Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
01/2006
01/04/2006EP1612204A1 Hydrazone derivative
01/04/2006EP1611902A1 Preventive and/or therapeutic agent for neuropathic pain
01/04/2006EP1611128A2 Positive allosteric modulators of the nicotinic acetylcholine receptor
01/04/2006EP1611127A2 4-substitued quinolein derivatives with antimicrobial activity
01/04/2006EP1611122A1 Substituted pyrazole compounds
01/04/2006EP1611121A1 Pyridazinone derivatives as cdk2-inhibitors
01/04/2006EP1611119A1 Pi-3 kinase inhibitor prodrugs
01/04/2006EP1611113A1 Process to produce enantiomerically enriched 1-aryl- and 1-heteroaryl-2-aminoethanols
01/04/2006EP1611112A1 Isoxazole compounds as inhibitors of heat shock proteins
01/04/2006EP1611109A1 Novel quinazoline derivatives and methods of treatment related to the use thereof
01/04/2006EP1611105A1 Isoquinoline-5-sulfonic acid amides as inhibitors of akt (protein kinase b)
01/04/2006EP1611088A2 Hydroxamates as therapeutic agents
01/04/2006EP1610812A1 Pharmaceutical preparations comprising acid-stabilised insulin
01/04/2006EP1610776A2 Ophthalmic compositions for treating ocular hypertension
01/04/2006EP1610774A2 Tie-2 modulators and methods of use
01/04/2006EP1363873A4 Peptide deformylase inhibitors
01/04/2006EP1296979B1 HETeroARYL-SUBSTITUTED HETEROCYCLES and their use as pesticides
01/04/2006EP1242403B1 2,4-diaminopyrimidine compounds usful as immunosuppressants
01/04/2006EP1102755B1 Substituted isoxazole derivatives as estrogen receptor modulators
01/04/2006EP0934288B1 Oxadiazoles, processes for their preparation and their use as medicaments
01/04/2006EP0885885B1 Pyridone derivatives and herbicides
01/04/2006CN1717407A Indolyl derivatives
01/04/2006CN1717401A Anilinopyrazole derivatives useful for the treatment of diabetes
01/04/2006CN1717396A Chk-, Pdk- and Akt-inhibitory pyrimidines, their production and use as pharmaceutical agents
01/04/2006CN1717393A Pyrazole derivatives useful as COX-I inhibitors
01/04/2006CN1234706C Oxygen nitride heterocyclic compounds and preparation thereof
01/04/2006CN1234705C New hydroxyl indoles, their use as phosphor diesterase 4 inhibitors and method for producing same
01/04/2006CN1234693C Indazol compound for inhibiting protein kinase and medicine composition and their application
01/03/2006US6982278 For modulating a peroxisome proliferator activated receptor, particularly in the treatment of diabetes mellitus
01/03/2006US6982272 E.g., 4-acetylamino-N-(1-((4-cyano-1-methylpiperidin-4-yl-carbamoyl)-2 -(cyclohexylethyl)benzamide; Alzheimer's, auto-immune and Crohn's diseases; atherosclerosis; antiarthritic agents; osteoporosis; atherosclerosis
01/03/2006US6982263 Peptidyl carbamates; treatments for osteoporosis and autoimmune diseases
01/03/2006US6982261 A progesterone receptor antagonist for providing progestational therapy, treating cancer of breast, uterine, ovarian, endometrial, or prostate, providing contraceptives, hormone replacement therapy
01/03/2006CA2343236C 4,4-biarylpiperidine derivatives
01/03/2006CA2247451C Carboxylic acid derivatives having fused rings as retinoic acid receptor agonist
01/03/2006CA2244695C Cyclic amic acid derivatives
12/2005
12/29/2005WO2005123727A1 3-aryl-3-hydroxy- and 3-aryl-3-oxopropionic acid esters as fungicides
12/29/2005WO2005123726A1 Pyridinyl-isoxazoles and their use as herbicides
12/29/2005WO2005123724A1 2,4-diaminoquinazolines for spinal muscular atrophy
12/29/2005WO2005123723A1 3-cycloalkylbenzazepines as histamine h3 antagonists
12/29/2005WO2005123718A2 Benzimidazolone carboxylic acid derivatives
12/29/2005WO2005123717A1 7-pyrazolylbenzazepines having affinity for d3 receptor
12/29/2005WO2005123715A1 Novel alkyl substituted piperidine derivatives as monoamine neurotransmitter re-uptake inhibitors
12/29/2005WO2005123703A2 Alkynyl derivatives as modulators of metabotropic glutamate receptors
12/29/2005WO2005123697A1 Quinazoline derivatives
12/29/2005WO2005123688A2 3-aminoindazoles
12/29/2005WO2005123687A1 Substituted tetrahydro-2h-isoquinolin-1-one derivatives, method for the production thereof, and use of the same as medicaments
12/29/2005WO2005123681A1 Saturated and unsaturated 3-pyridyl-benzocycloalkylmethyl-amines for use in the treatment of pains, depressions and anxiety states
12/29/2005WO2005123680A1 Six-membered heterocycles useful as serine protease inhibitors
12/29/2005WO2005123671A1 Pyrrole derivative
12/29/2005WO2005123089A2 Multicyclic sulfonamide compounds as inhibitors of histone deacetylase for the treatment of disease
12/29/2005WO2005123050A2 Five-membered heterocycles useful as serine protease inhibitors
12/29/2005WO2005105780A3 Compositions useful as inhibitors of rock and other protein kinases
12/29/2005WO2005047524A3 Compositions and methods for inducing cell dedifferentiation
12/29/2005WO2005012294A8 2,4-pyrimidinediamine compounds for use in the treatment or prevention of autoimmune diseases
12/29/2005WO2005007625A3 Heterocyclic amides with anti-tuberculosis activity
12/29/2005US20050288515 Chemical compounds
12/29/2005US20050288501 Reducing a 2-(protected amino)-3-(piperazin-1-yl, N-morpholinyl, or N-thiomorpholinyl) propanoate, deprotecting the amine, and reacting with t-butylisothiocyanate
12/29/2005US20050288376 Bicyclyl or heterobicyclylmethanesulfonylanimo-substituted N-hydroxyformamides
12/29/2005US20050288350 Useful in female hormone replacement therapy and as modulators of fertility; therapy of dysfunctional uterine bleeding, dysmenorrhea, endometriosis, leiomyomas (uterine fibroids), hot flashes, mood disorders, meningiomas, cancer; 6-(bis-2,2,2-Trifluoroethyl)amino-4-trifluoromethylcoumarin
12/29/2005US20050288336 Cysteine protease inhibitors
12/29/2005US20050288324 Aromatic sulfonamides as peroxynitrite-rearrangement catalysts
12/29/2005US20050288322 Cyclizing 2,6-diaminopyridine in sulfuric acid with malic acid to form 2-amino-7-hydroxy-1,8-naphthyridine; phthalimidating the naphthyridine and replacing the OH with Cl; reducing the product to form the hydroxyindolinone derivative and etherifying with 5-methyl-2-oxo-hexyltriphenylphosphonium halide
12/29/2005US20050288314 2,4-diaminoquinazolines for spinal muscular atrophy
12/29/2005US20050288308 11B-HSD1 inhibitors for the treatment of diabetes
12/29/2005US20050288305 N-biarylmethyl aminocycloalkanecarboxamide derivatives
12/29/2005US20050288287 Chiral cis-imidazolines
12/29/2005US20050288284 Specific binding is extremely high; low toxicity; high degree of activity; 2-(5-m-Tolyl-thiazol-2-yl )-7,8-dihydro-6H-quinolin-5-one, acute and/or chronic neurological disorders
12/29/2005US20050288281 Hetero isonipecotic modulators of vanilloid VR1 receptor
12/29/2005US20050288275 New compounds
12/29/2005US20050288273 Antibacterial agents
12/29/2005US20050288270 New aminopyridine derivatives and their use as pharmaceuticals
12/29/2005US20050287617 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
12/29/2005DE102004029309A1 Pyridinylisoxazole und ihre Verwendung als Herbizide Pyridinylisoxazole and their use as herbicides
12/29/2005DE102004028862A1 3-Aminoindazole 3 aminoindazoles
12/29/2005DE102004027358A1 Pyrimidinverbindungen und ihre Verwendung Pyrimidine compounds and their use
12/29/2005CA2570529A1 Pyridinyl-isoxazoles and their use as herbicides
12/29/2005CA2570472A1 Five-membered heterocycles useful as serine protease inhibitors
12/29/2005CA2570264A1 3-aminoindazoles
12/29/2005CA2570065A1 Novel alkyl substituted piperidine derivatives as monoamine neurotransmitter re-uptake inhibitors
12/28/2005EP1609790A2 Benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists
12/28/2005EP1609785A1 C-glycoside derivatives and salts thereof
12/28/2005EP1609784A1 Process for the preparation of 4-(benzimidazolylmethylamino)-benzamidines
12/28/2005EP1608648A1 Pyridyloxymethyl and benzisoxazole azabicyclic derivatives
12/28/2005EP1608646A1 Method for the production of pyrrolidine-1,2-dicarboxylic acid-1-(phenyl(-amide))-2-(phenyl(-amide)) derivatives and 1-(phenylcarbamoyl)-pyrrolidine-2-carboxylic acid derivatives as intermediate products
12/28/2005EP1608645A1 Pyrazolidine-1,2-dicarboxyldiphenylamide derivatives as coagulation factor xa inhibitors for the treatment of thromboses
12/28/2005EP1608639A2 Novel bicyclic urea derivatives useful in the treatment of cancer and other disorders
12/28/2005EP1608632A1 Quinazolines useful as modulators of ion channels
12/28/2005EP1608631A2 Bi-cyclic pyrimidine inhibitors of tgf beta
12/28/2005EP1608630A1 2, 3, 6-trisubstituted-4-pyrimidone derivatives
12/28/2005EP1608628A2 Histone deacetylase inhibitors
12/28/2005EP1608375A1 Methods for treating or preventing an inflammatory or metabolic condition by inhibiting jnk
12/28/2005EP1497240A4 Non-heating clay composites for building materials
12/28/2005EP1495011B1 A semi-synthetic process for the preparation of n debenzoylpaclitaxel
12/28/2005EP1461318B9 Tetrahydroquinoline analogues as muscarinic agonists
12/28/2005EP1382604B1 Quinoline derivative having azolyl group and quinazoline derivative
12/28/2005EP1303641B1 Method for recovery of copper from sulfidic ore materials using super-fine grinding and medium temperature pressure leaching
12/28/2005EP1224183B1 Heterocyclic sodium/proton exchange inhibitors and method
12/28/2005EP1173433B1 Cyanopyrroles as progesterone receptor agonists
12/28/2005EP0945445B9 1,5-benzodiazepine derivatives
12/28/2005CN1714084A Pyrimidine-2,4,6-trione metalloproteinase inhibitors