Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
10/2006
10/11/2006CN1845911A Condensed ring compound and use thereof
10/11/2006CN1845909A Quinoxaline derivatives as neutrophil elastase inhibitors and their use
10/11/2006CN1845905A PPAR-activating compound and pharmaceutical composition comprising the compound
10/11/2006CN1845900A Quinoline derivatives as neutrophil elastase inhibitors and their use
10/11/2006CN1845734A Benzimidazole derivatives and their use as protein kinases inhibitors
10/11/2006CN1279034C Dna-pk抑制剂 Dna-pk inhibitors
10/11/2006CN1279026C Prostaglandin endoperoxide H synthase biosynthesis inhibitors
10/10/2006US7119214 dibenzofuranyl, dibenzothiophenyl or fluorenyl thioacetamides used for prophylaxis of sleep disorders
10/10/2006US7119207 NK-1 receptor antagonists, (e.g., substance P receptor antagonists)
10/10/2006US7119203 Piperidinyl- and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
10/10/2006US7119201 Triaryl-oxy-aryloxy-pyrimidine-2,4,6-trione metalloproteinase inhibitors
10/10/2006US7119198 beta-aryl-alpha-oxysubstituted alkylcarboxylic acids, usch as Ethyl (E/Z)-3-[4-[2-(phenoxazin-10-yl)ethoxy]phenyl]-2-ethoxypropenoate, used as antilipemic or hypoglycemic agents
10/10/2006US7119120 A 2-benzenesulfonylamino-N-benzyl-benzamides for treating hyperphosphatemia, urogential disorders
10/10/2006US7119116 Direct aminolysis of a carbamate ester or hydrolysis to an acid followed by coupling with an amine; analgesics, disorders of eating, nervous system, psychology, sleep, urogenital, respiratory and gastrointestinal systems; antiischemic, anticarcinogenic, antiinflammatory agents, antiallergens
10/10/2006US7119115 For therapy of treating tumors or cancerous cells
10/10/2006US7119113 optionally halogenated N-(trifluoromethyloxazol-2-yl)xanthene-9-carboxamides; treatment of neurological disorders such as Alzheimer's disease and dementia
10/10/2006US7119105 Methods for treating neurodegenerative disorders using aspartyl protease inhibitors
10/10/2006US7119104 Alpha-(oxy-, sulfo- or amino-)[3-(imidazolyl, oxazolyl or thiazolyl)alkylene(indazolyl, benzisoxazolyl or benzisothiazolyl)]acetic acids, esters or alkali salts
10/10/2006US7119102 3-amino-6-{4-[2-hydroxy-2-(substituted heteroaryl)ethylamino]-piperidin-1-yl}thieno[2,3-b]pyridine-2-carboxylic acid amides; reductive amination; I kappa B kinase inhibitors; autoimmune diseases; antiinflammatory and anticarcinogenic agents
10/10/2006US7119099 DNA replication that interfere with the E1-E2-DNA complex during initiation of DNA replication; 1-(hydroxy, oxo, or epoxy)-3-oxo-3'-benzaminocarbonyl-4'-(carboxy or carboxylate)-1,2,3-trihydroindene-2-spiro-2'-tetrahydrofuran derivatives
10/10/2006US7119098 Antitumor agents; osteoporosis; antiarthritic agents; oral diseases
10/10/2006US7119090 Anticancer agents; antiinflammatory agents; autoimmune diseases; rheumatic diseases, enzyme inhibitors
10/10/2006US7119088 A bi-heterocycle-4H-2,3,5,10b-tetraaza-benzo[e]azulene derivatives; for therapy of dysmenorrhoea, anxiety disorder, asthma, atherosclerosis, cardiac failure, cardiovascular disease, cataract, central nervous system disease, motion sickness, Raynaud's disease, rheumatoid arthritis; chemical synthesis
10/10/2006US7119084 4-amino-6-cycloalkyloxy-7-substituted quinazolines; inhibition of signal transduction mediated by tyrosine kinases; antitumor agents, respiratory system and gastrointestinal disorders
10/10/2006US7119083 novel 2-(azetidin-2-on-1-yl)alkanedioic acid esters and amides useful for treating disease states that are associated with and responsive to antagonism of a vasopressin V1a receptor in a mammal
10/10/2006US7118811 Materials for light emitting devices consisting of novel compounds and light emitting devices using the same
10/10/2006CA2418778C Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives
10/10/2006CA2274594C Aminopyrazole derivatives
10/10/2006CA2255951C Substituted 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators
10/10/2006CA2158862C Taxanes having alkoxy, alkenoxy or aryloxy substituted side-chain and pharmaceutical compositions containing same
10/05/2006WO2006105289A1 Bicyclic pyrazole compounds as antibacterial agents
10/05/2006WO2006105262A1 HETEROARYL UREA DERIVATIVES USEFUL FOR INHIBITING CHKl
10/05/2006WO2006104280A1 Prophylactic/therapeutic agent for diabetes
10/05/2006WO2006104141A1 3-propenylcephem derivative
10/05/2006WO2006104008A1 Urea derivative, medicinal composition containing the same, and medicinal use of these
10/05/2006WO2006103511A1 Cyclopentapyridine and tetrahydroquinoline derivatives
10/05/2006WO2006103277A2 2 , 4 , 5-substituted piperidines as renin inhibitors
10/05/2006WO2006103275A1 3,4,5-substituted piperidines as renin inhibitors
10/05/2006WO2006103273A1 Substituted piperidines as renin inhibitors
10/05/2006WO2006103120A2 New heterocyclic compounds, their preparation and their use as medicaments, in particular as anti-alzheimer agents
10/05/2006WO2006103057A1 Compounds comprising an oxazoline or thiazoline moiety, processes for making them, and their uses
10/05/2006WO2006103045A1 Compounds comprising an oxazole or thiazole moiety, processes for making them, and their uses
10/05/2006WO2006102760A1 Inhibitors of histone deacetylase
10/05/2006WO2006078621A3 2-phenoxy-n- (1, 3 , 4-thiadizol-2-yl) pyridin-3-amine derivatives and related compounds as p2y1 receptor inhibitors for the treatment of thromboembolic disorders
10/05/2006WO2006071609A3 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
10/05/2006WO2006059245A3 Compounds for the treatment of cns and amyloid associated diseases
10/05/2006WO2006058012A3 Gonadotropin releasing hormone receptor antagonists
10/05/2006WO2006047196A3 Cgrp receptor antagonists
10/05/2006WO2006044825A3 Mitotic kinesin inhibitors and methods of use thereof
10/05/2006WO2005115392A8 3-(4-heteroarylcyclohexylamino) cyclopentanecarboxamides as modulators of chemokine receptors
10/05/2006WO2004060308A3 Thiosemicarbazones as anti-virals and immunopotentiators
10/05/2006US20060223996 IL-12 modulatory compounds
10/05/2006US20060223890 N-arylsulfonyl-3-substituted indoles having serotonin receptor affinity, process for their preparation and pharmaceutical composition containing them
10/05/2006US20060223873 Isoxazole derivatives and methods of treating nitric oxide mediated diseases
10/05/2006US20060223850 8-(3-Biaryl)phenylquinoline phosphodiesterase-4 inhibitors
10/05/2006US20060223849 Benzazole derivatives, compositions, and methods of use as beta-secretase inhibitors
10/05/2006US20060223848 Caspase inhibitors containing isoxazoline ring
10/05/2006US20060223822 Dehydrophenylahistins and analogs thereof and the synthesis of dehydrophenylahistins and analogs thereof
10/05/2006US20060223808 Spirocyclic thrombin receptor antagonists
10/05/2006US20060223804 NK1 antagonists
10/05/2006US20060223802 Derivatives of N-[phenyl(pyrrolidine-2-yl)methyl]benzamide and N-[(azepan-2-yl)phenylmethyl]benzamide, preparation method thereof and application of same in therapeutics
10/05/2006US20060223801 Pyrrol derivatives with antibacterial activity
10/05/2006US20060223746 Injecting an alpha v beta 3 and/or alpha v beta 5 inhibitor, sufficient to inhibit or reduce angiogenesis or neovascularization in the treated eye, into the sclera layer of the eye; (2S)-2-benzyloxycarboxamido-3-(2-guanidinomethyl-1,4-benzodioxan-6-yl)propionic acid
10/05/2006US20060223151 Production of polyketides
10/05/2006US20060223076 Cyanine dyes and their applications as luminescence quenching compounds
10/05/2006DE102005000666B3 Sulfonylpyrrolidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Sulfonylpyrrolidine, processes for their preparation and their use as medicaments
10/05/2006CA2603589A1 Inhibitors of histone deacetylase
10/05/2006CA2603345A1 New heterocyclic compounds, their preparation and their use as medicaments, in particular as anti-alzheimer agents
10/05/2006CA2603322A1 Bicyclic pyrazole compounds as antibacterial agents
10/05/2006CA2602546A1 Novel compounds
10/05/2006CA2602351A1 Urea derivative, medicinal composition containing the same, and medicinal use of these
10/05/2006CA2602339A1 Compounds comprising an oxazoline or thiazoline moiety, processes for making them, and their uses
10/05/2006CA2602336A1 Compounds comprising an oxazole or thiazole moiety, processes for making them, and their uses
10/05/2006CA2602257A1 Alkynyl pyrrolopyrimidines and related analogs as hsp90-inhibitors
10/05/2006CA2602254A1 Pharmacokinetically improved compounds
10/05/2006CA2601702A1 2, 4, 5-substituted piperidines as renin inhibitors
10/05/2006CA2601699A1 Substituted piperidines
10/05/2006CA2601108A1 3,4,5-substituted piperidines as renin inhibitors
10/04/2006EP1706409A1 Compounds useful in therapy
10/04/2006EP1706402A1 Cathepsin cysteine protease inhibitors
10/04/2006EP1706398A1 Amino-benzazoles as p2y1 receptor inhibitors
10/04/2006EP1706396A1 N-(4-carbamimidoyl-benzyl)-2-alkoxy-2-heterocyclyl acetamides as inhibitors of the formation of coagulation factors xa, ixa and thrombin induced by factor viia
10/04/2006EP1706390A2 Isoxazole derivatives and their use as cyclooxygenase inhibitors
10/04/2006EP1706385A1 Pyrazole derivatives as protein kinase modulators
10/04/2006EP1706372A1 Alpha-hydroxy amides as bradykinin antagonists or inverse agonists
10/04/2006EP1706129A1 Drug therapy for celiac sprue
10/04/2006EP1705989A1 Substituted arylpyrazoles as parasiticidal agents
10/04/2006EP1377290B1 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
10/04/2006EP1372653B1 Acylated piperidine derivatives as melanocortin-4 receptor agonists
10/04/2006CN1842522A Benzothiazole-4,7-diones and benzoxazole-4,7-diones with substituents in position 5 or 6 and method for production thereof
10/04/2006CN1842521A Caspase inhibitors containing isoxazoline ring
10/04/2006CN1842336A Aryloxy and arylalkyleneoxy substituted imidazoquinolines
10/04/2006CN1842272A Hydrazone derivatives for combatting harmful insects and arachnids
10/04/2006CN1277829C 3, 5-disubstituted-oxazolidine with antibiotic activity, its preparation method and use
10/04/2006CN1277824C Piperazine derivatives
10/04/2006CN1277820C Phthalimido derivatives as inhibitors of monoamine oxidase B
10/03/2006US7115750 Melanin concentrating hormone antagonist
10/03/2006US7115739 Triazole compounds useful as protein kinase inhibitors
10/03/2006US7115658 Compounds of formula I are hepatitis C virus (HCV) RNA-dependent RNA polymerase (RdRp) inhibitors, and are useful in therapeutic and prophylactic treatment of persons infected with hepatitis C virus.
10/03/2006US7115654 Caspase-1 inhibitors and methods for their use