triglyceride-lowering properties; metabolic disorders; antidiabetic agents (type II); therapy of syndrome X; eating disorders; cardiomyopathy
10/14/2004US20040204461 1,2,4-oxadiazole benzoic acid compounds and their use for nonsense suppression and the treatment of disease
10/14/2004US20040204454 Lactam-containing cyclic diamines and derivatives as factor Xa inhibitors
10/14/2004US20040204452 to decompose peroxynitrite anion into harmless nitrate or nitrite endproducts which prevents the free radical-mediated cell damage; cytoprotective; Alzheimer's disease; 3,5-dimethylisoxazole-4-sulfonic acid 4-pyrrolidin-1-ylphenylamide
10/14/2004US20040204450 For therapy of atherosclerosis, coronary artery disease, coronary heart disease, coronary vascular disease, peripheral vascular disease, dyslipidemia, hyperbetalipoproteinemia, hypoalphalipoproteinemia, hypercholesterolemia, hypertriglyceridemia, familial-hypercholesterolemia
10/14/2004US20040204437 Substituted arylamine derivatives and methods of use
10/14/2004US20040204421 Certain 1,3-disubstituted isoquinoline derivatives
10/14/2004US20040204417 For therapy of cancer
10/14/2004US20040204410 Such as 1-(4,5-Bis-(4-chloro-phenyl)-2-(2,4-dimethoxy-phenyl)-4,5-dihydro-imidazol-1-yl)-2-methyl-propan-1-one which inhibits the interaction of MDM2 protein with p53-like peptide; antiproliferative agents
10/14/2004US20040204408 Piperidinyl-morpholinyl derivatives as modulators of chemokine receptor activity
10/14/2004US20040204406 Pyrazole-derivatives as factor Xa inhibitors
10/14/2004US20040204386 for uses such as inhibiting the activity of lysophosphatidic acid acyltransferase beta and/or inhibiting the proliferation of a cell (e.g., tumor cell)
10/14/2004DE10315572A1 Substituierte Pyrazole Substituted pyrazoles
10/14/2004DE10315570A1 New 1-aryl-1,2,3-triazole derivatives useful for treating e.g. schizophrenia, depression, dementia, Parkinson's disease or Alzheimer's disease, are glycine transporter inhibitors
10/14/2004DE10315569A1 Substituierte Pyrazolverbindungen Substituted pyrazole
10/14/2004DE10315377A1 New carbonyl-substituted carbocyclic or heterocyclic compounds, are factor Xa and factor VIIa inhibitors useful e.g. for treating thrombosis, myocardial infarction, arteriosclerosis, inflammation or tumors
10/14/2004CA2521056A1 Hydrazone derivative
10/14/2004CA2520896A1 Indole acetamides as inhibitors of the hepatitis c virus ns5b polymerase
10/14/2004CA2520894A1 Pyrazolidine-1,2-dicarboxyldiphenylamide derivatives as coagulation factor xa inhibitors for the treatment of thromboses
10/14/2004CA2520764A1 4-substituted quinolein derivatives with antimicrobial activity
10/14/2004CA2520723A1 N-aryl-2-oxazolidinone-5-carboxamides derivatives with antibacterial activity
10/14/2004CA2520281A1 Benzimidazole derivatives and their use for modulating the gabaa recept or complex
10/14/2004CA2519899A1 Ophthalmic compositions for treating ocular hypertension
10/14/2004CA2518913A1 Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof
10/14/2004CA2518465A1 Dipeptidyl peptidase inhibitors
10/13/2004EP1466902A1 Androgen receptor antagonists
10/13/2004EP1466901A1 Serotonine reuptake inhibitor
10/13/2004EP1465892A1 Glycinamides as factor xa inhibitors
10/13/2004EP1465872A1 4-sulfide/sulfoxide/sulfonyl-1h-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor