Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
07/2005
07/20/2005CN1642599A ACC inhibitors
07/20/2005CN1642580A Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
07/20/2005CN1642552A 4-(N-phenylamino)-quinazolines / quinolines as tyrosine kinase inhibitors
07/20/2005CN1642551A Inhibitors of histone deacetylase
07/20/2005CN1642543A Parenteral, intravenous, and oral administration of oxazolidinones for treating diabetic foot infections
07/20/2005CN1211384C Thiadiazolyl and oxidiazolyl phenyl oxazolidinone antibacterial agent
07/20/2005CN1211383C Process for making substituted 8-arylquinolinium benzenesulfonate
07/20/2005CN1211367C Prostaglandin agonists and their use to treat bone disorders
07/19/2005US6919482 A 1,4-bis(N-(2-(4-hydroxy-3-hydroxymethylphenyl) -2-hydroxyethyl)amino)-cyclohexane or alkyl-cyclohexane or -pyrazine derivatives; treating respiratory diseases disorders, asthma, bronchitis, nervous system injury
07/19/2005US6919460 Making 2-bromo-1-pyridin-3-yl-ethanol by reducing the ketone, protecting the alcohol, condensing with a p-(heterocycle)-phenoxyethylamine, then deprotecting to form 2-(2-(4-heterocycyl-phenoxy)-ethylamino)-1-pyridin-3-ylethanol
07/19/2005US6919375 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
07/19/2005US6919371 Antidiabetic agents; dietetics; gastrointestinal disorders
07/19/2005US6919368 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
07/19/2005US6919367 Substituted thioacetamides
07/19/2005US6919365 Also oxazolidinediones; excellant enzyme inhibitors of chymase and/or tryptase; antiallergens; antiinflammatory agents; vascular circulatory system disease; vision defects, antidiabetic and -arthritic agents; pancreatitis; hepatitis
07/19/2005US6919359 Azabicyclic-substituted-heteroaryl compounds for the treatment of disease
07/19/2005US6919358 Substituted acid derivatives useful as antidiabetic and antiobesity agents and method
07/19/2005US6919356 Antihistamines, antiallergens, autoimmune disease, antiinflammatory agents
07/19/2005US6919353 Enzyme inhibitors of phosphordiesterase 4 having minimal side effects; antiinflammatory agents; antiallergens; asthma; neurodegenerative disorders; antidiabetic agents; pain; anti-tumor, -carcinogenic and -arthritic agents
07/19/2005US6919347 Antidiabetic agents; antiinflammatory agents; analgesics; antiallergens
07/19/2005US6919346 Isoxazolone compounds useful in treating diseases associated with unwanted cytokine activity
07/19/2005US6919343 N-biphenyl(substituted methyl) aminocycloalkane-carboxamide derivatives
07/19/2005US6919339 ABCA-1 elevating compounds
07/19/2005US6919338 Antiproliferative agents; anticancer agents
07/19/2005US6919335 Heterocycles that are inhibitors of IMPDH enzyme
07/19/2005US6919331 Substituted 2-methyl-benzimidazole respiratory syncytial virus antiviral agents
07/19/2005US6919329 Microorganisms; bactericides; human and veterinary medicine
07/14/2005WO2005063765A1 Inhibitors of cyclin-dependent kinases, compositions and uses related thereto
07/14/2005WO2005063754A1 Triazole derivatives as vasopressin antagonists
07/14/2005WO2005063742A2 Amidino compounds as cysteine protease inhibitors
07/14/2005WO2005063738A1 Novel 2-heteroaryl-substituted benzimidazole derivative
07/14/2005WO2005063736A1 Aminoalkylpyrazole derivative
07/14/2005WO2005063723A1 Benzo`1,4 ! diazepin-2-one derivatives as phosphodiesterase pde2 inhibitors, preparation and therapeutic use thereof
07/14/2005WO2005063715A1 Polymorph of birb 796, a p38map kinase inhibitor
07/14/2005WO2005063705A1 Benzene compounds disubstituted with cyclic groups at the 1- and 2-positions
07/14/2005WO2005063690A1 Alpha-hydroxy amides as bradykinin antagonists or inverse agonists
07/14/2005WO2005056550A3 Heterocyclic anti-migraine agents
07/14/2005WO2005049579A3 Immobilized n-substituted tricyclic 3-aminopyrazoles for the identification of biomolecular targets
07/14/2005WO2005040142B1 Novel keto-oxadiazole derivatives as cathepsin inhibitors
07/14/2005WO2004098528A3 Pyrazole-amine compounds useful as kinase inhibitors
07/14/2005US20050154200 Method for producing cyclic carbamate ester
07/14/2005US20050154056 Inhibitors of HCV NS5B polymerase
07/14/2005US20050154042 N-alkyl pyrroles as HMG-CoA reductase inhibitors
07/14/2005US20050154038 bicyclo[2.2.2]-oct-1-yl-1,2,4-triazoles; type 2 diabetes, lipid disorders, obesity, atherosclerosis, metabolic syndrome, hyperglycemia, insulin resistance; increase insulin sensitivity in muscle, liver and adipose tissue by correction of the elevated plasma levels of glucose without causing hypoglycemia
07/14/2005US20050154028 1-(3-Fluoro-phenyl)-3-[4-methoxy-3-(2-piperidin-1-yl-ethoxy)-phenyl]-imidazolidin-2-one; serotonin 5-ht2c receptor antagonist; antidepressant and anxiolytic agent
07/14/2005US20050154027 Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
07/14/2005US20050154023 1-(4-methoxynaphthalene-1-sulfonyl)-2,3-dihydro-1H-indole-3-carboxylic acid [2-(1-methyl-pyrrolidin-2-yl)-ethyl]amide; selective affinity for 5-HT6 receptor; psychosis, schizophrenia, depression, neurological disorders, cognitive enhancement, Parkinson's disease, ALS, Alzheimer's, Huntington's disease
07/14/2005US20050154019 Substituted cyclic amine metalloprotease inhibitors
07/14/2005US20050154012 Substituted 3-aryl-5-aryl-[1,2,4]-oxadiazoles and analogs as activators of caspases and inducers of apoptosis and the use thereof
07/14/2005US20050153997 Fredericamycin derivatives
07/14/2005US20050153996 Compounds that modulate ppar activity and methods for their preparation
07/14/2005US20050153987 Compounds
07/14/2005US20050153986 Psychiatric and mood disorders, Bipolar Disorder, Circadian rhythm disorders, sleep disorders, pain, Parkinson's disease, cognitive dysfunction, epilepsy, obesity, drug addiction, drug abuse, drug withdrawal; side effects reduction; 1-Methyl-3-[3-(5-pyridin-2-yl-2H-tetrazol-2-yl)phenyl]imidazolidin-2-one
07/14/2005US20050153979 Novel piperidine-substituted indoles-or heteroderivatives thereof
07/14/2005US20050153978 Medicaments
07/14/2005US20050153974 Heterocyclymethylpiperidines and -piperazines possessing affinity at 5ht-1 type receptors
07/14/2005US20050153972 Triazole compounds
07/14/2005US20050153971 Halogenated biaryl heterocyclic compounds and methods of making and using the same
07/14/2005US20050153963 exhibit a particular activity as specific inhibitors of the glycine transporters glyt1 and/or glyt2
07/14/2005US20050153960 Substituted arylamine derivatives and methods of use
07/14/2005US20050153959 Heterocyclic anti-migraine agents
07/14/2005US20050153951 Neurotrophic pyrrolidines and piperidines, and related compositions and methods
07/14/2005US20050153944 Oxazole derivatives of tetracyclines
07/14/2005US20050153942 Heterocyclic inhibitors of MEK and methods of use thereof
07/14/2005CA2548318A1 Benzo-1, 4 diazepin-2-one derivatives as phosphodiesterase pde2 inhibitors, preparation and therapeutic use thereof
07/14/2005CA2547837A1 Polymorph of birb 796, a p38map kinase inhibitor
07/13/2005EP1553097A1 Quinazoline derivatives as angiogenesis inhibitors and intermediates therefore
07/13/2005EP1553091A1 Heteroaromatic pentacyclic compound and medicinal use thereof
07/13/2005EP1553089A1 Antagonist of melanin-concentrating hormone receptor comprising benzimidazole derivative as active ingredient
07/13/2005EP1553085A1 Cyclic amine derivatives and their use as drugs
07/13/2005EP1553084A1 Piperidine derivative, process for producing the same, and use
07/13/2005EP1552836A1 Anti-neurodegenerative agents
07/13/2005EP1551831A1 Method for preparing risperidone
07/13/2005EP1551830A2 Heterocyclically substituted indolinones and their use as receptor tyrosine kinase inhibators
07/13/2005EP1551829A2 Novel compounds with antibacterial activity
07/13/2005EP1551813A2 Chemical compounds
07/13/2005EP1551812A2 Mitotic kinesin inhibitors
07/13/2005EP1551809A1 Pyrazole compounds for treatment of neurodegenerative disorders
07/13/2005EP1551804A1 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
07/13/2005EP1551803A1 Azabicyclo derivatives as muscarinic receptor antagonists
07/13/2005EP1551384A2 R-nsaid esters and their use
07/13/2005EP1427711B1 Oxazolidinone and/or isoxazoline derivatives as antibacterial agents
07/13/2005EP1235802B1 Carbamate derivatives having muscarinic receptor antagonist activity
07/13/2005EP1042291B1 Aryl-substituted pyridylalkane, alkene, and alkine carboxamides useful as cytostatic and immunosuppressive agents
07/13/2005CN1639159A N-aminoacetyl-pyrrolidine-2-carbonitriles and their use as DDP-IV inhibitors
07/13/2005CN1639156A 8'4-'3-(5-fluoro-1H-indol-3-yl)propyl!-1-piperazinyl!-2-methyl-2H-1, 4-benzoxazin -3(4H)-one methanesulfonate with high affinity for the dopamine D2 receptor and the seotonin reuptake site
07/13/2005CN1639155A Pyrrolidine oxadiazole- and thiadiazole derivatives
07/13/2005CN1639154A Pyranones useful as ATM inhibitors
07/13/2005CN1639149A Processes for the preparation of substituted bicyclic derivatives for the treatment of abnormal cell growth
07/13/2005CN1639146A Fused tricyclic heterocycles useful for treating hyper-proliferative disorders
07/13/2005CN1639145A Benzofuran and benzothiophene derivatives useful in the treatment of hyper-proliferative disorders
07/13/2005CN1639136A Oxazolidinone and/or isoxazoline as antibacterial agents
07/13/2005CN1639135A N-aryl-2-oxazolidinone-5-carboxamides and their derivatives and their use as antibacterials
07/13/2005CN1639133A Novel antibacterial compounds, process for their preparation and pharmaceutical compositions containing them
07/13/2005CN1639132A N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases
07/13/2005CN1639125A New inhibitors of histone deacetylase
07/13/2005CN1639124A Aminotetralin derivatives as muscarinic receptor antagonists
07/13/2005CN1639121A 3-azabicyclo (3.1.0) hexane derivatives having opioid receptor affinity
07/13/2005CN1639120A Indolamid derivatives which possess glycogenphosphorylase inhibitory activity
07/13/2005CN1639096A Process for producing trans-4-amino-1-cyclohexanecarboxylic acid derivative