Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
09/2006
09/12/2006US7105544 N-{3-[1-(3-{[BIS(4-FLUOROPHENYL)ACETYL]AMINO}PROPYL)-4-PIPERIDINYL]PHENYL}-2-METHYLPROPANAMIDE; antagonists for melanin concentrating hormone-1 (MCH1) receptors; treating depression, anxiety, obesity
09/12/2006US7105538 4-oxo-4-[2-(5-pyridin-4-yl-[1,3,4]oxadiazol-2-yl)-pyrrolidin-1-yl]-butyric acid ethyl ester; inhibition of serotonin re-uptake; analgesic effect
09/12/2006US7105535 Such as n-{4-[4-(1,3-benzoxazol-2-yl)pyrazol-3-yl]phenyl}-n'-methyl urea; synthesis; cancer, cell proliferative disorders, viral infections, autoimmune diseases, neurodegenerative disorders
09/12/2006US7105530 Pyrimidineamines as angiogenesis modulators
09/12/2006US7105529 A novel compound for treating alopecia induced by cancer chemotherapy or radiotherapy
09/12/2006US7105519 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
09/12/2006US7105518 Thiopyrane-4-ones as DNA protein kinase inhibitors
09/12/2006US7105516 Compounds for the treatment of premature ejaculation
09/12/2006US7105515 Such as N-[3-(2-diethylaminoethyl)-1H-indol-5-yl]-5-chloro-3-methylbenzo[b]thiophene-2-sulphonamide for treating anxiety, depression, cognitive memory disorders and senile dementia, psychosis, infant hyperkinesia (ADHD, attention deficit/hyperactivity disorder)
09/12/2006US7105509 Benzodiazepine derivatives as APP modulators
09/12/2006US7105505 Benzimidazole derivatives useful as histamine H3 antagonists
09/12/2006US7105503 Pyrazole compounds
09/12/2006CA2235986C Inhibitors of protein isoprenyl transferases
09/12/2006CA2167004C Agent for treating mental disorders associated with cerebrovascular disorders
09/08/2006WO2006094237A2 Acridine and quinoline dervatives as sirtuin modulators
09/08/2006WO2006094187A2 Phthalazine, aza- and diaza-phthalazine compounds and methods of use
09/08/2006WO2006093677A1 Tetracyclic sulfonamide compounds and methods of use thereof
09/08/2006WO2006093667A1 Tetracyclic amino and carboxamido compounds and methods of use thereof
09/08/2006WO2006093339A1 Use of cinnamoyl compound
09/08/2006WO2006093336A1 Use of cinnamoyl compound
09/08/2006WO2006093247A1 NOVEL AMINOPYRIDINE COMPOUND WITH Syk INHIBITORY ACTIVITY
09/08/2006WO2006092739A1 Anti-inflammatory conjugates of macrolides and coumarins
09/08/2006WO2006092599A2 Pyrrole derivatives as dna gyrase and topoisomerase inhibitors
09/08/2006WO2006092291A2 Method for producing alkyl anilides
09/08/2006WO2006092143A1 Substituted pyridine derivatives
09/08/2006WO2005086700A3 Hiv integrase inhibitors
09/08/2006CA2600933A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
09/08/2006CA2600287A1 Use of cinnamoyl compound
09/08/2006CA2599992A1 Acridine and quinoline dervatives as sirtuin modulators
09/08/2006CA2599544A1 Novel aminopyridine compound with syk inhibitory activity
09/08/2006CA2598647A1 Tetracyclic amino and carboxamido compounds and methods of use thereof
09/08/2006CA2597576A1 Isoquinoline compounds and methods of use thereof
09/07/2006US20060199964 preparation of 6-haloalkyl-3-nicotinic acid esters and also to novel enamine intermediates
09/07/2006US20060199958 Process and intermediates for the preparation of pyrrolidine carboxylic acids
09/07/2006US20060199949 Cyanine dyes as labeling reagents for detection of biological and other materials by luminescence methods
09/07/2006US20060199827 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
09/07/2006US20060199826 Cyclopropane compounds and pharmaceutical use thereof
09/07/2006US20060199825 4-Aminating a 4-chloro-2-hydroxy-3-nitrodihydroquinoline with a N-(hetero)cyclylpiperazine, and alkylating the remaining amine group in the quinoline ring to produce a 4-(4-(hetero)cyclylpiperazinyl)-3-nitro-1-alkyldihydroquinolinone
09/07/2006US20060199824 Treating or preventing pain, UI, an ulcer, IBD, IBS, an addictive disorder, Parkinson's disease, parkinsonism, anxiety, epilepsy, stroke, a seizure, a pruritic condition, psychosis, a cognitive disorder, a memory deficit, restricted brain function, Huntington's chorea, amyotrophic lateral sclerosis
09/07/2006US20060199821 Heterocyclic amides and sulfonamides
09/07/2006US20060199820 e.g. N1-hydroxy-N2-[(4-phenoxyphenyl)sulfonyl]-D-argininamide; metallopeptidase inhibitor; antiinflammation, anticarcinogenic, antidiabetic agent; angiogenesis inhibitor; atherosclerosis, stroke, ulcer, infertility, scleroderma, endometriosis, mesothelioma
09/07/2006US20060199818 Inhibiting the activity of a 5-hydroxytryptamine 2A by administering a N-heterocyclyl (preferably 1,3-dioxan-5-yl)-4-[(N-substituted)(hetero)arylamino]piperidine in which the N-substituant is arylalkanoyl, arylthioalkanoyl, arylalkylaminocarbonyl or arylalkylaminothiocarbonyl group
09/07/2006US20060199815 NK1 antagonists
09/07/2006US20060199813 Neurodegenerative diseases, psychological disorders; e.g. 1-[3-(4-Butyl-piperidin-1-yl)-propyl]-1,2,3,4-tetrahydroquinoline
09/07/2006US20060199810 Neurodegenerative diseases, psychological disorders; e.g. 1-[3-(4-Butyl-piperidin-1-yl)-propyl]-1,2,3,4-tetrahydro-quinoline
09/07/2006US20060199804 ATP-competitive inhibitors of serine/threonine kinase (mTOR); antifungal agents, anticancer agents, autoimmune diseases, inflammation, bone loss, bowel disorders, hepatic fibrosis/necrosis, rheumatoid arthritis, psoriasis
09/07/2006US20060199799 Benzimidazolidinone derivatives as muscarinic agents
09/07/2006DE102005009457A1 Verfahren zum Herstellen von Alkylaniliden A process for producing alkylanilides
09/06/2006EP1698628A1 Hydroxypyrimidinone derivative having hiv integrase inhibitory activity
09/06/2006EP1698627A1 Pyrazole compounds useful as protein kinase inhibitors
09/06/2006EP1698620A1 Benzene compounds disubstituted with cyclic groups at the 1- and 2-positions
09/06/2006EP1698334A1 Pharmaceutically active isoindoline derivatives
09/06/2006EP1697355A2 Amidino compounds as cysteine protease inhibitors
09/06/2006EP1697353A2 Aralkyl and aralkylidene heterocyclic lactams with affinity for 5-ht1 receptors
09/06/2006EP1697352A2 4-azole substituted imidazole compositions useful as inhibitors or c-met receptor tyrosine kinase
09/06/2006EP1697348A1 Hiv protease inhibiting compounds
09/06/2006EP1697345A1 Morpholinyl containing benzimidazoles as inhibitors of respiratory syncytial virus replication
09/06/2006EP1697333A1 (3,4-disubstituted)propanoic carboxylates as s1p (edg) receptor agonists
09/06/2006EP1697332A1 Benzo'1,4 ! diazepin-2-one derivatives as phosphodiesterase pde2 inhibitors, preparation and therapeutic use thereof
09/06/2006EP1697327A1 Insecticidal spiroindane derivatives
09/06/2006EP1697320A1 A synthetic methodology for the reductive alkylation at the c-3 position of indoles
09/06/2006EP1697312A2 Hydroxamic acid esters and pharmaceutical use thereof
09/06/2006EP1696919A2 3-cycloalkylaminopyrrolidine derivatives as modulators of chemokine receptors
09/06/2006EP1562935B1 Heteroaryloxy-substituted phenylaminopyrimidines as rho-kinase inhibitors
09/06/2006EP1455579B1 Pyrazoles-pyrimidine fungicides
09/06/2006EP1406609B1 Substituted aryl compounds as novel cyclooxygenase-2 selective inhibitors, compositions and methods of use
09/06/2006EP1223933B1 5-membered heterocycle derivatives and use thereof as monoaminoxidase inhibitors
09/06/2006CN1829714A Pna单体和前体 Pna monomers and precursors
09/06/2006CN1829713A 3,5 disubstituted indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation
09/06/2006CN1829712A Nicotinamide derivatives useful as PDE4 inhibitors
09/06/2006CN1829709A Bicyclic imidazol derivatives against flaviviridae
09/06/2006CN1829701A Piperazine derivatives and their use as therapeutic agents
09/06/2006CN1829698A Pyridazine derivatives and their use as therapeutic agents
09/06/2006CN1829506A Novel coumarin-amide derivatives and its preparation, its drug composition and use
09/06/2006CN1827642A Ofloxacin couple and its preparing method and use
09/06/2006CN1273466C Quinoline derivatives and quinazoline derivatives having azolyl group
09/06/2006CN1273463C (1-phenacy-3-phenyl-3-piperidylethyl)piperidine derivatives, method for production thereof and pharmaceutical compositions containing the same
09/06/2006CN1273456C Thiazole or oxazole derivatives
09/06/2006CN1273451C Piperidine MCH antagonists and their use in treatment of obesity
09/05/2006USRE39266 5-[4-[2-[2,4-dimethyl-6-oxo-1,6-dihydro-1-pyrimidinyl]ethoxy]phenyl methyl]thiazolidine-2,4-dione; intermediate compound for antidiabetic drug
09/05/2006USRE39265 Heteroarylpiperidines, and their use as antipsychotics and analgetics
09/05/2006USRE39263 2-2-fluoro-5-ethylsulphonylamino-4-thiocarbamoyl-phenyl)-5,6,7,8-tetrahydro-1,2,4triazolo[4,3-a]pyridin-3(2H)-one; post or preemergent
09/05/2006US7102009 For treating cancer and angiogenesis-related disorders
09/05/2006US7102001 Process for preparing pyrrolotriazine
09/05/2006US7102000 Heterocyclic amide derivatives for the treatment of diabetes and other diseases
09/05/2006US7101999 Red fluorescence dyes; labels
09/05/2006US7101896 Pharmaceutical compositions and methods for use
09/05/2006US7101892 2-(4-benzenesulfonyl-4-methyl-pentyl)-5-phenyl-2-aza-bicyclo[2.2.1]heptane; useful for treating sleep disorder, depression, anxiety
09/05/2006US7101885 1-(4-Bromo-phenyl)-3-[2-(4-methyl-piperazin-1-yl)-pyridin-3-yloxy]-pyrrolidin-2-one; antagonists of the serotonin 5HT1B receptor; treating depression
09/05/2006US7101882 Morpholin-acetamide derivatives for the treatment of inflammatory diseases
09/05/2006US7101881 N-(4-Chlorophenylacetyl)-8-(4-methylpiperazinyl)-tetrahydroisoquinoline; treating anxiety, depression, dysthymia, major depressive disorder, migraine, post-traumatic stress disorder, avoidant personality disorder, borderline personality disorder, phobias
09/05/2006US7101880 Peptidic compounds as cysteine protease inhibitors
09/05/2006US7101877 Trans-[2-(4-Morpholinyl)-1-(2-Naphthenethoxy)]Cyclohexane Monohydrochloride; selectively inhibiting cardiac early repolarising currents and cardiac sodium currents
09/05/2006US7101876 Substituted benzoxazines as integrin antagonists
09/05/2006US7101875 E.g., 4-(2-(1-Benzhydryl-2-(2-((benzylsulfonyl)amino)ethyl)-5-chloro-1H-indol-3 -yl)ethoxy)benzoic acid; inhibitors of phospholipase enzymes, esp. phospholipase A2; antiarthritic and -inflammatory agents; analgesics; rheumatoid diseases
09/05/2006US7101874 1) N-[[(5S)-3-[4-(2,3-dihydro-1,1-dioxido-4H-1,4-thiazin-4-yl)-3-fluorophenyl]-2-oxo-5-oxazolidinyl]methyl]acetamide; potent activities against Gram-positive and Gram-negative bacteria
09/05/2006US7101868 A 2-(((4-fluorophenyl)methyl)amino)-3-pyridinecarboxamide derivatives for treating cancer, angiogenesis, tumor
09/05/2006US7101533 Agent for inducing receptor potential
08/2006
08/31/2006WO2006091674A1 Pgd2 receptor antagonists for the treatment of inflammatory diseases
08/31/2006WO2006091592A1 Naphthalene derivatives as modulators of the glucocorticoid receptor